Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT197 | Protein-Protein Interaction | Menin/Histone-lysine N-methyltransferase MLL | Homo sapiens | Potency | = | 3981.1 | nM | PubChem BioAssay data set |
NPT533 | Protein-Protein Interaction | Runt-related transcription factor 1/Core-binding factor subunit beta | Homo sapiens | Potency | 35481.3 | nM | PubChem BioAssay data set | |
NPT49 | Individual Protein | DNA-(apurinic or apyrimidinic site) lyase | Homo sapiens | Potency | 5011.9 | nM | PubChem BioAssay data set |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC329496 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Natural Product ID |
---|---|---|
1.0 | High Similarity | NPC230452 |
0.92 | High Similarity | NPC317724 |
0.8519 | High Similarity | NPC238135 |
0.84 | Intermediate Similarity | NPC318912 |
0.84 | Intermediate Similarity | NPC237965 |
0.8077 | Intermediate Similarity | NPC304786 |
0.7778 | Intermediate Similarity | NPC128335 |
0.75 | Intermediate Similarity | NPC272307 |
0.68 | Remote Similarity | NPC43196 |
0.6667 | Remote Similarity | NPC149567 |
0.6538 | Remote Similarity | NPC321400 |
0.6486 | Remote Similarity | NPC152008 |
0.6389 | Remote Similarity | NPC197039 |
0.6207 | Remote Similarity | NPC140389 |
0.6176 | Remote Similarity | NPC227267 |
0.6129 | Remote Similarity | NPC301586 |
0.6129 | Remote Similarity | NPC33415 |
0.5946 | Remote Similarity | NPC473991 |
0.5926 | Remote Similarity | NPC61373 |
0.5862 | Remote Similarity | NPC114270 |
0.5862 | Remote Similarity | NPC157340 |
0.5833 | Remote Similarity | NPC103612 |
0.5833 | Remote Similarity | NPC24967 |
0.5833 | Remote Similarity | NPC313405 |
0.5806 | Remote Similarity | NPC320326 |
0.575 | Remote Similarity | NPC31121 |
0.5714 | Remote Similarity | NPC219266 |
0.5714 | Remote Similarity | NPC140229 |
0.5667 | Remote Similarity | NPC317545 |
0.5641 | Remote Similarity | NPC266553 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC329496 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
0.6667 | Remote Similarity | NPD7374 | Approved |
0.6486 | Remote Similarity | NPD7536 | Approved |
0.625 | Remote Similarity | NPD901 | Approved |
0.6129 | Remote Similarity | NPD8549 | Clinical (unspecified phase) |
0.5862 | Remote Similarity | NPD8226 | Approved |
0.5862 | Remote Similarity | NPD8225 | Phase 3 |
0.5625 | Remote Similarity | NPD30 | Approved |
0.5625 | Remote Similarity | NPD3216 | Phase 3 |
0.56 | Remote Similarity | NPD8547 | Phase 2 |
PubChem CID   | 17472 |
ChEMBL   | CHEMBL1235082 |
ZINC   |
Molecular Weight:   | 282.17 |
ALogP:   | -1.5519 |
MLogP:   | 2.01 |
XLogP:   | -2.158 |
# Rotatable Bonds:   | 18 |
Polar Surface Area:   | 86.61 |
# H-Bond Aceptor:   | 7 |
# H-Bond Donor:   | 2 |
# Rings:   | 0 |
# Heavy Atoms:   | 19 |