Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 15664814 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 15664814 |
NPT1062 | Individual Protein | Carbonic anhydrase IV | Homo sapiens | Ki | = | 5700000 | nM | 15664814 |
NPT1143 | Individual Protein | Carbonic anhydrase VA | Homo sapiens | Ki | = | 95000000 | nM | 15664814 |
NPT948 | Individual Protein | Carbonic anhydrase IX | Homo sapiens | Ki | = | 8600 | nM | 15664814 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 15357993 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 15357993 |
NPT1062 | Individual Protein | Carbonic anhydrase IV | Homo sapiens | Ki | = | 44000000 | nM | 15357993 |
NPT4793 | Individual Protein | Carbonic anhydrase | Methanosarcina thermophila | Ki | = | 42000000 | nM | 15357993 |
NPT1150 | Individual Protein | Carbonic anhydrase | Methanobacterium thermoautotrophicum | Ki | = | 44900000 | nM | 15357993 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 15357993 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 15357993 |
NPT4793 | Individual Protein | Carbonic anhydrase | Methanosarcina thermophila | Ki | = | 6700000 | nM | 15357993 |
NPT1150 | Individual Protein | Carbonic anhydrase | Methanobacterium thermoautotrophicum | Ki | = | 9600000 | nM | 15357993 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 15454240 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 15454240 |
NPT1060 | Protein Family | Carbonic anhydrase V | Homo sapiens | Ki | = | 82000000 | nM | 15454240 |
NPT1061 | Individual Protein | Carbonic anhydrase XIII | Mus musculus | Ki | = | 140000000 | nM | 15454240 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 15454240 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 15454240 |
NPT1060 | Protein Family | Carbonic anhydrase V | Homo sapiens | Ki | = | 95000000 | nM | 15454240 |
NPT1061 | Individual Protein | Carbonic anhydrase XIII | Mus musculus | Ki | = | 5500000 | nM | 15454240 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 15501038 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 15501038 |
NPT1062 | Individual Protein | Carbonic anhydrase IV | Homo sapiens | Ki | = | 6600000 | nM | 15501038 |
NPT1060 | Protein Family | Carbonic anhydrase V | Homo sapiens | Ki | = | 82000000 | nM | 15501038 |
NPT948 | Individual Protein | Carbonic anhydrase IX | Homo sapiens | Ki | = | 13000000 | nM | 15501038 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 15501038 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 15501038 |
NPT1062 | Individual Protein | Carbonic anhydrase IV | Homo sapiens | Ki | = | 5700000 | nM | 15501038 |
NPT1060 | Protein Family | Carbonic anhydrase V | Homo sapiens | Ki | = | 95000000 | nM | 15501038 |
NPT955 | Individual Protein | Carbonic anhydrase VII | Homo sapiens | Ki | = | 270000 | nM | 16621537 |
NPT955 | Individual Protein | Carbonic anhydrase VII | Homo sapiens | Ki | = | 160000 | nM | 16621537 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 21208801 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 21208801 |
NPT1063 | Individual Protein | Carbonic anhydrase VI | Homo sapiens | Ki | = | 800000 | nM | 21208801 |
NPT1064 | Individual Protein | Alpha carbonic anhydrase | Stylophora pistillata | Ki | = | 450000 | nM | 21208801 |
NPT1065 | Individual Protein | Carbonic anhydrase | Stylophora pistillata | Ki | = | 7810000 | nM | 21208801 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 21208801 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 21208801 |
NPT1063 | Individual Protein | Carbonic anhydrase VI | Homo sapiens | Ki | = | 690000 | nM | 21208801 |
NPT1064 | Individual Protein | Alpha carbonic anhydrase | Stylophora pistillata | Ki | = | 10000 | nM | 21208801 |
NPT1065 | Individual Protein | Carbonic anhydrase | Stylophora pistillata | Ki | = | 240000 | nM | 21208801 |
NPT2 | Others | Unspecified | Ki | = | 750000 | nM | 23078755 | |
NPT2 | Others | Unspecified | Ki | = | 15700000 | nM | 23078755 | |
NPT2 | Others | Unspecified | Ki | = | 33200000 | nM | 23078755 | |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 23078755 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 26525863 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 26525863 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 26525863 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 26525863 |
NPT2 | Others | Unspecified | Ki | = | 730000 | nM | 26525863 | |
NPT2 | Others | Unspecified | Ki | = | 1020000 | nM | 26525863 | |
NPT2 | Others | Unspecified | Ki | = | 6700000 | nM | 26853167 | |
NPT2 | Others | Unspecified | Ki | = | 5900000 | nM | 26853167 | |
NPT2 | Others | Unspecified | Ki | = | 4640000 | nM | 26853167 | |
NPT2 | Others | Unspecified | Ki | = | 5130000 | nM | 26853167 | |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 26853167 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 26853167 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 26853167 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 26853167 |
NPT2 | Others | Unspecified | Ki | = | 5900000 | nM | 27283786 | |
NPT2 | Others | Unspecified | Ki | = | 6700000 | nM | 27283786 | |
NPT2 | Others | Unspecified | Ki | = | 4640000 | nM | 27283786 | |
NPT2 | Others | Unspecified | Ki | = | 5130000 | nM | 27283786 | |
NPT2 | Others | Unspecified | Ki | = | 660000 | nM | 27283786 | |
NPT2 | Others | Unspecified | Ki | = | 750000 | nM | 27283786 | |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 73000000 | nM | 27283786 |
NPT233 | Individual Protein | Carbonic anhydrase II | Homo sapiens | Ki | = | 85000000 | nM | 27283786 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 15000000 | nM | 27283786 |
NPT947 | Individual Protein | Carbonic anhydrase I | Homo sapiens | Ki | = | 12000000 | nM | 27283786 |
NPT2 | Others | Unspecified | Ki | = | 3000000 | nM | 27283786 | |
NPT2 | Others | Unspecified | Ki | = | 8200000 | nM | 27283786 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC327795 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC327795 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
1.0 | High Similarity | NPD9749 | Approved |
1.0 | High Similarity | NPD9746 | Approved |
1.0 | High Similarity | NPD9748 | Approved |
0.75 | Intermediate Similarity | NPD9736 | Approved |
0.75 | Intermediate Similarity | NPD9737 | Approved |
0.75 | Intermediate Similarity | NPD9750 | Approved |
0.75 | Intermediate Similarity | NPD9740 | Approved |
0.75 | Intermediate Similarity | NPD9739 | Approved |
0.75 | Intermediate Similarity | NPD9743 | Approved |
0.75 | Intermediate Similarity | NPD9742 | Approved |
0.75 | Intermediate Similarity | NPD9738 | Approved |
0.75 | Intermediate Similarity | NPD9744 | Approved |
0.75 | Intermediate Similarity | NPD113 | Approved |
0.75 | Intermediate Similarity | NPD9745 | Approved |
0.75 | Intermediate Similarity | NPD9747 | Approved |
0.75 | Intermediate Similarity | NPD9741 | Approved |
0.5714 | Remote Similarity | NPD9752 | Clinical (unspecified phase) |
PubChem CID   | 767;3614646;22639876 |
ChEMBL   | CHEMBL1161632 |
ZINC   |
Molecular Weight:   | 62.00 |
ALogP:   | 0.1623 |
MLogP:   | 1.24 |
XLogP:   | -0.23 |
# Rotatable Bonds:   | 2 |
Polar Surface Area:   | 57.53 |
# H-Bond Aceptor:   | 3 |
# H-Bond Donor:   | 2 |
# Rings:   | 0 |
# Heavy Atoms:   | 4 |