Target ID |
Target Type |
Target Name |
Target Organism |
Activity Type |
Activity Relation |
Value |
Unit |
Reference |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
150000 |
nM |
9301668 |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
140000 |
nM |
9301668 |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
30000 |
nM |
9767632 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
CC50 |
= |
7400 |
nM |
9767632 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
CC50 |
= |
16000 |
nM |
9767632 |
NPT319 |
Cell Line |
B16 |
Mus musculus |
Inhibition |
= |
87 |
% |
14643343 |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
57500 |
nM |
10969990 |
NPT681 |
Cell Line |
PC-12 |
Rattus norvegicus |
ED50 |
= |
7.1 |
ug/ml |
11549465 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
ED50 |
= |
7.4 |
ug/ml |
11549465 |
NPT12 |
Individual Protein |
Human immunodeficiency virus type 1 integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
30199.52 |
nM |
11831895 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
71.2 |
% |
9871681 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
63.4 |
% |
9871681 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
-44.3 |
% |
9871681 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
98.8 |
% |
9871681 |
NPT681 |
Cell Line |
PC-12 |
Rattus norvegicus |
ED50 |
= |
17.1 |
nM |
14980683 |
NPT744 |
Cell Line |
IMR-32 |
Homo sapiens |
ED50 |
= |
23.9 |
nM |
14980683 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
IC50 |
= |
10.84 |
ug/ml |
15993583 |
NPT324 |
Individual Protein |
Cyclooxygenase-1 |
Ovis aries |
Inhibition |
= |
80.5 |
% |
15780608 |
NPT325 |
Individual Protein |
Cyclooxygenase-2 |
Ovis aries |
Inhibition |
= |
35 |
% |
15780608 |
NPT4243 |
Individual Protein |
Cyclooxygenase-2 |
Rattus norvegicus |
Inhibition |
= |
61.4 |
% |
15780608 |
NPT31 |
Individual Protein |
Cyclooxygenase-2 |
Homo sapiens |
IC50 |
= |
11060 |
nM |
15780608 |
NPT29 |
Organism |
Rattus norvegicus |
Rattus norvegicus |
Inhibition |
= |
80 |
% |
15878268 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
3800 |
nM |
16789753 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
7700 |
nM |
16789753 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Ki |
= |
0.208 |
nM |
17004725 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Activity |
= |
17.5 |
% |
17154519 |
NPT4244 |
Individual Protein |
RmtA |
Emericella nidulans |
IC50 |
= |
1100000 |
nM |
17323938 |
NPT4245 |
Individual Protein |
Protein-arginine N-methyltransferase 1 |
Homo sapiens |
IC50 |
= |
1070000 |
nM |
17323938 |
NPT1079 |
Individual Protein |
Histone acetyltransferase p300 |
Homo sapiens |
IC50 |
> |
400000 |
nM |
17348637 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
24690 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC90 |
= |
44450 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
22930 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC90 |
= |
41270 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
27450 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC90 |
= |
49420 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
29610 |
nM |
17145789 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC90 |
= |
53290 |
nM |
17145789 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
48000 |
nM |
17145789 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
95 |
% |
17145789 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
10000 |
nM |
17049256 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
0 |
% |
17503850 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
22.8 |
% |
17503850 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
81.7 |
% |
17503850 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
100 |
% |
17503850 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
IC50 |
= |
10.2 |
nM |
17503850 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
= |
60 |
% |
17503850 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
ED50 |
= |
0.75 |
ug/ml |
17643301 |
NPT1515 |
Organism |
SARS coronavirus |
SARS coronavirus |
EC50 |
> |
10000 |
nM |
17663539 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
CC50 |
> |
250000 |
nM |
17663539 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40000 |
nM |
17663539 |
NPT1515 |
Organism |
SARS coronavirus |
SARS coronavirus |
Inhibition |
= |
25 |
% |
17663539 |
NPT1515 |
Organism |
SARS coronavirus |
SARS coronavirus |
Inhibition |
= |
50 |
% |
17663539 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
0 |
% |
17316910 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
22.8 |
% |
17316910 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
81.7 |
% |
17316910 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
Inhibition |
= |
100 |
% |
17316910 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
= |
60 |
% |
17316910 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Survival |
> |
80 |
% |
17316910 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
EC50 |
= |
35000 |
nM |
17383188 |
NPT164 |
Organism |
Human herpesvirus 4 |
Human herpesvirus 4 |
IC50 |
= |
345000 |
nM |
17950604 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
65 |
% |
17973470 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Activity |
= |
90 |
% |
17973470 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
17973470 |
NPT4246 |
Cell Line |
LS174T |
Homo sapiens |
IC50 |
= |
6500 |
nM |
17973470 |
NPT783 |
Cell Line |
MIA PaCa-2 |
Homo sapiens |
IC50 |
= |
9000 |
nM |
17973470 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
2900 |
nM |
17973470 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
IC50 |
= |
800 |
nM |
17270435 |
NPT804 |
Cell Line |
HT-22 |
Mus musculus |
Activity |
= |
116 |
% |
17270435 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
9000 |
nM |
17768050 |
NPT404 |
Cell Line |
CCRF-CEM |
Homo sapiens |
IC50 |
= |
8700 |
nM |
17768050 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
0 |
% |
17685651 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
= |
70 |
% |
17685651 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
22.8 |
% |
17685651 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
81.8 |
% |
17685651 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
100 |
% |
17685651 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
6810 |
nM |
18076140 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17400 |
nM |
18039573 |
NPT2 |
Others |
Unspecified |
|
IC70 |
= |
24.6 |
nM |
18039573 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
29300 |
nM |
18039573 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC70 |
= |
51.7 |
nM |
18039573 |
NPT4247 |
Cell Line |
MCF7R |
Homo sapiens |
IC50 |
= |
26200 |
nM |
18039573 |
NPT4247 |
Cell Line |
MCF7R |
Homo sapiens |
IC70 |
= |
46.2 |
nM |
18039573 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
45 |
% |
18042380 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
10000 |
nM |
18042380 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
29 |
% |
17284452 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
361110 |
nM |
17284452 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
59.32 |
% |
18024584 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
228.38 |
% |
18024584 |
NPT1892 |
Cell Line |
H4 |
Rattus norvegicus |
Activity |
= |
249.22 |
% |
18024584 |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
8000 |
nM |
18077363 |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
IC50 |
= |
52000 |
nM |
18077363 |
NPT3517 |
Individual Protein |
Nitric oxide synthase, inducible |
Homo sapiens |
IC50 |
= |
6000 |
nM |
18077363 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3250 |
nM |
18194869 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
MIC |
= |
13200 |
nM |
18194869 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
MIC |
= |
14400 |
nM |
18194869 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
4210 |
nM |
18194869 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
Activity |
= |
89.2 |
% |
18295490 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
93.1 |
% |
18295490 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
820 |
nM |
18295490 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
420 |
nM |
18295490 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Activity |
= |
25 |
% |
18348515 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Activity |
= |
8.5 |
% |
18348515 |
NPT466 |
Cell Line |
U-937 |
Homo sapiens |
Activity |
= |
25.3 |
% |
18348515 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
46 |
% |
18434144 |
NPT521 |
Cell Line |
RBL-2H3 |
Rattus norvegicus |
Inhibition |
= |
62.6 |
% |
12398545 |
NPT521 |
Cell Line |
RBL-2H3 |
Rattus norvegicus |
Inhibition |
= |
14.2 |
% |
12398545 |
NPT521 |
Cell Line |
RBL-2H3 |
Rattus norvegicus |
Inhibition |
= |
2 |
% |
12398545 |
NPT521 |
Cell Line |
RBL-2H3 |
Rattus norvegicus |
IC50 |
= |
3000 |
nM |
12398545 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
23.2 |
nM |
11430002 |
NPT453 |
Cell Line |
HT-1080 |
Homo sapiens |
ED50 |
= |
23.4 |
nM |
11430002 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
38300 |
nM |
18678491 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4200 |
nM |
18678491 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
IZ |
= |
10 |
mm |
18201805 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
= |
20000000 |
nM |
18201805 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
IZ |
= |
15 |
mm |
18201805 |
NPT212 |
Individual Protein |
Cytochrome P450 2C9 |
Homo sapiens |
IC50 |
= |
4300 |
nM |
18249473 |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
IC50 |
= |
16300 |
nM |
18249473 |
NPT208 |
Individual Protein |
Cytochrome P450 1A2 |
Homo sapiens |
IC50 |
= |
40000 |
nM |
18249473 |
NPT627 |
Individual Protein |
Cytochrome P450 2B6 |
Homo sapiens |
IC50 |
= |
24500 |
nM |
18249473 |
NPT110 |
Individual Protein |
Cytochrome P450 2D6 |
Homo sapiens |
IC50 |
= |
50300 |
nM |
18249473 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
2110 |
nM |
19019687 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
5580 |
nM |
19019687 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
58.4 |
% |
19179077 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
7480 |
nM |
19179077 |
NPT1821 |
Individual Protein |
Sortase |
Staphylococcus aureus |
IC50 |
= |
13.8 |
ug/ml |
19269184 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
19800 |
nM |
19249204 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
19600 |
nM |
19249204 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
21500 |
nM |
19249204 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
25600 |
nM |
19249204 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1020 |
nM |
9599258 |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
IC50 |
= |
8800 |
nM |
16038536 |
NPT377 |
Cell Line |
OVCAR-3 |
Homo sapiens |
CD50 |
= |
4.4 |
ug/ml |
9868158 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
18419109 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
45.1 |
% |
19131254 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
19131254 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
22.8 |
% |
19131254 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
81.7 |
% |
19131254 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
19131254 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
331000 |
nM |
19131254 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
= |
60 |
% |
19131254 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
> |
80 |
% |
19131254 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
45 |
% |
19334715 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
19334715 |
NPT547 |
Cell Line |
BGC-823 |
Homo sapiens |
IC50 |
= |
16700 |
nM |
19243951 |
NPT3887 |
Cell Line |
CNE |
Homo sapiens |
IC50 |
= |
32800 |
nM |
19243951 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
11600 |
nM |
19243951 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
35900 |
nM |
19243951 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6400 |
nM |
19243951 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
19243951 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
17500 |
nM |
19243951 |
NPT35 |
Others |
n.a. |
|
Activity |
> |
64 |
% |
19243951 |
NPT35 |
Others |
n.a. |
|
Activity |
= |
92 |
% |
19243951 |
NPT1719 |
Cell Line |
2008 |
Homo sapiens |
Activity |
> |
90 |
% |
19329324 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
60 |
% |
19329324 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Activity |
> |
25 |
% |
19329324 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Activity |
= |
10 |
% |
19329324 |
NPT1719 |
Cell Line |
2008 |
Homo sapiens |
IC50 |
= |
5000 |
nM |
19329324 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17000 |
nM |
19329324 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Ratio IC50 |
= |
1.3 |
|
19329324 |
NPT1719 |
Cell Line |
2008 |
Homo sapiens |
Ratio IC50 |
= |
3.4 |
|
19329324 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
22000 |
nM |
19329324 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
IC50 |
= |
800 |
nM |
18793854 |
NPT1649 |
Cell Line |
MV4-11 |
Homo sapiens |
Activity |
= |
15 |
% |
19112019 |
NPT3701 |
Individual Protein |
CpG DNA methylase |
Spiroplasma monobiae |
IC50 |
= |
30 |
nM |
19112019 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
150000 |
nM |
19114310 |
NPT4248 |
Individual Protein |
Histone acetyltransferase KAT5 |
Homo sapiens |
IC50 |
> |
200000 |
nM |
19114310 |
NPT1079 |
Individual Protein |
Histone acetyltransferase p300 |
Homo sapiens |
IC50 |
> |
40000 |
nM |
19114310 |
NPT280 |
Individual Protein |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50 |
= |
8500 |
nM |
19128977 |
NPT1090 |
Individual Protein |
Matrix metalloproteinase 13 |
Homo sapiens |
IC50 |
= |
10300 |
nM |
18358729 |
NPT2 |
Others |
Unspecified |
|
Kd |
= |
1150 |
nM |
19329310 |
NPT2 |
Others |
Unspecified |
|
Kd |
= |
2450 |
nM |
19329310 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
15000 |
nM |
19329310 |
NPT681 |
Cell Line |
PC-12 |
Rattus norvegicus |
ED50 |
= |
7 |
ug/ml |
12350137 |
NPT681 |
Cell Line |
PC-12 |
Rattus norvegicus |
ED50 |
= |
10 |
ug/ml |
12350137 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
5.5 |
ug/ml |
17067159 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
3.1 |
ug/ml |
17067159 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
5.2 |
ug/ml |
17067159 |
NPT23 |
Individual Protein |
Integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
51.3 |
ug/ml |
16643034 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
96.5 |
% |
16038556 |
NPT116 |
Cell Line |
HL-60 |
Homo sapiens |
IC50 |
= |
34220 |
nM |
16038556 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
35530 |
nM |
16038556 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
10440 |
nM |
16038556 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
20600 |
nM |
16038556 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
27600 |
nM |
16038556 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Inhibition |
= |
10 |
% |
18439726 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Inhibition |
= |
20 |
% |
18439726 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
19481937 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
22.8 |
% |
19481937 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
81.7 |
% |
19481937 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
19481937 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
341 |
molar ratio |
19481937 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
= |
60 |
% |
19481937 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
> |
80 |
% |
19481937 |
NPT1310 |
Individual Protein |
Xanthine dehydrogenase |
Bos taurus |
Activity |
= |
160 |
nM/s |
19388706 |
NPT1310 |
Individual Protein |
Xanthine dehydrogenase |
Bos taurus |
Activity |
= |
150 |
nM/s |
19388706 |
NPT1310 |
Individual Protein |
Xanthine dehydrogenase |
Bos taurus |
Inhibition |
= |
60 |
% |
19388706 |
NPT1310 |
Individual Protein |
Xanthine dehydrogenase |
Bos taurus |
Inhibition |
> |
20 |
% |
19388706 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
8500 |
nM |
19725582 |
NPT1629 |
Cell Line |
CWR22R |
Homo sapiens |
IC50 |
= |
18300 |
nM |
19725582 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6100 |
nM |
19725582 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
16800 |
nM |
19725582 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
29500 |
nM |
19725582 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
20380 |
nM |
19359068 |
NPT35 |
Others |
n.a. |
|
IC50 |
> |
500000 |
nM |
19359068 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
109740 |
nM |
19359068 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
13000 |
nM |
19854644 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
950 |
nM |
19842664 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
10 |
nM |
19842664 |
NPT664 |
Protein Family |
Histone deacetylase |
Homo sapiens |
Activity |
= |
52 |
% |
19520580 |
NPT664 |
Protein Family |
Histone deacetylase |
Homo sapiens |
Ki |
= |
539 |
nM |
19520580 |
NPT664 |
Protein Family |
Histone deacetylase |
Homo sapiens |
IC50 |
= |
115000 |
nM |
19520580 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
8.9 |
% |
19674905 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
40.3 |
% |
19674905 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
74.5 |
% |
19674905 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
95.8 |
% |
19674905 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
345000 |
nM |
19674905 |
NPT80 |
Cell Line |
Raji |
Homo sapiens |
Activity |
= |
60 |
% |
19674905 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
Inhibition |
= |
25 |
% |
19775895 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
Inhibition |
= |
47 |
% |
19775895 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
Inhibition |
= |
52 |
% |
19775895 |
NPT1460 |
Cell Line |
L929 |
Mus musculus |
IC50 |
= |
20000 |
nM |
19775895 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
Inhibition |
= |
90 |
% |
19674910 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
2.1 |
|
19646881 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC90 |
= |
73.7 |
ug/ml |
19959361 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC90 |
> |
500 |
ug/ml |
19959361 |
NPT1573 |
Individual Protein |
Enoyl-[acyl-carrier-protein] reductase |
Escherichia coli K-12 |
Ki |
= |
14960 |
nM |
19959361 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
Ratio |
= |
7 |
|
19959361 |
NPT579 |
Cell Line |
DLD-1 |
Homo sapiens |
GI50 |
= |
8000 |
nM |
20060305 |
NPT881 |
Individual Protein |
Protein kinase C delta |
Homo sapiens |
EC50 |
= |
10670 |
nM |
20100661 |
NPT761 |
Individual Protein |
Protein kinase C epsilon |
Homo sapiens |
EC50 |
= |
8810 |
nM |
20100661 |
NPT887 |
Individual Protein |
Protein kinase C theta |
Homo sapiens |
EC50 |
= |
11080 |
nM |
20100661 |
NPT2752 |
Individual Protein |
DNA (cytosine-5)-methyltransferase 1 |
Homo sapiens |
Inhibition |
= |
66 |
% |
20006515 |
NPT3537 |
Individual Protein |
DNA (cytosine-5)-methyltransferase 3B |
Homo sapiens |
Inhibition |
= |
80 |
% |
20006515 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
23500 |
nM |
20167482 |
NPT338 |
Organism |
Sindbis virus |
Sindbis virus |
EC50 |
> |
10 |
nM |
20034711 |
NPT335 |
Organism |
Human coxsackievirus B4 |
Human coxsackievirus B4 |
EC50 |
> |
10 |
nM |
20034711 |
NPT341 |
Organism |
Punta Toro virus |
Punta Toro virus |
EC50 |
> |
10 |
nM |
20034711 |
NPT342 |
Organism |
Feline coronavirus |
Feline coronavirus |
EC50 |
> |
271 |
nM |
20034711 |
NPT343 |
Organism |
Felid herpesvirus 1 |
Felid herpesvirus 1 |
EC50 |
> |
271 |
nM |
20034711 |
NPT742 |
Organism |
Influenza A virus |
Influenza A virus |
EC50 |
> |
271 |
nM |
20034711 |
NPT4249 |
Organism |
Influenza B virus |
Influenza B virus |
EC50 |
> |
271 |
nM |
20034711 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
CC50 |
>= |
10 |
nM |
20034711 |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
CC50 |
>= |
10 |
nM |
20034711 |
NPT2192 |
Cell Line |
HEL |
Homo sapiens |
CC50 |
> |
2 |
nM |
20034711 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
CC50 |
= |
54 |
nM |
20034711 |
NPT616 |
Cell Line |
MDCK |
Canis lupus familiaris |
CC50 |
> |
92 |
nM |
20034711 |
NPT24 |
Organism |
Human immunodeficiency virus 1 |
Human immunodeficiency virus 1 |
IC50 |
= |
37 |
nM |
20034711 |
NPT3795 |
Organism |
Human immunodeficiency virus 2 |
Human immunodeficiency virus 2 |
IC50 |
= |
37 |
nM |
20034711 |
NPT25 |
Cell Line |
MT4 |
Homo sapiens |
CC50 |
> |
37 |
nM |
20034711 |
NPT2 |
Others |
Unspecified |
|
Ratio CC50/IC50 |
< |
1 |
|
20034711 |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
EC50 |
= |
2500 |
nM |
20004045 |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
EC50 |
= |
4700 |
nM |
20004045 |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
EC50 |
= |
2900 |
nM |
20004045 |
NPT841 |
Organism |
Leishmania major |
Leishmania major |
EC50 |
= |
33000 |
nM |
20004045 |
NPT842 |
Organism |
Leishmania mexicana |
Leishmania mexicana |
EC50 |
= |
16000 |
nM |
20004045 |
NPT71 |
Cell Line |
HEK293 |
Homo sapiens |
EC50 |
= |
37000 |
nM |
20004045 |
NPT843 |
Organism |
Trypanosoma evansi |
Trypanosoma evansi |
EC50 |
= |
2000 |
nM |
20004045 |
NPT471 |
Organism |
Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
EC50 |
= |
4800 |
nM |
20004045 |
NPT3843 |
Organism |
Streptococcus viridans |
Streptococcus viridans |
MIC |
= |
2470 |
nM |
20034711 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
= |
1230 |
nM |
20034711 |
NPT173 |
Organism |
Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
= |
1230 |
nM |
20034711 |
NPT172 |
Organism |
Proteus mirabilis |
Proteus mirabilis |
MIC |
= |
1230 |
nM |
20034711 |
NPT195 |
Organism |
Vesicular stomatitis virus |
Vesicular stomatitis virus |
EC50 |
> |
10 |
nM |
20034711 |
NPT70 |
Organism |
Respiratory syncytial virus |
Respiratory syncytial virus |
EC50 |
> |
10 |
nM |
20034711 |
NPT190 |
Organism |
Human herpesvirus 1 |
Human herpesvirus 1 |
EC50 |
> |
10 |
nM |
20034711 |
NPT1141 |
Organism |
Human herpesvirus 2 |
Human herpesvirus 2 |
EC50 |
= |
10 |
nM |
20034711 |
NPT334 |
Organism |
Vaccinia virus |
Vaccinia virus |
EC50 |
= |
10 |
nM |
20034711 |
NPT195 |
Organism |
Vesicular stomatitis virus |
Vesicular stomatitis virus |
EC50 |
= |
10 |
nM |
20034711 |
NPT190 |
Organism |
Human herpesvirus 1 |
Human herpesvirus 1 |
EC50 |
= |
10 |
nM |
20034711 |
NPT336 |
Organism |
Human parainfluenza virus 3 |
Human parainfluenza virus 3 |
EC50 |
> |
10 |
nM |
20034711 |
NPT3878 |
Organism |
Mammalian orthoreovirus 1 |
Mammalian orthoreovirus 1 |
EC50 |
> |
10 |
nM |
20034711 |
NPT23 |
Individual Protein |
Integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
40000 |
nM |
19813754 |
NPT23 |
Individual Protein |
Integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
30000 |
nM |
19813754 |
NPT202 |
Individual Protein |
Protease |
Human immunodeficiency virus 1 |
IC50 |
= |
100000 |
nM |
19813754 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
250000 |
nM |
19813754 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
81.1 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
92.4 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
91 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
92.9 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
96.8 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
59 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
99 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
94.5 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
31.9 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
41 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
53.3 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
89 |
% |
19653644 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
92 |
% |
19653644 |
NPT4250 |
Individual Protein |
Potassium channel subfamily K member 2 |
Bos taurus |
IC50 |
= |
930 |
nM |
19653644 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
2 |
|
19653644 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
8300 |
nM |
19778086 |
NPT848 |
Cell Line |
N9 |
Homo sapiens |
Inhibition |
= |
86.6 |
% |
19691309 |
NPT848 |
Cell Line |
N9 |
Homo sapiens |
Inhibition |
= |
75.6 |
% |
19691309 |
NPT848 |
Cell Line |
N9 |
Homo sapiens |
Inhibition |
= |
56.1 |
% |
19691309 |
NPT848 |
Cell Line |
N9 |
Homo sapiens |
Inhibition |
= |
35.2 |
% |
19691309 |
NPT848 |
Cell Line |
N9 |
Homo sapiens |
IC50 |
= |
13500 |
nM |
19691309 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
36 |
% |
20346654 |
NPT906 |
Individual Protein |
Testosterone 17-beta-dehydrogenase 3 |
Rattus norvegicus |
IC50 |
= |
9000 |
nM |
20346654 |
NPT906 |
Individual Protein |
Testosterone 17-beta-dehydrogenase 3 |
Rattus norvegicus |
IC50 |
= |
2300 |
nM |
20346654 |
NPT958 |
Individual Protein |
Estradiol 17-beta-dehydrogenase 3 |
Homo sapiens |
IC50 |
= |
67300 |
nM |
20346654 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
30 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
78 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
127 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
40 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
65 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
50 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
45 |
% |
20227282 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
75700 |
nM |
20297825 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
51500 |
nM |
20297825 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
43800 |
nM |
20297825 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
22700 |
nM |
20297825 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
48600 |
nM |
20297825 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
24.15 |
% |
20170988 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
79.9 |
% |
20170988 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
7.3 |
% |
20170988 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1.89 |
% |
20170988 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
45 |
% |
20452207 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
10000 |
nM |
20452207 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
24000 |
nM |
20466556 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
22000 |
nM |
20466556 |
NPT1125 |
Cell Line |
T98G |
Homo sapiens |
IC50 |
= |
25000 |
nM |
20466556 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18000 |
nM |
20466556 |
NPT169 |
Cell Line |
B16-F10 |
Mus musculus |
IC50 |
= |
10000 |
nM |
20466556 |
NPT2337 |
Cell Line |
OE33 |
Homo sapiens |
IC50 |
= |
35000 |
nM |
20466556 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
27000 |
nM |
20466556 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
33000 |
nM |
20466556 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
24000 |
nM |
20466556 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
27000 |
nM |
20466556 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
IC50 |
= |
1210 |
nM |
20561785 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
4.2 |
ug/ml |
19299148 |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
= |
3.5 |
ug/ml |
19299148 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
15000 |
nM |
20728364 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
EC50 |
= |
7600 |
nM |
20728364 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
EC50 |
= |
9700 |
nM |
20728364 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
2400 |
nM |
20728364 |
NPT947 |
Individual Protein |
Carbonic anhydrase I |
Homo sapiens |
Ki |
= |
2410 |
nM |
20674354 |
NPT233 |
Individual Protein |
Carbonic anhydrase II |
Homo sapiens |
Ki |
= |
380 |
nM |
20674354 |
NPT1146 |
Individual Protein |
Carbonic anhydrase III |
Homo sapiens |
Ki |
= |
11300 |
nM |
20674354 |
NPT1062 |
Individual Protein |
Carbonic anhydrase IV |
Homo sapiens |
Ki |
= |
4970 |
nM |
20674354 |
NPT1143 |
Individual Protein |
Carbonic anhydrase VA |
Homo sapiens |
Ki |
= |
10250 |
nM |
20674354 |
NPT1144 |
Individual Protein |
Carbonic anhydrase VB |
Homo sapiens |
Ki |
= |
9460 |
nM |
20674354 |
NPT1063 |
Individual Protein |
Carbonic anhydrase VI |
Homo sapiens |
Ki |
= |
9940 |
nM |
20674354 |
NPT955 |
Individual Protein |
Carbonic anhydrase VII |
Homo sapiens |
Ki |
= |
9300 |
nM |
20674354 |
NPT948 |
Individual Protein |
Carbonic anhydrase IX |
Homo sapiens |
Ki |
= |
4050 |
nM |
20674354 |
NPT949 |
Individual Protein |
Carbonic anhydrase XII |
Homo sapiens |
Ki |
= |
3480 |
nM |
20674354 |
NPT3101 |
Individual Protein |
Carbonic anhydrase XIII |
Homo sapiens |
Ki |
= |
6850 |
nM |
20674354 |
NPT954 |
Individual Protein |
Carbonic anhydrase XIV |
Homo sapiens |
Ki |
= |
11730 |
nM |
20674354 |
NPT1147 |
Individual Protein |
Carbonic anhydrase 15 |
Mus musculus |
Ki |
= |
5090 |
nM |
20674354 |
NPT4251 |
Individual Protein |
Cell division protein ftsZ |
Bacillus subtilis (strain 168) |
IC50 |
= |
30000 |
nM |
20615583 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
24460 |
nM |
20805034 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
FC |
= |
4 |
|
20805034 |
NPT115 |
Organism |
Mycobacterium tuberculosis H37Ra |
Mycobacterium tuberculosis H37Ra |
MIC |
= |
100 |
ug/ml |
20691508 |
NPT492 |
Cell Line |
Caco-2 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
20831222 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
12800 |
nM |
20831222 |
NPT76 |
Cell Line |
C6 |
Rattus norvegicus |
IC50 |
= |
16100 |
nM |
20831222 |
NPT941 |
Cell Line |
HaCaT |
Homo sapiens |
IC50 |
= |
21900 |
nM |
20831222 |
NPT886 |
Cell Line |
NIH3T3 |
Mus musculus |
IC50 |
= |
14200 |
nM |
20831222 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
< |
10 |
% |
20951593 |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT149 |
Individual Protein |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT48 |
Individual Protein |
Lysine-specific demethylase 4D-like |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT1038 |
Individual Protein |
Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
44668.4 |
nM |
PubChem BioAssay data set |
NPT50 |
Individual Protein |
Tyrosyl-DNA phosphodiesterase 1 |
Homo sapiens |
Potency |
= |
5623.4 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
28183.8 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
39810.7 |
nM |
PubChem BioAssay data set |
NPT791 |
Individual Protein |
Cruzipain |
Trypanosoma cruzi |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
7079.5 |
nM |
PubChem BioAssay data set |
NPT51 |
Individual Protein |
Microtubule-associated protein tau |
Homo sapiens |
Potency |
= |
3162.3 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
22387.2 |
nM |
PubChem BioAssay data set |
NPT94 |
Individual Protein |
Aldehyde dehydrogenase 1A1 |
Homo sapiens |
Potency |
= |
19952.6 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
14581 |
nM |
PubChem BioAssay data set |
NPT3 |
Individual Protein |
Thioredoxin glutathione reductase |
Schistosoma mansoni |
Potency |
= |
12589.3 |
nM |
PubChem BioAssay data set |
NPT792 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT282 |
Individual Protein |
MAP kinase ERK2 |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT2930 |
Individual Protein |
Hemoglobin beta chain |
Homo sapiens |
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT197 |
Protein-Protein Interaction |
Menin/Histone-lysine N-methyltransferase MLL |
Homo sapiens |
Potency |
= |
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
= |
31622.8 |
nM |
PubChem BioAssay data set |
NPT45 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 2 |
Homo sapiens |
Potency |
= |
10000 |
nM |
PubChem BioAssay data set |
NPT151 |
Individual Protein |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Homo sapiens |
Potency |
= |
22387.2 |
nM |
PubChem BioAssay data set |
NPT531 |
Individual Protein |
Nuclear receptor ROR-gamma |
Mus musculus |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
= |
15848.9 |
nM |
PubChem BioAssay data set |
NPT109 |
Individual Protein |
Cytochrome P450 3A4 |
Homo sapiens |
Potency |
= |
25118.9 |
nM |
PubChem BioAssay data set |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
35.6 |
% |
20934787 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
75.7 |
% |
20934787 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
96.8 |
% |
21190861 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
35 |
% |
21190861 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
106 |
% |
21190861 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
51.77 |
% |
21211982 |
NPT323 |
Cell Line |
SW-620 |
Homo sapiens |
GI50 |
= |
32000 |
nM |
21183341 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9600 |
nM |
21112783 |
NPT451 |
Organism |
Helicobacter pylori |
Helicobacter pylori |
MIC |
= |
5 |
ug/ml |
19204190 |
NPT451 |
Organism |
Helicobacter pylori |
Helicobacter pylori |
MIC |
= |
15 |
ug/ml |
19204190 |
NPT451 |
Organism |
Helicobacter pylori |
Helicobacter pylori |
MIC |
= |
50 |
ug/ml |
19204190 |
NPT2 |
Others |
Unspecified |
|
MIC |
= |
20 |
ug/ml |
19204190 |
NPT451 |
Organism |
Helicobacter pylori |
Helicobacter pylori |
MIC |
= |
30 |
ug/ml |
19204190 |
NPT3704 |
Individual Protein |
Multidrug resistance protein CDR1 |
Candida albicans |
IC50 |
= |
14200 |
nM |
19470507 |
NPT3704 |
Individual Protein |
Multidrug resistance protein CDR1 |
Candida albicans |
IC50 |
= |
40000 |
nM |
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
IC50 |
= |
421600 |
nM |
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
IC50 |
= |
492800 |
nM |
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
IC50 |
= |
410600 |
nM |
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
IC50 |
= |
498000 |
nM |
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
IC50 |
= |
454600 |
nM |
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Ratio IC50 |
= |
1.16 |
|
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Ratio IC50 |
= |
0.99 |
|
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Ratio IC50 |
= |
1.18 |
|
19470507 |
NPT20 |
Organism |
Candida albicans |
Candida albicans |
Ratio IC50 |
= |
1.07 |
|
19470507 |
NPT1566 |
Individual Protein |
Glyoxalase I |
Homo sapiens |
Ki |
= |
10000 |
nM |
21237663 |
NPT762 |
Cell Line |
A-431 |
Homo sapiens |
IC50 |
= |
13800 |
nM |
21215629 |
NPT380 |
Cell Line |
U-251 |
Homo sapiens |
IC50 |
= |
13800 |
nM |
21215629 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
27400 |
nM |
21215629 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
31600 |
nM |
21215629 |
NPT146 |
Cell Line |
SK-OV-3 |
Homo sapiens |
IC50 |
= |
37700 |
nM |
21215629 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
42600 |
nM |
21215629 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
48000 |
nM |
21215629 |
NPT1171 |
Cell Line |
HEp-2 |
Homo sapiens |
IC50 |
= |
56900 |
nM |
21215629 |
NPT1120 |
Individual Protein |
Pancreatic triacylglycerol lipase |
Sus scrofa |
IC50 |
> |
250000 |
nM |
21282056 |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
Inhibition |
= |
59.01 |
% |
21345672 |
NPT31 |
Individual Protein |
Cyclooxygenase-2 |
Homo sapiens |
Inhibition |
= |
20.32 |
% |
21345672 |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
IC50 |
= |
35090 |
nM |
21345672 |
NPT31 |
Individual Protein |
Cyclooxygenase-2 |
Homo sapiens |
IC50 |
= |
79200 |
nM |
21345672 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
Activity |
= |
3.4 |
% |
21188975 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
Activity |
= |
10.3 |
% |
21188975 |
NPT1083 |
Cell Line |
A-375 |
Homo sapiens |
Activity |
= |
30.5 |
% |
21188975 |
NPT532 |
Individual Protein |
Lysine-specific demethylase 4A |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT226 |
Individual Protein |
Beta-2 adrenergic receptor |
Homo sapiens |
Potency |
|
23109.3 |
nM |
PubChem BioAssay data set |
NPT1005 |
Individual Protein |
Tumor susceptibility gene 101 protein |
Homo sapiens |
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT539 |
Individual Protein |
Cellular tumor antigen p53 |
Homo sapiens |
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT799 |
Individual Protein |
Intestinal alkaline phosphatase |
Mus musculus |
IC50 |
= |
12000 |
nM |
PubChem BioAssay data set |
NPT801 |
Individual Protein |
Intestinal alkaline phosphatase |
Homo sapiens |
IC50 |
= |
7410 |
nM |
PubChem BioAssay data set |
NPT798 |
Individual Protein |
Alkaline phosphatase placental-like |
Homo sapiens |
IC50 |
= |
63500 |
nM |
PubChem BioAssay data set |
NPT63 |
Individual Protein |
Bromodomain adjacent to zinc finger domain protein 2B |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT1139 |
Individual Protein |
Arachidonate 15-lipoxygenase, type II |
Homo sapiens |
Potency |
|
10000 |
nM |
PubChem BioAssay data set |
NPT64 |
Individual Protein |
ATPase family AAA domain-containing protein 5 |
Homo sapiens |
Potency |
|
25918.5 |
nM |
PubChem BioAssay data set |
NPT802 |
Individual Protein |
Alkaline phosphatase, tissue-nonspecific isozyme |
Homo sapiens |
IC50 |
> |
100000 |
nM |
PubChem BioAssay data set |
NPT801 |
Individual Protein |
Intestinal alkaline phosphatase |
Homo sapiens |
IC50 |
= |
44100 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
80 |
% |
21435875 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
90 |
% |
21435875 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.1 |
% |
21397508 |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
49.8 |
nM |
21417461 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
34.4 |
% |
21236667 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
33.26 |
% |
21367493 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
2.71 |
ug/ml |
21600765 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
50 |
% |
21497959 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
20290 |
nM |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
70 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
12.02 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
87.91 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
7.97 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
3.66 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
0.46 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
89.15 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
8.57 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
2.06 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
0.23 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
83.6 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
4.06 |
% |
21504179 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
Activity |
= |
0.32 |
% |
21504179 |
NPT1 |
Others |
Radical scavenging activity |
|
EC50 |
= |
22600 |
nM |
21601463 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
10 |
% |
21601463 |
NPT1566 |
Individual Protein |
Glyoxalase I |
Homo sapiens |
Ki |
= |
10300 |
nM |
21689932 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
38 |
% |
21514701 |
NPT68 |
Individual Protein |
Aldose reductase |
Rattus norvegicus |
Inhibition |
= |
12 |
% |
21514701 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
16700 |
nM |
21514701 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
TGI |
= |
50100 |
nM |
21514701 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
GI50 |
= |
4700 |
nM |
21514701 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
TGI |
= |
8300 |
nM |
21514701 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
GI50 |
= |
5100 |
nM |
21514701 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
TGI |
= |
9200 |
nM |
21514701 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
LC50 |
= |
83400 |
nM |
21514701 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
LC50 |
= |
67200 |
nM |
21514701 |
NPT395 |
Cell Line |
SF-268 |
Homo sapiens |
LC50 |
= |
61000 |
nM |
21514701 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
15230 |
nM |
21070043 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
GI50 |
= |
9440 |
nM |
21070043 |
NPT2 |
Others |
Unspecified |
|
GI50 |
= |
16160 |
nM |
21070043 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
GI50 |
= |
12130 |
nM |
21070043 |
NPT1668 |
Cell Line |
NCI-H157 |
Homo sapiens |
GI50 |
= |
19250 |
nM |
21070043 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
9500 |
nM |
21070043 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
12100 |
nM |
21840724 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
71.3 |
% |
21840724 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
2.5 |
|
21840724 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
Activity |
= |
16 |
% |
21830815 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
8 |
% |
21830815 |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
5.01 |
10'5/M |
21830815 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
17000 |
nM |
21830815 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
18000 |
nM |
21830815 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
18 |
% |
21830815 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20000 |
nM |
21830815 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
34.5 |
% |
21871694 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
41.8 |
% |
21871694 |
NPT2 |
Others |
Unspecified |
|
Ki |
= |
3.57 |
nM |
21885280 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
44668.4 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
50118.7 |
nM |
PubChem BioAssay data set |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
Potency |
|
39810.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
5011.9 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
19011.5 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
2078.7 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT4252 |
Individual Protein |
Toll-like receptor 9 |
Homo sapiens |
IC50 |
= |
15266 |
nM |
PubChem BioAssay data set |
NPT803 |
Individual Protein |
Flap endonuclease 1 |
Homo sapiens |
Potency |
|
89125.1 |
nM |
PubChem BioAssay data set |
NPT8 |
Individual Protein |
DNA polymerase iota |
Homo sapiens |
Potency |
|
19952.6 |
nM |
PubChem BioAssay data set |
NPT199 |
Individual Protein |
DNA polymerase kappa |
Homo sapiens |
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
CC50 |
|
19880 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT6 |
Organism |
Plasmodium falciparum |
Plasmodium falciparum |
Potency |
|
18526 |
nM |
PubChem BioAssay data set |
NPT1161 |
Cell Line |
CHO |
Cricetulus griseus |
IC50 |
= |
34611 |
nM |
PubChem BioAssay data set |
NPT154 |
Individual Protein |
Mothers against decapentaplegic homolog 3 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT226 |
Individual Protein |
Beta-2 adrenergic receptor |
Homo sapiens |
Potency |
|
6513.1 |
nM |
PubChem BioAssay data set |
NPT4253 |
Individual Protein |
Beta Lactamase |
Pseudomonas aeruginosa |
IC50 |
= |
10769 |
nM |
PubChem BioAssay data set |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
|
31622.8 |
nM |
PubChem BioAssay data set |
NPT444 |
Individual Protein |
Ubiquitin carboxyl-terminal hydrolase 1 |
Homo sapiens |
Potency |
|
12589.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.1 |
% |
22019228 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
30.7 |
% |
22019228 |
NPT1 |
Others |
Radical scavenging activity |
|
EC50 |
= |
13000 |
nM |
22029378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18000 |
nM |
22029378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7000 |
nM |
22029378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4700 |
nM |
22029378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26000 |
nM |
22029378 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16000 |
nM |
22029378 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
38000 |
nM |
22029378 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
22029378 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
8000 |
nM |
22029378 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
28000 |
nM |
22029378 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
18000 |
nM |
22029378 |
NPT179 |
Cell Line |
A2780 |
Homo sapiens |
IC50 |
= |
11000 |
nM |
22029378 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
13000 |
nM |
22029378 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
4000 |
nM |
22029378 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
16000 |
nM |
22029378 |
NPT114 |
Cell Line |
LoVo |
Homo sapiens |
IC50 |
= |
10000 |
nM |
22029378 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
3.4 |
|
22029378 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
IC50 |
> |
100000 |
nM |
22041172 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.1 |
% |
22041172 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20300 |
nM |
22137846 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
49800 |
nM |
22222040 |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
IC50 |
= |
105000 |
nM |
22222040 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
87500 |
nM |
22222040 |
NPT397 |
Cell Line |
NCI-H460 |
Homo sapiens |
IC50 |
= |
51300 |
nM |
22222040 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
34.5 |
% |
22341944 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
2.1 |
% |
22341944 |
NPT445 |
Individual Protein |
Peripheral myelin protein 22 |
Rattus norvegicus |
Potency |
|
28695.4 |
nM |
PubChem BioAssay data set |
NPT484 |
Individual Protein |
Luciferin 4-monooxygenase |
Photinus pyralis |
Potency |
|
32196.8 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
48.76 |
% |
22444876 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
48.97 |
% |
22409967 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
5.62 |
% |
22409967 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
45.42 |
% |
22409967 |
NPT2907 |
Organism |
Burkholderia pseudomallei |
Burkholderia pseudomallei |
IZ |
= |
8 |
mm |
22440624 |
NPT2907 |
Organism |
Burkholderia pseudomallei |
Burkholderia pseudomallei |
IZ |
= |
9 |
mm |
22440624 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
IZ |
= |
8 |
mm |
22440624 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
IZ |
= |
10 |
mm |
22440624 |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
= |
11 |
mm |
22440624 |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
= |
9 |
mm |
22440624 |
NPT566 |
Organism |
Salmonella typhimurium |
Salmonella enterica subsp. enterica serovar Typhimurium |
IZ |
= |
12 |
mm |
22440624 |
NPT566 |
Organism |
Salmonella typhimurium |
Salmonella enterica subsp. enterica serovar Typhimurium |
IZ |
= |
10 |
mm |
22440624 |
NPT566 |
Organism |
Salmonella typhimurium |
Salmonella enterica subsp. enterica serovar Typhimurium |
IZ |
= |
9 |
mm |
22440624 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
= |
40000000 |
nM |
22440624 |
NPT2907 |
Organism |
Burkholderia pseudomallei |
Burkholderia pseudomallei |
MIC |
= |
80000000 |
nM |
22440624 |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
= |
80000000 |
nM |
22440624 |
NPT566 |
Organism |
Salmonella typhimurium |
Salmonella enterica subsp. enterica serovar Typhimurium |
MIC |
= |
80000000 |
nM |
22440624 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
80000000 |
nM |
22440624 |
NPT3540 |
Organism |
Cochliobolus lunatus |
Cochliobolus lunatus |
IZ |
= |
11 |
mm |
22440624 |
NPT3540 |
Organism |
Cochliobolus lunatus |
Cochliobolus lunatus |
IZ |
= |
9 |
mm |
22440624 |
NPT2567 |
Organism |
Trichoderma viride |
Hypocrea rufa |
IZ |
= |
9 |
mm |
22440624 |
NPT2567 |
Organism |
Trichoderma viride |
Hypocrea rufa |
MIC |
= |
80000000 |
nM |
22440624 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
50000000 |
nM |
22440624 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
50000000 |
nM |
22440624 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
100000000 |
nM |
22440624 |
NPT3540 |
Organism |
Cochliobolus lunatus |
Cochliobolus lunatus |
MIC |
= |
80000000 |
nM |
22440624 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.1 |
% |
22472046 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18700 |
nM |
22472046 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
19370 |
nM |
22551677 |
NPT461 |
Cell Line |
PANC-1 |
Homo sapiens |
IC50 |
= |
23680 |
nM |
22551677 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
18740 |
nM |
22551677 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
36400 |
nM |
22672984 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
36000 |
nM |
22672984 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
62590 |
nM |
22546674 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
38170 |
nM |
22546674 |
NPT373 |
Cell Line |
SK-MEL-5 |
Homo sapiens |
IC50 |
= |
50370 |
nM |
22546674 |
NPT1081 |
Cell Line |
BXPC-3 |
Homo sapiens |
IC50 |
= |
11430 |
nM |
22546674 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
59370 |
nM |
22546674 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
15900 |
nM |
22546674 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
65160 |
nM |
22546674 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
64670 |
nM |
22546674 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
37.93 |
% |
22546674 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2750 |
nM |
22832313 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
11580 |
nM |
22889562 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5760 |
nM |
22889562 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
10170 |
nM |
22889562 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
15660 |
nM |
22889562 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
20690 |
nM |
22889562 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
21360 |
nM |
22889562 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
35100 |
nM |
22884407 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
35 |
% |
22126405 |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
33498.3 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
18356.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT100 |
Individual Protein |
Glutaminase kidney isoform, mitochondrial |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT477 |
Individual Protein |
DNA dC->dU-editing enzyme APOBEC-3G |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
11220.2 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
23109.3 |
nM |
PubChem BioAssay data set |
NPT10 |
Individual Protein |
Geminin |
Homo sapiens |
Potency |
|
29855.4 |
nM |
PubChem BioAssay data set |
NPT478 |
Individual Protein |
Ataxin-2 |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT755 |
Individual Protein |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
Homo sapiens |
Potency |
|
19952.6 |
nM |
PubChem BioAssay data set |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT1417 |
Individual Protein |
Transcriptional regulator ERG |
Homo sapiens |
Potency |
|
15848.9 |
nM |
PubChem BioAssay data set |
NPT4255 |
Individual Protein |
Toll-like receptor 4 |
Mus musculus |
IC50 |
= |
6000 |
nM |
22985959 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
IC50 |
= |
13000 |
nM |
22989913 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
IC50 |
= |
21000 |
nM |
22989913 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
IC50 |
= |
45000 |
nM |
22989913 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
IC50 |
= |
34000 |
nM |
22989913 |
NPT1674 |
Individual Protein |
CaM kinase II alpha |
Homo sapiens |
IC50 |
= |
33000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
37000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
112000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
64000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
143000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
80000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
33000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
69000 |
nM |
22989913 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.2 |
% |
22944335 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
35100 |
nM |
22995623 |
NPT740 |
Individual Protein |
Beta-secretase 1 |
Homo sapiens |
IC50 |
= |
5700 |
nM |
23041347 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10400 |
nM |
23041347 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10000 |
nM |
23164658 |
NPT2 |
Others |
Unspecified |
|
Ratio CC50/IC50 |
= |
3.5 |
|
22742496 |
NPT2 |
Others |
Unspecified |
|
CC50 |
= |
14800 |
nM |
22742496 |
NPT194 |
Organism |
Dengue virus 2 |
Dengue virus 2 |
IC50 |
= |
4200 |
nM |
22742496 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
Inhibition |
= |
-2.21 |
% |
23062825 |
NPT67 |
Individual Protein |
Cholinesterase |
Equus caballus |
Inhibition |
= |
2.41 |
% |
23062825 |
NPT35 |
Others |
n.a. |
|
Activity |
= |
2.57 |
nmol |
22978824 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.1 |
% |
22978824 |
NPT4256 |
Individual Protein |
Islet amyloid polypeptide |
Homo sapiens |
Activity |
= |
15.1 |
/day |
24900390 |
NPT87 |
Organism |
Aspergillus fumigatus |
Aspergillus fumigatus |
MIC95 |
= |
20 |
uM/ml |
22683240 |
NPT21 |
Organism |
Aspergillus niger |
Aspergillus niger |
MIC95 |
= |
20 |
uM/ml |
22683240 |
NPT87 |
Organism |
Aspergillus fumigatus |
Aspergillus fumigatus |
IZ |
= |
12 |
mm |
22683240 |
NPT21 |
Organism |
Aspergillus niger |
Aspergillus niger |
IZ |
= |
9 |
mm |
22683240 |
NPT2894 |
Organism |
Providencia rettgeri |
Providencia rettgeri |
MIC95 |
= |
20 |
uM/ml |
22683240 |
NPT314 |
Organism |
Bacillus cereus |
Bacillus cereus |
MIC95 |
= |
10 |
uM/ml |
22683240 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC95 |
= |
20 |
uM/ml |
22683240 |
NPT1242 |
Organism |
Salmonella typhi |
Salmonella enterica subsp. enterica serovar Typhi |
MIC95 |
= |
20 |
uM/ml |
22683240 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC95 |
= |
20 |
uM/ml |
22683240 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
52.77 |
% |
23127891 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
37800 |
nM |
23153397 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
31300 |
nM |
23153397 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
49200 |
nM |
23153397 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
GI |
= |
70 |
% |
23245566 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
45 |
% |
23245566 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Activity |
= |
84 |
% |
23245566 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
22.4 |
% |
10.1007/s00044-011-9851-6 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
49.6 |
% |
10.1007/s00044-011-9851-6 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Activity |
= |
61.6 |
% |
10.1007/s00044-011-9851-6 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
Activity |
= |
56.5 |
% |
10.1007/s00044-011-9851-6 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
Activity |
= |
74 |
% |
10.1007/s00044-011-9851-6 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
Activity |
= |
53.7 |
% |
10.1007/s00044-011-9851-6 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
28 |
% |
10.1007/s00044-011-9851-6 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
53.7 |
% |
10.1007/s00044-011-9851-6 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Activity |
= |
78.3 |
% |
10.1007/s00044-011-9851-6 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
10000 |
nM |
10.1007/s00044-011-9851-6 |
NPT134 |
Cell Line |
SK-BR-3 |
Homo sapiens |
IC50 |
= |
27000 |
nM |
10.1007/s00044-011-9851-6 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
17000 |
nM |
10.1007/s00044-011-9851-6 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
44.7 |
% |
10.1007/s00044-011-9851-6 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
62.4 |
% |
10.1007/s00044-011-9851-6 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
86.1 |
% |
10.1007/s00044-011-9851-6 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Activity |
= |
50.2 |
% |
10.1007/s00044-011-9851-6 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Activity |
= |
72.3 |
% |
10.1007/s00044-011-9851-6 |
NPT1174 |
Cell Line |
A375 |
Homo sapiens |
Activity |
= |
92 |
% |
10.1007/s00044-011-9851-6 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
21580 |
nM |
10.1007/s00044-010-9521-0 |
NPT660 |
Cell Line |
SW480 |
Homo sapiens |
IC50 |
= |
18130 |
nM |
10.1007/s00044-010-9353-y |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
24590 |
nM |
10.1007/s00044-010-9353-y |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
21390 |
nM |
10.1007/s00044-010-9353-y |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
17310 |
nM |
10.1007/s00044-010-9353-y |
NPT1548 |
Organism |
Pseudomonas aeruginosa PAO1 |
Pseudomonas aeruginosa PAO1 |
FC |
= |
3 |
|
18284200 |
NPT1548 |
Organism |
Pseudomonas aeruginosa PAO1 |
Pseudomonas aeruginosa PAO1 |
Activity |
> |
2 |
% |
18284200 |
NPT1548 |
Organism |
Pseudomonas aeruginosa PAO1 |
Pseudomonas aeruginosa PAO1 |
Activity |
= |
25 |
% |
18284200 |
NPT1548 |
Organism |
Pseudomonas aeruginosa PAO1 |
Pseudomonas aeruginosa PAO1 |
FC |
= |
2 |
|
18284200 |
NPT1548 |
Organism |
Pseudomonas aeruginosa PAO1 |
Pseudomonas aeruginosa PAO1 |
Activity |
= |
60 |
% |
18284200 |
NPT1548 |
Organism |
Pseudomonas aeruginosa PAO1 |
Pseudomonas aeruginosa PAO1 |
MIC |
= |
30 |
ug/ml |
18284200 |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
54300 |
nM |
10.1007/s00044-010-9344-z |
NPT682 |
Cell Line |
SK-N-MC |
Homo sapiens |
IC50 |
= |
57400 |
nM |
10.1007/s00044-010-9344-z |
NPT111 |
Cell Line |
K562 |
Homo sapiens |
IC50 |
= |
49200 |
nM |
10.1007/s00044-010-9344-z |
NPT4257 |
Individual Protein |
Tubulin alpha 4a |
Ovis aries |
IC50 |
= |
26600 |
nM |
10.1007/s00044-010-9344-z |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
12000 |
nM |
10.1007/s00044-010-9344-z |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
13800 |
nM |
10.1007/s00044-010-9344-z |
NPT1044 |
Individual Protein |
DNA topoisomerase II alpha |
Homo sapiens |
IC50 |
= |
15000 |
nM |
10.1007/s00044-011-9587-3 |
NPT457 |
Cell Line |
BT-549 |
Homo sapiens |
IC50 |
= |
10500 |
nM |
10.1007/s00044-011-9587-3 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
> |
25000 |
nM |
10.1007/s00044-011-9587-3 |
NPT916 |
Cell Line |
SK-MEL |
Homo sapiens |
IC50 |
= |
13750 |
nM |
10.1007/s00044-011-9587-3 |
NPT2 |
Others |
Unspecified |
|
ED25 |
= |
4.8 |
nM |
10.1007/s00044-009-9199-3 |
NPT2 |
Others |
Unspecified |
|
ED50 |
= |
0.0001 |
nM |
10.1007/s00044-009-9199-3 |
NPT2564 |
Organism |
Blumeria graminis |
Blumeria graminis |
Activity |
= |
0 |
% |
12617587 |
NPT829 |
Organism |
Puccinia recondita |
Puccinia recondita |
Activity |
= |
63 |
% |
12617587 |
NPT829 |
Organism |
Puccinia recondita |
Puccinia recondita |
Activity |
= |
76 |
% |
12617587 |
NPT829 |
Organism |
Puccinia recondita |
Puccinia recondita |
Activity |
= |
100 |
% |
12617587 |
NPT825 |
Organism |
Phytophthora infestans |
Phytophthora infestans |
Activity |
= |
57 |
% |
12617587 |
NPT825 |
Organism |
Phytophthora infestans |
Phytophthora infestans |
Activity |
= |
85 |
% |
12617587 |
NPT825 |
Organism |
Phytophthora infestans |
Phytophthora infestans |
Activity |
= |
100 |
% |
12617587 |
NPT635 |
Organism |
Botryotinia fuckeliana |
Botryotinia fuckeliana |
Activity |
= |
0 |
% |
12617587 |
NPT635 |
Organism |
Botryotinia fuckeliana |
Botryotinia fuckeliana |
Activity |
= |
15 |
% |
12617587 |
NPT635 |
Organism |
Botryotinia fuckeliana |
Botryotinia fuckeliana |
Activity |
= |
40 |
% |
12617587 |
NPT635 |
Organism |
Botryotinia fuckeliana |
Botryotinia fuckeliana |
Activity |
= |
70 |
% |
12617587 |
NPT529 |
Organism |
Rhizoctonia solani |
Rhizoctonia solani |
Activity |
= |
26 |
% |
12617587 |
NPT529 |
Organism |
Rhizoctonia solani |
Rhizoctonia solani |
Activity |
= |
45 |
% |
12617587 |
NPT529 |
Organism |
Rhizoctonia solani |
Rhizoctonia solani |
Activity |
= |
63 |
% |
12617587 |
NPT529 |
Organism |
Rhizoctonia solani |
Rhizoctonia solani |
Activity |
= |
85 |
% |
12617587 |
NPT1198 |
Organism |
Magnaporthe grisea |
Magnaporthe grisea |
Activity |
= |
0 |
% |
12617587 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
Activity |
= |
19 |
% |
10.1007/s00044-012-0116-9 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
Activity |
= |
24 |
% |
10.1007/s00044-012-0116-9 |
NPT1374 |
Cell Line |
WI-38 |
Homo sapiens |
Activity |
= |
51 |
% |
10.1007/s00044-012-0116-9 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
18 |
% |
10.1007/s00044-012-0116-9 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
50.4 |
% |
10.1007/s00044-012-0116-9 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
87.64 |
% |
10.1007/s00044-012-0116-9 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
22000 |
nM |
10.1007/s00044-013-0510-y |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
16000 |
nM |
10.1007/s00044-013-0510-y |
NPT1718 |
Cell Line |
A431 |
Homo sapiens |
IC50 |
= |
22000 |
nM |
10.1007/s00044-013-0510-y |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
17000 |
nM |
10.1007/s00044-013-0510-y |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
26000 |
nM |
10.1007/s00044-013-0510-y |
NPT677 |
Individual Protein |
Coagulation factor III |
Homo sapiens |
IC50 |
= |
199.63 |
nM |
10.1007/s00044-012-0330-5 |
NPT285 |
Individual Protein |
Epidermal growth factor receptor erbB1 |
Homo sapiens |
IC50 |
= |
8600 |
nM |
23245570 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18650 |
nM |
23245570 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
26990 |
nM |
23245570 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
34 |
% |
23294827 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18000 |
nM |
23294827 |
NPT677 |
Individual Protein |
Coagulation factor III |
Homo sapiens |
IC50 |
= |
199.63 |
nM |
23199480 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
300000 |
nM |
23394144 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
73 |
% |
24900645 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
FC |
= |
8 |
|
23276449 |
NPT198 |
Individual Protein |
Vitamin D receptor |
Homo sapiens |
EC50 |
= |
20000 |
nM |
23276449 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
196500 |
nM |
23376248 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
Inhibition |
= |
3.88 |
% |
23376248 |
NPT38 |
Individual Protein |
Signal transducer and activator of transcription 3 |
Homo sapiens |
IC50 |
= |
19250 |
nM |
23376248 |
NPT38 |
Individual Protein |
Signal transducer and activator of transcription 3 |
Homo sapiens |
Inhibition |
= |
30.66 |
% |
23376248 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
IC50 |
= |
196500 |
nM |
23434226 |
NPT784 |
Cell Line |
MDA-MB-468 |
Homo sapiens |
Inhibition |
= |
3.88 |
% |
23434226 |
NPT38 |
Individual Protein |
Signal transducer and activator of transcription 3 |
Homo sapiens |
IC50 |
= |
19250 |
nM |
23434226 |
NPT38 |
Individual Protein |
Signal transducer and activator of transcription 3 |
Homo sapiens |
Inhibition |
= |
41 |
% |
23434226 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
16360.1 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
18356.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
29092.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
20596.2 |
nM |
PubChem BioAssay data set |
NPT861 |
Individual Protein |
Isocitrate dehydrogenase [NADP] cytoplasmic |
Homo sapiens |
Potency |
|
29092.9 |
nM |
PubChem BioAssay data set |
NPT920 |
Individual Protein |
Alpha-synuclein |
Homo sapiens |
Potency |
|
19952.6 |
nM |
PubChem BioAssay data set |
NPT160 |
Individual Protein |
TAR DNA-binding protein 43 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
79 |
% |
23524113 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
FC |
= |
1.4 |
|
23524113 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
FC |
= |
1.7 |
|
23524113 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
FC |
= |
2.1 |
|
23524113 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
35600 |
nM |
23501115 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.5 |
equiv |
23501115 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
2.8 |
equiv |
23501115 |
NPT66 |
Individual Protein |
Acetylcholinesterase |
Electrophorus electricus |
IC50 |
= |
81050 |
nM |
23583510 |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
= |
11 |
mm |
23685942 |
NPT1242 |
Organism |
Salmonella typhi |
Salmonella enterica subsp. enterica serovar Typhi |
MIC |
> |
80000 |
nM |
23685942 |
NPT1242 |
Organism |
Salmonella typhi |
Salmonella enterica subsp. enterica serovar Typhi |
IZ |
= |
9 |
mm |
23685942 |
NPT1242 |
Organism |
Salmonella typhi |
Salmonella enterica subsp. enterica serovar Typhi |
IZ |
= |
11 |
mm |
23685942 |
NPT314 |
Organism |
Bacillus cereus |
Bacillus cereus |
MIC |
> |
80000 |
nM |
23685942 |
NPT314 |
Organism |
Bacillus cereus |
Bacillus cereus |
IZ |
= |
9 |
mm |
23685942 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
= |
80000 |
nM |
23685942 |
NPT34 |
Cell Line |
BV-2 |
Mus musculus |
IC50 |
= |
3100 |
nM |
23734721 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Inhibition |
= |
12.9 |
% |
23685942 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
50000000 |
nM |
23685942 |
NPT3558 |
Cell Line |
QG-56 |
|
IC50 |
= |
100000000 |
nM |
23685942 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
50000000 |
nM |
23685942 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
50000000 |
nM |
23685942 |
NPT2567 |
Organism |
Trichoderma viride |
Hypocrea rufa |
MIC |
> |
80000 |
nM |
23685942 |
NPT2567 |
Organism |
Trichoderma viride |
Hypocrea rufa |
IZ |
= |
9 |
mm |
23685942 |
NPT3540 |
Organism |
Cochliobolus lunatus |
Cochliobolus lunatus |
MIC |
> |
80000 |
nM |
23685942 |
NPT3540 |
Organism |
Cochliobolus lunatus |
Cochliobolus lunatus |
IZ |
= |
9 |
mm |
23685942 |
NPT3540 |
Organism |
Cochliobolus lunatus |
Cochliobolus lunatus |
IZ |
= |
11 |
mm |
23685942 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
> |
80000 |
nM |
23685942 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
IZ |
= |
12 |
mm |
23685942 |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
> |
80000 |
nM |
23685942 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
50.12 |
% |
23511019 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
IC50 |
= |
13200 |
nM |
23644215 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
11540 |
nM |
23644215 |
NPT139 |
Cell Line |
HT-29 |
Homo sapiens |
Ratio IC50 |
= |
0.48 |
|
23644215 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
Ratio IC50 |
= |
0.39 |
|
23644215 |
NPT2 |
Others |
Unspecified |
|
IC50 |
> |
100000 |
nM |
23357628 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
4.6 |
% |
23357628 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
5.8 |
% |
23357628 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
13.7 |
% |
23357628 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
22.2 |
% |
23357628 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
45 |
% |
23357628 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
26500 |
nM |
23357628 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
0.3 |
% |
23357628 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
2.4 |
% |
23357628 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
23.1 |
% |
23357628 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
42 |
% |
23357628 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
87.2 |
% |
23357628 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
50.2 |
% |
23357628 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
29.33 |
% |
23357628 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
Activity |
= |
20.46 |
% |
23357628 |
NPT393 |
Cell Line |
HCT-116 |
Homo sapiens |
IC50 |
= |
41500 |
nM |
23357628 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
32200 |
nM |
23357628 |
NPT515 |
Cell Line |
SGC-7901 |
Homo sapiens |
IC50 |
= |
29000 |
nM |
23357628 |
NPT65 |
Cell Line |
HepG2 |
Homo sapiens |
IC50 |
= |
78700 |
nM |
23357628 |
NPT202 |
Individual Protein |
Protease |
Human immunodeficiency virus 1 |
IC50 |
= |
100000 |
nM |
23742639 |
NPT23 |
Individual Protein |
Integrase |
Human immunodeficiency virus 1 |
IC50 |
= |
40000 |
nM |
23742639 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
16400 |
nM |
23742639 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
42.4 |
% |
23685572 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
24000 |
nM |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
5.02 |
U/L |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
7.13 |
U/L |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
589 |
K/uL |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
485 |
K/uL |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
6.83 |
K/uL |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
4.69 |
K/uL |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
31.1 |
% |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
30.6 |
% |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.139 |
ug |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.129 |
ug |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
1.1 |
ug |
23145932 |
NPT32 |
Organism |
Mus musculus |
Mus musculus |
Activity |
= |
0.987 |
ug |
23145932 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
> |
50 |
% |
23145932 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
48 |
% |
23145932 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
53 |
% |
23145932 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
57 |
% |
23145932 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
Inhibition |
= |
51 |
% |
23145932 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
IC50 |
= |
12350 |
nM |
23799643 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
52.77 |
% |
23799643 |
NPT1137 |
Individual Protein |
11-beta-hydroxysteroid dehydrogenase 1 |
Homo sapiens |
IC50 |
= |
15983 |
nM |
23800686 |
NPT1138 |
Individual Protein |
11-beta-hydroxysteroid dehydrogenase 2 |
Homo sapiens |
Inhibition |
= |
15696 |
% |
23800686 |
NPT4259 |
Individual Protein |
11-beta-hydroxysteroid dehydrogenase 2 |
Rattus norvegicus |
Inhibition |
= |
14939 |
% |
23800686 |
NPT1137 |
Individual Protein |
11-beta-hydroxysteroid dehydrogenase 1 |
Homo sapiens |
IC50 |
= |
4501 |
nM |
23800686 |
NPT4260 |
Individual Protein |
11-beta-hydroxysteroid dehydrogenase 1 |
Rattus norvegicus |
IC50 |
= |
4125 |
nM |
23800686 |
NPT4260 |
Individual Protein |
11-beta-hydroxysteroid dehydrogenase 1 |
Rattus norvegicus |
IC50 |
= |
3921 |
nM |
23800686 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
11400 |
nM |
23830698 |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
IC50 |
= |
35500 |
nM |
23830698 |
NPT2489 |
Cell Line |
MeWo |
Homo sapiens |
Activity |
= |
90 |
% |
23830698 |
NPT2553 |
Individual Protein |
Aminopeptidase N |
Homo sapiens |
IC50 |
= |
10000 |
nM |
23860593 |
NPT1553 |
Individual Protein |
Aminopeptidase N |
Sus scrofa |
IC50 |
= |
15500 |
nM |
23860593 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
51.3 |
% |
23932451 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
FC |
= |
1.8 |
|
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
FC |
= |
1.5 |
|
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
FC |
= |
0.9 |
|
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
FC |
= |
0.5 |
|
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
Inhibition |
= |
1.5 |
% |
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
Inhibition |
= |
38 |
% |
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
Inhibition |
= |
95.5 |
% |
23933533 |
NPT1970 |
Cell Line |
THP-1 |
Homo sapiens |
Inhibition |
= |
102.5 |
% |
23933533 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
28.3 |
ug/ml |
23933533 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
17.03 |
ug/ml |
23933533 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
11.41 |
ug/ml |
23933533 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
5000 |
nM |
24094143 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
IC50 |
= |
20300 |
nM |
24095756 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
43.5 |
% |
24095756 |
NPT73 |
Individual Protein |
Solute carrier organic anion transporter family member 1B1 |
Homo sapiens |
Inhibition |
= |
82.72 |
% |
23571415 |
NPT72 |
Individual Protein |
Solute carrier organic anion transporter family member 1B3 |
Homo sapiens |
Inhibition |
= |
115.19 |
% |
23571415 |
NPT2028 |
Cell Line |
SK-N-FI |
Homo sapiens |
IC50 |
= |
11300 |
nM |
24183537 |
NPT136 |
Cell Line |
SK-N-SH |
Homo sapiens |
IC50 |
= |
6400 |
nM |
24183537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
8100 |
nM |
24183537 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3900 |
nM |
24256496 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
51.04 |
% |
24148835 |
NPT737 |
Cell Line |
HUVEC |
Homo sapiens |
Inhibition |
= |
45 |
% |
24332631 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
29 |
% |
24342238 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
24 |
% |
24342238 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
51.5 |
% |
24269515 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
20700 |
nM |
24275249 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Activity |
= |
34.8 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
59.4 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
27.1 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
62.8 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
82.5 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
89.3 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
99.4 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
98.2 |
% |
24275249 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Activity |
= |
42.4 |
% |
24275249 |
NPT1045 |
Cell Line |
U2OS |
Homo sapiens |
Activity |
= |
29 |
% |
24275249 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
93.3 |
% |
24467317 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
530 |
nM |
24467317 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
341 |
molar ratio |
24411124 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
100 |
% |
24411124 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
81.7 |
% |
24411124 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
22.8 |
% |
24411124 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0 |
% |
24411124 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
20 |
% |
24321865 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
64 |
% |
24589487 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
43.1 |
% |
24589487 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
29 |
% |
24594525 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
24 |
% |
24594525 |
NPT81 |
Cell Line |
A549 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
24531225 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
12600 |
nM |
24531225 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
880 |
nM |
24531225 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
1980 |
nM |
24531225 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
300 |
nM |
24531225 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
52.21 |
% |
10.1039/C3MD00376K |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
> |
1.26 |
|
10.1039/C3MD00376K |
NPT2 |
Others |
Unspecified |
|
Potency |
|
1995.3 |
nM |
PubChem BioAssay data set |
NPT161 |
Individual Protein |
Rap guanine nucleotide exchange factor 4 |
Homo sapiens |
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
25118.9 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
22387.2 |
nM |
PubChem BioAssay data set |
NPT831 |
Individual Protein |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
Potency |
|
1683.4 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
Potency |
|
35481.3 |
nM |
PubChem BioAssay data set |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6700 |
nM |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
37 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
33 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
12 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
17 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
70 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
13 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
44 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
82 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
17 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
25 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
58 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
71 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
54 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
66 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
75 |
% |
24689857 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
500 |
nM |
24593150 |
NPT1 |
Others |
Radical scavenging activity |
|
EC50 |
= |
26600 |
nM |
24657052 |
NPT983 |
Protein Complex |
Nuclear factor NF-kappa-B complex |
Homo sapiens |
IC50 |
= |
8000 |
nM |
24775915 |
NPT1 |
Others |
Radical scavenging activity |
|
Activity |
= |
63.9 |
% |
24920381 |
NPT1119 |
Individual Protein |
Arachidonate 12-lipoxygenase |
Homo sapiens |
Inhibition |
= |
65 |
% |
24920381 |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
3900 |
nM |
24920381 |
NPT30 |
Individual Protein |
Cyclooxygenase-1 |
Homo sapiens |
IC50 |
= |
8100 |
nM |
24920381 |
NPT38 |
Individual Protein |
Signal transducer and activator of transcription 3 |
Homo sapiens |
IC50 |
= |
33900 |
nM |
24920381 |
NPT983 |
Protein Complex |
Nuclear factor NF-kappa-B complex |
Homo sapiens |
IC50 |
= |
20900 |
nM |
24920381 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
36000 |
nM |
24920381 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
34800 |
nM |
24920381 |
NPT152 |
Individual Protein |
Nuclear factor erythroid 2-related factor 2 |
Homo sapiens |
EC50 |
= |
9900 |
nM |
24920381 |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
500 |
nM |
24920381 |
NPT956 |
Individual Protein |
Prostaglandin E synthase |
Homo sapiens |
IC50 |
= |
600 |
nM |
24920381 |
NPT956 |
Individual Protein |
Prostaglandin E synthase |
Homo sapiens |
IC50 |
= |
1200 |
nM |
24920381 |
NPT570 |
Individual Protein |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50 |
= |
600 |
nM |
24920381 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
1200 |
nM |
24920381 |
NPT792 |
Individual Protein |
Arachidonate 15-lipoxygenase |
Homo sapiens |
IC50 |
= |
1200 |
nM |
24920381 |
NPT91 |
Cell Line |
KB |
Homo sapiens |
IC50 |
= |
21360 |
nM |
24857542 |
NPT189 |
Cell Line |
Vero |
Chlorocebus aethiops |
IC50 |
= |
35050 |
nM |
24857542 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.64 |
|
24857542 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
25000 |
nM |
10.1039/C1MD00199J |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
34400 |
nM |
25453798 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
77.04 |
% |
25453803 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
6200 |
nM |
25453803 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
80 |
% |
25467149 |
NPT270 |
Individual Protein |
Nitric oxide synthase, inducible |
Mus musculus |
Inhibition |
= |
97 |
% |
25058929 |
NPT270 |
Individual Protein |
Nitric oxide synthase, inducible |
Mus musculus |
IC50 |
= |
800 |
nM |
25058929 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6010 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
7990 |
nM |
24960549 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
IC50 |
= |
11000 |
nM |
25088549 |
NPT740 |
Individual Protein |
Beta-secretase 1 |
Homo sapiens |
IC50 |
= |
5300 |
nM |
25088549 |
NPT2 |
Others |
Unspecified |
|
FC |
= |
2 |
|
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
40000 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26000 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
48000 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2500 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
4800 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3800 |
nM |
24960549 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
6000 |
nM |
25051453 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
45 |
% |
24961640 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
60 |
% |
24961640 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Ratio |
= |
2 |
|
24961640 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
53 |
% |
25093453 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6.9 |
nM |
24831826 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
480000 |
nM |
24831826 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
11020 |
nM |
25113933 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18520 |
nM |
25113933 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
1.25 |
ug/ml |
25113933 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
2.08 |
ug/ml |
25113933 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
6.44 |
ug/ml |
25113933 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
24.82 |
ug/ml |
25113933 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
11020 |
nM |
24909081 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18520 |
nM |
24909081 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
1.25 |
% |
24909081 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
2.08 |
% |
24909081 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
6.44 |
% |
24909081 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
24.82 |
% |
24909081 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6460 |
nM |
24657568 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
8160 |
nM |
24657568 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
21200 |
nM |
24657568 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
15100 |
nM |
24657568 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
10120 |
nM |
24938495 |
NPT324 |
Individual Protein |
Cyclooxygenase-1 |
Ovis aries |
IC50 |
= |
29650 |
nM |
24938495 |
NPT31 |
Individual Protein |
Cyclooxygenase-2 |
Homo sapiens |
IC50 |
> |
100000 |
nM |
24938495 |
NPT4261 |
Individual Protein |
Lipoxygenase |
Glycine max |
IC50 |
= |
59520 |
nM |
24938495 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
81.5 |
% |
24938495 |
NPT4261 |
Individual Protein |
Lipoxygenase |
Glycine max |
Inhibition |
= |
68.28 |
% |
24938495 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.53 |
|
25305717 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
6000 |
nM |
25277281 |
NPT1032 |
Individual Protein |
Neuraminidase |
Influenza A virus (strain A/USSR/90/1977 H1N1) |
IC50 |
= |
10000 |
nM |
25277281 |
NPT1032 |
Individual Protein |
Neuraminidase |
Influenza A virus (strain A/USSR/90/1977 H1N1) |
IC50 |
= |
8100 |
nM |
25277281 |
NPT804 |
Cell Line |
HT-22 |
Mus musculus |
Inhibition |
= |
36 |
% |
25313922 |
NPT804 |
Cell Line |
HT-22 |
Mus musculus |
Inhibition |
= |
18 |
% |
25313922 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
42.3 |
% |
25282654 |
NPT2 |
Others |
Unspecified |
|
Ratio |
= |
1.83 |
|
25282654 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Inhibition |
= |
19.2 |
% |
25420236 |
NPT621 |
Tissue |
Plasma |
Homo sapiens |
Inhibition |
= |
18.6 |
% |
25420236 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
50.2 |
% |
25542589 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
81 |
% |
25577709 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
55 |
% |
25577709 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
83.8 |
% |
25577709 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
53.6 |
% |
25577709 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
93.1 |
% |
25577709 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
90.2 |
% |
25577709 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
85.5 |
% |
25577709 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
43.1 |
% |
25678013 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
58 |
% |
25678013 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
51.8 |
% |
25624107 |
NPT333 |
Cell Line |
CEM |
Homo sapiens |
IC50 |
= |
15000 |
nM |
25577711 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
18000 |
nM |
25577711 |
NPT137 |
Cell Line |
L1210 |
Mus musculus |
IC50 |
= |
22000 |
nM |
25577711 |
NPT2 |
Others |
Unspecified |
|
Ratio IC50 |
= |
1.5 |
|
25577711 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1201.4 |
umol/ml |
25577711 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
1581.9 |
umol/ml |
25577711 |
NPT1 |
Others |
Radical scavenging activity |
|
Inhibition |
= |
96.8 |
% |
25577711 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
98.7 |
% |
25577711 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
47.8 |
% |
25724825 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
18520 |
nM |
25824662 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
11020 |
nM |
25824662 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
3400 |
nM |
25824662 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
5600 |
nM |
25824662 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
17500 |
nM |
25824662 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
67400 |
nM |
25824662 |
NPT878 |
Organism |
Streptococcus mutans |
Streptococcus mutans |
MIC |
> |
542900 |
nM |
25746812 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
91500 |
nM |
25746812 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
26.8 |
ug/ml |
25881826 |
NPT927 |
Cell Line |
PBMC |
Homo sapiens |
IC50 |
= |
12.3 |
ug/ml |
25881826 |
NPT983 |
Protein Complex |
Nuclear factor NF-kappa-B complex |
Homo sapiens |
IC50 |
= |
7.7 |
ug/ml |
25881826 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
20.7 |
% |
25881826 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
23 |
% |
25881826 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
23.3 |
% |
25881826 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
13530 |
nM |
25728027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
48630 |
nM |
25728027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
54350 |
nM |
25728027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
89820 |
nM |
25728027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
39420 |
nM |
25728027 |
NPT83 |
Cell Line |
MCF7 |
Homo sapiens |
IC50 |
= |
70200 |
nM |
25728027 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
59020 |
nM |
25728027 |
NPT1830 |
Organism |
Mycobacterium marinum |
Mycobacterium marinum |
IZ |
= |
1.1 |
mm |
25618016 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
35 |
% |
25791674 |
NPT2 |
Others |
Unspecified |
|
Kd |
= |
507000 |
nM |
25681711 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
78.8 |
|
25681711 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
36.4 |
|
25681711 |
NPT2704 |
Individual Protein |
Hemagglutinin |
Influenza A virus |
Activity |
= |
16.1 |
|
25681711 |
NPT2704 |
Individual Protein |
Hemagglutinin |
Influenza A virus |
Activity |
= |
6.8 |
|
25681711 |
NPT2704 |
Individual Protein |
Hemagglutinin |
Influenza A virus |
Activity |
= |
2.7 |
|
25681711 |
NPT2704 |
Individual Protein |
Hemagglutinin |
Influenza A virus |
Activity |
= |
0.8 |
|
25681711 |
NPT79 |
Organism |
Bacillus subtilis |
Bacillus subtilis |
MIC |
= |
16 |
ug/ml |
25938986 |
NPT19 |
Organism |
Escherichia coli |
Escherichia coli |
MIC |
> |
128 |
ug/ml |
25938986 |
NPT16 |
Organism |
Staphylococcus aureus |
Staphylococcus aureus |
MIC |
> |
128 |
ug/ml |
25938986 |
NPT1079 |
Individual Protein |
Histone acetyltransferase p300 |
Homo sapiens |
Inhibition |
= |
93.45 |
% |
25730130 |
NPT1079 |
Individual Protein |
Histone acetyltransferase p300 |
Homo sapiens |
IC50 |
= |
6500 |
nM |
25730130 |
NPT79 |
Organism |
Bacillus subtilis |
Bacillus subtilis |
MIC |
= |
32 |
ug/ml |
25938986 |
NPT18 |
Organism |
Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
> |
128 |
ug/ml |
25938986 |
NPT1228 |
Organism |
Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
> |
128 |
ug/ml |
25938986 |
NPT2 |
Others |
Unspecified |
|
Potency |
|
17782.8 |
nM |
PubChem BioAssay data set |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
43.1 |
% |
25778991 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
58 |
% |
25778991 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
56.5 |
% |
25778991 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
2.45 |
% |
25961334 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Inhibition |
= |
55.07 |
% |
25961334 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
58.49 |
% |
25961334 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Inhibition |
= |
7.25 |
% |
25961334 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Inhibition |
= |
65.45 |
% |
25961334 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Inhibition |
= |
28.78 |
% |
25961334 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
50.3 |
% |
25961334 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Inhibition |
= |
13.75 |
% |
25961334 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
25430 |
nM |
25961334 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
12360 |
nM |
25961334 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
26230 |
nM |
25961334 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
13610 |
nM |
25961334 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
12110 |
nM |
25961334 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
IC50 |
= |
10460 |
nM |
25961334 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
25961334 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
25961334 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
25961334 |
NPT165 |
Cell Line |
HeLa |
Homo sapiens |
Ratio IC50 |
= |
1 |
|
25961334 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
IC50 |
= |
3900 |
nM |
26099993 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
70 |
% |
26099993 |
NPT2794 |
Individual Protein |
Quinolone resistance protein norA |
Staphylococcus aureus |
MIC |
= |
1 |
ug/ml |
10.1039/C4MD00196F |
NPT2794 |
Individual Protein |
Quinolone resistance protein norA |
Staphylococcus aureus |
FC |
= |
8 |
|
10.1039/C4MD00196F |
NPT2 |
Others |
Unspecified |
|
MIC |
= |
32 |
ug/ml |
10.1039/C4MD00196F |
NPT2 |
Others |
Unspecified |
|
FC |
= |
0 |
|
10.1039/C4MD00196F |
NPT2 |
Others |
Unspecified |
|
MIC |
= |
64 |
ug/ml |
10.1039/C4MD00196F |
NPT2795 |
Individual Protein |
Fluoroquinolone resistance protein |
Staphylococcus aureus |
MIC |
= |
256 |
ug/ml |
10.1039/C4MD00196F |
NPT2795 |
Individual Protein |
Fluoroquinolone resistance protein |
Staphylococcus aureus |
FC |
= |
0 |
|
10.1039/C4MD00196F |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
22910 |
nM |
26048786 |
NPT668 |
Individual Protein |
P-glycoprotein 1 |
Homo sapiens |
IC50 |
= |
62000 |
nM |
10.1039/C4MD00196F |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
14700 |
nM |
26071636 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
Inhibition |
= |
99.3 |
% |
26071636 |
NPT113 |
Cell Line |
RAW264.7 |
Mus musculus |
IC50 |
= |
28800 |
nM |
26071636 |
NPT35 |
Others |
n.a. |
|
Inhibition |
= |
88.3 |
% |
26071636 |
NPT1 |
Others |
Radical scavenging activity |
|
Inhibition |
= |
84.2 |
% |
26071636 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
23600 |
nM |
26071636 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
0.803 |
mmolequiv/L |
26071636 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
3900 |
nM |
26241103 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
86.6 |
% |
26197162 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
51.5 |
% |
26337018 |
NPT2 |
Others |
Unspecified |
|
Inhibition |
= |
65.9 |
% |
26337018 |
NPT1 |
Others |
Radical scavenging activity |
|
IC50 |
= |
14.83 |
ug/ml |
26264500 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
34.71 |
ug/ml |
26264500 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
50 |
% |
26288690 |
NPT90 |
Cell Line |
DU-145 |
Homo sapiens |
IC50 |
= |
26200 |
nM |
26341135 |
NPT306 |
Cell Line |
PC-3 |
Homo sapiens |
IC50 |
= |
25400 |
nM |
26341135 |
NPT858 |
Cell Line |
LNCaP |
Homo sapiens |
IC50 |
= |
12100 |
nM |
26341135 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
7480 |
nM |
26386817 |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
58.4 |
% |
26386817 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
70.6 |
% |
10.1039/C4MD00305E |
NPT519 |
Cell Line |
SH-SY5Y |
Homo sapiens |
Inhibition |
= |
37.87 |
% |
10.1039/C4MD00305E |
NPT2 |
Others |
Unspecified |
|
Activity |
= |
8.5 |
% |
26386817 |
NPT2 |
Others |
Unspecified |
|
EC50 |
= |
48500 |
nM |
26386817 |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
48.74 |
% |
10.1039/C4MD00305E |
NPT78 |
Individual Protein |
Beta amyloid A4 protein |
Homo sapiens |
Inhibition |
= |
42.3 |
% |
26514744 |
NPT82 |
Cell Line |
MDA-MB-231 |
Homo sapiens |
IC50 |
= |
15000 |
nM |
26561365 |
NPT3722 |
Cell Line |
4T1 |
Mus musculus |
IC50 |
= |
20000 |
nM |
26561365 |
NPT2 |
Others |
Unspecified |
|
IC50 |
= |
20000 |
nM |
26561365 |