Plant ingredients against the target with activities between 10uM and 50uM
Ingredient ID | Target (Gene Symbol) | No. of Activity Values | Activity Value (nM) | Activity Type | Activity Reference |
---|---|---|---|---|---|
NPC1075 | CYP2C9 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC110899 | CA5B | 1 | 35400 | Ki |
PMID: 20185318 |
NPC112701 | GAA | 2 |
Median: 35481.3 Range: 35481.3 to 35481.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC112701 | KDM4E | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC116146 | GLI1 | 2 |
Median: 38000 Range: 38000 to 38000 |
IC50 |
PMID: 18842418 PMID: 19309080 |
NPC119949 | ALDH1A1 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC119949 | SMN1;SMN2 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC126029 | TSHR | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC142415 | ACP1 | 4 |
Median: 22050 Range: 21200 to 22900 |
IC50 |
PMID: 21453996 PMID: 21453996 PMID: 25264584 PMID: 25264584 |
NPC142415 | PTPN6 | 2 |
Median: 22760 Range: 14190 to 31330 |
IC50 |
PMID: 18707891 PMID: 27123900 |
NPC14330 | ALDH1A1 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC149184 | PPARG | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC149184 | PPARD | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC149184 | PPARA | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC156461 | GAPDH | 7 |
Median: 35000000 Range: 35000 to 100000000 |
IC50 |
PMID: 7562915 PMID: 7562915 PMID: 7562915 PMID: 7932587 PMID: 7932587 PMID: 7932587 PMID: 9822549 |
NPC156461 | ADORA2B | 3 |
Median: 24000 Range: 24000 to 24000 |
EC50 |
PMID: 20541935 PMID: 21388809 PMID: 24164628 |
NPC156461 | SLC29A1 | 1 | 17000 | IC50 |
PMID: 23388705 |
NPC156654 | L3MBTL1 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC156654 | KDM4E | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC156654 | POLB | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC161659 | ALDH1A1 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC167400 | ALDH1A1 | 1 | 18029.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC171736 | PPARG | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC171736 | PPARA | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC171736 | PPARD | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC176740 | MAPT | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC176740 | EPHX2 | 1 | 24300 | IC50 |
PMID: 24679441 |
NPC176740 | KDM4E | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC17810 | LMNA | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC17810 | ALDH1A1 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CYP2C9 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CYP2C19 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | THRB | 2 |
Median: 32464.8 Range: 25118.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CARM1 | 1 | 25000 | IC50 |
DOI: 10.1039/C1MD00199J |
NPC178134 | GSR | 1 | 22800 | IC50 |
PMID: 19015351 |
NPC178134 | EPHX2 | 1 | 20700 | IC50 |
PMID: 24679441 |
NPC178134 | ATM | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | MAPK1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC179950 | EPHX2 | 1 | 28430 | IC50 |
PMID: 24679441 |
NPC179950 | XDH | 1 | 26310 | IC50 |
PMID: 12444671 |
NPC179950 | MAPT | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC181465 | XDH | 1 | 14800 | IC50 |
PMID: 9461655 |
NPC183950 | POLB | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC183950 | ALDH1A1 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC183950 | MAPT | 1 | 22387.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC183950 | KMT2A | 1 | 17782.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC187770 | TYR | 1 | 32500 | IC50 |
PMID: 25726329 |
NPC192744 | SMN1;SMN2 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC201844 | PPARA | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC201844 | PPARD | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC201844 | PPARG | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC204932 | CA14 | 2 |
Median: 48900 Range: 48900 to 48900 |
Ki |
PMID: 18579385 PMID: 20185318 |
NPC204932 | BLM | 2 |
Median: 44668.4 Range: 44668.4 to 44668.4 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | POLB | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | APEX1 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | EGFR | 1 | 26043 | IC50 |
DrugMatrix in vitro pharmacology data CHEMBL1909046 |
NPC204932 | MMP9 | 1 | 23367 | IC50 |
DrugMatrix in vitro pharmacology data CHEMBL1909046 |
NPC204932 | TDP1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | L3MBTL1 | 1 | 17782.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | FYN | 1 | 17431 | IC50 |
DrugMatrix in vitro pharmacology data CHEMBL1909046 |
NPC204932 | RECQL | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | ALOX15 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | KDM4E | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | PMP22 | 1 | 47754.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | THRB | 1 | 44668.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | GALK1 | 1 | 42128.5 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CDK2 | 1 | 40000 | IC50 |
PMID: 17178224 |
NPC20791 | CD38 | 1 | 37900 | IC50 |
PMID: 21641214 |
NPC20791 | SORD | 2 |
Median: 106300 Range: 35600 to 177000 |
IC50 |
PMID: 8893834 PMID: 12672241 |
NPC20791 | SMN1;SMN2 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | EPHX2 | 1 | 33540 | IC50 |
PMID: 24679441 |
NPC20791 | DPP4 | 2 |
Median: 81365 Range: 32730 to 130000 |
IC50 |
PMID: 18650094 DOI: 10.1039/C0MD00245C |
NPC20791 | MAPK1 | 2 |
Median: 35716.75 Range: 31622.8 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | ADORA3 | 1 | 30000 | Ki |
PMID: 8576921 |
NPC20791 | PTGS2 | 1 | 28600 | IC50 |
PMID: 17378609 |
NPC20791 | BLM | 3 |
Median: 28183.8 Range: 28183.8 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | TDP1 | 2 |
Median: 26651.35 Range: 25118.9 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | ALDH1A1 | 6 |
Median: 37646 Range: 25118.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CDK6 | 2 |
Median: 25000 Range: 25000 to 25000 |
IC50 |
PMID: 15689157 DOI: 10.1007/s00044-009-9233-5 |
NPC20791 | PTPN1 | 2 |
Median: 23300 Range: 23300 to 23300 |
IC50 |
PMID: 12419367 PMID: 19297174 |
NPC20791 | KMT2A | 1 | 22387.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | AMY1A;AMY1B;AMY1C | 1 | 21400 | IC50 |
PMID: 18507367 |
NPC20791 | SYK | 1 | 20000 | IC50 |
PMID: 22257213 |
NPC20791 | HPGD | 2 |
Median: 21169.9 Range: 19952.6 to 22387.2 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | APEX1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CYP2D6 | 1 | 18800 | IC50 |
PMID: 22328583 |
NPC20791 | USP2 | 2 |
Median: 25057.75 Range: 18492.7 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | GPR35 | 1 | 15400 | IC50 |
PMID: 24900447 |
NPC20791 | APP | 1 | 15300 | IC50 |
PMID: 26719209 |
NPC209970 | ALOX15 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC209970 | PPARG | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC209970 | TDP1 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC209970 | HSD17B10 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC212551 | RAPGEF4 | 2 |
Median: 40000 Range: 40000 to 40000 |
IC50 |
PMID: 23286832 PMID: 24256330 |
NPC212551 | GMNN | 1 | 22387.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC216630 | PPARG | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC219876 | HSD17B10 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | PTGS1 | 2 |
Median: 58350 Range: 36700 to 80000 |
IC50 |
PMID: 11858749 PMID: 16038536 |
NPC219876 | SMN1;SMN2 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | NPSR1 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | BLM | 2 |
Median: 28183.8 Range: 28183.8 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | ALDH1A1 | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | RECQL | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | MAPT | 2 |
Median: 19952.6 Range: 19952.6 to 19952.6 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | APEX1 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC220498 | GLI1 | 2 |
Median: 42000 Range: 42000 to 42000 |
IC50 |
PMID: 18842418 PMID: 19309080 |
NPC225710 | SELL | 1 | 27600 | IC50 |
PMID: 17302397 |
NPC225710 | GAPDH | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | MAPK1 | 2 |
Median: 23753.05 Range: 22387.2 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | SELP | 1 | 19100 | IC50 |
PMID: 17302397 |
NPC225710 | SMN1;SMN2 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC235059 | MAPK1 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC257124 | AR | 2 |
Median: 19027.305 Range: 19000 to 19054.61 |
IC50 |
PMID: 20226658 PMID: 20226658 |
NPC261619 | BACE1 | 2 |
Median: 25500 Range: 23000 to 28000 |
IC50 |
PMID: 14592472 PMID: 14592472 |
NPC261831 | BLM | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC261831 | CYP19A1 | 1 | 32700 | IC50 |
PMID: 16643058 |
NPC261831 | TOP1 | 1 | 31000 | IC50 |
PMID: 12444712 |
NPC261831 | MAPT | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC261831 | FABP4 | 1 | 26100 | IC50 |
PMID: 20471252 |
NPC261831 | KMT2A | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC261831 | ATM | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC261831 | HSD17B10 | 2 |
Median: 17900.75 Range: 15848.9 to 19952.6 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC264317 | POLB | 2 |
Median: 44925 Range: 43600 to 46250 |
IC50 |
PMID: 14640519 PMID: 18343122 |
NPC264317 | GLI1 | 2 |
Median: 32000 Range: 32000 to 32000 |
IC50 |
PMID: 18842418 PMID: 19309080 |
NPC267691 | NOS2 | 1 | 37000 | IC50 |
PMID: 15837296 |
NPC281131 | MAPK1 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC281131 | GLA | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC281131 | MAPT | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC281131 | LMNA | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC281131 | EPHX2 | 1 | 21760 | IC50 |
PMID: 24679441 |
NPC287331 | RECQL | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC287331 | LMNA | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC287331 | TSHR | 2 |
Median: 15848.9 Range: 15848.9 to 15848.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC289774 | TDP1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | CYP19A1 | 1 | 44200 | IC50 |
PMID: 16643058 |
NPC294548 | BLM | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | L3MBTL1 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | F3 | 1 | 30000 | IC50 |
PMID: 9834151 |
NPC294548 | HPGD | 2 |
Median: 28183.8 Range: 28183.8 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | MAPT | 3 |
Median: 28183.8 Range: 28183.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | LMNA | 1 | 22387.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | PLA2G1B | 1 | 22300 | IC50 |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | KDM4E | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | PPARD | 1 | 16000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC294548 | CYP3A4 | 2 |
Median: 15848.9 Range: 15848.9 to 15848.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | ATG4B | 1 | 15300 | IC50 |
PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | HPGD | 3 |
Median: 39810.7 Range: 39810.7 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | ALDH1A1 | 2 |
Median: 39810.7 Range: 39810.7 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | APEX1 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | APP | 1 | 32800 | IC50 |
PMID: 22921742 |
NPC294902 | AKR1B1 | 1 | 32000 | IC50 |
PMID: 22236472 |
NPC294902 | CYP3A4 | 2 |
Median: 25118.9 Range: 25118.9 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | POLB | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC301585 | PPARD | 1 | 24000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC301585 | PPARG | 1 | 21000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC301696 | ALDH1A1 | 1 | 44668.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC328740 | RECQL | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC328740 | GAA | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC328740 | KDM4E | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC328740 | ALDH1A1 | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC328740 | L3MBTL1 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | POLB | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | GLA | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | GAA | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | BLM | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | HPGD | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | ALDH1A1 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | RECQL | 2 |
Median: 27005 Range: 22387.2 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | MAPT | 2 |
Median: 19622.15 Range: 14125.4 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC43246 | SLC28A2 | 1 | 32000 | IC50 |
PMID: 23388705 |
NPC51700 | PPARA | 1 | 41310 | EC50 |
PMID: 21855333 |
NPC51700 | AKR1B1 | 1 | 41000 | IC50 |
PMID: 21561086 |
NPC51700 | CYP19A1 | 1 | 32000 | IC50 |
PMID: 18192087 |
NPC51700 | PTPN6 | 1 | 25780 | IC50 |
PMID: 18707891 |
NPC51700 | POLB | 1 | 18600 | IC50 |
PMID: 15165161 |
NPC51700 | CTSD | 1 | 18200 | IC50 |
DOI: 10.1007/s00044-012-0397-z |
NPC51700 | SLCO1B1 | 1 | 15848.93 | IC50 |
PMID: 23571415 |
NPC58616 | ALDH1A1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | HPGD | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | MAPK1 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | RECQL | 2 |
Median: 77689.6 Range: 14125.4 to 141253.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC70744 | KDM4E | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC71074 | PTPN6 | 1 | 24560 | IC50 |
PMID: 18707891 |
NPC71074 | PYGM | 1 | 20000 | IC50 |
PMID: 16169219 |
NPC7491 | CYP2C9 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC76336 | GLA | 2 |
Median: 40074.85 Range: 35481.3 to 44668.4 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC76336 | GAA | 2 |
Median: 40074.85 Range: 35481.3 to 44668.4 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC76336 | RECQL | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC76336 | CA13 | 1 | 17800 | Ki |
PMID: 22892213 |
NPC81010 | ESR1 | 1 | 16120 | EC50 |
PMID: 23608764 |
NPC84319 | PYGM | 1 | 28000 | IC50 |
PMID: 16169219 |
NPC84319 | PTPN2 | 1 | 19470 | IC50 |
PMID: 19846303 |
NPC85813 | CYP19A1 | 1 | 48000 | IC50 |
PMID: 16643058 |
NPC85813 | F3 | 1 | 41000 | IC50 |
PMID: 9834151 |
NPC85813 | HSD17B10 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC85813 | TSHR | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC85813 | CYP3A4 | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC85813 | ALDH1A1 | 1 | 17782.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | RECQL | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | ALOX15 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | CASP7 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | CASP1 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | MAPK1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | CYP3A4 | 2 |
Median: 19952.6 Range: 19952.6 to 19952.6 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC94167 | HSD17B10 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC1075 | KDM4E | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC110899 | CA4 | 1 | 10600 | Ki |
PMID: 20185318 |
NPC126029 | CYP3A4 | 2 |
Median: 12589.3 Range: 12589.3 to 12589.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC126029 | KDM4E | 2 |
Median: 16803.7 Range: 11220.2 to 22387.2 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC142415 | PTPRF | 2 |
Median: 17055 Range: 11800 to 22310 |
IC50 |
PMID: 21453996 PMID: 27123900 |
NPC142415 | PTPN11 | 1 | 11620 | IC50 |
PMID: 27123900 |
NPC156461 | MAPK1 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CA5B | 1 | 12700 | Ki |
PMID: 20185318 |
NPC178134 | MAPT | 8 |
Median: 21169.9 Range: 12589.3 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | TP53 | 2 |
Median: 22106.05 Range: 12589.3 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | KMT2A | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CA3 | 1 | 10500 | Ki |
PMID: 20185318 |
NPC179950 | ALPL | 1 | 14000 | IC50 |
PubChem BioAssay data set CHEMBL1201862 |
NPC179950 | KDM4E | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC18335 | XDH | 1 | 10890 | IC50 |
PMID: 17379526 |
NPC201844 | ALDH1A1 | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | ALDH1A1 | 2 |
Median: 15954.1 Range: 14125.4 to 17782.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | CA3 | 2 |
Median: 13000 Range: 13000 to 13000 |
Ki |
PMID: 18579385 PMID: 20185318 |
NPC204932 | SMN1;SMN2 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | HIF1A | 2 |
Median: 12589.3 Range: 12589.3 to 12589.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | LMNA | 2 |
Median: 23350.75 Range: 11220.2 to 35481.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | HPGD | 2 |
Median: 14501.5 Range: 11220.2 to 17782.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | GMNN | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC204932 | CA4 | 3 |
Median: 10900 Range: 10900 to 10900 |
Ki |
PMID: 18579385 PMID: 20185318 PMID: 22245047 |
NPC20791 | LMNA | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | PIK3CG | 1 | 13790 | IC50 |
PMID: 25050878 |
NPC20791 | PREP | 1 | 13000 | IC50 |
PMID: 18650094 |
NPC20791 | LCK | 2 |
Median: 13000 Range: 13000 to 13000 |
IC50 |
PMID: 1995903 PMID: 16441060 |
NPC20791 | CALM1;CALM2;CALM3 | 1 | 12970 | IC50 |
PMID: 21129983 |
NPC20791 | PLAU | 1 | 12100 | IC50 |
PMID: 24610996 |
NPC20791 | CA5B | 1 | 11900 | Ki |
PMID: 20185318 |
NPC20791 | CYP2C19 | 1 | 10500 | IC50 |
PMID: 22328583 |
NPC20791 | MMP12 | 1 | 10230 | IC50 |
PMID: 22658537 |
NPC20791 | HIF1AN | 1 | 10200 | IC50 |
PMID: 19822432 |
NPC20791 | CYP2C9 | 1 | 10200 | IC50 |
PMID: 22328583 |
NPC219876 | KDM4E | 2 |
Median: 19622.15 Range: 14125.4 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | POLB | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | FUT4 | 1 | 14000 | IC50 |
DOI: 10.1039/C4MD00086B |
NPC257124 | ALDH1A1 | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC257124 | PTGS1 | 1 | 11000 | IC50 |
PMID: 16038536 |
NPC261831 | KCNH2 | 1 | 10410 | EC50 |
PubChem BioAssay data set CHEMBL1201862 |
NPC264317 | AKR1B1 | 1 | 11000 | IC50 |
PMID: 21561086 |
NPC293378 | ALDH1A1 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294548 | HSD17B10 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | THRB | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | CA4 | 1 | 10100 | Ki |
PMID: 20185318 |
NPC29883 | CA2 | 2 |
Median: 10600 Range: 10600 to 10600 |
Ki |
PMID: 18501600 PMID: 18579385 |
NPC328740 | APEX1 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | LMNA | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC41326 | NR1I2 | 1 | 12000 | IC50 |
PMID: 24828006 |
NPC51700 | SLCO1B3 | 1 | 11481.54 | IC50 |
PMID: 23571415 |
NPC61477 | MAPT | 2 |
Median: 14125.4 Range: 14125.4 to 14125.4 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | ALOX15 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | CA14 | 1 | 11550 | Ki |
PMID: 20674354 |
NPC61477 | KDM4E | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | CA13 | 1 | 10510 | Ki |
PMID: 20674354 |
NPC70744 | CA3 | 1 | 11100 | Ki |
PMID: 20185318 |
NPC70744 | CA4 | 1 | 10800 | Ki |
PMID: 20185318 |
NPC70744 | CA5B | 1 | 10500 | Ki |
PMID: 20185318 |
NPC71074 | POLB | 1 | 12600 | IC50 |
PMID: 15165161 |
NPC71074 | HTT | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC71074 | PTPN2 | 1 | 11310 | IC50 |
PMID: 18707891 |
NPC7491 | CYP2C19 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC76336 | HIF1A | 2 |
Median: 12589.3 Range: 12589.3 to 12589.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC76336 | CA1 | 1 | 10560 | Ki |
PMID: 22892213 |
NPC81010 | HCAR2 | 1 | 14000 | Ki |
PMID: 21167710 |
NPC85813 | FABP4 | 2 |
Median: 15650 Range: 13600 to 17700 |
IC50 |
PMID: 20471252 PMID: 25461324 |
NPC85813 | PTGS1 | 1 | 13000 | IC50 |
PMID: 16038536 |
NPC94167 | HPGD | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |