Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC138113 TSHR 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC13826 POLB 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC13826 MAPT 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC13826 RAD52 1 15210 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC13991 MAPK1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC149184 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC149184 PPARD 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC149184 PPARA 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC158853 KDM4E 2 Median: 25665.1
Range: 15848.9 to 35481.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC195268 ALOX15 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC195268 ACHE 1 24330 IC50 PMID: 16483771
NPC202605 CYP3A4 1 30600 IC50 PMID: 17994701
NPC203719 HPGD 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC203719 ABAT 1 17100 IC50 PMID: 16290145
NPC203719 ALDH5A1 1 15600 IC50 PMID: 16290145
NPC203719 ALDH1A1 2 Median: 19622.15
Range: 14125.4 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC208936 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC208936 TSHR 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC209970 ALOX15 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC209970 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC209970 TDP1 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC209970 HSD17B10 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC216630 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC261831 BLM 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC261831 CYP19A1 1 32700 IC50 PMID: 16643058
NPC261831 TOP1 1 31000 IC50 PMID: 12444712
NPC261831 MAPT 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC261831 FABP4 1 26100 IC50 PMID: 20471252
NPC261831 KMT2A 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC261831 ATM 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC261831 HSD17B10 2 Median: 17900.75
Range: 15848.9 to 19952.6
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC273410 PTPN1 1 23600 IC50 PMID: 23177789
NPC294548 CYP19A1 1 44200 IC50 PMID: 16643058
NPC294548 BLM 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294548 L3MBTL1 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294548 F3 1 30000 IC50 PMID: 9834151
NPC294548 HPGD 2 Median: 28183.8
Range: 28183.8 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC294548 MAPT 3 Median: 28183.8
Range: 28183.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC294548 LMNA 1 22387.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294548 PLA2G1B 1 22300 IC50 PubChem BioAssay data set
CHEMBL1201862
NPC294548 KDM4E 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294548 PPARD 1 16000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC294548 CYP3A4 2 Median: 15848.9
Range: 15848.9 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC294548 ATG4B 1 15300 IC50 PubChem BioAssay data set
CHEMBL1201862
NPC301585 PPARD 1 24000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC301585 PPARG 1 21000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC301696 ALDH1A1 1 44668.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC49075 HSD17B10 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC49075 PDE1A 1 22000 IC50 PMID: 1955879
NPC49075 CYP3A4 2 Median: 19952.6
Range: 19952.6 to 19952.6
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC53069 ALDH1A1 1 44668.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC53069 TERT 1 37000 IC50 PMID: 22336246
NPC6095 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC75179 CYP2D6 1 32000 Ki PMID: 16248836
NPC85813 CYP19A1 1 48000 IC50 PMID: 16643058
NPC85813 F3 1 41000 IC50 PMID: 9834151
NPC85813 HSD17B10 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC85813 TSHR 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC85813 CYP3A4 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC85813 ALDH1A1 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC13826 KDM4E 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC13826 LMNA 1 11220.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC16452 HIF1A 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC16452 CYP2D6 1 12589.25 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC195268 CYP2C9 2 Median: 26200
Range: 12589.3 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC195268 THPO 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC195268 USP2 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC261831 KCNH2 1 10410 EC50 PubChem BioAssay data set
CHEMBL1201862
NPC294548 HSD17B10 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC51758 ALOX15 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC53069 CYP3A4 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC53069 TSHR 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC53069 MAPT 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC66775 MIF 1 11000 IC50 PMID: 25743213
NPC85813 FABP4 2 Median: 15650
Range: 13600 to 17700
IC50 PMID: 20471252
PMID: 25461324
NPC85813 PTGS1 1 13000 IC50 PMID: 16038536