Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC127447 TSHR 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC187432 CYP2D6 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC187432 ADORA2A 2 Median: 17400
Range: 16700 to 18100
Ki PMID: 9258366
PMID: 9258366
NPC187432 CYP3A4 2 Median: 15848.9
Range: 15848.9 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC78540 CALM1;CALM2;CALM3 1 33430 IC50 PMID: 21129983
NPC78540 MAPK1 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC78540 KDM4E 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC78540 PTGS2 1 25500 IC50 PMID: 24332492
NPC78540 TP53 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC94045 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC94045 CYP3A4 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC94045 HPGD 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC94045 SMN1;SMN2 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC94045 USP2 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC94045 KDM4E 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC94045 HSD17B10 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC94045 MAPT 2 Median: 24068.2
Range: 19952.6 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC94045 TRPV1 3 Median: 23700
Range: 15000 to 30000
IC50 PMID: 26750258
PMID: 26750258
PMID: 26750258
NPC187432 MAPT 2 Median: 14501.5
Range: 11220.2 to 17782.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC78540 CYP2D6 1 12589.25 AC50 PubChem BioAssay data set
CHEMBL1201862