Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC137419 KDM4E 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC158028 CYP2A6 2 Median: 26000.8
Range: 26000 to 26001.6
IC50 PMID: 15658857
PMID: 19110342
NPC182570 MAPT 2 Median: 22387.2
Range: 22387.2 to 22387.2
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC182570 CHRNA1 1 21000 IC50 PMID: 11312774
NPC182570 TRPA1 1 17000 EC50 PMID: 20356305
NPC182570 ALDH1A1 3 Median: 28183.8
Range: 15848.9 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC256853 KDM4E 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC256853 CYP3A4 2 Median: 19952.6
Range: 19952.6 to 19952.6
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC260491 MAPT 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC260491 RECQL 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC260491 KDM4E 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862