Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC117237 ALDH1A1 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC117237 AOX1 1 15000 IC50 PMID: 20853847
NPC157340 ALDH1A1 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC158853 KDM4E 2 Median: 25665.1
Range: 15848.9 to 35481.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC163984 ALDH1A1 2 Median: 25285.5
Range: 22387.2 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC216630 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC235059 MAPK1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC243728 POLB 1 26500 IC50 PMID: 15165161
NPC250999 MAPT 2 Median: 35716.75
Range: 31622.8 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC250999 HPGD 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC2518 ATM 1 44668.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC2518 THRB 2 Median: 34893.65
Range: 25118.9 to 44668.4
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC257124 AR 2 Median: 19027.305
Range: 19000 to 19054.61
IC50 PMID: 20226658
PMID: 20226658
NPC305039 SMN1;SMN2 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC305039 LMNA 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC86412 L3MBTL1 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC86412 LMNA 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC250999 HSD17B10 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC257124 ALDH1A1 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC257124 PTGS1 1 11000 IC50 PMID: 16038536
NPC259134 CYP3A4 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC29883 CA2 2 Median: 10600
Range: 10600 to 10600
Ki PMID: 18501600
PMID: 18579385
NPC305039 MAPT 1 11220.2 Potency PubChem BioAssay data set
CHEMBL1201862