Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC246162 APP 1 33000 IC50 PMID: 26719209
NPC246162 BACE1 2 Median: 32500
Range: 30000 to 35000
IC50 PMID: 14592472
PMID: 14592472
NPC246162 RECQL 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC246162 KDM4E 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC246162 MAPT 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC246162 KIT 2 Median: 18800
Range: 15700 to 21900
IC50 PMID: 26807861
PMID: 26807861
NPC32441 GSK3B 1 45700 IC50 DOI: 10.1007/s00044-012-0353-y
NPC32441 AKR1B1 1 28870 IC50 PMID: 22261024
NPC32441 CYP1A2 1 26339 IC50 PMID: 20696580
NPC32441 CALM1;CALM2;CALM3 1 22010 IC50 PMID: 21129983
NPC32441 CBR1 1 21480 IC50 PMID: 19097799
NPC32441 HSD17B10 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC32441 CYP1A1 1 15167 IC50 PMID: 20696580
NPC32441 HSD17B2 1 14400 IC50 PMID: 18533708
NPC32441 ESR2 1 13473 IC50 PMID: 17149865
NPC32441 CYP2C9 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862