Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC293454 PNLIP 1 36000 IC50 PMID: 17521912
NPC293454 HPGD 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC293454 ALDH1A1 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC315634 TDP1 2 Median: 49489.2
Range: 28183.8 to 70794.6
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC315634 KDM4E 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC315634 MAPT 2 Median: 22016.35
Range: 15848.9 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC471593 CYP3A4 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PMID: 20155971
DrugMatrix in vitro pharmacology data
CHEMBL1909046
NPC471593 BLM 2 Median: 28183.8
Range: 28183.8 to 28183.8
Potency PMID: 14640513
PMID: 20384317
NPC471593 CYP2C9 1 25118.86 AC50 PMID: 23327759
NPC471593 TSHR 2 Median: 19952.6
Range: 19952.6 to 19952.6
Potency PMID: 19128055
PMID: 22280481
NPC71074 PTPN6 1 24560 IC50 PMID: 18707891
NPC71074 PYGM 1 20000 IC50 PMID: 16169219
NPC88923 PMP22 1 47754.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 THPO 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC88923 HBB 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 POLB 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 L3MBTL1 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 KMT2A 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 ABCG2 1 26302.68 IC50 PMID: 18678495
NPC88923 HSD17B10 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 KDM4E 1 22387.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 ALDH1A1 2 Median: 29881.65
Range: 19952.6 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC88923 ALOX15 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 LMNA 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 BLM 2 Median: 17782.8
Range: 17782.8 to 17782.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC88923 TSHR 2 Median: 15848.9
Range: 15848.9 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC71074 POLB 1 12600 IC50 PMID: 15165161
NPC71074 HTT 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC71074 PTPN2 1 11310 IC50 PMID: 18707891
NPC84786 PNLIP 1 13000 IC50 PMID: 17521912
NPC88923 MAPT 2 Median: 13357.35
Range: 12589.3 to 14125.4
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC88923 GMNN 1 11220.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC88923 ABCB11 1 10200 IC50 PMID: 12739759