Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC100079 RAB9A 1 46109.1 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 CYP2C9 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 CYP3A4 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC100079 MAPK1 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 HIF1A 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC100079 USP2 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 TSHR 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC100079 CYP2D6 1 25118.86 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC100079 HPGD 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 ALOX15 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 HSD17B10 2 Median: 22535.75
Range: 19952.6 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC100079 ALDH1A1 2 Median: 19118.05
Range: 15848.9 to 22387.2
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC100079 MAPT 4 Median: 15848.9
Range: 14125.4 to 17782.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC1075 CYP2C9 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC111132 TSHR 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC118633 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC118633 LMNA 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC125732 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC125732 CYP2C19 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC125732 KDM4E 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC125732 HTR3A 1 26000 EC50 PMID: 18033297
NPC133671 P4HB 1 19020 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC173637 PIM2 1 25000 IC50 PMID: 18163587
NPC173637 L3MBTL1 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC173637 XDH 1 14740 IC50 PMID: 12444671
NPC176740 MAPT 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC176740 EPHX2 1 24300 IC50 PMID: 24679441
NPC176740 KDM4E 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC179950 EPHX2 1 28430 IC50 PMID: 24679441
NPC179950 XDH 1 26310 IC50 PMID: 12444671
NPC179950 MAPT 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC181465 XDH 1 14800 IC50 PMID: 9461655
NPC265885 RECQL 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC265885 GAA 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC265885 L3MBTL1 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294902 HPGD 3 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC294902 ALDH1A1 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC294902 APEX1 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294902 APP 1 32800 IC50 PMID: 22921742
NPC294902 AKR1B1 1 32000 IC50 PMID: 22236472
NPC294902 CYP3A4 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC294902 POLB 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC303581 KDM4E 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC308267 KDM4E 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC308267 CYP3A4 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC46451 RAB9A 1 46109.1 Potency PubChem BioAssay data set
CHEMBL1201862
NPC46451 RGS12 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC46451 MAPK1 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC46451 USP2 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC46451 ALDH1A1 1 22387.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC46451 BAD 1 19000 IC50 PMID: 18925736
NPC46451 MAPT 2 Median: 22983.3
Range: 17782.8 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC46451 CYP2C9 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC53069 ALDH1A1 1 44668.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC53069 TERT 1 37000 IC50 PMID: 22336246
NPC67978 KMT2A 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC70744 KDM4E 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC81010 ESR1 1 16120 EC50 PMID: 23608764
NPC93730 MAPK1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93730 CYP3A4 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC93730 KDM4E 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93730 LMNA 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93730 AR 1 23500 IC50 PMID: 19592245
NPC100079 ALOX12 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC100079 NFKB1 2 Median: 11220.2
Range: 11220.2 to 11220.2
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC1075 KDM4E 1 11220.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC125732 L3MBTL1 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC179950 ALPL 1 14000 IC50 PubChem BioAssay data set
CHEMBL1201862
NPC179950 KDM4E 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC293378 ALDH1A1 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294902 THRB 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC294902 CA4 1 10100 Ki PMID: 20185318
NPC29883 CA2 2 Median: 10600
Range: 10600 to 10600
Ki PMID: 18501600
PMID: 18579385
NPC308267 TSHR 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC46451 HPGD 2 Median: 21154.6
Range: 14125.4 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC46451 TSHR 4 Median: 18854.1
Range: 12589.3 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC46451 SMN1;SMN2 2 Median: 16803.7
Range: 11220.2 to 22387.2
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC53069 CYP3A4 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC53069 TSHR 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC53069 MAPT 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC70744 CA3 1 11100 Ki PMID: 20185318
NPC70744 CA4 1 10800 Ki PMID: 20185318
NPC70744 CA5B 1 10500 Ki PMID: 20185318
NPC81010 HCAR2 1 14000 Ki PMID: 21167710
NPC93730 TP53 2 Median: 14219.1
Range: 12589.3 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862