Plant ingredients against the target with activities between 10uM and 50uM
Ingredient ID | Target (Gene Symbol) | No. of Activity Values | Activity Value (nM) | Activity Type | Activity Reference |
---|---|---|---|---|---|
NPC116775 | BCHE | 1 | 43100 | Ki |
PMID: 19879672 |
NPC116775 | ALDH1A1 | 2 |
Median: 35716.75 Range: 31622.8 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | HPGD | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | CDK6 | 2 |
Median: 22000 Range: 22000 to 22000 |
IC50 |
PMID: 15689157 DOI: 10.1007/s00044-009-9233-5 |
NPC116775 | GLO1 | 1 | 20600 | IC50 |
PMID: 18258440 |
NPC116775 | KDM4E | 2 |
Median: 27829.8 Range: 15848.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | HSD17B10 | 2 |
Median: 15848.9 Range: 15848.9 to 15848.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | BACE1 | 1 | 14700 | IC50 |
DOI: 10.1007/s00044-012-0353-y |
NPC142415 | ACP1 | 4 |
Median: 22050 Range: 21200 to 22900 |
IC50 |
PMID: 21453996 PMID: 21453996 PMID: 25264584 PMID: 25264584 |
NPC142415 | PTPN6 | 2 |
Median: 22760 Range: 14190 to 31330 |
IC50 |
PMID: 18707891 PMID: 27123900 |
NPC161571 | POLB | 1 | 44668.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC161571 | PMP22 | 1 | 42561.5 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC161571 | GAA | 1 | 39506.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC161571 | CYP1A1 | 1 | 34000 | IC50 |
PMID: 27265259 |
NPC161571 | HSD17B10 | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC161571 | ALDH1A1 | 4 |
Median: 37646 Range: 31622.8 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC161571 | MAOB | 1 | 29370 | IC50 |
DOI: 10.1039/C3MD00376K |
NPC161571 | BCR | 1 | 28000 | IC50 |
PMID: 16686543 |
NPC161571 | CYP19A1 | 2 |
Median: 25000 Range: 25000 to 25000 |
IC50 |
PMID: 22115839 PMID: 22386564 |
NPC161571 | SIRT1 | 3 |
Median: 46200 Range: 23600 to 87200 |
EC50 |
PMID: 18046409 PMID: 23316803 PMID: 23316803 |
NPC161571 | KDM4E | 4 |
Median: 28370.85 Range: 22387.2 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC161571 | RELA | 1 | 20000 | IC50 |
Patent: Patent: US20130178536 A1 |
NPC161571 | ODC1 | 1 | 19000 | IC50 |
PMID: 10075742 |
NPC20791 | PMP22 | 1 | 47754.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | THRB | 1 | 44668.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | GALK1 | 1 | 42128.5 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CDK2 | 1 | 40000 | IC50 |
PMID: 17178224 |
NPC20791 | CD38 | 1 | 37900 | IC50 |
PMID: 21641214 |
NPC20791 | SORD | 2 |
Median: 106300 Range: 35600 to 177000 |
IC50 |
PMID: 8893834 PMID: 12672241 |
NPC20791 | SMN1;SMN2 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | EPHX2 | 1 | 33540 | IC50 |
PMID: 24679441 |
NPC20791 | DPP4 | 2 |
Median: 81365 Range: 32730 to 130000 |
IC50 |
PMID: 18650094 DOI: 10.1039/C0MD00245C |
NPC20791 | MAPK1 | 2 |
Median: 35716.75 Range: 31622.8 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | ADORA3 | 1 | 30000 | Ki |
PMID: 8576921 |
NPC20791 | PTGS2 | 1 | 28600 | IC50 |
PMID: 17378609 |
NPC20791 | BLM | 3 |
Median: 28183.8 Range: 28183.8 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | TDP1 | 2 |
Median: 26651.35 Range: 25118.9 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | ALDH1A1 | 6 |
Median: 37646 Range: 25118.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CDK6 | 2 |
Median: 25000 Range: 25000 to 25000 |
IC50 |
PMID: 15689157 DOI: 10.1007/s00044-009-9233-5 |
NPC20791 | PTPN1 | 2 |
Median: 23300 Range: 23300 to 23300 |
IC50 |
PMID: 12419367 PMID: 19297174 |
NPC20791 | KMT2A | 1 | 22387.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | AMY1A;AMY1B;AMY1C | 1 | 21400 | IC50 |
PMID: 18507367 |
NPC20791 | SYK | 1 | 20000 | IC50 |
PMID: 22257213 |
NPC20791 | HPGD | 2 |
Median: 21169.9 Range: 19952.6 to 22387.2 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | APEX1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CYP2D6 | 1 | 18800 | IC50 |
PMID: 22328583 |
NPC20791 | USP2 | 2 |
Median: 25057.75 Range: 18492.7 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | GPR35 | 1 | 15400 | IC50 |
PMID: 24900447 |
NPC20791 | APP | 1 | 15300 | IC50 |
PMID: 26719209 |
NPC229649 | FASN | 1 | 25400 | IC50 |
PMID: 16870425 |
NPC248573 | ALOX15 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC248573 | HPGD | 2 |
Median: 25665.1 Range: 15848.9 to 35481.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC248573 | SMN1;SMN2 | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC290466 | FASN | 1 | 31000 | IC50 |
PMID: 16870425 |
NPC4154 | BACE1 | 1 | 36470 | IC50 |
PMID: 20462757 |
NPC473210 | FASN | 1 | 28700 | IC50 |
PMID: 20886871 |
NPC473211 | FASN | 1 | 23100 | IC50 |
PMID: 20886871 |
NPC473212 | FASN | 1 | 29700 | IC50 |
PMID: 20886871 |
NPC473213 | FASN | 1 | 32600 | IC50 |
PMID: 23270663 |
NPC71074 | PTPN6 | 1 | 24560 | IC50 |
PMID: 18707891 |
NPC71074 | PYGM | 1 | 20000 | IC50 |
PMID: 16169219 |
NPC84319 | PYGM | 1 | 28000 | IC50 |
PMID: 16169219 |
NPC84319 | PTPN2 | 1 | 19470 | IC50 |
PMID: 19846303 |
NPC84772 | FASN | 1 | 49100 | IC50 |
PMID: 16870425 |
NPC85813 | CYP19A1 | 1 | 48000 | IC50 |
PMID: 16643058 |
NPC85813 | F3 | 1 | 41000 | IC50 |
PMID: 9834151 |
NPC85813 | HSD17B10 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC85813 | TSHR | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC85813 | CYP3A4 | 2 |
Median: 31622.8 Range: 31622.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC85813 | ALDH1A1 | 1 | 17782.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | MAPT | 2 |
Median: 14219.1 Range: 12589.3 to 15848.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC142415 | PTPRF | 2 |
Median: 17055 Range: 11800 to 22310 |
IC50 |
PMID: 21453996 PMID: 27123900 |
NPC142415 | PTPN11 | 1 | 11620 | IC50 |
PMID: 27123900 |
NPC20791 | LMNA | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | PIK3CG | 1 | 13790 | IC50 |
PMID: 25050878 |
NPC20791 | PREP | 1 | 13000 | IC50 |
PMID: 18650094 |
NPC20791 | LCK | 2 |
Median: 13000 Range: 13000 to 13000 |
IC50 |
PMID: 1995903 PMID: 16441060 |
NPC20791 | CALM1;CALM2;CALM3 | 1 | 12970 | IC50 |
PMID: 21129983 |
NPC20791 | PLAU | 1 | 12100 | IC50 |
PMID: 24610996 |
NPC20791 | CA5B | 1 | 11900 | Ki |
PMID: 20185318 |
NPC20791 | CYP2C19 | 1 | 10500 | IC50 |
PMID: 22328583 |
NPC20791 | MMP12 | 1 | 10230 | IC50 |
PMID: 22658537 |
NPC20791 | HIF1AN | 1 | 10200 | IC50 |
PMID: 19822432 |
NPC20791 | CYP2C9 | 1 | 10200 | IC50 |
PMID: 22328583 |
NPC248573 | MAPT | 2 |
Median: 14125.4 Range: 14125.4 to 14125.4 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC248573 | THPO | 2 |
Median: 12589.3 Range: 12589.3 to 12589.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC248573 | KDM4E | 2 |
Median: 20386.55 Range: 12589.3 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC248573 | HSD17B10 | 4 |
Median: 12589.3 Range: 12589.3 to 12589.3 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC71074 | POLB | 1 | 12600 | IC50 |
PMID: 15165161 |
NPC71074 | HTT | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC71074 | PTPN2 | 1 | 11310 | IC50 |
PMID: 18707891 |
NPC85813 | FABP4 | 2 |
Median: 15650 Range: 13600 to 17700 |
IC50 |
PMID: 20471252 PMID: 25461324 |
NPC85813 | PTGS1 | 1 | 13000 | IC50 |
PMID: 16038536 |