Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC476440 HTT 1 35481.3 Potency PMID: 22260257
NPC476440 TSHR 1 31622.8 Potency PMID: 26355532
NPC476440 PMP22 1 30131.3 Potency PMID: 19064900
NPC476440 HIF1A 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PMID: 11543673
DrugMatrix in vitro pharmacology data
CHEMBL1909046
NPC476440 MAPK1 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC476440 CYP2C9 1 19952.6 Potency PMID: 9733489
NPC476440 HPGD 2 Median: 18867.7
Range: 17782.8 to 19952.6
Potency PMID: 19459694
DrugMatrix in vitro pharmacology data
CHEMBL1909046
NPC476440 MTOR 4 Median: 19620.9
Range: 16481.6 to 23280.9
Potency PMID: 2578192
PMID: 11931609
PMID: 18417256
PMID: 22070654
NPC476440 PADI4 1 13000 IC50 PMID: 9461657
NPC476440 NPSR1 2 Median: 16270.95
Range: 12589.3 to 19952.6
Potency PMID: 18183025
PMID: 19105653
NPC476440 CYP1A2 1 12589.25 AC50 PMID: 18332176