Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC116775 BCHE 1 43100 Ki PMID: 19879672
NPC116775 ALDH1A1 2 Median: 35716.75
Range: 31622.8 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC116775 HPGD 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC116775 CDK6 2 Median: 22000
Range: 22000 to 22000
IC50 PMID: 15689157
DOI: 10.1007/s00044-009-9233-5
NPC116775 GLO1 1 20600 IC50 PMID: 18258440
NPC116775 KDM4E 2 Median: 27829.8
Range: 15848.9 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC116775 HSD17B10 2 Median: 15848.9
Range: 15848.9 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC116775 BACE1 1 14700 IC50 DOI: 10.1007/s00044-012-0353-y
NPC278175 ALOX12 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC278175 HPGD 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC278175 ALOX15 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC278175 USP2 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC278175 CYP1A2 1 31622.78 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC278175 ALDH1A1 1 22387.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC278175 KDM4E 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC312929 KDM4E 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC312929 GLA 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC312929 ALDH1A1 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC3224 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC70622 EPHX2 1 26800 IC50 PMID: 26372074
NPC116775 MAPT 2 Median: 14219.1
Range: 12589.3 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC278175 TDP1 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC278175 TP53 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC312929 HPGD 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC312929 ALOX15 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862