Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC107482 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC110899 CA5B 1 35400 Ki PMID: 20185318
NPC125417 TPMT 1 19952.62 IC50 PMID: 3950915
NPC131885 ALDH1A1 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC131885 KDM4E 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC131885 HPGD 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC144682 ALDH1A1 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC156654 L3MBTL1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC156654 KDM4E 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC156654 POLB 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC201844 PPARA 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC201844 PPARD 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC201844 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC203719 HPGD 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC203719 ABAT 1 17100 IC50 PMID: 16290145
NPC203719 ALDH5A1 1 15600 IC50 PMID: 16290145
NPC203719 ALDH1A1 2 Median: 19622.15
Range: 14125.4 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC209970 ALOX15 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC209970 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC209970 TDP1 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC209970 HSD17B10 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC210460 ABCB1 1 32000 IC50 DOI: 10.1039/C4MD00196F
NPC210460 MAPT 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC216630 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC230301 DPP4 1 28840 IC50 DOI: 10.1039/C0MD00245C
NPC230301 POLB 1 26300 IC50 PMID: 14640519
NPC234536 HPGD 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC234536 KDM4E 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC234536 POLB 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC257490 HPGD 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC27633 ESR1 1 38200 EC50 PMID: 23608764
NPC279026 TSHR 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC279026 PPARD 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC279026 PPARA 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC279026 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC301585 PPARD 1 24000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC301585 PPARG 1 21000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC34770 ALDH1A1 2 Median: 29903.3
Range: 28183.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC34770 TP53 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC34770 CYP2D6 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC41721 MAPT 1 44668.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC41721 HSD17B10 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC41721 HPGD 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC41721 ALDH1A1 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC41721 CYP3A4 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC41721 KDM4E 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC70290 CYP1A2 1 25118.86 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC70744 KDM4E 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC74458 ALDH1A1 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC74539 KDM4E 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC74539 HSD17B10 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC74539 ALDH1A1 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC76336 GLA 2 Median: 40074.85
Range: 35481.3 to 44668.4
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC76336 GAA 2 Median: 40074.85
Range: 35481.3 to 44668.4
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC76336 RECQL 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC76336 CA13 1 17800 Ki PMID: 22892213
NPC81010 ESR1 1 16120 EC50 PMID: 23608764
NPC85813 CYP19A1 1 48000 IC50 PMID: 16643058
NPC85813 F3 1 41000 IC50 PMID: 9834151
NPC85813 HSD17B10 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC85813 TSHR 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC85813 CYP3A4 2 Median: 31622.8
Range: 31622.8 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC85813 ALDH1A1 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93653 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93653 SMN1;SMN2 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93653 KDM4E 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC93653 HPGD 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC110899 CA4 1 10600 Ki PMID: 20185318
NPC201844 ALDH1A1 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC29883 CA2 2 Median: 10600
Range: 10600 to 10600
Ki PMID: 18501600
PMID: 18579385
NPC34770 HPGD 2 Median: 14125.4
Range: 14125.4 to 14125.4
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC34770 HSD17B10 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC34770 KDM4E 2 Median: 13357.35
Range: 12589.3 to 14125.4
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC70290 TSHR 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC70744 CA3 1 11100 Ki PMID: 20185318
NPC70744 CA4 1 10800 Ki PMID: 20185318
NPC70744 CA5B 1 10500 Ki PMID: 20185318
NPC74539 MAOA 1 13800 IC50 PMID: 23517722
NPC74539 CYP2A6 1 12000 Ki PMID: 16248836
NPC76336 HIF1A 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC76336 CA1 1 10560 Ki PMID: 22892213
NPC81010 HCAR2 1 14000 Ki PMID: 21167710
NPC85813 FABP4 2 Median: 15650
Range: 13600 to 17700
IC50 PMID: 20471252
PMID: 25461324
NPC85813 PTGS1 1 13000 IC50 PMID: 16038536