Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC146373 CYP2A6 1 32400 IC50 Patent: Patent: US8609708 B2
NPC15864 PKM 2 Median: 28183.8
Range: 28183.8 to 28183.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC166424 SMN1;SMN2 1 14125.4 Potency PubChem BioAssay data set
CHEMBL1201862
NPC188231 KDM4E 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC193536 CA12 1 44100 Ki PMID: 20590092
NPC193536 TSHR 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC193536 CYP1A2 1 31622.78 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC193536 MTOR 2 Median: 24701.25
Range: 23280.9 to 26121.6
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC207554 KMT2A 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC207554 MAPT 1 17782.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC208936 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC208936 TSHR 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC209296 KMT2A 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC209296 POLB 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC249797 CYP1A2 1 15848.93 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC249797 CASP1 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC48564 CYP2A6 1 26300 IC50 Patent: Patent: US8609708 B2
NPC81010 ESR1 1 16120 EC50 PMID: 23608764
NPC96102 CYP3A4 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC96102 CYP2D6 1 31622.78 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC96102 CYP2A13 1 16000 Ki PMID: 22696418
NPC96102 CTSK 1 15000 IC50 PMID: 11975521
NPC193536 ALOX15 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC193536 CYP2C9 1 12589.25 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC193536 CA3 1 11500 Ki PMID: 20590092
NPC207554 HTT 1 11220.2 Potency PubChem BioAssay data set
CHEMBL1201862
NPC245244 CYP2D6 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC249797 KDM4E 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC249797 CYP3A4 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC81010 HCAR2 1 14000 Ki PMID: 21167710
NPC96102 NFKB1 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862