Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC10251 L3MBTL1 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC107482 ALDH1A1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC137958 CYP1A2 1 39810.72 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC137958 SLC1A3 1 35000 Ki PMID: 18578477
NPC142415 ACP1 4 Median: 22050
Range: 21200 to 22900
IC50 PMID: 21453996
PMID: 21453996
PMID: 25264584
PMID: 25264584
NPC142415 PTPN6 2 Median: 22760
Range: 14190 to 31330
IC50 PMID: 18707891
PMID: 27123900
NPC216630 PPARG 1 30000 IC50 DOI: 10.1007/s00044-012-0285-6
NPC230301 DPP4 1 28840 IC50 DOI: 10.1039/C0MD00245C
NPC230301 POLB 1 26300 IC50 PMID: 14640519
NPC243728 POLB 1 26500 IC50 PMID: 15165161
NPC273330 CYP1A2 1 31622.78 AC50 PubChem BioAssay data set
CHEMBL1201862
NPC273330 CYP3A4 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC282923 BRCA1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC282923 CYP3A4 2 Median: 25118.9
Range: 25118.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC282923 USP2 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC282923 KDM4E 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC282923 TDP1 1 19952.6 Potency PubChem BioAssay data set
CHEMBL1201862
NPC282923 ELANE 1 18000 IC50 PMID: 1578486
NPC282923 TSHR 2 Median: 15848.9
Range: 15848.9 to 15848.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC10251 TSHR 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC141953 TSHR 2 Median: 12589.3
Range: 12589.3 to 12589.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC142415 PTPRF 2 Median: 17055
Range: 11800 to 22310
IC50 PMID: 21453996
PMID: 27123900
NPC142415 PTPN11 1 11620 IC50 PMID: 27123900
NPC153556 RGS12 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC282923 ALDH1A1 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862