Putative targets based on weak experimental activity

Plant ingredients against the target with activities between 10uM and 50uM


Ingredient ID Target (Gene Symbol) No. of Activity Values Activity Value (nM) Activity Type Activity Reference
NPC102810 MAPK1 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC102810 KDM4E 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC102810 MAPT 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC102810 HSD17B10 1 31622.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC102810 ALDH1A1 1 29906.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC102810 TP53 2 Median: 25787.7
Range: 19952.6 to 31622.8
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC102810 USP2 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC264317 POLB 2 Median: 44925
Range: 43600 to 46250
IC50 PMID: 14640519
PMID: 18343122
NPC264317 GLI1 2 Median: 32000
Range: 32000 to 32000
IC50 PMID: 18842418
PMID: 19309080
NPC55422 CYP3A4 2 Median: 39810.7
Range: 39810.7 to 39810.7
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC55422 KDM4E 1 39810.7 Potency PubChem BioAssay data set
CHEMBL1201862
NPC55422 HPGD 1 35481.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC55422 BLM 1 28183.8 Potency PubChem BioAssay data set
CHEMBL1201862
NPC55422 HSD17B10 1 25118.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC55422 MAPT 2 Median: 28934.25
Range: 22387.2 to 35481.3
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC55422 ALOX15 1 15848.9 Potency PubChem BioAssay data set
CHEMBL1201862
NPC55422 MAPK1 2 Median: 20483.9
Range: 15848.9 to 25118.9
Potency PubChem BioAssay data set
CHEMBL1201862
PubChem BioAssay data set
CHEMBL1201862
NPC102810 ALOX15 1 12589.3 Potency PubChem BioAssay data set
CHEMBL1201862
NPC264317 AKR1B1 1 11000 IC50 PMID: 21561086