Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT79 | Organism | Bacillus subtilis | Bacillus subtilis | MIC | = | 112201845.4 | nM | 17869511 |
NPT16 | Organism | Staphylococcus aureus | Staphylococcus aureus | MIC | = | 141253754.5 | nM | 17869511 |
NPT19 | Organism | Escherichia coli | Escherichia coli | MIC | = | 177827941 | nM | 17869511 |
NPT20 | Organism | Candida albicans | Candida albicans | MIC | = | 112201845.4 | nM | 17869511 |
NPT21 | Organism | Aspergillus niger | Aspergillus niger | MIC | = | 125892541.2 | nM | 17869511 |
NPT664 | Protein Family | Histone deacetylase | Homo sapiens | Activity | = | 91 | % | 19520580 |
NPT3 | Individual Protein | Thioredoxin glutathione reductase | Schistosoma mansoni | Potency | = | 39810.7 | nM | PubChem BioAssay data set |
NPT443 | Individual Protein | Histone acetyltransferase GCN5 | Homo sapiens | Potency | 35481.3 | nM | PubChem BioAssay data set | |
NPT2 | Others | Unspecified | Potency | 29092.9 | nM | PubChem BioAssay data set | ||
NPT32 | Organism | Mus musculus | Mus musculus | IC50 | = | 210 | nM | 21388814 |
NPT135 | Individual Protein | Chromobox protein homolog 1 | Homo sapiens | Potency | 89125.1 | nM | PubChem BioAssay data set | |
NPT153 | Individual Protein | Androgen Receptor | Homo sapiens | Potency | 22.4 | nM | PubChem BioAssay data set | |
NPT249 | Individual Protein | Glucocorticoid receptor | Homo sapiens | Potency | 50118.7 | nM | PubChem BioAssay data set | |
NPT10 | Individual Protein | Geminin | Homo sapiens | Potency | 183.6 | nM | PubChem BioAssay data set | |
NPT774 | Organism | Zygosaccharomyces bailii | Zygosaccharomyces bailii | MIC | = | 1600 | ug/ml | 15969495 |
NPT774 | Organism | Zygosaccharomyces bailii | Zygosaccharomyces bailii | MFC | = | 800 | ug/ml | 15969495 |
NPT312 | Organism | Saccharomyces cerevisiae | Saccharomyces cerevisiae | MFC | = | 3200 | ug/ml | 12083872 |
NPT312 | Organism | Saccharomyces cerevisiae | Saccharomyces cerevisiae | MFC | = | 1600 | ug/ml | 12083872 |
NPT312 | Organism | Saccharomyces cerevisiae | Saccharomyces cerevisiae | MIC | > | 1600 | ug/ml | 12083872 |
NPT312 | Organism | Saccharomyces cerevisiae | Saccharomyces cerevisiae | MIC | = | 800 | ug/ml | 12083872 |
NPT312 | Organism | Saccharomyces cerevisiae | Saccharomyces cerevisiae | MIC | = | 400 | ug/ml | 12083872 |
NPT2 | Others | Unspecified | Potency | 21872.4 | nM | PubChem BioAssay data set | ||
NPT2 | Others | Unspecified | Potency | 27056.3 | nM | PubChem BioAssay data set | ||
NPT152 | Individual Protein | Nuclear factor erythroid 2-related factor 2 | Homo sapiens | Potency | 24336.5 | nM | PubChem BioAssay data set | |
NPT2 | Others | Unspecified | Potency | 27306 | nM | PubChem BioAssay data set | ||
NPT153 | Individual Protein | Androgen Receptor | Homo sapiens | Potency | 194.9 | nM | PubChem BioAssay data set | |
NPT2 | Others | Unspecified | Potency | 48966.2 | nM | PubChem BioAssay data set | ||
NPT153 | Individual Protein | Androgen Receptor | Homo sapiens | Potency | 33491.5 | nM | PubChem BioAssay data set | |
NPT2 | Others | Unspecified | Potency | 68589.6 | nM | PubChem BioAssay data set | ||
NPT2 | Others | Unspecified | Potency | 61130.6 | nM | PubChem BioAssay data set | ||
NPT2 | Others | Unspecified | Potency | 54482.7 | nM | PubChem BioAssay data set | ||
NPT2 | Others | Unspecified | Potency | 30357.7 | nM | PubChem BioAssay data set |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC63598 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Natural Product ID |
---|---|---|
0.9167 | High Similarity | NPC107877 |
0.9143 | High Similarity | NPC60675 |
0.9143 | High Similarity | NPC297363 |
0.8974 | High Similarity | NPC102879 |
0.8462 | Intermediate Similarity | NPC8270 |
0.8378 | Intermediate Similarity | NPC308418 |
0.8333 | Intermediate Similarity | NPC224651 |
0.8333 | Intermediate Similarity | NPC98098 |
0.825 | Intermediate Similarity | NPC221250 |
0.775 | Intermediate Similarity | NPC298413 |
0.7619 | Intermediate Similarity | NPC41409 |
0.7609 | Intermediate Similarity | NPC221467 |
0.7556 | Intermediate Similarity | NPC128520 |
0.7447 | Intermediate Similarity | NPC43053 |
0.7429 | Intermediate Similarity | NPC20903 |
0.7222 | Intermediate Similarity | NPC323552 |
0.7143 | Intermediate Similarity | NPC297608 |
0.7021 | Intermediate Similarity | NPC126184 |
0.6923 | Remote Similarity | NPC217161 |
0.6889 | Remote Similarity | NPC6963 |
0.6889 | Remote Similarity | NPC304079 |
0.6809 | Remote Similarity | NPC90490 |
0.6744 | Remote Similarity | NPC250954 |
0.6744 | Remote Similarity | NPC281043 |
0.6731 | Remote Similarity | NPC324224 |
0.6731 | Remote Similarity | NPC472808 |
0.6667 | Remote Similarity | NPC82446 |
0.6667 | Remote Similarity | NPC144407 |
0.6596 | Remote Similarity | NPC87137 |
0.6596 | Remote Similarity | NPC308331 |
0.6512 | Remote Similarity | NPC147824 |
0.65 | Remote Similarity | NPC146507 |
0.65 | Remote Similarity | NPC310810 |
0.6481 | Remote Similarity | NPC189700 |
0.6346 | Remote Similarity | NPC474127 |
0.6346 | Remote Similarity | NPC218486 |
0.6341 | Remote Similarity | NPC122676 |
0.625 | Remote Similarity | NPC130953 |
0.619 | Remote Similarity | NPC65353 |
0.6111 | Remote Similarity | NPC51846 |
0.6098 | Remote Similarity | NPC63354 |
0.6047 | Remote Similarity | NPC8416 |
0.6038 | Remote Similarity | NPC322461 |
0.6034 | Remote Similarity | NPC77891 |
0.6034 | Remote Similarity | NPC473737 |
0.6 | Remote Similarity | NPC137419 |
0.6 | Remote Similarity | NPC234084 |
0.6 | Remote Similarity | NPC203382 |
0.6 | Remote Similarity | NPC129150 |
0.6 | Remote Similarity | NPC313553 |
0.6 | Remote Similarity | NPC122212 |
0.6 | Remote Similarity | NPC294938 |
0.5965 | Remote Similarity | NPC98519 |
0.5962 | Remote Similarity | NPC191643 |
0.5897 | Remote Similarity | NPC8466 |
0.5897 | Remote Similarity | NPC280312 |
0.5893 | Remote Similarity | NPC474084 |
0.5893 | Remote Similarity | NPC254095 |
0.5893 | Remote Similarity | NPC223679 |
0.5882 | Remote Similarity | NPC275316 |
0.5882 | Remote Similarity | NPC15789 |
0.5862 | Remote Similarity | NPC326645 |
0.5862 | Remote Similarity | NPC317177 |
0.5862 | Remote Similarity | NPC317025 |
0.5862 | Remote Similarity | NPC329416 |
0.5818 | Remote Similarity | NPC325977 |
0.5818 | Remote Similarity | NPC150717 |
0.5818 | Remote Similarity | NPC86948 |
0.5789 | Remote Similarity | NPC97570 |
0.5789 | Remote Similarity | NPC302564 |
0.5789 | Remote Similarity | NPC82465 |
0.5763 | Remote Similarity | NPC2328 |
0.575 | Remote Similarity | NPC242117 |
0.5745 | Remote Similarity | NPC57923 |
0.5741 | Remote Similarity | NPC478120 |
0.5738 | Remote Similarity | NPC255781 |
0.5738 | Remote Similarity | NPC146811 |
0.5714 | Remote Similarity | NPC135863 |
0.5714 | Remote Similarity | NPC249850 |
0.5714 | Remote Similarity | NPC472445 |
0.5714 | Remote Similarity | NPC245650 |
0.5714 | Remote Similarity | NPC283502 |
0.5714 | Remote Similarity | NPC44542 |
0.5714 | Remote Similarity | NPC293437 |
0.5714 | Remote Similarity | NPC270706 |
0.5714 | Remote Similarity | NPC250734 |
0.5652 | Remote Similarity | NPC323278 |
0.5645 | Remote Similarity | NPC254886 |
0.5636 | Remote Similarity | NPC478117 |
0.5636 | Remote Similarity | NPC173157 |
0.5625 | Remote Similarity | NPC270796 |
0.5614 | Remote Similarity | NPC471619 |
0.5614 | Remote Similarity | NPC21946 |
0.5614 | Remote Similarity | NPC34416 |
0.561 | Remote Similarity | NPC273054 |
0.56 | Remote Similarity | NPC128280 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC63598 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
0.8333 | Intermediate Similarity | NPD8573 | Approved |
0.7429 | Intermediate Similarity | NPD8187 | Phase 3 |
0.7391 | Intermediate Similarity | NPD4220 | Pre-registration |
0.725 | Intermediate Similarity | NPD9115 | Approved |
0.6154 | Remote Similarity | NPD9114 | Clinical (unspecified phase) |
0.5957 | Remote Similarity | NPD9411 | Phase 1 |
0.5862 | Remote Similarity | NPD4191 | Approved |
0.5862 | Remote Similarity | NPD4194 | Approved |
0.5862 | Remote Similarity | NPD4192 | Approved |
0.5862 | Remote Similarity | NPD4193 | Approved |
0.5625 | Remote Similarity | NPD5326 | Phase 3 |
PubChem CID   | 643460 |
ChEMBL   | CHEMBL250212 |
ZINC   |
Molecular Weight:   | 112.05 |
ALogP:   | 1.0286 |
MLogP:   | 1.9 |
XLogP:   | 1.43 |
# Rotatable Bonds:   | 4 |
Polar Surface Area:   | 37.3 |
# H-Bond Aceptor:   | 2 |
# H-Bond Donor:   | 1 |
# Rings:   | 0 |
# Heavy Atoms:   | 8 |