Target ID | Target Type | Target Name | Target Organism | Activity Type | Activity Relation | Value | Unit | Reference |
---|---|---|---|---|---|---|---|---|
NPT165 | Cell Line | HeLa | Homo sapiens | IC50 | = | 33500 | nM | PubChem BioAssay data set |
NPT177 | Tissue | Aorta | Rattus norvegicus | IC50 | > | 80000 | nM | 21807513 |
NPT137 | Cell Line | L1210 | Mus musculus | IC50 | = | 103000 | nM | 17618115 |
NPT177 | Tissue | Aorta | Rattus norvegicus | Activity | = | 65.6 | % | 22264115 |
NPT88 | Organism | Mycobacterium tuberculosis | Mycobacterium tuberculosis | MIC90 | = | 173000 | nM | 18710917 |
NPT165 | Cell Line | HeLa | Homo sapiens | IC50 | = | 131000 | nM | 18973387 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules. Tc lies between [0, 1] where '1' indicates the highest similarity. What is Tanimoto coefficient
●  The left chart: Distribution of similarity level between NPC474105 and all remaining natural products in the NPASS database.
●  The right table: Most similar natural products (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Natural Product ID |
---|---|---|
0.9434 | High Similarity | NPC184819 |
0.9259 | High Similarity | NPC151464 |
0.9259 | High Similarity | NPC143597 |
0.9245 | High Similarity | NPC53245 |
0.9245 | High Similarity | NPC288296 |
0.8525 | High Similarity | NPC96812 |
0.8525 | High Similarity | NPC107704 |
0.8525 | High Similarity | NPC39462 |
0.8525 | High Similarity | NPC189917 |
0.8525 | High Similarity | NPC168824 |
0.8333 | Intermediate Similarity | NPC274182 |
0.8269 | Intermediate Similarity | NPC98246 |
0.8269 | Intermediate Similarity | NPC285814 |
0.8269 | Intermediate Similarity | NPC83187 |
0.8125 | Intermediate Similarity | NPC477857 |
0.8125 | Intermediate Similarity | NPC474962 |
0.807 | Intermediate Similarity | NPC307063 |
0.8 | Intermediate Similarity | NPC477856 |
0.8 | Intermediate Similarity | NPC214770 |
0.7963 | Intermediate Similarity | NPC293343 |
0.7963 | Intermediate Similarity | NPC247786 |
0.7963 | Intermediate Similarity | NPC258672 |
0.7937 | Intermediate Similarity | NPC43300 |
0.7879 | Intermediate Similarity | NPC473267 |
0.7812 | Intermediate Similarity | NPC130459 |
0.7812 | Intermediate Similarity | NPC474221 |
0.7812 | Intermediate Similarity | NPC478180 |
0.7778 | Intermediate Similarity | NPC294440 |
0.7761 | Intermediate Similarity | NPC474123 |
0.7692 | Intermediate Similarity | NPC473225 |
0.7667 | Intermediate Similarity | NPC127798 |
0.7593 | Intermediate Similarity | NPC131981 |
0.7593 | Intermediate Similarity | NPC40249 |
0.7593 | Intermediate Similarity | NPC173996 |
0.7536 | Intermediate Similarity | NPC255650 |
0.7536 | Intermediate Similarity | NPC273366 |
0.7463 | Intermediate Similarity | NPC40574 |
0.7463 | Intermediate Similarity | NPC108131 |
0.7463 | Intermediate Similarity | NPC477850 |
0.7424 | Intermediate Similarity | NPC20610 |
0.7391 | Intermediate Similarity | NPC255021 |
0.7385 | Intermediate Similarity | NPC42060 |
0.7385 | Intermediate Similarity | NPC323005 |
0.7385 | Intermediate Similarity | NPC477931 |
0.7385 | Intermediate Similarity | NPC268736 |
0.7353 | Intermediate Similarity | NPC151018 |
0.7353 | Intermediate Similarity | NPC197701 |
0.7353 | Intermediate Similarity | NPC110615 |
0.7353 | Intermediate Similarity | NPC156277 |
0.7353 | Intermediate Similarity | NPC58057 |
0.7353 | Intermediate Similarity | NPC320549 |
0.7344 | Intermediate Similarity | NPC128608 |
0.7324 | Intermediate Similarity | NPC264602 |
0.7324 | Intermediate Similarity | NPC475031 |
0.7313 | Intermediate Similarity | NPC324607 |
0.7313 | Intermediate Similarity | NPC182815 |
0.7313 | Intermediate Similarity | NPC327728 |
0.7313 | Intermediate Similarity | NPC196197 |
0.7313 | Intermediate Similarity | NPC321732 |
0.7313 | Intermediate Similarity | NPC213178 |
0.7313 | Intermediate Similarity | NPC131892 |
0.7313 | Intermediate Similarity | NPC6120 |
0.7286 | Intermediate Similarity | NPC72444 |
0.7246 | Intermediate Similarity | NPC232112 |
0.7246 | Intermediate Similarity | NPC310766 |
0.7222 | Intermediate Similarity | NPC478128 |
0.7206 | Intermediate Similarity | NPC307176 |
0.7206 | Intermediate Similarity | NPC159577 |
0.7206 | Intermediate Similarity | NPC282593 |
0.7206 | Intermediate Similarity | NPC476731 |
0.7206 | Intermediate Similarity | NPC35734 |
0.7183 | Intermediate Similarity | NPC69408 |
0.717 | Intermediate Similarity | NPC18397 |
0.7164 | Intermediate Similarity | NPC474954 |
0.7143 | Intermediate Similarity | NPC254340 |
0.7143 | Intermediate Similarity | NPC20017 |
0.7143 | Intermediate Similarity | NPC270042 |
0.7143 | Intermediate Similarity | NPC472854 |
0.7143 | Intermediate Similarity | NPC159497 |
0.7123 | Intermediate Similarity | NPC52951 |
0.7115 | Intermediate Similarity | NPC45270 |
0.7115 | Intermediate Similarity | NPC215118 |
0.7115 | Intermediate Similarity | NPC59570 |
0.7115 | Intermediate Similarity | NPC135077 |
0.7101 | Intermediate Similarity | NPC305501 |
0.7101 | Intermediate Similarity | NPC234707 |
0.7101 | Intermediate Similarity | NPC115023 |
0.7101 | Intermediate Similarity | NPC126642 |
0.7101 | Intermediate Similarity | NPC472309 |
0.7101 | Intermediate Similarity | NPC89310 |
0.7101 | Intermediate Similarity | NPC470078 |
0.7059 | Intermediate Similarity | NPC319671 |
0.7059 | Intermediate Similarity | NPC64466 |
0.7059 | Intermediate Similarity | NPC469941 |
0.7059 | Intermediate Similarity | NPC476734 |
0.7059 | Intermediate Similarity | NPC252032 |
0.7059 | Intermediate Similarity | NPC139397 |
0.7042 | Intermediate Similarity | NPC21220 |
0.7042 | Intermediate Similarity | NPC125767 |
0.7042 | Intermediate Similarity | NPC293803 |
0.7042 | Intermediate Similarity | NPC195155 |
0.7042 | Intermediate Similarity | NPC97534 |
0.7042 | Intermediate Similarity | NPC472311 |
0.7042 | Intermediate Similarity | NPC174964 |
0.7037 | Intermediate Similarity | NPC171783 |
0.7 | Intermediate Similarity | NPC303613 |
0.7 | Intermediate Similarity | NPC474228 |
0.7 | Intermediate Similarity | NPC251705 |
0.6957 | Remote Similarity | NPC2634 |
0.6957 | Remote Similarity | NPC265782 |
0.6957 | Remote Similarity | NPC477929 |
0.6957 | Remote Similarity | NPC260040 |
0.6957 | Remote Similarity | NPC251929 |
0.6944 | Remote Similarity | NPC472487 |
0.6944 | Remote Similarity | NPC475742 |
0.6944 | Remote Similarity | NPC472486 |
0.6944 | Remote Similarity | NPC5767 |
0.6933 | Remote Similarity | NPC77311 |
0.6933 | Remote Similarity | NPC469745 |
0.6923 | Remote Similarity | NPC472306 |
0.6901 | Remote Similarity | NPC167702 |
0.6901 | Remote Similarity | NPC280026 |
0.6901 | Remote Similarity | NPC133922 |
0.6857 | Remote Similarity | NPC54123 |
0.6857 | Remote Similarity | NPC223187 |
0.6857 | Remote Similarity | NPC469940 |
0.6857 | Remote Similarity | NPC5701 |
0.6849 | Remote Similarity | NPC470557 |
0.6849 | Remote Similarity | NPC221420 |
0.6849 | Remote Similarity | NPC477918 |
0.6849 | Remote Similarity | NPC474404 |
0.6849 | Remote Similarity | NPC91665 |
0.6849 | Remote Similarity | NPC23884 |
0.6842 | Remote Similarity | NPC477858 |
0.6818 | Remote Similarity | NPC469662 |
0.6806 | Remote Similarity | NPC24014 |
0.6806 | Remote Similarity | NPC27349 |
0.6806 | Remote Similarity | NPC212733 |
0.6806 | Remote Similarity | NPC159789 |
0.68 | Remote Similarity | NPC477851 |
0.6765 | Remote Similarity | NPC220210 |
0.6765 | Remote Similarity | NPC20181 |
0.6761 | Remote Similarity | NPC470044 |
0.6761 | Remote Similarity | NPC52667 |
0.6761 | Remote Similarity | NPC470045 |
0.6757 | Remote Similarity | NPC185465 |
0.6757 | Remote Similarity | NPC63020 |
0.6753 | Remote Similarity | NPC15821 |
0.6753 | Remote Similarity | NPC472744 |
0.6731 | Remote Similarity | NPC223315 |
0.6712 | Remote Similarity | NPC20466 |
0.6712 | Remote Similarity | NPC471046 |
0.6712 | Remote Similarity | NPC4209 |
0.6711 | Remote Similarity | NPC12933 |
0.6667 | Remote Similarity | NPC281203 |
0.6667 | Remote Similarity | NPC142754 |
0.6667 | Remote Similarity | NPC31302 |
0.6667 | Remote Similarity | NPC245029 |
0.6667 | Remote Similarity | NPC477930 |
0.6667 | Remote Similarity | NPC260319 |
0.6667 | Remote Similarity | NPC215843 |
0.6667 | Remote Similarity | NPC178025 |
0.6667 | Remote Similarity | NPC202118 |
0.6667 | Remote Similarity | NPC469724 |
0.6667 | Remote Similarity | NPC296697 |
0.6667 | Remote Similarity | NPC103647 |
0.6667 | Remote Similarity | NPC39157 |
0.6667 | Remote Similarity | NPC470956 |
0.6667 | Remote Similarity | NPC31187 |
0.6667 | Remote Similarity | NPC320144 |
0.6667 | Remote Similarity | NPC2568 |
0.6667 | Remote Similarity | NPC309852 |
0.6667 | Remote Similarity | NPC192744 |
0.6667 | Remote Similarity | NPC180777 |
0.6667 | Remote Similarity | NPC474996 |
0.6667 | Remote Similarity | NPC319909 |
0.6667 | Remote Similarity | NPC201459 |
0.6667 | Remote Similarity | NPC16287 |
0.6667 | Remote Similarity | NPC82477 |
0.6667 | Remote Similarity | NPC197238 |
0.6667 | Remote Similarity | NPC475977 |
0.6667 | Remote Similarity | NPC181743 |
0.6667 | Remote Similarity | NPC100917 |
0.6623 | Remote Similarity | NPC271163 |
0.6622 | Remote Similarity | NPC477919 |
0.6622 | Remote Similarity | NPC143133 |
0.6622 | Remote Similarity | NPC212661 |
0.6622 | Remote Similarity | NPC207010 |
0.6622 | Remote Similarity | NPC298168 |
0.6622 | Remote Similarity | NPC180199 |
0.6622 | Remote Similarity | NPC471035 |
0.6622 | Remote Similarity | NPC317913 |
0.6622 | Remote Similarity | NPC66105 |
0.6622 | Remote Similarity | NPC106078 |
0.6613 | Remote Similarity | NPC200258 |
0.6582 | Remote Similarity | NPC60350 |
0.6582 | Remote Similarity | NPC76518 |
0.6579 | Remote Similarity | NPC472853 |
0.6579 | Remote Similarity | NPC474509 |
0.6579 | Remote Similarity | NPC470609 |
Similarity level is defined by Tanimoto coefficient (Tc) between two molecules.
●  The left chart: Distribution of similarity level between NPC474105 and all drugs/candidates.
●  The right table: Most similar clinical/approved drugs (Tc>=0.56 or Top200).
Similarity Score | Similarity Level | Drug ID | Developmental Stage |
---|---|---|---|
0.7692 | Intermediate Similarity | NPD5360 | Phase 3 |
0.7692 | Intermediate Similarity | NPD5361 | Clinical (unspecified phase) |
0.7656 | Intermediate Similarity | NPD4224 | Phase 2 |
0.7593 | Intermediate Similarity | NPD345 | Approved |
0.7593 | Intermediate Similarity | NPD344 | Approved |
0.7593 | Intermediate Similarity | NPD343 | Approved |
0.75 | Intermediate Similarity | NPD3171 | Clinical (unspecified phase) |
0.7463 | Intermediate Similarity | NPD4789 | Approved |
0.7353 | Intermediate Similarity | NPD4808 | Clinical (unspecified phase) |
0.7353 | Intermediate Similarity | NPD4809 | Clinical (unspecified phase) |
0.7353 | Intermediate Similarity | NPD4758 | Discontinued |
0.7353 | Intermediate Similarity | NPD6081 | Approved |
0.7313 | Intermediate Similarity | NPD3698 | Phase 2 |
0.7313 | Intermediate Similarity | NPD3700 | Clinical (unspecified phase) |
0.7313 | Intermediate Similarity | NPD3699 | Clinical (unspecified phase) |
0.7206 | Intermediate Similarity | NPD4747 | Approved |
0.7206 | Intermediate Similarity | NPD4244 | Approved |
0.7206 | Intermediate Similarity | NPD4245 | Approved |
0.7164 | Intermediate Similarity | NPD3621 | Clinical (unspecified phase) |
0.7101 | Intermediate Similarity | NPD5777 | Approved |
0.7059 | Intermediate Similarity | NPD4137 | Phase 3 |
0.6957 | Remote Similarity | NPD4691 | Approved |
0.6901 | Remote Similarity | NPD6113 | Clinical (unspecified phase) |
0.6806 | Remote Similarity | NPD3703 | Phase 2 |
0.6757 | Remote Similarity | NPD5364 | Discontinued |
0.6712 | Remote Similarity | NPD6117 | Approved |
0.6667 | Remote Similarity | NPD4687 | Approved |
0.6667 | Remote Similarity | NPD5733 | Approved |
0.6667 | Remote Similarity | NPD4058 | Approved |
0.6622 | Remote Similarity | NPD6116 | Phase 1 |
0.662 | Remote Similarity | NPD5276 | Approved |
0.6575 | Remote Similarity | NPD3702 | Approved |
0.6533 | Remote Similarity | NPD3671 | Phase 1 |
0.6533 | Remote Similarity | NPD6697 | Approved |
0.6533 | Remote Similarity | NPD6115 | Approved |
0.6533 | Remote Similarity | NPD6118 | Approved |
0.6533 | Remote Similarity | NPD4777 | Suspended |
0.6533 | Remote Similarity | NPD4776 | Phase 2 |
0.6533 | Remote Similarity | NPD6114 | Approved |
0.6329 | Remote Similarity | NPD4788 | Approved |
0.6316 | Remote Similarity | NPD3617 | Approved |
0.6203 | Remote Similarity | NPD4221 | Approved |
0.6203 | Remote Similarity | NPD4223 | Phase 3 |
0.6076 | Remote Similarity | NPD4139 | Approved |
0.6076 | Remote Similarity | NPD4692 | Approved |
0.6049 | Remote Similarity | NPD4197 | Approved |
0.6049 | Remote Similarity | NPD4786 | Approved |
0.6026 | Remote Similarity | NPD7155 | Clinical (unspecified phase) |
0.6 | Remote Similarity | NPD3667 | Approved |
0.5976 | Remote Similarity | NPD5329 | Approved |
0.5976 | Remote Similarity | NPD7520 | Clinical (unspecified phase) |
0.5904 | Remote Similarity | NPD5205 | Approved |
0.5904 | Remote Similarity | NPD4138 | Approved |
0.5904 | Remote Similarity | NPD6098 | Approved |
0.5904 | Remote Similarity | NPD4693 | Phase 3 |
0.5904 | Remote Similarity | NPD4689 | Approved |
0.5904 | Remote Similarity | NPD4690 | Approved |
0.5904 | Remote Similarity | NPD4688 | Approved |
0.5854 | Remote Similarity | NPD3665 | Phase 1 |
0.5854 | Remote Similarity | NPD3133 | Approved |
0.5854 | Remote Similarity | NPD3666 | Approved |
0.5854 | Remote Similarity | NPD3668 | Phase 3 |
0.5795 | Remote Similarity | NPD6001 | Approved |
0.5765 | Remote Similarity | NPD6672 | Approved |
0.5765 | Remote Similarity | NPD5737 | Approved |
0.5765 | Remote Similarity | NPD7513 | Clinical (unspecified phase) |
0.5765 | Remote Similarity | NPD5208 | Approved |
0.5732 | Remote Similarity | NPD3527 | Clinical (unspecified phase) |
0.573 | Remote Similarity | NPD6356 | Clinical (unspecified phase) |
0.5714 | Remote Similarity | NPD7146 | Approved |
0.5714 | Remote Similarity | NPD5690 | Phase 2 |
0.5714 | Remote Similarity | NPD6684 | Approved |
0.5714 | Remote Similarity | NPD6409 | Approved |
0.5714 | Remote Similarity | NPD3574 | Clinical (unspecified phase) |
0.5714 | Remote Similarity | NPD3618 | Phase 1 |
0.5714 | Remote Similarity | NPD7521 | Approved |
0.5714 | Remote Similarity | NPD5330 | Approved |
0.5714 | Remote Similarity | NPD4694 | Approved |
0.5714 | Remote Similarity | NPD7334 | Approved |
0.5714 | Remote Similarity | NPD5280 | Approved |
0.5698 | Remote Similarity | NPD6904 | Approved |
0.5698 | Remote Similarity | NPD6080 | Approved |
0.5698 | Remote Similarity | NPD6673 | Approved |
0.5698 | Remote Similarity | NPD5328 | Approved |
0.5698 | Remote Similarity | NPD4753 | Phase 2 |
0.5682 | Remote Similarity | NPD5133 | Approved |
0.5679 | Remote Similarity | NPD8028 | Phase 2 |
0.5676 | Remote Similarity | NPD4267 | Clinical (unspecified phase) |
0.56 | Remote Similarity | NPD4787 | Phase 1 |
PubChem CID   | 44566738 |
ChEMBL   | CHEMBL461825 |
ZINC   |
Molecular Weight:   | 286.23 |
ALogP:   | 1.7496 |
MLogP:   | 3.55 |
XLogP:   | 6.566 |
# Rotatable Bonds:   | 4 |
Polar Surface Area:   | 17.07 |
# H-Bond Aceptor:   | 1 |
# H-Bond Donor:   | 0 |
# Rings:   | 4 |
# Heavy Atoms:   | 21 |