Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT176 | Acyl coenzyme A:cholesterol acyltransferase 1 | Homo sapiens |
IC50: 3700 (nM), Ref: 23419736 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 9100 (nM), Ref: 15679319 |
|
TCMT559 | Beta-2 adrenergic receptor | Homo sapiens |
Ki: 1 (nM), Ref: 24454993 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
Ki: 5100 (nM), Ref: 16248836 Ki: 6460 (nM), Ref: 16248836 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 4400 (nM), Ref: 15634016 |
|
TCMT241 | Neuronal acetylcholine receptor protein alpha-7 subunit | Homo sapiens |
Ki: 7200 (nM), Ref: 15686879 Ki: 6300 (nM), Ref: 15908213 Ki: 630 (nM), Ref: 16171993 Ki: 10000 (nM), Ref: 17722904 Ki: 1000 (nM), Ref: 19331415 Ki: 1023.29 (nM), Ref: 20828128 Ki: 1000 (nM), Ref: 21920761 Ki: 1000 (nM), Ref: 22243960 Ki: 3000 (nM), Ref: 22793665 Ki: 3000 (nM), Ref: 23126648 Ki: 3800 (nM), Ref: 23561269 IC50: 7600 (nM), Ref: 23561269 Ki: 3000 (nM), Ref: 23692872 |
|
TCMT552 | Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens |
IC50: 45 (nM), Ref: 11312774 |
|
TCMT643 | Alpha-1a adrenergic receptor | Homo sapiens |
Ki: 0.2 (nM), Ref: 15664832 Ki: 0.19 (nM), Ref: 17517507 Ki: 0.19 (nM), Ref: 17452102 Ki: 0.19 (nM), Ref: 18055202 Ki: 0.05012 (nM), Ref: 20934789 |
|
TCMT650 | Alpha-1b adrenergic receptor | Homo sapiens |
Ki: 2 (nM), Ref: 17517507 Ki: 2 (nM), Ref: 17452102 Ki: 2 (nM), Ref: 18055202 Ki: 0.631 (nM), Ref: 20934789 |
|
TCMT642 | Alpha-1d adrenergic receptor | Homo sapiens |
Ki: 0.2 (nM), Ref: 17517507 Ki: 0.2 (nM), Ref: 17452102 Ki: 0.2 (nM), Ref: 18055202 Ki: 0.1 (nM), Ref: 20934789 Ki: 0.18 (nM), Ref: 26954848 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
Ki: 1390 (nM), Ref: 16248836 Ki: 2970 (nM), Ref: 16248836 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 52 (nM), Ref: 17497806 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT314 | Serotonin 2c (5-HT2c) receptor | Homo sapiens |
Ki: 10 (nM), Ref: 24491146 |
|
TCMT307 | HERG | Homo sapiens |
IC50: 143 (nM), Ref: 12190308 IC50: 143 (nM), Ref: 12729675 IC50: 141.25 (nM), Ref: 12873512 IC50: 144.54 (nM), Ref: 15745831 IC50: 141.25 (nM), Ref: 18448342 IC50: 144.54 (nM), Ref: 19110341 IC50: 141.25 (nM), Ref: 21185626 IC50: 10 (nM), Ref: 23919353 |
|
TCMT232 | P-glycoprotein 1 | Homo sapiens |
IC50: 6606.93 (nM), Ref: 17890094 IC50: 4570.88 (nM), Ref: 17890094 IC50: 6606.93 (nM), Ref: 18083034 IC50: 4570.88 (nM), Ref: 18083034 IC50: 4570.88 (nM), Ref: 18678495 IC50: 5420 (nM), Ref: 18707884 IC50: 5200 (nM), Ref: 19250834 IC50: 500 (nM), Ref: 22112208 IC50: 575.44 (nM), Ref: 22452412 Ki: 1750 (nM), Ref: 22320402 Ki: 1750 (nM), Ref: 22320402 IC50: 1600 (nM), Ref: 23245571 IC50: 1700 (nM), Ref: 10.1039/C2MD20286G IC50: 29 (nM), Ref: 25282263 IC50: 740 (nM), Ref: 25282263 IC50: 38 (nM), Ref: 25985195 |
|
TCMT629 | Multidrug resistance-associated protein 1 | Homo sapiens |
IC50: 9660 (nM), Ref: 18707884 IC50: 3500 (nM), Ref: 25093931 |
|
TCMT213 | Solute carrier family 22 member 1 | Homo sapiens |
IC50: 6800 (nM), Ref: 18788725 |