TCM Putative Target References: TCMH494


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
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Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC2091
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7610 (nM), Ref: 21402476
TCMC2091
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7280 (nM), Ref: 21402476
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC983
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2800 (nM), Ref: 15887952
IC50: 2800 (nM), Ref: 15887952
IC50: 1200 (nM), Ref: 12502307
IC50: 2800 (nM), Ref:
TCMC983
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 7300 (nM), Ref: 21030469
TCMC983
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 718.7 (nM), Ref: 26498393
TCMC983
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.2 (nM), Ref: 26498393
TCMC983
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 56.4 (nM), Ref: 26498393
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC412
TCMT683 Macrophage migration inhibitory factor Homo sapiens Ki: 38 (nM), Ref: 19090668
IC50: 38 (nM), Ref: 27156768
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC515
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 15 (nM), Ref: 17560111
TCMC1236
TCMT236 Estrogen receptor beta Homo sapiens IC50: 10 (nM), Ref: 15341953
IC50: 10 (nM), Ref: 15456246
IC50: 98.7 (nM), Ref: 15887952
IC50: 98.7 (nM), Ref: 15887952
IC50: 9.7 (nM), Ref: 15943471
IC50: 10 (nM), Ref: 16098741
IC50: 1.3 (nM), Ref: 16219463
IC50: 61 (nM), Ref: 16610787
IC50: 25 (nM), Ref: 17149865
IC50: 395 (nM), Ref: 17049855
IC50: 9.7 (nM), Ref: 17188490
IC50: 6.8 (nM), Ref: 17574424
IC50: 18 (nM), Ref: 12502307
IC50: 98.7 (nM), Ref:
TCMC1236
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 395 (nM), Ref: 15341953
IC50: 395 (nM), Ref: 15456246
IC50: 4660 (nM), Ref: 15887952
IC50: 4660 (nM), Ref: 15887952
IC50: 395 (nM), Ref: 15943471
IC50: 395 (nM), Ref: 16098741
IC50: 29.4 (nM), Ref: 16219463
IC50: 1973 (nM), Ref: 16610787
IC50: 1145 (nM), Ref: 17149865
IC50: 2150 (nM), Ref: 17696335
IC50: 9.7 (nM), Ref: 17049855
IC50: 395 (nM), Ref: 17188490
IC50: 580 (nM), Ref: 17574424
IC50: 300 (nM), Ref: 12502307
IC50: 4680 (nM), Ref:
TCMC1236
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 10 (nM), Ref: 17482813
TCMC1236
TCMT910 Estrogen-related receptor beta Homo sapiens IC50: 395 (nM), Ref: 17482813
TCMC1236
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 2210 (nM), Ref: 18533708
TCMC1236
TCMT344 Aldehyde oxidase Homo sapiens IC50: 340 (nM), Ref: 20853847
TCMC1236
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 7720 (nM), Ref:
TCMC1297
TCMT632 Purine nucleoside phosphorylase Homo sapiens Ki: 5000 (nM), Ref: 31484
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC983
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.43 (ug/ml), Ref: 20116898
TCMC1236
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.84 (ug/ml), Ref: 20116898
TCMC2302
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 2.2 (ug/ml), Ref: 22197393
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC2540
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 16.3 (ug/ml), Ref: 26099531
TCMC2540
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 18.2 (ug/ml), Ref: 26099531
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2587
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 10.2 (ug/ml), Ref: 26099531
TCMC2587
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 8.7 (ug/ml), Ref: 26099531
TCMC2657
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 15.1 (ug/ml), Ref: 26099531
TCMC2657
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 17.2 (ug/ml), Ref: 26099531
TCMC1236
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (ug/ml), Ref: 19299148
TCMC2826
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 17869507
MIC: 100 (ug/ml), Ref: 20542692
TCMC2826
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 17869507
MIC: 100 (ug/ml), Ref: 20542692
TCMC2302
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 15.9 (nM), Ref: 23631483