Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 5930 (nM), Ref: 19846303 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 630 (nM), Ref: 21561086 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 560 (nM), Ref: 18258440 IC50: 560 (nM), Ref: 21669529 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18778944 |
|
TCMT737 | DNA dC->dU-editing enzyme APOBEC-3G | Homo sapiens | IC50: 2390 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 2120 (nM), Ref: 24900447 |
|
TCMT558 | DNA topoisomerase II alpha | Homo sapiens |
IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1690 (nM), Ref: 23411073 |
|
TCMT2 | Microtubule-associated protein tau | Homo sapiens |
IC50: 1200 (nM), Ref: 23484434 IC50: 3000 (nM), Ref: 25086914 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 3000 (nM), Ref: 25086914 |
|
TCMT740 | PI3-kinase p110-gamma subunit | Homo sapiens |
IC50: 4720 (nM), Ref: 25050878 |
|
TCMT13 | DNA-(apurinic or apyrimidinic site) lyase | Homo sapiens |
IC50: 320 (nM), Ref: 25280182 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT304 | Matrix metalloproteinase 14 | Homo sapiens |
IC50: 6800 (nM), Ref: 19524436 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 9600 (nM), Ref: 19524436 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 757 (nM), Ref: 22225636 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 1000 (nM), Ref: 22413845 IC50: 1080 (nM), Ref: 22413845 IC50: 1180 (nM), Ref: 22413845 IC50: 1000 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT47 | Apoptosis regulator Bcl-2 | Homo sapiens |
Ki: 335 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT2 | Microtubule-associated protein tau | Homo sapiens |
IC50: 1800 (nM), Ref: 23484434 |
|
TCMT751 | Dual-specificity tyrosine-phosphorylation regulated kinase 1A | Homo sapiens |
IC50: 330 (nM), Ref: 24188002 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 4600 (nM), Ref: 24878198 IC50: 3000 (nM), Ref: 24878198 IC50: 500 (nM), Ref: 25978520 |
|
TCMT567 | DNA (cytosine-5)-methyltransferase 1 | Homo sapiens |
IC50: 500 (nM), Ref: 25406944 |
|
TCMT232 | P-glycoprotein 1 | Homo sapiens |
IC50: 124.1 (nM), Ref: 25985195 IC50: 122.6 (nM), Ref: 25985195 |