TCM Putative Target References: TCMFx6433


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC417
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 7585.78 (nM), Ref: 23574272
IC50: 7500 (nM), Ref: 23574272
TCMC417
TCMT128 Tankyrase-2 Homo sapiens IC50: 870.96 (nM), Ref: 23574272
IC50: 870 (nM), Ref: 23574272
TCMC417
TCMT129 Tankyrase-1 Homo sapiens IC50: 645.65 (nM), Ref: 23574272
IC50: 630 (nM), Ref: 23574272
TCMC417
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2000 (nM), Ref: 24368208
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC444
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 5200 (nM), Ref: 20100662
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1537
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 5930 (nM), Ref: 19846303
TCMC1537
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 630 (nM), Ref: 21561086
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2126
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 1410 (nM), Ref: 23286284
TCMC2126
TCMT171 Protein-tyrosine phosphatase 1C Homo sapiens IC50: 1970 (nM), Ref: 23957426
TCMC2126
TCMT233 Protein-tyrosine phosphatase 2C Homo sapiens IC50: 2570 (nM), Ref: 23957426
TCMC1180
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5210 (nM), Ref: 22487176
Ki: 5100 (nM), Ref: 22487176
TCMC1180
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9300 (nM), Ref: 22487176
Ki: 9200 (nM), Ref: 22487176
TCMC1180
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5540 (nM), Ref: 22487176
Ki: 5630 (nM), Ref: 22487176
TCMC1180
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 6590 (nM), Ref: 22487176
Ki: 6650 (nM), Ref: 22487176
TCMC1803
TCMT337 Exportin-1 Homo sapiens IC50: 1600 (nM), Ref: 20493693
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC619
TCMT293 Muscarinic acetylcholine receptor M2 Homo sapiens Ki: 158.49 (nM), Ref: 18077164
TCMC619
TCMT291 Muscarinic acetylcholine receptor M3 Homo sapiens Ki: 7079.46 (nM), Ref: 18077164
TCMC619
TCMT551 Muscarinic acetylcholine receptor M4 Homo sapiens Ki: 8511.38 (nM), Ref: 18077164
TCMC619
TCMT290 Muscarinic acetylcholine receptor M5 Homo sapiens Ki: 9772.37 (nM), Ref: 18077164
TCMC619
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens Ki: 7943.28 (nM), Ref: 21920761
TCMC487
TCMT561 5'-nucleotidase Homo sapiens IC50: 8200 (nM), Ref: 24215819
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC2188
TCMT223 Aldose reductase Homo sapiens IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC2054
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 9640 (nM), Ref: 18507367
TCMC2054
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 6610 (nM), Ref:
TCMC2054
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 600 (nM), Ref: 26602279
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC2025
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2025.72 (nM), Ref:
TCMC1041
TCMT636 DNA polymerase alpha subunit Homo sapiens Ki: 830 (nM), Ref: 1705574
TCMC1041
TCMT17 DNA polymerase beta Homo sapiens Ki: 390 (nM), Ref: 1705574
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC2124
TCMT39 Phosphodiesterase 5A Homo sapiens IC50: 4703 (nM), Ref:
TCMC2124
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 325 (nM), Ref:
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC2025
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 5600 (nM), Ref: 23353736
TCMC2025
TCMT359 Tyrosine-protein kinase FYN Homo sapiens IC50: 1300 (nM), Ref: 17315853
IC50: 3600 (nM), Ref: 17315853
Ki: 7500 (nM), Ref: 17315853
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC614
TCMT151 Protein kinase C alpha Homo sapiens IC50: 9300 (nM), Ref: 9834166
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC1268
TCMT278 Solute carrier organic anion transporter family member 1B1 Homo sapiens IC50: 1400 (nM), Ref: 22587986
IC50: 2200 (nM), Ref: 22587986
TCMC1268
TCMT221 Bile salt export pump Homo sapiens IC50: 5300 (nM), Ref: 21965623
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC755
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens Ki: 600 (nM), Ref: 21739938
TCMC755
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens Ki: 1600 (nM), Ref: 21739938
TCMC755
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4400 (nM), Ref: 21030469
IC50: 7000 (nM), Ref: 21030469
TCMC755
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 8700 (nM), Ref:
TCMC1428
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 509 (nM), Ref: 20696580
TCMC1428
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 88 (nM), Ref: 20696580
TCMC1428
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1565
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 4440 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 4440 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC937
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 11.5 (nM), Ref: 23332369
IC50: 6.6 (nM), Ref: 23895532
TCMC937
TCMT801 Tubulin beta-3 chain Homo sapiens IC50: 5.2 (nM), Ref: 23332369
IC50: 5.7 (nM), Ref: 23895532
TCMC1078
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC1798
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1480 (nM), Ref: 23411073
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC1123
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1284 (nM), Ref: 20696580
TCMC1123
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 72.8 (nM), Ref: 26498393
TCMC1123
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1123
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 31.1 (nM), Ref: 26498393
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2018
TCMT907 Farnesyl diphosphate synthase Homo sapiens IC50: 452.9 (nM), Ref: 18327899
Ki: 82.2 (nM), Ref: 18327899
IC50: 5.7 (nM), Ref: 18327899
Ki: 0.36 (nM), Ref: 18327899
IC50: 5.7 (nM), Ref: 18434151
IC50: 300 (nM), Ref: 20801032
IC50: 11 (nM), Ref: 22390415
IC50: 860 (nM), Ref: 22390415
IC50: 11 (nM), Ref: 22884353
IC50: 10 (nM), Ref: 21780776
IC50: 5.2 (nM), Ref: 23998921
IC50: 11 (nM), Ref: 23998921
IC50: 6 (nM), Ref: 24911527
IC50: 11 (nM), Ref: 25630225
IC50: 6 (nM), Ref: 25935643
IC50: 0.36 (nM), Ref: 25815158
IC50: 82 (nM), Ref: 25815158
TCMC2055
TCMT747 ATP-binding cassette sub-family G member 2 Homo sapiens IC50: 10000 (nM), Ref: 22822035
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC1403
TCMT223 Aldose reductase Homo sapiens IC50: 1910 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC1803
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 2 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC2054
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 14.48 (ug/ml), Ref: 20116898
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2124
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 50 (ug/ml), Ref: 1710653
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC2281
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 0.00342 (ug/ml), Ref: 21334901
IC50: 0.00356 (ug/ml), Ref: 21334901
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC2292
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.15 (ug/ml), Ref: 20116898
TCMC1491
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 0.00423 (ug/ml), Ref: 21334901
IC50: 0.00211 (ug/ml), Ref: 21334901
TCMC2123
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1537
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 21288041
TCMC1537
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1901
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1236 Mycobacterium bovis Mycobacterium bovis BCG MIC: 26 (ug/ml), Ref: 18849164
TCMC1901
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1191 Bacillus megaterium Bacillus megaterium MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1286 Bacillus cereus Bacillus cereus MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1260 Streptococcus agalactiae Streptococcus agalactiae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1322 Streptococcus mitis Streptococcus mitis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1323 Corynebacterium pseudodiphtheriticum Corynebacterium pseudodiphtheriticum MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1324 Corynebacterium diphtheriae Corynebacterium diphtheriae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1319 Corynebacterium xerosis Corynebacterium xerosis MIC: 16 (ug/ml), Ref: 18849164
TCMC1803
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 23369537
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2411
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 16 (ug/ml), Ref: 11141098
TCMC2411
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 64 (ug/ml), Ref: 12608857
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC2459
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 37.5 (ug/ml), Ref: 9748372
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC749
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 16945527
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC614
TCMT1454 Bacillus subtilis Bacillus subtilis IC50: 98.5 (ug/ml), Ref: 25981688
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC2578
TCMT1251 Candida albicans Candida albicans IC50: 82.98 (ug/ml), Ref: 25686593
TCMC2182
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 12.5 (ug/ml), Ref: 22280816
TCMC2281
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 13 (ug/ml), Ref: 21334901
TCMC2281
TCMT1318 Human T-lymphotropic virus 1 Human T-lymphotropic virus 1 IC50: 3.98 (ug/ml), Ref: 21334901
TCMC755
TCMT1251 Candida albicans Candida albicans IC50: 6 (ug/ml), Ref: 12502337
TCMC755
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC755
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 6.46 (ug/ml), Ref: 25564380
TCMC1428
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1428
TCMT1286 Bacillus cereus Bacillus cereus MIC: 25 (ug/ml), Ref: 12762812
TCMC1428
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 32.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 26 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2613
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 15 (ug/ml), Ref: 9748372
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2660
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 6.25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2014
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 10 (ug/ml), Ref: 17220400
TCMC2025
TCMT1218 Staphylococcus aureus Staphylococcus aureus MBC: 0.12 (ug/ml), Ref: 18004816
TCMC2025
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MBC: 0.12 (ug/ml), Ref: 18004816
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2025
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MBC: 0.12 (ug/ml), Ref: 18004816
TCMC1123
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1123
TCMT1442 Leishmania donovani Leishmania donovani IC50: 25 (ug/ml), Ref: 15679330
TCMC2025
TCMT1246 Escherichia coli Escherichia coli MBC: 0.12 (ug/ml), Ref: 18004816
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1491
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 0.92 (ug/ml), Ref: 21334901
TCMC1491
TCMT1318 Human T-lymphotropic virus 1 Human T-lymphotropic virus 1 IC50: 1.07 (ug/ml), Ref: 21334901
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1403
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC2018
TCMT1155 Farnesyl pyrophosphate synthase Leishmania major Ki: 17 (nM), Ref: 15828834
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850