References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC1112
|
TCMT203 |
Glucose-6-phosphate 1-dehydrogenase |
Homo sapiens |
Ki: 3400 (nM), Ref: 19231202 Ki: 3000 (nM), Ref: 19231202 IC50: 9400 (nM), Ref: 22506561 |
TCMC1982
|
TCMT239 |
Serine/threonine-protein kinase PIM1 |
Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
TCMC1982
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
TCMC1982
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
TCMC1982
|
TCMT44 |
Glyoxalase I |
Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
TCMC1982
|
TCMT66 |
Estradiol 17-beta-dehydrogenase 2 |
Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
TCMC1982
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
TCMC1982
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
TCMC1982
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
TCMC1982
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
TCMC1982
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
TCMC1982
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
TCMC1982
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
TCMC1982
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
TCMC1982
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
TCMC1982
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
TCMC1982
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
TCMC1982
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
TCMC1982
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
TCMC1982
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
TCMC1982
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
TCMC1982
|
TCMT320 |
Matrix metalloproteinase 3 |
Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
TCMC1982
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
TCMC1982
|
TCMT322 |
Matrix metalloproteinase 13 |
Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
TCMC1982
|
TCMT422 |
CaM kinase II beta |
Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
TCMC1982
|
TCMT265 |
Glycogen synthase kinase-3 beta |
Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
TCMC1982
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
TCMC1982
|
TCMT784 |
Vasopressin V2 receptor |
Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
TCMC1982
|
TCMT785 |
Interleukin-8 receptor A |
Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
TCMC1982
|
TCMT786 |
C-C chemokine receptor type 4 |
Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
TCMC1982
|
TCMT260 |
Tyrosine-protein kinase receptor FLT3 |
Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
TCMC1982
|
TCMT601 |
Thrombin |
Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
TCMC1982
|
TCMT370 |
Vascular endothelial growth factor receptor 2 |
Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
TCMC1982
|
TCMT212 |
Tyrosine-protein kinase SRC |
Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
TCMC1982
|
TCMT791 |
Protein kinase N1 |
Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
TCMC1982
|
TCMT484 |
Serine/threonine-protein kinase PLK1 |
Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
TCMC1982
|
TCMT462 |
Serine/threonine-protein kinase NEK6 |
Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
TCMC1982
|
TCMT445 |
Serine/threonine-protein kinase NEK2 |
Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
TCMC1982
|
TCMT401 |
Hepatocyte growth factor receptor |
Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
TCMC1982
|
TCMT369 |
Insulin-like growth factor I receptor |
Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
TCMC1982
|
TCMT441 |
Focal adhesion kinase 1 |
Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
TCMC1982
|
TCMT388 |
Tyrosine-protein kinase receptor UFO |
Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
TCMC1982
|
TCMT374 |
Serine/threonine-protein kinase Aurora-B |
Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
TCMC1982
|
TCMT436 |
NUAK family SNF1-like kinase 1 |
Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
TCMC1982
|
TCMT402 |
ALK tyrosine kinase receptor |
Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
TCMC1982
|
TCMT479 |
Serine/threonine-protein kinase AKT |
Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
TCMC1982
|
TCMT592 |
Xanthine dehydrogenase |
Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
TCMC1982
|
TCMT793 |
Liver glycogen phosphorylase |
Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
TCMC1982
|
TCMT33 |
Cytochrome P450 3A4 |
Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
TCMC1982
|
TCMT217 |
Cytochrome P450 2C8 |
Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
TCMC1982
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
TCMC1155
|
TCMT230 |
Estradiol 17-beta-dehydrogenase 3 |
Homo sapiens |
IC50: 330 (nM), Ref: 11086723 IC50: 330 (nM), Ref: 16078844 |
TCMC1597
|
TCMT807 |
Solute carrier family 22 member 12 |
Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
TCMC1597
|
TCMT236 |
Estrogen receptor beta |
Homo sapiens |
IC50: 2927.18 (nM), Ref: |
TCMC1597
|
TCMT61 |
Induced myeloid leukemia cell differentiation protein Mcl-1 |
Homo sapiens |
IC50: 2988.26 (nM), Ref: |
TCMC1597
|
TCMT739 |
G-protein coupled receptor 35 |
Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
TCMC1597
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
TCMC1597
|
TCMT283 |
Receptor-type tyrosine-protein phosphatase S |
Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
TCMC2111
|
TCMT614 |
Egl nine homolog 1 |
Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
TCMC1898
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
TCMC1898
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
TCMC1898
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
TCMC1898
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
TCMC732
|
TCMT280 |
Aldo-keto reductase family 1 member B10 |
Homo sapiens |
IC50: 5900 (nM), Ref: 21561086 |
TCMC847
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
TCMC847
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
TCMC847
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
TCMC847
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
TCMC847
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
TCMC847
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
TCMC847
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
TCMC847
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
TCMC847
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
TCMC847
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
TCMC847
|
TCMT101 |
Protein-tyrosine phosphatase 1B |
Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
TCMC847
|
TCMT321 |
Matrix metalloproteinase 9 |
Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
TCMC847
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
TCMC847
|
TCMT295 |
Matrix metalloproteinase-1 |
Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
TCMC847
|
TCMT130 |
Arachidonate 5-lipoxygenase |
Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
TCMC2018
|
TCMT907 |
Farnesyl diphosphate synthase |
Homo sapiens |
IC50: 452.9 (nM), Ref: 18327899 Ki: 82.2 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18327899 Ki: 0.36 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18434151 IC50: 300 (nM), Ref: 20801032 IC50: 11 (nM), Ref: 22390415 IC50: 860 (nM), Ref: 22390415 IC50: 11 (nM), Ref: 22884353 IC50: 10 (nM), Ref: 21780776 IC50: 5.2 (nM), Ref: 23998921 IC50: 11 (nM), Ref: 23998921 IC50: 6 (nM), Ref: 24911527 IC50: 11 (nM), Ref: 25630225 IC50: 6 (nM), Ref: 25935643 IC50: 0.36 (nM), Ref: 25815158 IC50: 82 (nM), Ref: 25815158 |
TCMC1133
|
TCMT82 |
Estrogen receptor alpha |
Homo sapiens |
IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030 |
TCMC1133
|
TCMT236 |
Estrogen receptor beta |
Homo sapiens |
IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030 |
TCMC1133
|
TCMT187 |
Androgen Receptor |
Homo sapiens |
IC50: 19.1 (nM), Ref: 16309907 |
TCMC1133
|
TCMT99 |
Testis-specific androgen-binding protein |
Homo sapiens |
IC50: 50 (nM), Ref: 17149875 |
TCMC1133
|
TCMT591 |
Estrogen-related receptor alpha |
Homo sapiens |
IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346 |
TCMC1133
|
TCMT910 |
Estrogen-related receptor beta |
Homo sapiens |
IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346 |
TCMC1133
|
TCMT344 |
Aldehyde oxidase |
Homo sapiens |
IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261 |
TCMC1133
|
TCMT974 |
G-protein coupled estrogen receptor 1 |
Homo sapiens |
Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A |