References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC1881
|
TCMT151 |
Protein kinase C alpha |
Homo sapiens |
Ki: 2.5 (nM), Ref: 11327599 Ki: 6.4 (nM), Ref: 21596562 |
TCMC1881
|
TCMT152 |
Protein kinase C beta |
Homo sapiens |
Ki: 1.8 (nM), Ref: 11327599 |
TCMC1881
|
TCMT153 |
Protein kinase C gamma |
Homo sapiens |
Ki: 4.9 (nM), Ref: 11327599 |
TCMC1881
|
TCMT154 |
Protein kinase C delta |
Homo sapiens |
Ki: 0.8 (nM), Ref: 11327599 |
TCMC1881
|
TCMT155 |
Protein kinase C epsilon |
Homo sapiens |
Ki: 0.45 (nM), Ref: 11327599 |
TCMC1495
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
TCMC1495
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
TCMC1495
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1112
|
TCMT203 |
Glucose-6-phosphate 1-dehydrogenase |
Homo sapiens |
Ki: 3400 (nM), Ref: 19231202 Ki: 3000 (nM), Ref: 19231202 IC50: 9400 (nM), Ref: 22506561 |
TCMC2105
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2105
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1155
|
TCMT230 |
Estradiol 17-beta-dehydrogenase 3 |
Homo sapiens |
IC50: 330 (nM), Ref: 11086723 IC50: 330 (nM), Ref: 16078844 |
TCMC1597
|
TCMT807 |
Solute carrier family 22 member 12 |
Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
TCMC1597
|
TCMT236 |
Estrogen receptor beta |
Homo sapiens |
IC50: 2927.18 (nM), Ref: |
TCMC1597
|
TCMT61 |
Induced myeloid leukemia cell differentiation protein Mcl-1 |
Homo sapiens |
IC50: 2988.26 (nM), Ref: |
TCMC1597
|
TCMT739 |
G-protein coupled receptor 35 |
Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
TCMC1597
|
TCMT261 |
Death-associated protein kinase 1 |
Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
TCMC1597
|
TCMT283 |
Receptor-type tyrosine-protein phosphatase S |
Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
TCMC1830
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
TCMC1830
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
TCMC1830
|
TCMT808 |
Fatty acid binding protein epidermal |
Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
TCMC1830
|
TCMT809 |
Fatty acid binding protein intestinal |
Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
TCMC1830
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1830
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1898
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
TCMC1898
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
TCMC1898
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
TCMC1898
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
TCMC1788
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT126 |
Telomerase reverse transcriptase |
Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
TCMC1788
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
TCMC1496
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1496
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1496
|
TCMT164 |
Cyclooxygenase-1 |
Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
TCMC897
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
TCMC897
|
TCMT280 |
Aldo-keto reductase family 1 member B10 |
Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
TCMC1676
|
TCMT30 |
Cyclooxygenase-2 |
Homo sapiens |
IC50: 8500 (nM), Ref: 23869482 |
TCMC1133
|
TCMT82 |
Estrogen receptor alpha |
Homo sapiens |
IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030 |
TCMC1133
|
TCMT236 |
Estrogen receptor beta |
Homo sapiens |
IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030 |
TCMC1133
|
TCMT187 |
Androgen Receptor |
Homo sapiens |
IC50: 19.1 (nM), Ref: 16309907 |
TCMC1133
|
TCMT99 |
Testis-specific androgen-binding protein |
Homo sapiens |
IC50: 50 (nM), Ref: 17149875 |
TCMC1133
|
TCMT591 |
Estrogen-related receptor alpha |
Homo sapiens |
IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346 |
TCMC1133
|
TCMT910 |
Estrogen-related receptor beta |
Homo sapiens |
IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346 |
TCMC1133
|
TCMT344 |
Aldehyde oxidase |
Homo sapiens |
IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261 |
TCMC1133
|
TCMT974 |
G-protein coupled estrogen receptor 1 |
Homo sapiens |
Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A |