References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
Ingredient ID & Structure |
Target ID |
Target Name |
Target Organism |
Activity Records & Reference |
TCMC1173
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
TCMC1173
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
TCMC1173
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
TCMC1173
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
TCMC1173
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
TCMC1173
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
TCMC1173
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
TCMC1173
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
TCMC1187
|
TCMT151 |
Protein kinase C alpha |
Homo sapiens |
IC50: 1900 (nM), Ref: 9834166 |
TCMC1495
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
TCMC1495
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
TCMC1495
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1495
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2037
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
TCMC2037
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
TCMC2037
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
TCMC795
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 8000 (nM), Ref: 24341381 |
TCMC737
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 168 (nM), Ref: 26498393 |
TCMC737
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 5591.2 (nM), Ref: 26498393 |
TCMC737
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 423.7 (nM), Ref: 26498393 |
TCMC737
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4.9 (nM), Ref: 26498393 |
TCMC1480
|
TCMT107 |
Glutamate receptor ionotropic kainate 2 |
Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
TCMC1480
|
TCMT108 |
Glutamate receptor ionotropic, AMPA 1 |
Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
TCMC1480
|
TCMT109 |
Glutamate receptor ionotropic, AMPA 2 |
Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
TCMC1480
|
TCMT110 |
Glutamate receptor ionotropic, AMPA 4 |
Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
TCMC1480
|
TCMT111 |
Glutamate receptor ionotropic kainate 5 |
Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
TCMC1480
|
TCMT660 |
Metabotropic glutamate receptor 8 |
Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
TCMC1480
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
TCMC1480
|
TCMT653 |
Metabotropic glutamate receptor 1 |
Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT654 |
Metabotropic glutamate receptor 5 |
Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT657 |
Metabotropic glutamate receptor 4 |
Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT655 |
Metabotropic glutamate receptor 2 |
Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
TCMC1480
|
TCMT664 |
Excitatory amino acid transporter 3 |
Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
TCMC1480
|
TCMT656 |
Metabotropic glutamate receptor 3 |
Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
TCMC1083
|
TCMT38 |
Dopamine D2 receptor |
Homo sapiens |
Ki: 1.89 (nM), Ref: 10465538 Ki: 759 (nM), Ref: 10465538 Ki: 572 (nM), Ref: 8893836 Ki: 20 (nM), Ref: 10691700 Ki: 17 (nM), Ref: 10691700 Ki: 450 (nM), Ref: 18834111 Ki: 360 (nM), Ref: 18834111 Ki: 2100 (nM), Ref: 20155917 Ki: 2.9 (nM), Ref: 20155917 Ki: 2100 (nM), Ref: 22846798 Ki: 422 (nM), Ref: 23134120 Ki: 110 (nM), Ref: 23428965 Ki: 190 (nM), Ref: 23428965 Ki: 2100 (nM), Ref: 23727194 Ki: 8 (nM), Ref: 24138311 Ki: 8.73 (nM), Ref: 27035329 Ki: 3690 (nM), Ref: 27035329 Ki: 48 (nM), Ref: 27132867 |
TCMC1083
|
TCMT651 |
Dopamine D3 receptor |
Homo sapiens |
Ki: 13.2 (nM), Ref: 8893836 Ki: 50 (nM), Ref: 10691700 Ki: 240 (nM), Ref: 18834111 Ki: 72 (nM), Ref: 18834111 Ki: 15 (nM), Ref: 22846798 Ki: 20 (nM), Ref: 23134120 Ki: 21 (nM), Ref: 23428965 Ki: 15 (nM), Ref: 23727194 Ki: 7.58 (nM), Ref: 27035329 Ki: 293 (nM), Ref: 27035329 |
TCMC1083
|
TCMT635 |
Dopamine transporter |
Homo sapiens |
Ki: 6400 (nM), Ref: 14592523 IC50: 460 (nM), Ref: 14592523 |
TCMC1083
|
TCMT634 |
Norepinephrine transporter |
Homo sapiens |
IC50: 6.63 (nM), Ref: 14592523 |
TCMC1083
|
TCMT648 |
Dopamine D4 receptor |
Homo sapiens |
Ki: 1.2 (nM), Ref: 10691700 Ki: 6.2 (nM), Ref: 18834111 Ki: 8.9 (nM), Ref: 23428965 |
TCMC1083
|
TCMT316 |
Melatonin receptor 1A |
Homo sapiens |
Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
TCMC1083
|
TCMT317 |
Melatonin receptor 1B |
Homo sapiens |
Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
TCMC1083
|
TCMT27 |
Dopamine D1 receptor |
Homo sapiens |
Ki: 4470 (nM), Ref: 23134120 |
TCMC1083
|
TCMT8 |
Lysine-specific demethylase 4D-like |
Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
TCMC632
|
TCMT597 |
Solute carrier family 28 member 3 |
Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
TCMC632
|
TCMT709 |
Sodium/nucleoside cotransporter 2 |
Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
TCMC632
|
TCMT710 |
Sodium/nucleoside cotransporter 1 |
Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
TCMC632
|
TCMT296 |
Adenosine A1 receptor |
Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
TCMC632
|
TCMT112 |
Adenosine A3 receptor |
Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
TCMC1956
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
TCMC1956
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
TCMC1956
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
TCMC1956
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
TCMC1956
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
TCMC1956
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
TCMC1956
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
TCMC1956
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
TCMC876
|
TCMT560 |
Coagulation factor X |
Homo sapiens |
IC50: 720 (nM), Ref: 9834152 Ki: 450 (nM), Ref: 9834152 |
TCMC1624
|
TCMT560 |
Coagulation factor X |
Homo sapiens |
IC50: 280 (nM), Ref: 9834152 Ki: 690 (nM), Ref: 9834152 |
TCMC2031
|
TCMT131 |
Acetylcholinesterase |
Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
TCMC1409
|
TCMT22 |
Intestinal alkaline phosphatase |
Homo sapiens |
IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref: |
TCMC1409
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 4500 (nM), Ref: 22261024 |
TCMC1409
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393 |
TCMC1409
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 75.7 (nM), Ref: 26498393 |
TCMC1409
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 3.8 (nM), Ref: 26498393 |
TCMC1409
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393 |
TCMC1158
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 3100 (nM), Ref: 24835197 Ki: 6840 (nM), Ref: 24835197 |
TCMC614
|
TCMT151 |
Protein kinase C alpha |
Homo sapiens |
IC50: 9300 (nM), Ref: 9834166 |
TCMC916
|
TCMT161 |
Hydroxycarboxylic acid receptor 2 |
Homo sapiens |
Ki: 4900 (nM), Ref: 21167710 |
TCMC2105
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2105
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
TCMC1830
|
TCMT298 |
Fatty acid binding protein muscle |
Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
TCMC1830
|
TCMT808 |
Fatty acid binding protein epidermal |
Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
TCMC1830
|
TCMT809 |
Fatty acid binding protein intestinal |
Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
TCMC1830
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1830
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1830
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1202
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
TCMC1202
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1202
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
TCMC1202
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
TCMC1202
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
TCMC1202
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
TCMC1202
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1202
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
TCMC1202
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
TCMC1202
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
TCMC1202
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
TCMC1202
|
TCMT822 |
Alpha-(1,3)-fucosyltransferase 7 |
Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
TCMC2111
|
TCMT614 |
Egl nine homolog 1 |
Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
TCMC1839
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
TCMC1839
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
TCMC1839
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
TCMC1839
|
TCMT135 |
Carbonic anhydrase XIV |
Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
TCMC1839
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
TCMC1839
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
TCMC1839
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
TCMC1839
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
TCMC1839
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
TCMC1839
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
TCMC1839
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
TCMC2139
|
TCMT560 |
Coagulation factor X |
Homo sapiens |
IC50: 210 (nM), Ref: 9834152 Ki: 440 (nM), Ref: 9834152 |
TCMC1788
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1788
|
TCMT126 |
Telomerase reverse transcriptase |
Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
TCMC1788
|
TCMT297 |
Fatty acid binding protein adipocyte |
Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
TCMC1845
|
TCMT560 |
Coagulation factor X |
Homo sapiens |
IC50: 560 (nM), Ref: 9834152 Ki: 990 (nM), Ref: 9834152 |
TCMC1356
|
TCMT223 |
Aldose reductase |
Homo sapiens |
IC50: 3000 (nM), Ref: 22261024 |
TCMC2201
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 8700 (nM), Ref: 21332115 |
TCMC1611
|
TCMT810 |
Toll-like receptor 2 |
Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
TCMC1611
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1832
|
TCMT63 |
Peroxisome proliferator-activated receptor alpha |
Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1832
|
TCMT64 |
Peroxisome proliferator-activated receptor delta |
Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC1832
|
TCMT67 |
Peroxisome proliferator-activated receptor gamma |
Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
TCMC2018
|
TCMT907 |
Farnesyl diphosphate synthase |
Homo sapiens |
IC50: 452.9 (nM), Ref: 18327899 Ki: 82.2 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18327899 Ki: 0.36 (nM), Ref: 18327899 IC50: 5.7 (nM), Ref: 18434151 IC50: 300 (nM), Ref: 20801032 IC50: 11 (nM), Ref: 22390415 IC50: 860 (nM), Ref: 22390415 IC50: 11 (nM), Ref: 22884353 IC50: 10 (nM), Ref: 21780776 IC50: 5.2 (nM), Ref: 23998921 IC50: 11 (nM), Ref: 23998921 IC50: 6 (nM), Ref: 24911527 IC50: 11 (nM), Ref: 25630225 IC50: 6 (nM), Ref: 25935643 IC50: 0.36 (nM), Ref: 25815158 IC50: 82 (nM), Ref: 25815158 |
TCMC1236
|
TCMT236 |
Estrogen receptor beta |
Homo sapiens |
IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref: |
TCMC1236
|
TCMT82 |
Estrogen receptor alpha |
Homo sapiens |
IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref: |
TCMC1236
|
TCMT591 |
Estrogen-related receptor alpha |
Homo sapiens |
IC50: 10 (nM), Ref: 17482813 |
TCMC1236
|
TCMT910 |
Estrogen-related receptor beta |
Homo sapiens |
IC50: 395 (nM), Ref: 17482813 |
TCMC1236
|
TCMT65 |
Estradiol 17-beta-dehydrogenase 1 |
Homo sapiens |
IC50: 2210 (nM), Ref: 18533708 |
TCMC1236
|
TCMT344 |
Aldehyde oxidase |
Homo sapiens |
IC50: 340 (nM), Ref: 20853847 |
TCMC1236
|
TCMT289 |
Thromboxane-A synthase |
Homo sapiens |
IC50: 7720 (nM), Ref: |
TCMC547
|
TCMT313 |
Serotonin 2b (5-HT2b) receptor |
Homo sapiens |
IC50: 8912.51 (nM), Ref: 24582985 Ki: 2454.71 (nM), Ref: 24582985 |
TCMC547
|
TCMT644 |
Serotonin 3a (5-HT3a) receptor |
Homo sapiens |
Ki: 2511.89 (nM), Ref: 24582985 |
TCMC90
|
TCMT207 |
Beta-secretase 1 |
Homo sapiens |
IC50: 2400 (nM), Ref: 14592472 |
TCMC2209
|
TCMT597 |
Solute carrier family 28 member 3 |
Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
TCMC2209
|
TCMT710 |
Sodium/nucleoside cotransporter 1 |
Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
TCMC1064
|
TCMT219 |
Cytochrome P450 1A2 |
Homo sapiens |
IC50: 2437 (nM), Ref: 20696580 |
TCMC1064
|
TCMT215 |
Cytochrome P450 1A1 |
Homo sapiens |
IC50: 140 (nM), Ref: 20696580 |
TCMC1064
|
TCMT257 |
Cytochrome P450 1B1 |
Homo sapiens |
IC50: 29 (nM), Ref: 20696580 |
TCMC1228
|
TCMT156 |
Cytochrome P450 19A1 |
Homo sapiens |
IC50: 5200 (nM), Ref: 18558747 |
TCMC878
|
TCMT133 |
Carbonic anhydrase I |
Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
TCMC878
|
TCMT134 |
Carbonic anhydrase II |
Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
TCMC878
|
TCMT143 |
Carbonic anhydrase III |
Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
TCMC878
|
TCMT142 |
Carbonic anhydrase IV |
Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
TCMC878
|
TCMT141 |
Carbonic anhydrase VA |
Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
TCMC878
|
TCMT140 |
Carbonic anhydrase VB |
Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
TCMC878
|
TCMT139 |
Carbonic anhydrase VI |
Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
TCMC878
|
TCMT138 |
Carbonic anhydrase VII |
Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
TCMC878
|
TCMT137 |
Carbonic anhydrase IX |
Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
TCMC878
|
TCMT136 |
Carbonic anhydrase XII |
Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |
TCMC770
|
TCMT588 |
D-amino-acid oxidase |
Homo sapiens |
Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755 |
TCMC1378
|
TCMT306 |
Matrix metalloproteinase-2 |
Homo sapiens |
IC50: 8960 (nM), Ref: 22658537 |
TCMC1378
|
TCMT734 |
Matrix metalloproteinase 12 |
Homo sapiens |
IC50: 8220 (nM), Ref: 22658537 |