TCM Putative Target References: TCMF7177


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC879
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC417
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 7585.78 (nM), Ref: 23574272
IC50: 7500 (nM), Ref: 23574272
TCMC417
TCMT128 Tankyrase-2 Homo sapiens IC50: 870.96 (nM), Ref: 23574272
IC50: 870 (nM), Ref: 23574272
TCMC417
TCMT129 Tankyrase-1 Homo sapiens IC50: 645.65 (nM), Ref: 23574272
IC50: 630 (nM), Ref: 23574272
TCMC417
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2000 (nM), Ref: 24368208
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1372
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2330 (nM), Ref: 22245047
TCMC1372
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 3630 (nM), Ref: 22245047
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC704
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4000 (nM), Ref: 21030469
IC50: 3600 (nM), Ref: 21030469
TCMC2061
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 9550 (nM), Ref:
TCMC424
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 550 (nM), Ref: 21282059
TCMC424
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 21282059
TCMC424
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4410 (nM), Ref: 21282059
TCMC424
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3670 (nM), Ref: 21282059
TCMC424
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 650 (nM), Ref: 22668600
TCMC424
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7170 (nM), Ref: 22668600
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC1851
TCMT560 Coagulation factor X Homo sapiens IC50: 170 (nM), Ref: 9834152
Ki: 570 (nM), Ref: 9834152
TCMC1851
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3760 (nM), Ref: 24835197
Ki: 5130 (nM), Ref: 24835197
TCMC1851
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 2350 (nM), Ref: 26395057
Ki: 2600 (nM), Ref: 26395057
TCMC795
TCMT223 Aldose reductase Homo sapiens IC50: 8000 (nM), Ref: 24341381
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC882
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 780 (nM), Ref: 25812966
TCMC1773
TCMT575 Phospholipase A2 group IIA Homo sapiens IC50: 3500 (nM), Ref: 16504502
TCMC416
TCMT207 Beta-secretase 1 Homo sapiens IC50: 4500 (nM), Ref: 14592472
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC231
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 4800 (nM), Ref: 20806783
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC891
TCMT598 DNA topoisomerase I Homo sapiens IC50: 50 (nM), Ref: 1324981
IC50: 100 (nM), Ref: 1324981
TCMC2188
TCMT223 Aldose reductase Homo sapiens IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC1620
TCMT223 Aldose reductase Homo sapiens IC50: 88 (nM), Ref: 22236472
TCMC1620
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 130 (nM), Ref: 22236472
TCMC2054
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 9640 (nM), Ref: 18507367
TCMC2054
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 6610 (nM), Ref:
TCMC2054
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 600 (nM), Ref: 26602279
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC845
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 630 (nM), Ref: 19231207
TCMC1376
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 40 (nM), Ref: 11678654
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1113
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC2003
TCMT82 Estrogen receptor alpha Homo sapiens Ki: 785 (nM), Ref: 15634023
TCMC2003
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 2840 (nM), Ref: 16814546
IC50: 4120 (nM), Ref: 18063374
IC50: 625 (nM), Ref:
TCMC2003
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 996 (nM), Ref: 17604631
IC50: 750 (nM), Ref: 20527891
IC50: 996 (nM), Ref: 26850006
TCMC2003
TCMT329 Quinone reductase 2 Homo sapiens IC50: 960 (nM), Ref: 19265439
IC50: 450 (nM), Ref: 20036559
IC50: 450 (nM), Ref: 20356739
IC50: 960 (nM), Ref: 21261296
IC50: 6900 (nM), Ref: 23953689
Ki: 88 (nM), Ref: 23953689
IC50: 1400 (nM), Ref: 26854376
IC50: 913 (nM), Ref: 26854376
TCMC2003
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2210 (nM), Ref: 20674354
TCMC2003
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2770 (nM), Ref: 20674354
TCMC2003
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 9090 (nM), Ref: 20674354
TCMC2003
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4470 (nM), Ref: 20674354
TCMC2003
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4750 (nM), Ref: 20674354
TCMC2003
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4640 (nM), Ref: 20674354
TCMC2003
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8070 (nM), Ref: 20674354
TCMC2003
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4350 (nM), Ref: 20674354
TCMC2003
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 20674354
TCMC2003
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 950 (nM), Ref: 20674354
TCMC2003
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4090 (nM), Ref: 20674354
TCMC2003
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 830 (nM), Ref: 20674354
TCMC2003
TCMT729 PI3-kinase p110-alpha subunit Homo sapiens IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT730 PI3-kinase p110-beta subunit Homo sapiens IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4100 (nM), Ref: 27190601
IC50: 2600 (nM), Ref: 27190601
TCMC1446
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 6300 (nM), Ref: 21641214
TCMC1334
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 4200 (nM), Ref: 19481465
TCMC1334
TCMT114 Cannabinoid CB2 receptor Homo sapiens Ki: 5610 (nM), Ref: 24900561
Ki: 5.61 (nM), Ref: 27078864
TCMC1334
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 6460 (nM), Ref: 24900561
Ki: 6.46 (nM), Ref: 27078864
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC143
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 1610 (nM), Ref:
TCMC706
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 9510 (nM), Ref: 19028102
TCMC1986
TCMT223 Aldose reductase Homo sapiens IC50: 150 (nM), Ref: 18165015
IC50: 2000 (nM), Ref: 22261024
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 7500 (nM), Ref: 16610779
TCMC1102
TCMT752 Casein kinase II alpha Homo sapiens IC50: 40 (nM), Ref: 19414254
TCMC1102
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2320 (nM), Ref: 20185318
TCMC1102
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2180 (nM), Ref: 20185318
TCMC1102
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC1102
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7590 (nM), Ref: 20185318
TCMC1102
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7060 (nM), Ref: 20185318
TCMC1102
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6320 (nM), Ref: 20185318
Ki: 8790 (nM), Ref: 22892213
TCMC1102
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9370 (nM), Ref: 20185318
TCMC1102
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8910 (nM), Ref: 20185318
TCMC1102
TCMT753 Mothers against decapentaplegic homolog 3 Homo sapiens IC50: 142 (nM), Ref:
TCMC1102
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 760 (nM), Ref:
TCMC1102
TCMT189 Dual specificity protein phosphatase 3 Homo sapiens IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102
TCMT223 Aldose reductase Homo sapiens IC50: 200 (nM), Ref: 22261024
TCMC1102
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 510 (nM), Ref: 22377675
TCMC1102
TCMT354 Serine/threonine-protein kinase Aurora-A Homo sapiens IC50: 2480 (nM), Ref: 22377675
TCMC1102
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 2500 (nM), Ref: 22377675
TCMC1102
TCMT626 Serine/threonine-protein kinase B-raf Homo sapiens IC50: 1760 (nM), Ref: 22377675
TCMC1102
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 690 (nM), Ref: 22377675
TCMC1102
TCMT418 Ephrin type-B receptor 4 Homo sapiens IC50: 1830 (nM), Ref: 22377675
TCMC1102
TCMT704 Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50: 3540 (nM), Ref: 22377675
TCMC1102
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 3110 (nM), Ref: 22377675
TCMC1102
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 250 (nM), Ref: 22377675
TCMC1102
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 800 (nM), Ref: 22377675
TCMC1102
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 790 (nM), Ref: 22377675
TCMC1102
TCMT457 Vascular endothelial growth factor receptor 3 Homo sapiens IC50: 1540 (nM), Ref: 22377675
TCMC1102
TCMT377 Insulin receptor Homo sapiens IC50: 340 (nM), Ref: 22377675
TCMC1102
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 22377675
TCMC1102
TCMT536 Platelet-derived growth factor receptor beta Homo sapiens IC50: 1300 (nM), Ref: 22377675
TCMC1102
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT755 Serine/threonine-protein kinase PLK4 Homo sapiens IC50: 2970 (nM), Ref: 22377675
TCMC1102
TCMT502 Tyrosine-protein kinase TIE-2 Homo sapiens IC50: 260 (nM), Ref: 22377675
TCMC1102
TCMT756 Mitogen-activated protein kinase kinase kinase 8 Homo sapiens IC50: 2370 (nM), Ref: 22377675
TCMC1102
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 100 (nM), Ref: 24900447
TCMC1102
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8150 (nM), Ref: 22892213
TCMC1102
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1102
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3900 (nM), Ref: 24835197
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC910
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1118 (nM), Ref: 20696580
TCMC910
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 95 (nM), Ref: 20696580
TCMC910
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 20 (nM), Ref: 20696580
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC2183
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens IC50: 7000 (nM), Ref: 23713606
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC614
TCMT151 Protein kinase C alpha Homo sapiens IC50: 9300 (nM), Ref: 9834166
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC1281
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 10 (nM), Ref: 19564108
IC50: 18.6 (nM), Ref: 22148241
IC50: 6 (nM), Ref: 22360639
TCMC1281
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 1 (nM), Ref: 19564108
IC50: 0.7 (nM), Ref: 22148241
IC50: 0.4 (nM), Ref: 22360639
TCMC469
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 100 (nM), Ref: 22921742
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC1015
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 4320 (nM), Ref:
TCMC2196
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 64 (nM), Ref: 22819942
IC50: 64 (nM), Ref: 23146282
TCMC2196
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 150 (nM), Ref: 22819942
TCMC2196
TCMT336 Indoleamine 2,3-dioxygenase Homo sapiens IC50: 53.7 (nM), Ref: 24099220
IC50: 7150 (nM), Ref: 24099220
Ki: 4810 (nM), Ref: 24099220
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2063
TCMT646 Serotonin 5a (5-HT5a) receptor Homo sapiens Ki: 126 (nM), Ref: 12825922
IC50: 180 (nM), Ref: 18983139
Ki: 110 (nM), Ref: 18983139
IC50: 184 (nM), Ref: 18588282
Ki: 170 (nM), Ref: 21726069
IC50: 280 (nM), Ref: 23582449
Ki: 82 (nM), Ref: 23466604
IC50: 160 (nM), Ref: 23466604
IC50: 180 (nM), Ref: 26988801
TCMC2063
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 65 (nM), Ref: 12825922
Ki: 100 (nM), Ref: 15357994
IC50: 200 (nM), Ref: 18983139
Ki: 93 (nM), Ref: 18983139
IC50: 262 (nM), Ref: 18588282
IC50: 27.5 (nM), Ref: 20170099
Ki: 84 (nM), Ref: 21726069
Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
IC50: 180 (nM), Ref: 23582449
Ki: 50 (nM), Ref: 23466604
IC50: 100 (nM), Ref: 23466604
Ki: 33 (nM), Ref: 24805037
Ki: 33 (nM), Ref: 25557493
IC50: 120 (nM), Ref: 26988801
Ki: 100 (nM), Ref: 26996373
TCMC2063
TCMT160 Serotonin 7 (5-HT7) receptor Homo sapiens Ki: 8.1 (nM), Ref: 12825922
IC50: 0.61 (nM), Ref: 18983139
Ki: 0.22 (nM), Ref: 18983139
IC50: 2.55 (nM), Ref: 12713409
IC50: 1.5 (nM), Ref: 18588282
Ki: 0.13 (nM), Ref: 21726069
IC50: 0.49 (nM), Ref: 23582449
Ki: 0.11 (nM), Ref: 23466604
IC50: 0.29 (nM), Ref: 23466604
Ki: 1.4 (nM), Ref: 24763360
Ki: 0.8 (nM), Ref: 24805037
Ki: 0.8 (nM), Ref: 25557493
IC50: 0.25 (nM), Ref: 26988801
TCMC2063
TCMT37 Serotonin 2a (5-HT2a) receptor Homo sapiens Ki: 14 (nM), Ref: 15081042
Ki: 8.2 (nM), Ref: 16392816
Ki: 14 (nM), Ref: 16257207
Ki: 120 (nM), Ref: 18468904
Ki: 160 (nM), Ref: 18468904
Ki: 130 (nM), Ref: 18468904
Ki: 150 (nM), Ref: 18468904
Ki: 320 (nM), Ref: 11975483
Ki: 690 (nM), Ref: 17067154
Ki: 323.59 (nM), Ref: 23301527
Ki: 320 (nM), Ref: 23301527
TCMC2063
TCMT313 Serotonin 2b (5-HT2b) receptor Homo sapiens Ki: 12 (nM), Ref: 15081042
Ki: 13 (nM), Ref: 12954071
Ki: 13 (nM), Ref: 16392816
Ki: 12 (nM), Ref: 16257207
Ki: 13.49 (nM), Ref: 24582985
TCMC2063
TCMT314 Serotonin 2c (5-HT2c) receptor Homo sapiens Ki: 6.9 (nM), Ref: 15081042
Ki: 8.3 (nM), Ref: 12954071
Ki: 8.3 (nM), Ref: 16392816
Ki: 6.9 (nM), Ref: 16257207
Ki: 130 (nM), Ref: 11975483
Ki: 20 (nM), Ref: 17067154
Ki: 79.43 (nM), Ref: 23301527
Ki: 79 (nM), Ref: 23301527
TCMC2063
TCMT815 Serotonin 1d (5-HT1d) receptor Homo sapiens Ki: 5.5 (nM), Ref: 8071931
Ki: 0.5 (nM), Ref: 18507369
TCMC2063
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens Ki: 2.5 (nM), Ref: 7658447
IC50: 1.2 (nM), Ref: 12954071
Ki: 1.259 (nM), Ref: 18433113
Ki: 10000 (nM), Ref: 18433113
Ki: 0.62 (nM), Ref: 22748706
Ki: 0.9 (nM), Ref: 23332346
Ki: 9.5 (nM), Ref: 24161678
Ki: 2.08 (nM), Ref: 25128671
TCMC2063
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 79 (nM), Ref: 16250647
TCMC2063
TCMT816 Serotonin 1b (5-HT1b) receptor Homo sapiens Ki: 1.1 (nM), Ref: 18507369
IC50: 29 (nM), Ref: 18983139
Ki: 18 (nM), Ref: 18983139
Ki: 14 (nM), Ref: 21726069
IC50: 12 (nM), Ref: 23582449
Ki: 4 (nM), Ref: 23466604
IC50: 6.5 (nM), Ref: 23466604
TCMC2063
TCMT817 Serotonin 4 (5-HT4) receptor Homo sapiens Ki: 1049 (nM), Ref: 19334715
Ki: 500 (nM), Ref: 17067154
Ki: 29.51 (nM), Ref: 19223092
Ki: 109.65 (nM), Ref: 19223092
TCMC2063
TCMT645 Serotonin 1e (5-HT1e) receptor Homo sapiens Ki: 10.72 (nM), Ref: 24365159
Ki: 11 (nM), Ref: 24365159
TCMC418
TCMT223 Aldose reductase Homo sapiens IC50: 78 (nM), Ref: 22236472
TCMC418
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 240 (nM), Ref: 22236472
TCMC418
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4700 (nM), Ref: 22921742
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC183
TCMT188 Dihydrofolate reductase Homo sapiens IC50: 500 (nM), Ref: 26979156
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC755
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens Ki: 600 (nM), Ref: 21739938
TCMC755
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens Ki: 1600 (nM), Ref: 21739938
TCMC755
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4400 (nM), Ref: 21030469
IC50: 7000 (nM), Ref: 21030469
TCMC755
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 8700 (nM), Ref:
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1377
TCMT186 Monoamine oxidase B Homo sapiens Ki: 3000 (nM), Ref: 16137882
Ki: 3000 (nM), Ref: 19342233
IC50: 7943.28 (nM), Ref: 20934874
Ki: 5340 (nM), Ref: 21134756
Ki: 3000 (nM), Ref: 21778064
Ki: 2000 (nM), Ref: 24140951
TCMC1377
TCMT208 Monoamine oxidase A Homo sapiens Ki: 8380 (nM), Ref: 21134756
TCMC1105
TCMT752 Casein kinase II alpha Homo sapiens IC50: 2000 (nM), Ref: 19414254
TCMC1105
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2500 (nM), Ref: 27173800
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC937
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 11.5 (nM), Ref: 23332369
IC50: 6.6 (nM), Ref: 23895532
TCMC937
TCMT801 Tubulin beta-3 chain Homo sapiens IC50: 5.2 (nM), Ref: 23332369
IC50: 5.7 (nM), Ref: 23895532
TCMC1203
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 8000 (nM), Ref: 10.1039/C4MD00086B
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC1179
TCMT187 Androgen Receptor Homo sapiens IC50: 5900 (nM), Ref: 19592245
IC50: 5900 (nM), Ref: 19592245
TCMC1179
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8 (nM), Ref: 20413308
IC50: 10000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1179
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1890 (nM), Ref: 22487176
Ki: 1880 (nM), Ref: 22487176
TCMC1179
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8710 (nM), Ref: 22487176
Ki: 8800 (nM), Ref: 22487176
TCMC1179
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4130 (nM), Ref: 22487176
Ki: 4220 (nM), Ref: 22487176
TCMC1179
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7220 (nM), Ref: 22487176
Ki: 7330 (nM), Ref: 22487176
TCMC1179
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 1380.38 (nM), Ref: 23574272
IC50: 1400 (nM), Ref: 23574272
TCMC1179
TCMT128 Tankyrase-2 Homo sapiens IC50: 147.91 (nM), Ref: 23574272
IC50: 140 (nM), Ref: 23574272
TCMC1179
TCMT129 Tankyrase-1 Homo sapiens IC50: 323.59 (nM), Ref: 23574272
IC50: 320 (nM), Ref: 23574272
IC50: 323.59 (nM), Ref: 24116873
IC50: 330 (nM), Ref: 24116873
TCMC1523
TCMT114 Cannabinoid CB2 receptor Homo sapiens Ki: 1440 (nM), Ref: 24900561
TCMC1523
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 3150 (nM), Ref: 24900561
TCMC4
TCMT207 Beta-secretase 1 Homo sapiens IC50: 6000 (nM), Ref: 14592472
TCMC1798
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1480 (nM), Ref: 23411073
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC1123
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1284 (nM), Ref: 20696580
TCMC1123
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 72.8 (nM), Ref: 26498393
TCMC1123
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1123
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 31.1 (nM), Ref: 26498393
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC2004
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 800 (nM), Ref: 10.1039/C3MD00317E
Ki: 2100 (nM), Ref: 10.1039/C0MD00242A
TCMC2004
TCMT215 Cytochrome P450 1A1 Homo sapiens Ki: 160 (nM), Ref: 10.1039/C0MD00242A
TCMC1892
TCMT508 Tyrosine-protein kinase SYK Homo sapiens IC50: 10000 (nM), Ref: 23917087
TCMC1371
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 4 (nM), Ref: 26562543
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1940
TCMT187 Androgen Receptor Homo sapiens Ki: 8.5 (nM), Ref: 12954062
IC50: 37 (nM), Ref: 12954062
IC50: 37 (nM), Ref: 12781197
IC50: 37 (nM), Ref: 8627601
Ki: 8.5 (nM), Ref: 8627601
Ki: 8.5 (nM), Ref: 9873735
IC50: 37 (nM), Ref: 9784110
Ki: 35 (nM), Ref: 20510622
TCMC1940
TCMT613 Glucocorticoid receptor Homo sapiens Ki: 30.5 (nM), Ref: 12954062
Ki: 30.5 (nM), Ref: 9873735
Ki: 30.5 (nM), Ref: 9784110
TCMC1940
TCMT783 Mineralocorticoid receptor Homo sapiens IC50: 14 (nM), Ref: 12954062
IC50: 14 (nM), Ref: 12781197
IC50: 14 (nM), Ref: 9784110
IC50: 30 (nM), Ref: 8709117
TCMC1940
TCMT904 Progesterone receptor Homo sapiens Ki: 3.5 (nM), Ref: 10212133
IC50: 3.5 (nM), Ref: 11859003
Ki: 3.5 (nM), Ref: 9464361
IC50: 5 (nM), Ref: 8523399
Ki: 3.8 (nM), Ref: 9667968
Ki: 3.467 (nM), Ref: 16821785
Ki: 3.4 (nM), Ref: 18553958
Ki: 5.1 (nM), Ref: 20510622
TCMC1521
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3880 (nM), Ref: 22658537
TCMC1521
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 1200 (nM), Ref: 22658537
TCMC1521
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 7620 (nM), Ref: 22658537
TCMC2055
TCMT747 ATP-binding cassette sub-family G member 2 Homo sapiens IC50: 10000 (nM), Ref: 22822035
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC1063
TCMT277 Solute carrier organic anion transporter family member 1B3 Homo sapiens Ki: 1430 (nM), Ref: 23396419
Ki: 4550 (nM), Ref: 23396419
Ki: 8290 (nM), Ref: 23396419
Ki: 1030 (nM), Ref: 23396419
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC1851
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28 (ug/ml), Ref: 9461665
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1620
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 0.66 (ug/ml), Ref: 11430019
IC50: 5.9 (ug/ml), Ref: 16643034
TCMC2054
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 14.48 (ug/ml), Ref: 20116898
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC1986
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 75.2 (ug/ml), Ref: 9461665
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC469
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 5.4 (ug/ml), Ref: 16643034
TCMC914
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 7.4 (ug/ml), Ref: 16643034
TCMC2063
TCMT1086 Isocitrate lyase Candida albicans IC50: 53 (ug/ml), Ref: 21035332
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1203
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.5 (ug/ml), Ref: 9461665
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC2292
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.15 (ug/ml), Ref: 20116898
TCMC2304
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.3 (ug/ml), Ref: 9461665
TCMC1801
TCMT1136 Neuraminidase Influenza A virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1901
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1236 Mycobacterium bovis Mycobacterium bovis BCG MIC: 26 (ug/ml), Ref: 18849164
TCMC1901
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1191 Bacillus megaterium Bacillus megaterium MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1286 Bacillus cereus Bacillus cereus MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1260 Streptococcus agalactiae Streptococcus agalactiae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1322 Streptococcus mitis Streptococcus mitis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1323 Corynebacterium pseudodiphtheriticum Corynebacterium pseudodiphtheriticum MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1324 Corynebacterium diphtheriae Corynebacterium diphtheriae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1319 Corynebacterium xerosis Corynebacterium xerosis MIC: 16 (ug/ml), Ref: 18849164
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC795
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.6 (ug/ml), Ref: 15844943
TCMC882
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 0.1809 (ug/ml), Ref: 9644053
TCMC882
TCMT1438 Plasmodium falciparum Plasmodium falciparum NF54 IC50: 0.2542 (ug/ml), Ref: 9644053
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC2414
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1.95 (ug/ml), Ref: 12713410
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC845
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 1522419
MIC: 6.25 (ug/ml), Ref: 1522419
TCMC845
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 1522419
MIC: 1.57 (ug/ml), Ref: 1522419
TCMC1113
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 15863332
TCMC2003
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1251 Candida albicans Candida albicans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1246 Escherichia coli Escherichia coli MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12036362
TCMC2003
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
TCMC2003
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 25 (ug/ml), Ref: 20022753
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2477
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 72.5 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1986
TCMT1442 Leishmania donovani Leishmania donovani IC50: 17.7 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2479
TCMT1251 Candida albicans Candida albicans MIC: 6.25 (ug/ml), Ref: 11170676
TCMC2479
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 11170676
TCMC2481
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 12.5 (ug/ml), Ref: 17027268
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1102
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 5.5 (ug/ml), Ref: 12502337
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2493
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20004575
MIC: 1.56 (ug/ml), Ref: 22280816
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1515
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC614
TCMT1454 Bacillus subtilis Bacillus subtilis IC50: 98.5 (ug/ml), Ref: 25981688
TCMC2519
TCMT1283 Human enterovirus 71 Human enterovirus 71 IC50: 10 (ug/ml), Ref: 22342145
TCMC2196
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 10 (ug/ml), Ref: 22819942
MIC: 0.5 (ug/ml), Ref: 26253635
TCMC2196
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 1 (ug/ml), Ref: 23360475
MIC: 1 (ug/ml), Ref: 26253635
TCMC2196
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 6 (ug/ml), Ref: 26253635
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC1117
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 100 (ug/ml), Ref: 10425115
TCMC1117
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.89 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC1572
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC2182
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 12.5 (ug/ml), Ref: 22280816
TCMC755
TCMT1251 Candida albicans Candida albicans IC50: 6 (ug/ml), Ref: 12502337
TCMC755
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC755
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 6.46 (ug/ml), Ref: 25564380
TCMC2591
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 6.25 (ug/ml), Ref: 8864235
TCMC2591
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 0.78 (ug/ml), Ref: 8864235
TCMC2591
TCMT1210 Streptococcus sobrinus Streptococcus sobrinus MIC: 1.56 (ug/ml), Ref: 8864235
TCMC2591
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 0.39 (ug/ml), Ref: 8864235
TCMC2591
TCMT1370 Prevotella melaninogenica Prevotella melaninogenica MIC: 0.78 (ug/ml), Ref: 8864235
TCMC1105
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 51.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 50.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1105
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 23534483
TCMC1105
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 1 (ug/ml), Ref: 23534483
TCMC1105
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 23534483
MIC: 4 (ug/ml), Ref: 23534483
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2040
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.03 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC348
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 62 (ug/ml), Ref: 25813159
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC1203
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 22.6 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 0.087 (ug/ml), Ref: 9249972
TCMC2660
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 6.25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2661
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 11 (ug/ml), Ref: 19904996
TCMC2014
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 10 (ug/ml), Ref: 17220400
TCMC1523
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 18611050
MIC: 25 (ug/ml), Ref: 21131198
MIC: 25 (ug/ml), Ref: 21401117
MIC: 16 (ug/ml), Ref: 22424614
MIC: 32 (ug/ml), Ref: 22424614
MBC: 32 (ug/ml), Ref: 22424614
TCMC1523
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 6.25 (ug/ml), Ref: 18611050
MIC: 12.5 (ug/ml), Ref: 21131198
TCMC1523
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 12.5 (ug/ml), Ref: 18611050
MIC: 12.5 (ug/ml), Ref: 21131198
MIC: 12.5 (ug/ml), Ref: 21401117
TCMC1523
TCMT1201 Staphylococcus epidermidis ATCC 12228 Staphylococcus epidermidis ATCC 12228 MIC: 12.5 (ug/ml), Ref: 21401117
TCMC1523
TCMT1286 Bacillus cereus Bacillus cereus MIC: 12.5 (ug/ml), Ref: 21401117
TCMC1523
TCMT1219 Enterococcus Enterococcus MIC: 32 (ug/ml), Ref: 22424614
MBC: 32 (ug/ml), Ref: 22424614
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1123
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1123
TCMT1442 Leishmania donovani Leishmania donovani IC50: 25 (ug/ml), Ref: 15679330
TCMC1892
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC1892
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2681
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 16 (ug/ml), Ref: 19904996
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC2699
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 6.3 (ug/ml), Ref: 14995101
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC1889
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2709
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 59.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1063
TCMT1251 Candida albicans Candida albicans MIC: 1.56 (ug/ml), Ref: 3373231
MIC: 3.12 (ug/ml), Ref: 3373231
MIC: 6.25 (ug/ml), Ref: 3373231
MIC: 2 (ug/ml), Ref: 15921418
TCMC1063
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 3373231
MIC: 1 (ug/ml), Ref: 15921418
TCMC1063
TCMT1243 Aspergillus flavus Aspergillus flavus MIC: 100 (ug/ml), Ref: 3373231
TCMC1063
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 32 (ug/ml), Ref: 15921418
TCMC1915
TCMT1347 Human rhinovirus 16 Human rhinovirus 16 IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1333 Human rhinovirus 1A Human rhinovirus 1A IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1241 Human rhinovirus 14 Human rhinovirus 14 IC50: 0.02 (ug/ml), Ref: 17116681
IC50: 100 (nM), Ref: 23977995
TCMC1801
TCMT1449 Influenza A virus Influenza A virus IC50: 1 (ug/ml), Ref: 14987066
IC50: 2.4 (nM), Ref: 19919060
IC50: 3.41 (nM), Ref: 15974612
IC50: 3.79 (nM), Ref: 16532013
IC50: 7.03 (nM), Ref: 19101157
IC50: 30 (nM), Ref: 25305333
IC50: 1.08 (nM), Ref: 9784165
IC50: 0.85 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 2.27 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 93.92 (nM), Ref: 20430633
IC50: 99.57 (nM), Ref: 20430633
IC50: 0.54 (nM), Ref: 20430633
IC50: 94.4 (nM), Ref: 20430633
IC50: 0.49 (nM), Ref: 20411974
IC50: 0.25 (nM), Ref: 20384296
IC50: 1 (nM), Ref: IC50: 95.43 (nM), Ref: 9461668
IC50: 78.12 (nM), Ref: 9461668
IC50: 75.29 (nM), Ref: 9461668
IC50: 1.84 (nM), Ref: 20166736
IC50: 1.59 (nM), Ref: 24673739
IC50: 0.34 (nM), Ref: 23675610
IC50: 0.25 (nM), Ref: 1431945
IC50: 3.64 (nM), Ref: 11170656
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC1915
TCMT1348 Human rhinovirus 2 Human rhinovirus 2 IC50: 0.01 (ug/ml), Ref: 23920485
IC50: 100 (nM), Ref: 23977995
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC2806
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.5 (ug/ml), Ref: 18524594
TCMC2808
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 27 (ug/ml), Ref: 10425115
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1113
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 16 (nM), Ref: 17263522
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC1117
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 17.56 (nM), Ref: 17263522
TCMC2282
TCMT1090 Human immunodeficiency virus type 1 integrase Human immunodeficiency virus 1 IC50: 70 (nM), Ref: 9986720
TCMC4
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 40 (nM), Ref: 16722653
TCMC1801
TCMT1162 Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1)) Ki: 1.1 (nM), Ref: IC50: 0.1 (nM), Ref: 23398362
IC50: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1164 Neuraminidase Influenza A virus (A/chicken/Yogjakarta/BBVet-IX/2004(H5N1)) Ki: 4.9 (nM), Ref: 20579892
IC50: 4.9 (nM), Ref: 19708637
IC50: 3.7 (nM), Ref:
TCMC1801
TCMT1161 Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1)) Ki: 7.9 (nM), Ref: 20579892
IC50: 10.8 (nM), Ref: 10.6019/CHEMBL1201861
TCMC1801
TCMT1163 Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1)) IC50: 0.3 (nM), Ref: 9322359
IC50: 0.2 (nM), Ref: Ki: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/swine/Belzig/2/2001(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/New Caledonia/20/1999(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Yamagata/32/1989(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC1801
TCMT1151 Neuraminidase Influenza B virus IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Hong Kong/1/1968(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1160 Neuraminidase Influenza A virus (A/Aichi/2/1968(H3N2)) IC50: 1.55 (nM), Ref: 20185316
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/whooper swan/Mongolia/1/2009(H5N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Wisconsin/67/2005(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Shandong/LY/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/Perth/16/2009(H3N2)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1151 Neuraminidase Influenza B virus (B/Memphis/3/89) IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Sandong/Li/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850
TCMC1179
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (nM), Ref: 19097788
TCMC1801
TCMT1296 Influenza A virus H3N2 Influenza A virus H3N2 IC50: 18.5 (nM), Ref: 12542349
TCMC1915
TCMT1285 Human coxsackievirus B3 Human coxsackievirus B3 IC50: 2.5 (nM), Ref: 13678412