TCM Putative Target References: TCMF662


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC879
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC417
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 7585.78 (nM), Ref: 23574272
IC50: 7500 (nM), Ref: 23574272
TCMC417
TCMT128 Tankyrase-2 Homo sapiens IC50: 870.96 (nM), Ref: 23574272
IC50: 870 (nM), Ref: 23574272
TCMC417
TCMT129 Tankyrase-1 Homo sapiens IC50: 645.65 (nM), Ref: 23574272
IC50: 630 (nM), Ref: 23574272
TCMC417
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2000 (nM), Ref: 24368208
TCMC1881
TCMT151 Protein kinase C alpha Homo sapiens Ki: 2.5 (nM), Ref: 11327599
Ki: 6.4 (nM), Ref: 21596562
TCMC1881
TCMT152 Protein kinase C beta Homo sapiens Ki: 1.8 (nM), Ref: 11327599
TCMC1881
TCMT153 Protein kinase C gamma Homo sapiens Ki: 4.9 (nM), Ref: 11327599
TCMC1881
TCMT154 Protein kinase C delta Homo sapiens Ki: 0.8 (nM), Ref: 11327599
TCMC1881
TCMT155 Protein kinase C epsilon Homo sapiens Ki: 0.45 (nM), Ref: 11327599
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC1445
TCMT238 Sodium/glucose cotransporter 2 Homo sapiens IC50: 1700 (nM), Ref: 17374486
TCMC1445
TCMT207 Beta-secretase 1 Homo sapiens Ki: 7200 (nM), Ref: 18565755
IC50: 3300 (nM), Ref: 18565755
TCMC981
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens Ki: 4200 (nM), Ref: 15908213
Ki: 1420 (nM), Ref: 16171993
Ki: 5890 (nM), Ref: 24901260
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1187
TCMT151 Protein kinase C alpha Homo sapiens IC50: 1900 (nM), Ref: 9834166
TCMC1447
TCMT207 Beta-secretase 1 Homo sapiens Ki: 3000 (nM), Ref: 18565755
IC50: 2600 (nM), Ref: 18565755
TCMC1372
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2330 (nM), Ref: 22245047
TCMC1372
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 3630 (nM), Ref: 22245047
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC824
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 5000 (nM), Ref: 24844534
TCMC1957
TCMT34 Cytochrome P450 2D6 Homo sapiens Ki: 78 (nM), Ref: 26125082
TCMC244
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 7900 (nM), Ref: 15916432
TCMC244
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 8300 (nM), Ref: 15658857
IC50: 8298.51 (nM), Ref: 19110342
TCMC2013
TCMT223 Aldose reductase Homo sapiens IC50: 2700 (nM), Ref: 22261024
TCMC218
TCMT307 HERG Homo sapiens IC50: 6025.6 (nM), Ref: 21185626
TCMC2001
TCMT116 Mu opioid receptor Homo sapiens Ki: 6.9 (nM), Ref: 19027293
Ki: 3.9 (nM), Ref: 20055417
TCMC2001
TCMT113 Delta opioid receptor Homo sapiens Ki: 180 (nM), Ref: 19027293
Ki: 49 (nM), Ref: 20055417
TCMC2001
TCMT117 Kappa opioid receptor Homo sapiens Ki: 3 (nM), Ref: 19027293
Ki: 2.2 (nM), Ref: 20055417
TCMC37
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC2198
TCMT311 Multidrug and toxin extrusion protein 1 Homo sapiens IC50: 9400 (nM), Ref: 23241029
TCMC704
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4000 (nM), Ref: 21030469
IC50: 3600 (nM), Ref: 21030469
TCMC88
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 3400 (nM), Ref: 11678652
TCMC2061
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 9550 (nM), Ref:
TCMC1433
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6863.3 (nM), Ref: 26498393
TCMC1433
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 62.2 (nM), Ref: 26498393
TCMC1433
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 26.6 (nM), Ref: 26498393
TCMC1433
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 399.7 (nM), Ref: 26498393
TCMC1803
TCMT337 Exportin-1 Homo sapiens IC50: 1600 (nM), Ref: 20493693
TCMC2052
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9110 (nM), Ref: 22892213
TCMC2052
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8720 (nM), Ref: 22892213
TCMC2052
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 8430 (nM), Ref: 22892213
TCMC2052
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5930 (nM), Ref: 22892213
TCMC2052
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 780 (nM), Ref: 22892213
TCMC1258
TCMT37 Serotonin 2a (5-HT2a) receptor Homo sapiens Ki: 966 (nM), Ref: 25695425
TCMC1258
TCMT160 Serotonin 7 (5-HT7) receptor Homo sapiens Ki: 43 (nM), Ref: 25695425
TCMC1258
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens Ki: 171 (nM), Ref: 25695425
TCMC505
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 4880 (nM), Ref: 15658857
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC1851
TCMT560 Coagulation factor X Homo sapiens IC50: 170 (nM), Ref: 9834152
Ki: 570 (nM), Ref: 9834152
TCMC1851
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3760 (nM), Ref: 24835197
Ki: 5130 (nM), Ref: 24835197
TCMC1851
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 2350 (nM), Ref: 26395057
Ki: 2600 (nM), Ref: 26395057
TCMC415
TCMT207 Beta-secretase 1 Homo sapiens IC50: 1800 (nM), Ref: 14592472
TCMC1464
TCMT207 Beta-secretase 1 Homo sapiens Ki: 3900 (nM), Ref: 18565755
IC50: 8400 (nM), Ref: 18565755
TCMC795
TCMT223 Aldose reductase Homo sapiens IC50: 8000 (nM), Ref: 24341381
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1773
TCMT575 Phospholipase A2 group IIA Homo sapiens IC50: 3500 (nM), Ref: 16504502
TCMC416
TCMT207 Beta-secretase 1 Homo sapiens IC50: 4500 (nM), Ref: 14592472
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC1339
TCMT117 Kappa opioid receptor Homo sapiens Ki: 260 (nM), Ref: 22439881
TCMC1339
TCMT116 Mu opioid receptor Homo sapiens Ki: 9.5 (nM), Ref: 22439881
TCMC1439
TCMT588 D-amino-acid oxidase Homo sapiens IC50: 2000 (nM), Ref: 23683589
TCMC1439
TCMT159 Tyrosinase Homo sapiens IC50: 9150 (nM), Ref: 26386819
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC2188
TCMT223 Aldose reductase Homo sapiens IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC1795
TCMT116 Mu opioid receptor Homo sapiens Ki: 286 (nM), Ref: 17616524
TCMC1411
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1261 (nM), Ref: 20696580
TCMC1411
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 56 (nM), Ref: 20696580
TCMC1411
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 17 (nM), Ref: 20696580
TCMC1411
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 212.9 (nM), Ref: 26498393
TCMC1411
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.4 (nM), Ref: 26498393
TCMC1411
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 54.9 (nM), Ref: 26498393
Ki: 220 (nM), Ref: 26498393
TCMC1411
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 440 (nM), Ref: 26498393
TCMC895
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 7630 (nM), Ref: 20053563
TCMC895
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 7630 (nM), Ref: 20053563
TCMC895
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 8990 (nM), Ref:
TCMC895
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 3012 (nM), Ref: IC50: 2197 (nM), Ref:
TCMC895
TCMT608 Solute carrier family 22 member 3 Homo sapiens IC50: 410 (nM), Ref: 23241029
TCMC895
TCMT213 Solute carrier family 22 member 1 Homo sapiens IC50: 210 (nM), Ref: 23241029
TCMC895
TCMT309 Solute carrier family 22 member 2 Homo sapiens IC50: 400 (nM), Ref: 23241029
TCMC895
TCMT310 Multidrug and toxin extrusion protein 2 Homo sapiens IC50: 500 (nM), Ref: 23241029
TCMC895
TCMT311 Multidrug and toxin extrusion protein 1 Homo sapiens IC50: 700 (nM), Ref: 23241029
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC1620
TCMT223 Aldose reductase Homo sapiens IC50: 88 (nM), Ref: 22236472
TCMC1620
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 130 (nM), Ref: 22236472
TCMC1424
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2100 (nM), Ref: 17994701
TCMC2054
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 9640 (nM), Ref: 18507367
TCMC2054
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 6610 (nM), Ref:
TCMC2054
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 600 (nM), Ref: 26602279
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC1041
TCMT636 DNA polymerase alpha subunit Homo sapiens Ki: 830 (nM), Ref: 1705574
TCMC1041
TCMT17 DNA polymerase beta Homo sapiens Ki: 390 (nM), Ref: 1705574
TCMC1413
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7370 (nM), Ref: 22892213
TCMC1413
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 5270 (nM), Ref: 22892213
TCMC1413
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4140 (nM), Ref: 22892213
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC1506
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 101.2 (nM), Ref: 26498393
TCMC1506
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 268.3 (nM), Ref: 26498393
TCMC1506
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.8 (nM), Ref: 26498393
TCMC845
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 630 (nM), Ref: 19231207
TCMC315
TCMT46 Coagulation factor III Homo sapiens IC50: 14.98 (nM), Ref: 23199480
TCMC130
TCMT615 Sentrin-specific protease 8 Homo sapiens IC50: 2470 (nM), Ref:
TCMC130
TCMT616 Sentrin-specific protease 7 Homo sapiens IC50: 1670 (nM), Ref:
TCMC130
TCMT617 Sentrin-specific protease 6 Homo sapiens IC50: 805 (nM), Ref:
TCMC262
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 8040 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 8040 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC262
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 3000 (nM), Ref: 24844534
TCMC837
TCMT690 Histone deacetylase 3 Homo sapiens IC50: 9000 (nM), Ref: 21874153
TCMC1844
TCMT113 Delta opioid receptor Homo sapiens Ki: 8400 (nM), Ref: 26035635
TCMC1844
TCMT510 Stem cell growth factor receptor Homo sapiens IC50: 600 (nM), Ref: 26807861
IC50: 1500 (nM), Ref: 26807861
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1113
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC2003
TCMT82 Estrogen receptor alpha Homo sapiens Ki: 785 (nM), Ref: 15634023
TCMC2003
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 2840 (nM), Ref: 16814546
IC50: 4120 (nM), Ref: 18063374
IC50: 625 (nM), Ref:
TCMC2003
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 996 (nM), Ref: 17604631
IC50: 750 (nM), Ref: 20527891
IC50: 996 (nM), Ref: 26850006
TCMC2003
TCMT329 Quinone reductase 2 Homo sapiens IC50: 960 (nM), Ref: 19265439
IC50: 450 (nM), Ref: 20036559
IC50: 450 (nM), Ref: 20356739
IC50: 960 (nM), Ref: 21261296
IC50: 6900 (nM), Ref: 23953689
Ki: 88 (nM), Ref: 23953689
IC50: 1400 (nM), Ref: 26854376
IC50: 913 (nM), Ref: 26854376
TCMC2003
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2210 (nM), Ref: 20674354
TCMC2003
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2770 (nM), Ref: 20674354
TCMC2003
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 9090 (nM), Ref: 20674354
TCMC2003
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4470 (nM), Ref: 20674354
TCMC2003
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4750 (nM), Ref: 20674354
TCMC2003
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4640 (nM), Ref: 20674354
TCMC2003
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8070 (nM), Ref: 20674354
TCMC2003
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4350 (nM), Ref: 20674354
TCMC2003
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 20674354
TCMC2003
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 950 (nM), Ref: 20674354
TCMC2003
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4090 (nM), Ref: 20674354
TCMC2003
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 830 (nM), Ref: 20674354
TCMC2003
TCMT729 PI3-kinase p110-alpha subunit Homo sapiens IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT730 PI3-kinase p110-beta subunit Homo sapiens IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4100 (nM), Ref: 27190601
IC50: 2600 (nM), Ref: 27190601
TCMC963
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 500 (nM), Ref: 15357993
Ki: 500 (nM), Ref: 15454240
Ki: 500 (nM), Ref: 15501038
Ki: 500 (nM), Ref: 21208801
Ki: 500 (nM), Ref: 26525863
Ki: 500 (nM), Ref: 26853167
Ki: 500 (nM), Ref: 27283786
TCMC963
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4000 (nM), Ref: 15501038
TCMC2070
TCMT327 Vanilloid receptor Homo sapiens IC50: 290 (nM), Ref: 22257892
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC1446
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 6300 (nM), Ref: 21641214
TCMC1334
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 4200 (nM), Ref: 19481465
TCMC1334
TCMT114 Cannabinoid CB2 receptor Homo sapiens Ki: 5610 (nM), Ref: 24900561
Ki: 5.61 (nM), Ref: 27078864
TCMC1334
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 6460 (nM), Ref: 24900561
Ki: 6.46 (nM), Ref: 27078864
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC143
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 1610 (nM), Ref:
TCMC706
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 9510 (nM), Ref: 19028102
TCMC1986
TCMT223 Aldose reductase Homo sapiens IC50: 150 (nM), Ref: 18165015
IC50: 2000 (nM), Ref: 22261024
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1102
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 7500 (nM), Ref: 16610779
TCMC1102
TCMT752 Casein kinase II alpha Homo sapiens IC50: 40 (nM), Ref: 19414254
TCMC1102
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2320 (nM), Ref: 20185318
TCMC1102
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2180 (nM), Ref: 20185318
TCMC1102
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC1102
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7590 (nM), Ref: 20185318
TCMC1102
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7060 (nM), Ref: 20185318
TCMC1102
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6320 (nM), Ref: 20185318
Ki: 8790 (nM), Ref: 22892213
TCMC1102
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9370 (nM), Ref: 20185318
TCMC1102
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8910 (nM), Ref: 20185318
TCMC1102
TCMT753 Mothers against decapentaplegic homolog 3 Homo sapiens IC50: 142 (nM), Ref:
TCMC1102
TCMT721 Heat shock 70 kDa protein 1 Homo sapiens IC50: 760 (nM), Ref:
TCMC1102
TCMT189 Dual specificity protein phosphatase 3 Homo sapiens IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref:
TCMC1102
TCMT223 Aldose reductase Homo sapiens IC50: 200 (nM), Ref: 22261024
TCMC1102
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 510 (nM), Ref: 22377675
TCMC1102
TCMT354 Serine/threonine-protein kinase Aurora-A Homo sapiens IC50: 2480 (nM), Ref: 22377675
TCMC1102
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 2500 (nM), Ref: 22377675
TCMC1102
TCMT626 Serine/threonine-protein kinase B-raf Homo sapiens IC50: 1760 (nM), Ref: 22377675
TCMC1102
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 690 (nM), Ref: 22377675
TCMC1102
TCMT418 Ephrin type-B receptor 4 Homo sapiens IC50: 1830 (nM), Ref: 22377675
TCMC1102
TCMT704 Receptor protein-tyrosine kinase erbB-2 Homo sapiens IC50: 3540 (nM), Ref: 22377675
TCMC1102
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 3110 (nM), Ref: 22377675
TCMC1102
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 250 (nM), Ref: 22377675
TCMC1102
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 800 (nM), Ref: 22377675
TCMC1102
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 790 (nM), Ref: 22377675
TCMC1102
TCMT457 Vascular endothelial growth factor receptor 3 Homo sapiens IC50: 1540 (nM), Ref: 22377675
TCMC1102
TCMT377 Insulin receptor Homo sapiens IC50: 340 (nM), Ref: 22377675
TCMC1102
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 22377675
TCMC1102
TCMT536 Platelet-derived growth factor receptor beta Homo sapiens IC50: 1300 (nM), Ref: 22377675
TCMC1102
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 3340 (nM), Ref: 22377675
TCMC1102
TCMT755 Serine/threonine-protein kinase PLK4 Homo sapiens IC50: 2970 (nM), Ref: 22377675
TCMC1102
TCMT502 Tyrosine-protein kinase TIE-2 Homo sapiens IC50: 260 (nM), Ref: 22377675
TCMC1102
TCMT756 Mitogen-activated protein kinase kinase kinase 8 Homo sapiens IC50: 2370 (nM), Ref: 22377675
TCMC1102
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 100 (nM), Ref: 24900447
TCMC1102
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8150 (nM), Ref: 22892213
TCMC1102
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4240 (nM), Ref: 22892213
TCMC1102
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3900 (nM), Ref: 24835197
TCMC1248
TCMT759 SUMO-activating enzyme subunit 1 Homo sapiens IC50: 3000 (nM), Ref: 23360215
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC1964
TCMT726 Bcr/Abl fusion protein Homo sapiens IC50: 10000 (nM), Ref: 16686543
TCMC1964
TCMT329 Quinone reductase 2 Homo sapiens IC50: 5100 (nM), Ref: 23953689
TCMC1964
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1400 (nM), Ref: 10.1039/C3MD00317E
Ki: 900 (nM), Ref: 10.1039/C0MD00242A
TCMC1964
TCMT215 Cytochrome P450 1A1 Homo sapiens Ki: 570 (nM), Ref: 10.1039/C0MD00242A
TCMC2155
TCMT116 Mu opioid receptor Homo sapiens Ki: 7400 (nM), Ref: 17616524
TCMC910
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1118 (nM), Ref: 20696580
TCMC910
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 95 (nM), Ref: 20696580
TCMC910
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 20 (nM), Ref: 20696580
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1158
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3100 (nM), Ref: 24835197
Ki: 6840 (nM), Ref: 24835197
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC2053
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 22 (nM), Ref: 23332346
TCMC2053
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 214 (nM), Ref: 23332346
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1837
TCMT789 Phosphodiesterase 3A Homo sapiens Ki: 279 (nM), Ref: 17228859
TCMC1837
TCMT790 Phosphodiesterase 3B Homo sapiens Ki: 417 (nM), Ref: 17228859
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1837
TCMT792 Phosphodiesterase 10A Homo sapiens IC50: 56.9 (nM), Ref: 20450197
IC50: 76 (nM), Ref: 20450197
IC50: 17 (nM), Ref: 21087867
IC50: 21 (nM), Ref: 21705115
IC50: 36 (nM), Ref: 22321214
IC50: 210 (nM), Ref: 23978358
IC50: 36 (nM), Ref: 24721831
IC50: 36 (nM), Ref: 25592707
IC50: 92.3 (nM), Ref: 10.1039/C5MD00419E
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1837
TCMT307 HERG Homo sapiens IC50: 7244.36 (nM), Ref: 21185626
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC614
TCMT151 Protein kinase C alpha Homo sapiens IC50: 9300 (nM), Ref: 9834166
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC1724
TCMT113 Delta opioid receptor Homo sapiens Ki: 41 (nM), Ref: 10741545
Ki: 33 (nM), Ref: 14643346
Ki: 33 (nM), Ref: 17149859
Ki: 33 (nM), Ref: 17149858
Ki: 76 (nM), Ref: 17407276
IC50: 138 (nM), Ref: 17388627
IC50: 138 (nM), Ref: 17451272
IC50: 138 (nM), Ref: 18039010
Ki: 33 (nM), Ref: 18313920
Ki: 120 (nM), Ref: 19027293
IC50: 138 (nM), Ref: 16989522
Ki: 51 (nM), Ref: 20055417
Ki: 38 (nM), Ref: 21482470
Ki: 21.38 (nM), Ref: 19527931
Ki: 103 (nM), Ref: 25062506
Ki: 1516 (nM), Ref: 25268943
Ki: 30 (nM), Ref: 26035635
Ki: 103 (nM), Ref: 10.1039/C5MD00414D
TCMC1724
TCMT117 Kappa opioid receptor Homo sapiens Ki: 1.2 (nM), Ref: 10741545
Ki: 9.2 (nM), Ref: 17149859
Ki: 9.2 (nM), Ref: 17149858
Ki: 1.1 (nM), Ref: 17407276
IC50: 320 (nM), Ref: 17407276
Ki: 9.2 (nM), Ref: 18313920
Ki: 1.2 (nM), Ref: 19027293
Ki: 3 (nM), Ref: 20055417
Ki: 14.7 (nM), Ref: 20441176
Ki: 0.25 (nM), Ref: 21482470
Ki: 4.467 (nM), Ref: 19527931
Ki: 362 (nM), Ref: 25268943
Ki: 15 (nM), Ref: 10.1039/C5MD00414D
TCMC1724
TCMT116 Mu opioid receptor Homo sapiens IC50: 7.3 (nM), Ref: 14643346
Ki: 3.7 (nM), Ref: 17149859
IC50: 7.3 (nM), Ref: 17149859
Ki: 3.7 (nM), Ref: 17149858
IC50: 7.3 (nM), Ref: 17149858
Ki: 0.79 (nM), Ref: 17407276
IC50: 23 (nM), Ref: 17407276
Ki: 3.7 (nM), Ref: 18313920
IC50: 7.3 (nM), Ref: 18313920
Ki: 0.66 (nM), Ref: 19027293
Ki: 0.98 (nM), Ref: 20055417
Ki: 0.23 (nM), Ref: 21482470
Ki: 0.5623 (nM), Ref: 19527931
IC50: 1.87 (nM), Ref: 24171469
Ki: 2.3 (nM), Ref: 25062506
Ki: 354 (nM), Ref: 25268943
Ki: 1.148 (nM), Ref: 26632862
Ki: 1.259 (nM), Ref: 26632862
Ki: 2.3 (nM), Ref: 10.1039/C5MD00414D
TCMC1724
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.6 (nM), Ref: 16250647
TCMC1281
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 10 (nM), Ref: 19564108
IC50: 18.6 (nM), Ref: 22148241
IC50: 6 (nM), Ref: 22360639
TCMC1281
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 1 (nM), Ref: 19564108
IC50: 0.7 (nM), Ref: 22148241
IC50: 0.4 (nM), Ref: 22360639
TCMC1763
TCMT309 Solute carrier family 22 member 2 Homo sapiens IC50: 2600 (nM), Ref: 23241029
TCMC880
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9910 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 20185318
Ki: 9900 (nM), Ref: 22245047
Ki: 9900 (nM), Ref: 26073005
Ki: 9900 (nM), Ref: 26520662
TCMC880
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4200 (nM), Ref: 18579385
Ki: 4200 (nM), Ref: 20185318
TCMC880
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 18579385
Ki: 8900 (nM), Ref: 20185318
TCMC469
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 100 (nM), Ref: 22921742
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC264
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 105 (nM), Ref: 23332346
TCMC264
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 6.6 (nM), Ref: 23332346
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2150
TCMT46 Coagulation factor III Homo sapiens IC50: 22.78 (nM), Ref: 23199480
TCMC2150
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 231 (nM), Ref: 23332346
TCMC1886
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 670 (nM), Ref: 26498394
TCMC1886
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 770 (nM), Ref: 26498394
TCMC1886
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 620 (nM), Ref: 26498394
TCMC1886
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8470 (nM), Ref: 26498394
TCMC1886
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 720 (nM), Ref: 26498394
TCMC1768
TCMT131 Acetylcholinesterase Homo sapiens IC50: 7200 (nM), Ref: 22445674
Ki: 8400 (nM), Ref: 22445674
TCMC930
TCMT116 Mu opioid receptor Homo sapiens Ki: 459 (nM), Ref: 17616524
TCMC858
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 66 (nM), Ref: 23332346
TCMC858
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 119 (nM), Ref: 23332346
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1432
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8790.2 (nM), Ref: 26498393
TCMC1432
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 344.2 (nM), Ref: 26498393
TCMC1432
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1432
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 408.9 (nM), Ref: 26498393
TCMC2063
TCMT646 Serotonin 5a (5-HT5a) receptor Homo sapiens Ki: 126 (nM), Ref: 12825922
IC50: 180 (nM), Ref: 18983139
Ki: 110 (nM), Ref: 18983139
IC50: 184 (nM), Ref: 18588282
Ki: 170 (nM), Ref: 21726069
IC50: 280 (nM), Ref: 23582449
Ki: 82 (nM), Ref: 23466604
IC50: 160 (nM), Ref: 23466604
IC50: 180 (nM), Ref: 26988801
TCMC2063
TCMT315 Serotonin 6 (5-HT6) receptor Homo sapiens Ki: 65 (nM), Ref: 12825922
Ki: 100 (nM), Ref: 15357994
IC50: 200 (nM), Ref: 18983139
Ki: 93 (nM), Ref: 18983139
IC50: 262 (nM), Ref: 18588282
IC50: 27.5 (nM), Ref: 20170099
Ki: 84 (nM), Ref: 21726069
Ki: 70 (nM), Ref: 10.1007/s00044-004-0121-8
IC50: 180 (nM), Ref: 23582449
Ki: 50 (nM), Ref: 23466604
IC50: 100 (nM), Ref: 23466604
Ki: 33 (nM), Ref: 24805037
Ki: 33 (nM), Ref: 25557493
IC50: 120 (nM), Ref: 26988801
Ki: 100 (nM), Ref: 26996373
TCMC2063
TCMT160 Serotonin 7 (5-HT7) receptor Homo sapiens Ki: 8.1 (nM), Ref: 12825922
IC50: 0.61 (nM), Ref: 18983139
Ki: 0.22 (nM), Ref: 18983139
IC50: 2.55 (nM), Ref: 12713409
IC50: 1.5 (nM), Ref: 18588282
Ki: 0.13 (nM), Ref: 21726069
IC50: 0.49 (nM), Ref: 23582449
Ki: 0.11 (nM), Ref: 23466604
IC50: 0.29 (nM), Ref: 23466604
Ki: 1.4 (nM), Ref: 24763360
Ki: 0.8 (nM), Ref: 24805037
Ki: 0.8 (nM), Ref: 25557493
IC50: 0.25 (nM), Ref: 26988801
TCMC2063
TCMT37 Serotonin 2a (5-HT2a) receptor Homo sapiens Ki: 14 (nM), Ref: 15081042
Ki: 8.2 (nM), Ref: 16392816
Ki: 14 (nM), Ref: 16257207
Ki: 120 (nM), Ref: 18468904
Ki: 160 (nM), Ref: 18468904
Ki: 130 (nM), Ref: 18468904
Ki: 150 (nM), Ref: 18468904
Ki: 320 (nM), Ref: 11975483
Ki: 690 (nM), Ref: 17067154
Ki: 323.59 (nM), Ref: 23301527
Ki: 320 (nM), Ref: 23301527
TCMC2063
TCMT313 Serotonin 2b (5-HT2b) receptor Homo sapiens Ki: 12 (nM), Ref: 15081042
Ki: 13 (nM), Ref: 12954071
Ki: 13 (nM), Ref: 16392816
Ki: 12 (nM), Ref: 16257207
Ki: 13.49 (nM), Ref: 24582985
TCMC2063
TCMT314 Serotonin 2c (5-HT2c) receptor Homo sapiens Ki: 6.9 (nM), Ref: 15081042
Ki: 8.3 (nM), Ref: 12954071
Ki: 8.3 (nM), Ref: 16392816
Ki: 6.9 (nM), Ref: 16257207
Ki: 130 (nM), Ref: 11975483
Ki: 20 (nM), Ref: 17067154
Ki: 79.43 (nM), Ref: 23301527
Ki: 79 (nM), Ref: 23301527
TCMC2063
TCMT815 Serotonin 1d (5-HT1d) receptor Homo sapiens Ki: 5.5 (nM), Ref: 8071931
Ki: 0.5 (nM), Ref: 18507369
TCMC2063
TCMT36 Serotonin 1a (5-HT1a) receptor Homo sapiens Ki: 2.5 (nM), Ref: 7658447
IC50: 1.2 (nM), Ref: 12954071
Ki: 1.259 (nM), Ref: 18433113
Ki: 10000 (nM), Ref: 18433113
Ki: 0.62 (nM), Ref: 22748706
Ki: 0.9 (nM), Ref: 23332346
Ki: 9.5 (nM), Ref: 24161678
Ki: 2.08 (nM), Ref: 25128671
TCMC2063
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 79 (nM), Ref: 16250647
TCMC2063
TCMT816 Serotonin 1b (5-HT1b) receptor Homo sapiens Ki: 1.1 (nM), Ref: 18507369
IC50: 29 (nM), Ref: 18983139
Ki: 18 (nM), Ref: 18983139
Ki: 14 (nM), Ref: 21726069
IC50: 12 (nM), Ref: 23582449
Ki: 4 (nM), Ref: 23466604
IC50: 6.5 (nM), Ref: 23466604
TCMC2063
TCMT817 Serotonin 4 (5-HT4) receptor Homo sapiens Ki: 1049 (nM), Ref: 19334715
Ki: 500 (nM), Ref: 17067154
Ki: 29.51 (nM), Ref: 19223092
Ki: 109.65 (nM), Ref: 19223092
TCMC2063
TCMT645 Serotonin 1e (5-HT1e) receptor Homo sapiens Ki: 10.72 (nM), Ref: 24365159
Ki: 11 (nM), Ref: 24365159
TCMC2094
TCMT238 Sodium/glucose cotransporter 2 Homo sapiens IC50: 4100 (nM), Ref: 17374486
TCMC2094
TCMT207 Beta-secretase 1 Homo sapiens Ki: 1100 (nM), Ref: 18565755
IC50: 5200 (nM), Ref: 18565755
TCMC846
TCMT207 Beta-secretase 1 Homo sapiens Ki: 6200 (nM), Ref: 22222157
TCMC418
TCMT223 Aldose reductase Homo sapiens IC50: 78 (nM), Ref: 22236472
TCMC418
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 240 (nM), Ref: 22236472
TCMC418
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4700 (nM), Ref: 22921742
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1143
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 860 (nM), Ref: 22668600
TCMC1143
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 830 (nM), Ref: 22668600
TCMC1143
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 780 (nM), Ref: 22668600
TCMC1143
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 750 (nM), Ref: 22668600
TCMC1143
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 610 (nM), Ref: 22668600
TCMC1143
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 650 (nM), Ref: 22668600
TCMC1869
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 4410 (nM), Ref: 15658857
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC1600
TCMT116 Mu opioid receptor Homo sapiens Ki: 3.96 (nM), Ref: 12372519
Ki: 0.88 (nM), Ref: 16392810
Ki: 1.1 (nM), Ref: 16913723
Ki: 1.1 (nM), Ref: 17887741
Ki: 4 (nM), Ref: 17616524
Ki: 2.55 (nM), Ref: 19627147
Ki: 2.55 (nM), Ref: 21684752
Ki: 2.6 (nM), Ref: 21570305
Ki: 2.6 (nM), Ref: 22341895
Ki: 2.2 (nM), Ref: 24900459
Ki: 0.88 (nM), Ref: 22439881
IC50: 4.3 (nM), Ref: 22995061
Ki: 2.6 (nM), Ref: 23618710
Ki: 2.6 (nM), Ref: 23880358
IC50: 2.5 (nM), Ref: 24171469
Ki: 5.2 (nM), Ref: 25062506
Ki: 2.6 (nM), Ref: 25599950
Ki: 22 (nM), Ref: 25494650
IC50: 6.3 (nM), Ref: 26789491
Ki: 0.53 (nM), Ref: 26390077
Ki: 5.2 (nM), Ref: 10.1039/C5MD00414D
TCMC1600
TCMT113 Delta opioid receptor Homo sapiens Ki: 140 (nM), Ref: 16392810
Ki: 140 (nM), Ref: 16913723
Ki: 140 (nM), Ref: 17887741
Ki: 605 (nM), Ref: 22341895
Ki: 140 (nM), Ref: 22439881
Ki: 605 (nM), Ref: 23618710
Ki: 605 (nM), Ref: 23880358
Ki: 605 (nM), Ref: 25599950
TCMC1600
TCMT117 Kappa opioid receptor Homo sapiens Ki: 24 (nM), Ref: 16392810
Ki: 46.9 (nM), Ref: 16913723
Ki: 46.9 (nM), Ref: 17887741
Ki: 6.9 (nM), Ref: 19932964
Ki: 299 (nM), Ref: 22341895
Ki: 24 (nM), Ref: 22439881
Ki: 60.9 (nM), Ref: 23419026
Ki: 299 (nM), Ref: 23618710
Ki: 299 (nM), Ref: 23880358
Ki: 299 (nM), Ref: 25599950
Ki: 120 (nM), Ref: 26390077
TCMC435
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 1100 (nM), Ref: 24844534
TCMC84
TCMT207 Beta-secretase 1 Homo sapiens IC50: 6700 (nM), Ref: 18565755
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC755
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens Ki: 600 (nM), Ref: 21739938
TCMC755
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens Ki: 1600 (nM), Ref: 21739938
TCMC755
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4400 (nM), Ref: 21030469
IC50: 7000 (nM), Ref: 21030469
TCMC755
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 8700 (nM), Ref:
TCMC1329
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2710 (nM), Ref: 26275107
TCMC412
TCMT683 Macrophage migration inhibitory factor Homo sapiens Ki: 38 (nM), Ref: 19090668
IC50: 38 (nM), Ref: 27156768
TCMC1723
TCMT117 Kappa opioid receptor Homo sapiens Ki: 0.38 (nM), Ref: 19027293
Ki: 2 (nM), Ref: 26390077
TCMC1723
TCMT113 Delta opioid receptor Homo sapiens Ki: 120 (nM), Ref: 19027293
TCMC1723
TCMT116 Mu opioid receptor Homo sapiens Ki: 0.19 (nM), Ref: 19027293
Ki: 0.36 (nM), Ref: 26390077
TCMC726
TCMT167 Aldo-keto-reductase family 1 member C3 Homo sapiens IC50: 1000 (nM), Ref: 22506594
Ki: 680 (nM), Ref: 22506594
Ki: 680 (nM), Ref: 22506594
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC1168
TCMT117 Kappa opioid receptor Homo sapiens Ki: 2515 (nM), Ref: 18166466
TCMC2239
TCMT226 3-phosphoinositide dependent protein kinase-1 Homo sapiens IC50: 6600 (nM), Ref: 22537682
TCMC2239
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2100 (nM), Ref: 26918635
IC50: 2900 (nM), Ref: 26918635
TCMC38
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 529 (nM), Ref: 23332346
TCMC1118
TCMT304 Matrix metalloproteinase 14 Homo sapiens IC50: 6800 (nM), Ref: 19524436
TCMC1118
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 9600 (nM), Ref: 19524436
TCMC1118
TCMT207 Beta-secretase 1 Homo sapiens IC50: 757 (nM), Ref: 22225636
TCMC1118
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 1000 (nM), Ref: 22413845
IC50: 1080 (nM), Ref: 22413845
IC50: 1180 (nM), Ref: 22413845
IC50: 1000 (nM), Ref: 10.1039/C0MD00241K
TCMC1118
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 335 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1118
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1800 (nM), Ref: 23484434
TCMC1118
TCMT751 Dual-specificity tyrosine-phosphorylation regulated kinase 1A Homo sapiens IC50: 330 (nM), Ref: 24188002
TCMC1118
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4600 (nM), Ref: 24878198
IC50: 3000 (nM), Ref: 24878198
IC50: 500 (nM), Ref: 25978520
TCMC1118
TCMT567 DNA (cytosine-5)-methyltransferase 1 Homo sapiens IC50: 500 (nM), Ref: 25406944
TCMC1118
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 124.1 (nM), Ref: 25985195
IC50: 122.6 (nM), Ref: 25985195
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1105
TCMT752 Casein kinase II alpha Homo sapiens IC50: 2000 (nM), Ref: 19414254
TCMC1105
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2500 (nM), Ref: 27173800
TCMC2139
TCMT560 Coagulation factor X Homo sapiens IC50: 210 (nM), Ref: 9834152
Ki: 440 (nM), Ref: 9834152
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC937
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 11.5 (nM), Ref: 23332369
IC50: 6.6 (nM), Ref: 23895532
TCMC937
TCMT801 Tubulin beta-3 chain Homo sapiens IC50: 5.2 (nM), Ref: 23332369
IC50: 5.7 (nM), Ref: 23895532
TCMC732
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 5900 (nM), Ref: 21561086
TCMC1203
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 8000 (nM), Ref: 10.1039/C4MD00086B
TCMC804
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 2000 (nM), Ref: 21561086
TCMC1845
TCMT560 Coagulation factor X Homo sapiens IC50: 560 (nM), Ref: 9834152
Ki: 990 (nM), Ref: 9834152
TCMC1204
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2500 (nM), Ref: 14592472
TCMC28
TCMT853 Sigma opioid receptor Homo sapiens Ki: 36 (nM), Ref: 24617836
IC50: 8.24 (nM), Ref: 26717207
IC50: 7.59 (nM), Ref: 26717207
TCMC1078
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC313
TCMT46 Coagulation factor III Homo sapiens IC50: 187.26 (nM), Ref: 23199480
TCMC2151
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 443 (nM), Ref: 23332346
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC392
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 2400 (nM), Ref: 15658857
IC50: 2398.83 (nM), Ref: 19110342
TCMC1977
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7410 (nM), Ref: 21669522
TCMC1977
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 540 (nM), Ref: 21669522
TCMC1977
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 520 (nM), Ref: 21669522
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC17
TCMT241 Neuronal acetylcholine receptor protein alpha-7 subunit Homo sapiens Ki: 7943.28 (nM), Ref: 22243960
TCMC2228
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 6830 (nM), Ref: 21282059
TCMC2228
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6180 (nM), Ref: 21282059
TCMC2228
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8250 (nM), Ref: 21282059
TCMC2228
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 6700 (nM), Ref: 21282059
TCMC2228
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 6480 (nM), Ref: 22687439
TCMC2228
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 740 (nM), Ref: 22668600
TCMC2228
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7150 (nM), Ref: 22668600
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC192
TCMT176 Acyl coenzyme A:cholesterol acyltransferase 1 Homo sapiens IC50: 600 (nM), Ref: 17157006
TCMC192
TCMT263 Acyl coenzyme A:cholesterol acyltransferase 2 Homo sapiens IC50: 800 (nM), Ref: 17157006
TCMC1523
TCMT114 Cannabinoid CB2 receptor Homo sapiens Ki: 1440 (nM), Ref: 24900561
TCMC1523
TCMT115 Cannabinoid CB1 receptor Homo sapiens Ki: 3150 (nM), Ref: 24900561
TCMC4
TCMT207 Beta-secretase 1 Homo sapiens IC50: 6000 (nM), Ref: 14592472
TCMC341
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 19231207
TCMC1551
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 1900 (nM), Ref: 16248836
Ki: 1900 (nM), Ref: 16248836
Ki: 800 (nM), Ref: 16248836
Ki: 250 (nM), Ref: 22696418
TCMC1551
TCMT131 Acetylcholinesterase Homo sapiens IC50: 760 (nM), Ref: 23746477
TCMC1551
TCMT268 Cytochrome P450 2A13 Homo sapiens Ki: 40 (nM), Ref: 22696418
TCMC1798
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1480 (nM), Ref: 23411073
TCMC811
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 2030 (nM), Ref: 19097799
TCMC811
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 9900 (nM), Ref: 18533708
TCMC811
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10.2 (nM), Ref: 20413308
TCMC811
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7078.5 (nM), Ref: 26498393
TCMC811
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 371.5 (nM), Ref: 26498393
TCMC811
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.5 (nM), Ref: 26498393
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC1123
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1284 (nM), Ref: 20696580
TCMC1123
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 72.8 (nM), Ref: 26498393
TCMC1123
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1123
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 31.1 (nM), Ref: 26498393
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC785
TCMT131 Acetylcholinesterase Homo sapiens IC50: 610 (nM), Ref: 23062825
TCMC2004
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 800 (nM), Ref: 10.1039/C3MD00317E
Ki: 2100 (nM), Ref: 10.1039/C0MD00242A
TCMC2004
TCMT215 Cytochrome P450 1A1 Homo sapiens Ki: 160 (nM), Ref: 10.1039/C0MD00242A
TCMC1892
TCMT508 Tyrosine-protein kinase SYK Homo sapiens IC50: 10000 (nM), Ref: 23917087
TCMC2201
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8700 (nM), Ref: 21332115
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1003
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 15 (nM), Ref: 20413308
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC1148
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 800 (nM), Ref: 22668600
TCMC1148
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 490 (nM), Ref: 22668600
TCMC1148
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 610 (nM), Ref: 22668600
TCMC1148
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 850 (nM), Ref: 22668600
TCMC1148
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 710 (nM), Ref: 22668600
TCMC1148
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 320 (nM), Ref: 22668600
TCMC1657
TCMT116 Mu opioid receptor Homo sapiens Ki: 1.585 (nM), Ref: 26632862
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1828
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 900 (nM), Ref: 17994701
TCMC1940
TCMT187 Androgen Receptor Homo sapiens Ki: 8.5 (nM), Ref: 12954062
IC50: 37 (nM), Ref: 12954062
IC50: 37 (nM), Ref: 12781197
IC50: 37 (nM), Ref: 8627601
Ki: 8.5 (nM), Ref: 8627601
Ki: 8.5 (nM), Ref: 9873735
IC50: 37 (nM), Ref: 9784110
Ki: 35 (nM), Ref: 20510622
TCMC1940
TCMT613 Glucocorticoid receptor Homo sapiens Ki: 30.5 (nM), Ref: 12954062
Ki: 30.5 (nM), Ref: 9873735
Ki: 30.5 (nM), Ref: 9784110
TCMC1940
TCMT783 Mineralocorticoid receptor Homo sapiens IC50: 14 (nM), Ref: 12954062
IC50: 14 (nM), Ref: 12781197
IC50: 14 (nM), Ref: 9784110
IC50: 30 (nM), Ref: 8709117
TCMC1940
TCMT904 Progesterone receptor Homo sapiens Ki: 3.5 (nM), Ref: 10212133
IC50: 3.5 (nM), Ref: 11859003
Ki: 3.5 (nM), Ref: 9464361
IC50: 5 (nM), Ref: 8523399
Ki: 3.8 (nM), Ref: 9667968
Ki: 3.467 (nM), Ref: 16821785
Ki: 3.4 (nM), Ref: 18553958
Ki: 5.1 (nM), Ref: 20510622
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC1175
TCMT186 Monoamine oxidase B Homo sapiens IC50: 2870 (nM), Ref: 20045650
TCMC1175
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC1236
TCMT236 Estrogen receptor beta Homo sapiens IC50: 10 (nM), Ref: 15341953
IC50: 10 (nM), Ref: 15456246
IC50: 98.7 (nM), Ref: 15887952
IC50: 98.7 (nM), Ref: 15887952
IC50: 9.7 (nM), Ref: 15943471
IC50: 10 (nM), Ref: 16098741
IC50: 1.3 (nM), Ref: 16219463
IC50: 61 (nM), Ref: 16610787
IC50: 25 (nM), Ref: 17149865
IC50: 395 (nM), Ref: 17049855
IC50: 9.7 (nM), Ref: 17188490
IC50: 6.8 (nM), Ref: 17574424
IC50: 18 (nM), Ref: 12502307
IC50: 98.7 (nM), Ref:
TCMC1236
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 395 (nM), Ref: 15341953
IC50: 395 (nM), Ref: 15456246
IC50: 4660 (nM), Ref: 15887952
IC50: 4660 (nM), Ref: 15887952
IC50: 395 (nM), Ref: 15943471
IC50: 395 (nM), Ref: 16098741
IC50: 29.4 (nM), Ref: 16219463
IC50: 1973 (nM), Ref: 16610787
IC50: 1145 (nM), Ref: 17149865
IC50: 2150 (nM), Ref: 17696335
IC50: 9.7 (nM), Ref: 17049855
IC50: 395 (nM), Ref: 17188490
IC50: 580 (nM), Ref: 17574424
IC50: 300 (nM), Ref: 12502307
IC50: 4680 (nM), Ref:
TCMC1236
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 10 (nM), Ref: 17482813
TCMC1236
TCMT910 Estrogen-related receptor beta Homo sapiens IC50: 395 (nM), Ref: 17482813
TCMC1236
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 2210 (nM), Ref: 18533708
TCMC1236
TCMT344 Aldehyde oxidase Homo sapiens IC50: 340 (nM), Ref: 20853847
TCMC1236
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 7720 (nM), Ref:
TCMC273
TCMT332 Amine oxidase, copper containing Homo sapiens IC50: 4100 (nM), Ref: 23664164
TCMC547
TCMT313 Serotonin 2b (5-HT2b) receptor Homo sapiens IC50: 8912.51 (nM), Ref: 24582985
Ki: 2454.71 (nM), Ref: 24582985
TCMC547
TCMT644 Serotonin 3a (5-HT3a) receptor Homo sapiens Ki: 2511.89 (nM), Ref: 24582985
TCMC234
TCMT615 Sentrin-specific protease 8 Homo sapiens IC50: 5470 (nM), Ref:
TCMC234
TCMT616 Sentrin-specific protease 7 Homo sapiens IC50: 4630 (nM), Ref:
TCMC234
TCMT617 Sentrin-specific protease 6 Homo sapiens IC50: 1860 (nM), Ref:
TCMC2146
TCMT46 Coagulation factor III Homo sapiens IC50: 8.35 (nM), Ref: 23199480
TCMC90
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2400 (nM), Ref: 14592472
TCMC929
TCMT116 Mu opioid receptor Homo sapiens Ki: 6300 (nM), Ref: 17616524
TCMC1521
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3880 (nM), Ref: 22658537
TCMC1521
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 1200 (nM), Ref: 22658537
TCMC1521
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 7620 (nM), Ref: 22658537
TCMC2055
TCMT747 ATP-binding cassette sub-family G member 2 Homo sapiens IC50: 10000 (nM), Ref: 22822035
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC1961
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 600 (nM), Ref: 16248836
TCMC1961
TCMT131 Acetylcholinesterase Homo sapiens IC50: 6480 (nM), Ref: 23746477
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC1064
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 2437 (nM), Ref: 20696580
TCMC1064
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 140 (nM), Ref: 20696580
TCMC1064
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 29 (nM), Ref: 20696580
TCMC784
TCMT131 Acetylcholinesterase Homo sapiens IC50: 100 (nM), Ref: 26003344
TCMC784
TCMT132 Butyrylcholinesterase Homo sapiens IC50: 1090 (nM), Ref: 26003344
TCMC265
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 91 (nM), Ref: 23332346
TCMC265
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 4.5 (nM), Ref: 23332346
TCMC702
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 5150 (nM), Ref: 15658857
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755
TCMC1378
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 8960 (nM), Ref: 22658537
TCMC1378
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 8220 (nM), Ref: 22658537
TCMC1343
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 90 (nM), Ref: 18501600
Ki: 90 (nM), Ref: 18579385
TCMC1343
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7800 (nM), Ref: 18579385
TCMC1343
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8200 (nM), Ref: 18579385
TCMC1857
TCMT853 Sigma opioid receptor Homo sapiens Ki: 36 (nM), Ref: 27156565

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC2252
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 19.4 (ug/ml), Ref: 16643034
TCMC1803
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 2 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1851
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28 (ug/ml), Ref: 9461665
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1620
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 0.66 (ug/ml), Ref: 11430019
IC50: 5.9 (ug/ml), Ref: 16643034
TCMC2054
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 14.48 (ug/ml), Ref: 20116898
TCMC2177
TCMT1120 Cell division protein ftsZ Staphylococcus aureus MIC: 4 (ug/ml), Ref: 25791674
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2259
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 47.4 (ug/ml), Ref: 16643034
TCMC2265
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 23.6 (ug/ml), Ref: 16643034
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC1986
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 75.2 (ug/ml), Ref: 9461665
TCMC2271
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 43.5 (ug/ml), Ref: 16643034
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC1425
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 71 (ug/ml), Ref: 1710653
IC50: 71 (ug/ml), Ref: 21295891
TCMC2275
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 44.5 (ug/ml), Ref: 16643034
TCMC469
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 5.4 (ug/ml), Ref: 16643034
TCMC1866
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC2063
TCMT1086 Isocitrate lyase Candida albicans IC50: 53 (ug/ml), Ref: 21035332
TCMC1329
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.9 (ug/ml), Ref: 20116898
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1118
TCMT1092 Fatty acid synthase Plasmodium falciparum IC50: 0.03 (ug/ml), Ref: 20855214
IC50: 30 (nM), Ref: 24063369
TCMC1118
TCMT1094 3-oxoacyl-acyl-carrier protein reductase Plasmodium falciparum IC50: 0.32 (ug/ml), Ref: 20855214
TCMC1203
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.5 (ug/ml), Ref: 9461665
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC785
TCMT1104 Sortase Staphylococcus aureus IC50: 8.7 (ug/ml), Ref: 17716892
IC50: 8.7 (ug/ml), Ref: 19269184
TCMC785
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 100 (ug/ml), Ref: 1710653
IC50: 100 (ug/ml), Ref: 21295891
TCMC785
TCMT1154 Sortase Staphylococcus aureus IC50: 40.6 (ug/ml), Ref: 26551342
TCMC2292
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.15 (ug/ml), Ref: 20116898
TCMC1491
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 0.00423 (ug/ml), Ref: 21334901
IC50: 0.00211 (ug/ml), Ref: 21334901
TCMC1236
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.84 (ug/ml), Ref: 20116898
TCMC2299
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 20.1 (ug/ml), Ref: 16643034
TCMC2123
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1514
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 2.1 (ug/ml), Ref: 19515569
TCMC2304
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.3 (ug/ml), Ref: 9461665
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC1711
TCMT1257 Colletotrichum lagenarium Colletotrichum lagenarium MIC: 12.5 (ug/ml), Ref: 17190464
TCMC1793
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1251 Candida albicans Candida albicans MIC: 12.5 (ug/ml), Ref: 9392889
TCMC1793
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 61.5 (ug/ml), Ref: 20218656
TCMC2322
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 20 (ug/ml), Ref: 3204384
TCMC2322
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 5 (ug/ml), Ref: 3204384
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC1445
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2.5 (ug/ml), Ref: 10654410
TCMC1445
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 2.5 (ug/ml), Ref: 10654410
TCMC2325
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 71.7 (ug/ml), Ref: 15104496
TCMC2325
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 53.8 (ug/ml), Ref: 15104496
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC1957
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.13 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2013
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1395
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 23369537
TCMC2347
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 0.398 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2351
TCMT1190 Plasmodium falciparum (isolate FcB1 / Columbia) Plasmodium falciparum FcB1/Columbia IC50: 16.7 (ug/ml), Ref: 21985060
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC1901
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1236 Mycobacterium bovis Mycobacterium bovis BCG MIC: 26 (ug/ml), Ref: 18849164
TCMC1901
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1191 Bacillus megaterium Bacillus megaterium MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1286 Bacillus cereus Bacillus cereus MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1260 Streptococcus agalactiae Streptococcus agalactiae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1322 Streptococcus mitis Streptococcus mitis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1323 Corynebacterium pseudodiphtheriticum Corynebacterium pseudodiphtheriticum MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1324 Corynebacterium diphtheriae Corynebacterium diphtheriae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1319 Corynebacterium xerosis Corynebacterium xerosis MIC: 16 (ug/ml), Ref: 18849164
TCMC2108
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 0.5 (ug/ml), Ref: 10571160
MIC: 0.5 (ug/ml), Ref: 9873376
MIC: 2 (ug/ml), Ref: 10966749
MIC: 0.5 (ug/ml), Ref: 9873650
MIC: 0.5 (ug/ml), Ref: 16884306
MIC: 0.2 (ug/ml), Ref: 17331717
MIC: 1 (ug/ml), Ref: 17888665
MIC: 0.5 (ug/ml), Ref: 18494459
MIC: 4 (ug/ml), Ref: 18494459
MIC: 16 (ug/ml), Ref: 18494459
MIC: 2 (ug/ml), Ref: 9428161
MIC: 1.56 (ug/ml), Ref: 17132069
MIC: 0.78 (ug/ml), Ref: 17132069
MIC: 0.156 (ug/ml), Ref: 19555123
MIC: 0.5 (ug/ml), Ref: 19595488
MIC: 32 (ug/ml), Ref: 20516287
MIC: 0.125 (ug/ml), Ref: 20516287
MIC: 0.5 (ug/ml), Ref: 20934344
MIC: 16 (ug/ml), Ref: 20713679
MIC: 0.125 (ug/ml), Ref: 20713679
MIC: 0.5 (ug/ml), Ref: 20713679
MIC: 2 (ug/ml), Ref: 22418278
MIC: 2.5 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 2 (ug/ml), Ref: 25462220
MIC: 100 (nM), Ref: 17562368
TCMC2108
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 8 (ug/ml), Ref: 10571160
MIC: 8 (ug/ml), Ref: 9873376
MIC: 8 (ug/ml), Ref: 9873650
MIC: 0.5 (ug/ml), Ref: 15603950
MIC: 8 (ug/ml), Ref: 16884306
MIC: 1.56 (ug/ml), Ref: 1800634
MIC: 0.78 (ug/ml), Ref: 6361218
MIC: 8 (ug/ml), Ref: 18494459
MIC: 3.12 (ug/ml), Ref: 2746258
MIC: 0.39 (ug/ml), Ref: 19828313
MIC: 4 (ug/ml), Ref: 10.1007/s00044-013-0498-3
MIC: 4 (ug/ml), Ref: 23807823
MIC: 4 (ug/ml), Ref: 23871903
MIC: 1.25 (ug/ml), Ref: 10.1007/s00044-013-0737-7
MIC: 0.125 (ug/ml), Ref: 24835198
TCMC2108
TCMT1239 Mycobacterium marinum Mycobacterium marinum MIC: 32 (ug/ml), Ref: 10571160
MIC: 32 (ug/ml), Ref: 9873376
MIC: 32 (ug/ml), Ref: 9873650
MIC: 32 (ug/ml), Ref: 16884306
MIC: 32 (ug/ml), Ref: 18494459
MIC: 0.5 (ug/ml), Ref: 24835198
TCMC2108
TCMT1325 Mycobacterium gordonae Mycobacterium gordonae MIC: 16 (ug/ml), Ref: 10571160
MIC: 16 (ug/ml), Ref: 9873376
MIC: 16 (ug/ml), Ref: 9873650
TCMC2108
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2.1 (ug/ml), Ref: 11858989
IC50: 0.3 (ug/ml), Ref: 14741287
MIC: 4 (ug/ml), Ref: 15603950
MIC: 2 (ug/ml), Ref: 15603950
MIC: 3 (ug/ml), Ref: 15780612
MIC: 6.25 (ug/ml), Ref: 15686925
MIC: 6.25 (ug/ml), Ref: 16213726
MIC: 3.12 (ug/ml), Ref: 17337097
MIC: 100 (ug/ml), Ref: 17331717
MIC: 12.5 (ug/ml), Ref: 17822297
MIC: 1.562 (ug/ml), Ref: 18160285
MIC: 12.5 (ug/ml), Ref: 1800634
MIC: 5 (ug/ml), Ref: 16180824
MIC: 5 (ug/ml), Ref: 4031898
MIC: 1 (ug/ml), Ref: 4031898
MIC: 3.1 (ug/ml), Ref: 6361218
MIC: 6.25 (ug/ml), Ref: 2746258
MIC: 6.25 (ug/ml), Ref: 8289060
MIC: 100 (ug/ml), Ref: 12762812
MIC: 14 (ug/ml), Ref: 10514301
MIC: 10 (ug/ml), Ref: 16643045
MIC: 25 (ug/ml), Ref: 19477639
MIC: 3 (ug/ml), Ref: 17923494
MIC: 12 (ug/ml), Ref: 17923494
MIC: 8 (ug/ml), Ref: 17923494
MIC: 6 (ug/ml), Ref: 17923494
MIC: 16 (ug/ml), Ref: 17923494
MIC: 24 (ug/ml), Ref: 17923494
MIC: 32 (ug/ml), Ref: 17923494
MIC: 64 (ug/ml), Ref: 17923494
MIC: 96 (ug/ml), Ref: 17923494
MIC: 48 (ug/ml), Ref: 17923494
MIC: 50 (ug/ml), Ref: 19361987
MIC: 1.56 (ug/ml), Ref: 19931223
MIC: 50 (ug/ml), Ref: 19828313
MIC: 6.25 (ug/ml), Ref: 19647904
MIC: 7.8 (ug/ml), Ref: 19948407
MIC: 1.56 (ug/ml), Ref: 20457477
MIC: 10 (ug/ml), Ref: 20570024
MIC: 50 (ug/ml), Ref: 20933408
MIC: 4 (ug/ml), Ref: 18519725
MIC: 1.5 (ug/ml), Ref: 18541730
MIC: 50 (ug/ml), Ref: 20822833
MIC: 6.25 (ug/ml), Ref: 21067928
MIC: 50 (ug/ml), Ref: 20947223
MIC: 50 (ug/ml), Ref: 21232949
MIC: 50 (ug/ml), Ref: 21397368
MIC: 6.25 (ug/ml), Ref: 21641208
MIC: 50 (ug/ml), Ref: 21958543
MIC: 6.25 (ug/ml), Ref: 21924612
MIC: 6.25 (ug/ml), Ref: 22405285
MIC: 6.25 (ug/ml), Ref: 22742908
MIC: 32 (ug/ml), Ref: 22902657
MIC: 50 (ug/ml), Ref: 23031593
MIC: 5 (ug/ml), Ref: 23079521
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-010-9446-7
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9354-x
MIC: 2 (ug/ml), Ref: 10.1007/s00044-010-9360-z
MIC: 2 (ug/ml), Ref: 10.1007/s00044-009-9288-3
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9367-5
MIC: 6.25 (ug/ml), Ref: 19571412
MIC: 25 (ug/ml), Ref: 10.1007/s00044-010-9528-6
MIC: 25 (ug/ml), Ref: 10.1007/s00044-006-0032-y
MIC: 25 (ug/ml), Ref: 10.1007/s00044-007-9029-4
MIC: 25 (ug/ml), Ref: 10.1007/s00044-006-0014-0
MIC: 25 (ug/ml), Ref: 10.1007/s00044-007-9023-x
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0168-x
MIC: 50 (ug/ml), Ref: 10.1007/s00044-013-0533-4
MIC: 0.125 (ug/ml), Ref: 10.1007/s00044-013-0568-6
MIC: 30 (ug/ml), Ref: 10.1007/s00044-013-0494-7
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0408-0
MIC: 5 (ug/ml), Ref: 10.1007/s00044-012-0269-6
MIC: 1.56 (ug/ml), Ref: 10.1007/s00044-012-0332-3
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0290-9
MIC: 0.002 (ug/ml), Ref: 23265883
MIC: 6.25 (ug/ml), Ref: 23395665
MIC: 32 (ug/ml), Ref: 10.1007/s00044-013-0813-z
MIC: 6.25 (ug/ml), Ref: 23973825
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
MIC: 10 (ug/ml), Ref: 10.1007/s00044-013-0728-8
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-013-0737-7
MIC: 31.25 (ug/ml), Ref: 24144849
MIC: 31.25 (ug/ml), Ref: 24480358
MIC: 6.25 (ug/ml), Ref: 24956555
MIC: 6.25 (ug/ml), Ref: 24894558
MIC: 25 (ug/ml), Ref: 25096298
MIC: 3.9 (ug/ml), Ref: 24913712
MIC: 6.25 (ug/ml), Ref: 26028159
MIC: 5 (ug/ml), Ref: 26186257
MIC: 6.25 (ug/ml), Ref: 26296475
MIC: 32 (ug/ml), Ref: 26414807
TCMC2108
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 2.1 (ug/ml), Ref: 11858989
IC50: 0.12 (ug/ml), Ref: 14741287
MIC: 1 (ug/ml), Ref: 17979247
MIC: 1.562 (ug/ml), Ref: 18160285
MIC: 1.562 (ug/ml), Ref: 19931223
MIC: 1.562 (ug/ml), Ref: 20457477
MIC: 3.125 (ug/ml), Ref: 21067928
MIC: 3.125 (ug/ml), Ref: 21641208
MIC: 3.125 (ug/ml), Ref: 21924612
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-010-9367-5
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-0168-x
MIC: 1.562 (ug/ml), Ref: 10.1007/s00044-012-0332-3
MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 6.35 (ug/ml), Ref: 10.1007/s00044-013-0809-8
MIC: 3.125 (ug/ml), Ref: 23973825
MIC: 6.25 (ug/ml), Ref: 24956555
TCMC2108
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 0.6 (ug/ml), Ref: 11858989
MIC: 25 (ug/ml), Ref: 17241703
MIC: 6.25 (ug/ml), Ref: 17189665
MIC: 3.125 (ug/ml), Ref: 18160285
MIC: 1.56 (ug/ml), Ref: 6361218
MIC: 25 (ug/ml), Ref: 19477639
MIC: 25 (ug/ml), Ref: 19361987
MIC: 1.562 (ug/ml), Ref: 20705370
MIC: 25 (ug/ml), Ref: 20933408
MIC: 50 (ug/ml), Ref: 20822833
MIC: 3.125 (ug/ml), Ref: 21067928
MIC: 25 (ug/ml), Ref: 20947223
MIC: 1.562 (ug/ml), Ref: 21211971
MIC: 25 (ug/ml), Ref: 21397368
MIC: 3.125 (ug/ml), Ref: 21641208
MIC: 25 (ug/ml), Ref: 21958543
MIC: 3.125 (ug/ml), Ref: 21924612
MIC: 6.25 (ug/ml), Ref: 22405285
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9446-7
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-010-9367-5
MIC: 20 (ug/ml), Ref: 10.1007/s00044-010-9528-6
MIC: 25 (ug/ml), Ref: 10.1007/s00044-004-0035-5
MIC: 25 (ug/ml), Ref: 10.1007/s00044-005-0134-y
MIC: 3.1 (ug/ml), Ref: 23229055
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-0168-x
MIC: 20 (ug/ml), Ref: 10.1007/s00044-013-0533-4
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 6.25 (ug/ml), Ref: 23395665
MIC: 25 (ug/ml), Ref: 23639539
MIC: 3.125 (ug/ml), Ref: 23973825
MIC: 2.71 (ug/ml), Ref: 10.1007/s00044-013-0809-8
MIC: 5 (ug/ml), Ref: 10.1007/s00044-013-0728-8
MIC: 6.25 (ug/ml), Ref: 24956555
MIC: 6.25 (ug/ml), Ref: 24894558
MIC: 50 (ug/ml), Ref: 25096298
MIC: 6.25 (ug/ml), Ref: 26028159
MIC: 25 (ug/ml), Ref: 26296475
TCMC2108
TCMT1246 Escherichia coli Escherichia coli MIC: 0.6 (ug/ml), Ref: 11858989
IC50: 1.25 (ug/ml), Ref: 14741287
MIC: 6 (ug/ml), Ref: 15780612
MIC: 0.312 (ug/ml), Ref: 17315959
MIC: 1 (ug/ml), Ref: 17158944
MIC: 0.5 (ug/ml), Ref: 17158944
MIC: 8 (ug/ml), Ref: 17210778
MIC: 20 (ug/ml), Ref: 17210778
MIC: 4 (ug/ml), Ref: 17210778
MIC: 12.5 (ug/ml), Ref: 17241703
MIC: 1.56 (ug/ml), Ref: 17337097
MIC: 6.25 (ug/ml), Ref: 17189665
MIC: 12.5 (ug/ml), Ref: 17822297
MIC: 0.5 (ug/ml), Ref: 17979247
MIC: 100 (ug/ml), Ref: 18053730
MIC: 2.35 (ug/ml), Ref: 18160285
MIC: 80 (ug/ml), Ref: 4031898
MIC: 0.5 (ug/ml), Ref: 4031898
MIC: 12.5 (ug/ml), Ref: 6361218
MIC: 3.12 (ug/ml), Ref: 8289060
MIC: 28 (ug/ml), Ref: 10514301
MIC: 20 (ug/ml), Ref: 19477639
MIC: 2 (ug/ml), Ref: 17724159
MIC: 8 (ug/ml), Ref: 17724159
MIC: 1 (ug/ml), Ref: 17724159
MIC: 4 (ug/ml), Ref: 18657340
MIC: 32 (ug/ml), Ref: 17875999
MIC: 1 (ug/ml), Ref: 17875999
MIC: 12.5 (ug/ml), Ref: 19361987
MIC: 6.25 (ug/ml), Ref: 19683840
IC50: 0.73 (ug/ml), Ref: 19655779
MIC: 3.125 (ug/ml), Ref: 19931223
MIC: 50 (ug/ml), Ref: 19828313
MIC: 1.562 (ug/ml), Ref: 19647904
MIC: 5 (ug/ml), Ref: 20036039
MIC: 100 (ug/ml), Ref: 20112996
MIC: 5 (ug/ml), Ref: 20435389
MIC: 3.125 (ug/ml), Ref: 20457477
MIC: 2 (ug/ml), Ref: 19901088
MIC: 8 (ug/ml), Ref: 20570024
MIC: 1.562 (ug/ml), Ref: 20705370
MIC: 12.5 (ug/ml), Ref: 20933408
MIC: 2 (ug/ml), Ref: 20547812
MIC: 32 (ug/ml), Ref: 20547812
MIC: 1 (ug/ml), Ref: 20547812
MIC: 12.5 (ug/ml), Ref: 20822833
MIC: 6.25 (ug/ml), Ref: 21067928
MIC: 32 (ug/ml), Ref: 19029319
MIC: 12.5 (ug/ml), Ref: 20947223
MIC: 1 (ug/ml), Ref: 19687243
MIC: 32 (ug/ml), Ref: 19687243
MIC: 2 (ug/ml), Ref: 19687243
MIC: 0.5 (ug/ml), Ref: 19687243
MIC: 1.562 (ug/ml), Ref: 21211971
MIC: 50 (ug/ml), Ref: 21232949
MIC: 6.25 (ug/ml), Ref: 20855745
MIC: 0.78 (ug/ml), Ref: 20855745
MIC: 8 (ug/ml), Ref: 20855745
MIC: 2 (ug/ml), Ref: 20696876
MIC: 4 (ug/ml), Ref: 20696876
MIC: 12.5 (ug/ml), Ref: 21397368
MIC: 6.25 (ug/ml), Ref: 21641208
MIC: 12.5 (ug/ml), Ref: 21958543
MIC: 6.25 (ug/ml), Ref: 21924612
MIC: 6.25 (ug/ml), Ref: 22742908
MIC: 16 (ug/ml), Ref: 22902657
MIC: 12.5 (ug/ml), Ref: 23031593
MIC: 5 (ug/ml), Ref: 23079521
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9446-7
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9354-x
MIC: 4 (ug/ml), Ref: 10.1007/s00044-010-9360-z
MIC: 4 (ug/ml), Ref: 10.1007/s00044-009-9288-3
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9367-5
MIC: 0.7 (ug/ml), Ref: 10.1007/s00044-011-9755-5
MIC: 13 (ug/ml), Ref: 10.1007/s00044-006-0015-z
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-007-9029-4
MIC: 50 (ug/ml), Ref: 10.1007/s00044-010-9528-6
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-004-0035-5
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-005-0134-y
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-006-0014-0
MIC: 50 (ug/ml), Ref: 10.1007/s00044-007-9023-x
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0168-x
MIC: 50 (ug/ml), Ref: 10.1007/s00044-013-0533-4
MIC: 1 (ug/ml), Ref: 10.1007/s00044-013-0568-6
MIC: 30 (ug/ml), Ref: 10.1007/s00044-013-0494-7
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-0408-0
MIC: 5 (ug/ml), Ref: 10.1007/s00044-012-0269-6
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-0332-3
MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0290-9
MIC: 12.5 (ug/ml), Ref: 23639539
MIC: 6.25 (ug/ml), Ref: 23973825
MIC: 1.35 (ug/ml), Ref: 10.1007/s00044-013-0809-8
MIC: 64 (ug/ml), Ref: 10.1007/s00044-013-0813-z
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-013-0737-7
MIC: 15.63 (ug/ml), Ref: 24144849
MIC: 31.25 (ug/ml), Ref: 24480358
MIC: 5 (ug/ml), Ref: 24992076
MIC: 1 (ug/ml), Ref: 25356913
MIC: 1 (ug/ml), Ref: 26186257
MIC: 32 (ug/ml), Ref: 26414807
TCMC2108
TCMT1462 Streptococcus mutans Streptococcus mutans IC50: 0.12 (ug/ml), Ref: 14741287
MIC: 6.35 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2108
TCMT1229 Enterococcus faecalis Enterococcus faecalis IC50: 1.25 (ug/ml), Ref: 14741287
MIC: 50 (ug/ml), Ref: 17241703
MIC: 32 (ug/ml), Ref: 17371822
MIC: 32 (ug/ml), Ref: 19029325
MIC: 50 (ug/ml), Ref: 10.1007/s00044-007-9029-4
MIC: 50 (ug/ml), Ref: 10.1007/s00044-006-0032-y
MIC: 50 (ug/ml), Ref: 10.1007/s00044-004-0035-5
MIC: 50 (ug/ml), Ref: 10.1007/s00044-005-0134-y
MIC: 50 (ug/ml), Ref: 10.1007/s00044-006-0014-0
MIC: 50 (ug/ml), Ref: 23639539
MIC: 0.36 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2108
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium IC50: 1.25 (ug/ml), Ref: 14741287
MIC: 50 (ug/ml), Ref: 18053730
MIC: 30 (ug/ml), Ref: 22405285
MIC: 25 (ug/ml), Ref: 10.1007/s00044-010-9528-6
MIC: 30 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 30 (ug/ml), Ref: 23395665
MIC: 62.5 (ug/ml), Ref: 24144849
MIC: 30 (ug/ml), Ref: 24956555
MIC: 30 (ug/ml), Ref: 24894558
MIC: 30 (ug/ml), Ref: 26028159
MIC: 6.25 (ug/ml), Ref: 26296475
TCMC2108
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes IC50: 1.25 (ug/ml), Ref: 14741287
MIC: 1.562 (ug/ml), Ref: 15686925
MIC: 1.562 (ug/ml), Ref: 16213726
MIC: 2 (ug/ml), Ref: 20547812
MIC: 16 (ug/ml), Ref: 20547812
MIC: 25 (ug/ml), Ref: 22405285
MIC: 1.56 (ug/ml), Ref: 19571412
MIC: 25 (ug/ml), Ref: 23395665
MIC: 2.71 (ug/ml), Ref: 10.1007/s00044-013-0809-8
MIC: 25 (ug/ml), Ref: 24956555
MIC: 25 (ug/ml), Ref: 24894558
MIC: 25 (ug/ml), Ref: 26028159
MIC: 25 (ug/ml), Ref: 26296475
TCMC2108
TCMT1271 Shigella flexneri Shigella flexneri IC50: 1.25 (ug/ml), Ref: 14741287
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 6.25 (ug/ml), Ref: 23395665
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-013-0737-7
MIC: 6.25 (ug/ml), Ref: 24956555
MIC: 6.25 (ug/ml), Ref: 24894558
MIC: 6.25 (ug/ml), Ref: 26028159
MIC: 6.25 (ug/ml), Ref: 26296475
TCMC2108
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 32 (ug/ml), Ref: 15603950
TCMC2108
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 3 (ug/ml), Ref: 15780612
MIC: 6.25 (ug/ml), Ref: 15686925
MIC: 6.25 (ug/ml), Ref: 16213726
MIC: 2.5 (ug/ml), Ref: 17315959
MIC: 12.5 (ug/ml), Ref: 17241703
MIC: 50 (ug/ml), Ref: 17337097
MIC: 12.5 (ug/ml), Ref: 17822297
MIC: 0.5 (ug/ml), Ref: 17979247
MIC: 100 (ug/ml), Ref: 18053730
MIC: 6.25 (ug/ml), Ref: 18160285
MIC: 0.78 (ug/ml), Ref: 1800634
MIC: 3.12 (ug/ml), Ref: 1812213
MIC: 1 (ug/ml), Ref: 4031898
MIC: 0.2 (ug/ml), Ref: 4031898
MIC: 0.78 (ug/ml), Ref: 2746258
MIC: 1.56 (ug/ml), Ref: 8289060
MIC: 2 (ug/ml), Ref: 18657340
MIC: 2 (ug/ml), Ref: 18996622
MIC: 12.5 (ug/ml), Ref: 19361987
MIC: 3.125 (ug/ml), Ref: 19683840
MIC: 6.25 (ug/ml), Ref: 19931223
MIC: 6.25 (ug/ml), Ref: 19647904
MIC: 15.6 (ug/ml), Ref: 19948407
MIC: 5 (ug/ml), Ref: 20036039
MIC: 5 (ug/ml), Ref: 20435389
MIC: 6.25 (ug/ml), Ref: 20457477
MIC: 12 (ug/ml), Ref: 20570024
MIC: 12.5 (ug/ml), Ref: 20933408
MIC: 12.5 (ug/ml), Ref: 20822833
MIC: 6.25 (ug/ml), Ref: 21067928
MIC: 5 (ug/ml), Ref: 19001112
MIC: 12.5 (ug/ml), Ref: 20947223
MIC: 12.5 (ug/ml), Ref: 21397368
MIC: 6.25 (ug/ml), Ref: 21641208
MIC: 12.5 (ug/ml), Ref: 21958543
MIC: 6.25 (ug/ml), Ref: 21924612
MIC: 6.25 (ug/ml), Ref: 22742908
MIC: 32 (ug/ml), Ref: 22902657
MIC: 12.5 (ug/ml), Ref: 23031593
MIC: 5 (ug/ml), Ref: 23079521
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9446-7
MIC: 32 (ug/ml), Ref: 10.1007/s00044-009-9288-3
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9367-5
MIC: 6.25 (ug/ml), Ref: 19571412
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-010-9528-6
MIC: 1 (ug/ml), Ref: 10.1007/s00044-011-9755-5
MIC: 19 (ug/ml), Ref: 10.1007/s00044-006-0015-z
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-007-9029-4
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-006-0032-y
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-004-0035-5
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-005-0134-y
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-006-0014-0
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-007-9023-x
MIC: 16 (ug/ml), Ref: 10.1007/s00044-011-9951-3
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0168-x
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-013-0533-4
MIC: 0.25 (ug/ml), Ref: 10.1007/s00044-013-0568-6
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0408-0
MIC: 5 (ug/ml), Ref: 10.1007/s00044-012-0269-6
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0332-3
MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-012-0290-9
MIC: 12.5 (ug/ml), Ref: 23639539
MIC: 6.25 (ug/ml), Ref: 23973825
MIC: 32 (ug/ml), Ref: 10.1007/s00044-013-0813-z
MIC: 20 (ug/ml), Ref: 10.1007/s00044-013-0728-8
MIC: 1.5 (ug/ml), Ref: 10.1007/s00044-013-0737-7
MIC: 31.25 (ug/ml), Ref: 24144849
MIC: 15.63 (ug/ml), Ref: 24480358
MIC: 5 (ug/ml), Ref: 24992076
MIC: 64 (ug/ml), Ref: 24941130
MIC: 6.25 (ug/ml), Ref: 24894558
MIC: 5 (ug/ml), Ref: 25356913
MIC: 32 (ug/ml), Ref: 25461317
MIC: 5 (ug/ml), Ref: 26186257
MIC: 25 (ug/ml), Ref: 26296475
TCMC2108
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 3.125 (ug/ml), Ref: 15686925
MIC: 1.562 (ug/ml), Ref: 16213726
MIC: 25 (ug/ml), Ref: 17241703
MIC: 100 (ug/ml), Ref: 17337097
MIC: 6.25 (ug/ml), Ref: 17189665
MIC: 3.125 (ug/ml), Ref: 18160285
MIC: 7 (ug/ml), Ref: 4031898
MIC: 12 (ug/ml), Ref: 4031898
MIC: 45 (ug/ml), Ref: 19477639
MIC: 6.25 (ug/ml), Ref: 19683840
MIC: 3.125 (ug/ml), Ref: 19931223
MIC: 3.125 (ug/ml), Ref: 19647904
MIC: 3.125 (ug/ml), Ref: 20457477
MIC: 1.562 (ug/ml), Ref: 20705370
MIC: 8 (ug/ml), Ref: 20547812
MIC: 64 (ug/ml), Ref: 20547812
MIC: 25 (ug/ml), Ref: 20822833
MIC: 1.562 (ug/ml), Ref: 21067928
MIC: 1.562 (ug/ml), Ref: 21211971
MIC: 1.562 (ug/ml), Ref: 21641208
MIC: 1.562 (ug/ml), Ref: 21924612
MIC: 6.25 (ug/ml), Ref: 22742908
MIC: 5 (ug/ml), Ref: 23079521
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-010-9446-7
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-010-9354-x
MIC: 2 (ug/ml), Ref: 10.1007/s00044-010-9360-z
MIC: 2 (ug/ml), Ref: 10.1007/s00044-009-9288-3
MIC: 1.562 (ug/ml), Ref: 10.1007/s00044-010-9367-5
MIC: 1.56 (ug/ml), Ref: 19571412
MIC: 50 (ug/ml), Ref: 10.1007/s00044-010-9528-6
MIC: 25 (ug/ml), Ref: 10.1007/s00044-007-9029-4
MIC: 25 (ug/ml), Ref: 10.1007/s00044-006-0032-y
MIC: 25 (ug/ml), Ref: 10.1007/s00044-004-0035-5
MIC: 25 (ug/ml), Ref: 10.1007/s00044-005-0134-y
MIC: 25 (ug/ml), Ref: 10.1007/s00044-006-0014-0
MIC: 50 (ug/ml), Ref: 10.1007/s00044-007-9023-x
MIC: 64 (ug/ml), Ref: 10.1007/s00044-011-9951-3
MIC: 1.562 (ug/ml), Ref: 10.1007/s00044-012-0168-x
MIC: 50 (ug/ml), Ref: 10.1007/s00044-013-0533-4
MIC: 0.5 (ug/ml), Ref: 10.1007/s00044-013-0568-6
MIC: 30 (ug/ml), Ref: 10.1007/s00044-013-0494-7
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-0408-0
MIC: 5 (ug/ml), Ref: 10.1007/s00044-012-0269-6
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-0332-3
MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0393-3
MIC: 12.5 (ug/ml), Ref: 10.1007/s00044-012-0290-9
MIC: 25 (ug/ml), Ref: 23639539
MIC: 1.562 (ug/ml), Ref: 23973825
MIC: 64 (ug/ml), Ref: 10.1007/s00044-013-0813-z
MIC: 3.15 (ug/ml), Ref: 10.1007/s00044-013-0737-7
MIC: 25 (ug/ml), Ref: 24894558
MIC: 12.5 (ug/ml), Ref: 25096298
MIC: 10 (ug/ml), Ref: 26186257
MIC: 25 (ug/ml), Ref: 26296475
TCMC2108
TCMT1311 Pseudomonas tolaasii Pseudomonas tolaasii MIC: 1 (ug/ml), Ref: 17979247
TCMC2108
TCMT1305 Salmonella enteritidis Salmonella enterica subsp. enterica serovar Enteritidis MIC: 1 (ug/ml), Ref: 17979247
MIC: 50 (ug/ml), Ref: 18053730
TCMC2108
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 50 (ug/ml), Ref: 18053730
MIC: 1 (ug/ml), Ref: 10.1007/s00044-011-9755-5
TCMC2108
TCMT1286 Bacillus cereus Bacillus cereus MIC: 0.1 (ug/ml), Ref: 16180824
MIC: 100 (ug/ml), Ref: 12762812
MIC: 7.8 (ug/ml), Ref: 19948407
MIC: 50 (ug/ml), Ref: 20112996
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-010-9446-7
MIC: 15.63 (ug/ml), Ref: 24144849
MIC: 64 (ug/ml), Ref: 24941130
TCMC2108
TCMT1461 Salmonella enterica subsp. enterica serovar Gallinarum Salmonella enterica subsp. enterica serovar Gallinarum MIC: 25 (ug/ml), Ref: 6361218
MIC: 1 (ug/ml), Ref: 10.1007/s00044-011-9755-5
TCMC2108
TCMT1195 Streptococcus pasteurianus Streptococcus pasteurianus MIC: 32 (ug/ml), Ref: 17371822
MIC: 64 (ug/ml), Ref: 17371822
TCMC2108
TCMT1269 Mycobacterium ulcerans Mycobacterium ulcerans MIC: 0.5 (ug/ml), Ref: 17664316
MIC: 0.25 (ug/ml), Ref: 20421401
MIC: 1 (ug/ml), Ref: 20421401
MIC: 0.13 (ug/ml), Ref: 20421401
MIC: 0.5 (ug/ml), Ref: 20421401
TCMC2108
TCMT1460 Mycobacterium intracellulare Mycobacterium intracellulare MIC: 1.56 (ug/ml), Ref: 8289060
MIC: 2 (ug/ml), Ref: 23850570
TCMC2108
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 0.5 (ug/ml), Ref: 10571160
MIC: 0.5 (ug/ml), Ref: 9873376
MIC: 2 (ug/ml), Ref: 10966749
MIC: 0.5 (ug/ml), Ref: 9873650
MIC: 0.5 (ug/ml), Ref: 16884306
MIC: 0.2 (ug/ml), Ref: 17331717
MIC: 1 (ug/ml), Ref: 17888665
MIC: 0.5 (ug/ml), Ref: 18494459
MIC: 4 (ug/ml), Ref: 18494459
MIC: 16 (ug/ml), Ref: 18494459
MIC: 2 (ug/ml), Ref: 9428161
MIC: 1.56 (ug/ml), Ref: 17132069
MIC: 0.78 (ug/ml), Ref: 17132069
MIC: 0.156 (ug/ml), Ref: 19555123
MIC: 0.5 (ug/ml), Ref: 19595488
MIC: 32 (ug/ml), Ref: 20516287
MIC: 0.125 (ug/ml), Ref: 20516287
MIC: 0.5 (ug/ml), Ref: 20934344
MIC: 16 (ug/ml), Ref: 20713679
MIC: 0.125 (ug/ml), Ref: 20713679
MIC: 0.5 (ug/ml), Ref: 20713679
MIC: 2 (ug/ml), Ref: 22418278
MIC: 2.5 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 2 (ug/ml), Ref: 25462220
MIC: 100 (nM), Ref: 17562368
TCMC2108
TCMT1262 Mycoplasma putrefaciens Mycoplasma putrefaciens MIC: 64 (ug/ml), Ref: 17638695
TCMC2108
TCMT1216 Vibrio cholerae Vibrio cholerae MIC: 25 (ug/ml), Ref: 19477639
MIC: 50 (ug/ml), Ref: 10.1007/s00044-010-9528-6
TCMC2108
TCMT1197 Shigella sp. Shigella sp. MIC: 25 (ug/ml), Ref: 19477639
TCMC2108
TCMT1273 Pseudomonas putida Pseudomonas putida MIC: 4 (ug/ml), Ref: 18657340
TCMC2108
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Ra MIC: 0.5 (ug/ml), Ref: 10571160
MIC: 0.5 (ug/ml), Ref: 9873376
MIC: 2 (ug/ml), Ref: 10966749
MIC: 0.5 (ug/ml), Ref: 9873650
MIC: 0.5 (ug/ml), Ref: 16884306
MIC: 0.2 (ug/ml), Ref: 17331717
MIC: 1 (ug/ml), Ref: 17888665
MIC: 0.5 (ug/ml), Ref: 18494459
MIC: 4 (ug/ml), Ref: 18494459
MIC: 16 (ug/ml), Ref: 18494459
MIC: 2 (ug/ml), Ref: 9428161
MIC: 1.56 (ug/ml), Ref: 17132069
MIC: 0.78 (ug/ml), Ref: 17132069
MIC: 0.156 (ug/ml), Ref: 19555123
MIC: 0.5 (ug/ml), Ref: 19595488
MIC: 32 (ug/ml), Ref: 20516287
MIC: 0.125 (ug/ml), Ref: 20516287
MIC: 0.5 (ug/ml), Ref: 20934344
MIC: 16 (ug/ml), Ref: 20713679
MIC: 0.125 (ug/ml), Ref: 20713679
MIC: 0.5 (ug/ml), Ref: 20713679
MIC: 2 (ug/ml), Ref: 22418278
MIC: 2.5 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 2 (ug/ml), Ref: 25462220
MIC: 100 (nM), Ref: 17562368
TCMC2108
TCMT1200 Bacillus thuringiensis Bacillus thuringiensis MIC: 6.25 (ug/ml), Ref: 19683840
MIC: 3 (ug/ml), Ref: 10.1007/s00044-011-9755-5
MIC: 64 (ug/ml), Ref: 24941130
TCMC2108
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 0.39 (ug/ml), Ref: 19828313
MIC: 0.5 (ug/ml), Ref: 19595488
MIC: 2 (ug/ml), Ref: 20004575
MIC: 2 (ug/ml), Ref: 20584563
MIC: 0.5 (ug/ml), Ref: 20934344
MIC: 4 (ug/ml), Ref: 21130647
MIC: 1 (ug/ml), Ref: 21145625
MIC: 0.39 (ug/ml), Ref: 21232949
MIC: 1 (ug/ml), Ref: 20713679
MIC: 6 (ug/ml), Ref: 21440336
MIC: 2 (ug/ml), Ref: 21641212
MIC: 7.5 (ug/ml), Ref: 21802797
MIC: 0.5 (ug/ml), Ref: 21859082
MIC: 10 (ug/ml), Ref: 10.1007/s00044-010-9522-z
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-012-0080-4
MIC: 4.95 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 3.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 6.25 (ug/ml), Ref: 10.1007/s00044-013-0576-6
MIC: 2 (ug/ml), Ref: 10.1007/s00044-012-0268-7
MIC: 2 (ug/ml), Ref: 23369537
MIC: 6.25 (ug/ml), Ref: 24044875
MIC: 6.25 (ug/ml), Ref: 24463645
MIC: 0.83 (ug/ml), Ref: 25372601
TCMC2108
TCMT1289 Shigella dysenteriae Shigella dysenteriae MIC: 15.6 (ug/ml), Ref: 19948407
TCMC2108
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 31.3 (ug/ml), Ref: 19948407
TCMC2108
TCMT1268 Nocardia farcinica Nocardia farcinica MIC: 64 (ug/ml), Ref: 20308368
TCMC2108
TCMT1236 Mycobacterium bovis Mycobacterium bovis MIC: 0.25 (ug/ml), Ref: 18955515
MIC: 2 (ug/ml), Ref: 18955515
TCMC2108
TCMT1174 Mycobacterium bovis BCG Mycobacterium bovis BCG MIC: 0.5 (ug/ml), Ref: 18458127
MIC: 16 (ug/ml), Ref: 18458127
TCMC2108
TCMT1172 Staphylococcus aureus subsp. aureus RN4220 Staphylococcus aureus subsp. aureus RN4220 MIC: 4 (ug/ml), Ref: 18519725
TCMC2108
TCMT1270 Streptomyces coelicolor Streptomyces coelicolor MIC: 1 (ug/ml), Ref: 19104019
MIC: 100 (ug/ml), Ref: 19104019
MIC: 20 (ug/ml), Ref: 19104019
TCMC2108
TCMT1198 Serratia marcescens Serratia marcescens MIC: 3.13 (ug/ml), Ref: 19752278
MIC: 1.56 (ug/ml), Ref: 19752278
TCMC2108
TCMT1267 Mycobacterium chelonae Mycobacterium chelonae MIC: 10 (ug/ml), Ref: 19581465
TCMC2108
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 1 (ug/ml), Ref: 21145625
MIC: 0.625 (ug/ml), Ref: 25734623
TCMC2108
TCMT1303 Bacillus Bacillus MIC: 64 (ug/ml), Ref: 22902657
MIC: 16 (ug/ml), Ref: 10.1007/s00044-013-0813-z
TCMC2108
TCMT1278 Pseudomonas Pseudomonas MIC: 25 (ug/ml), Ref: 23031593
TCMC2108
TCMT1287 Bacillus subtilis subsp. spizizenii ATCC 6633 Bacillus subtilis subsp. spizizenii ATCC 6633 MIC: 32 (ug/ml), Ref: 10.1007/s00044-010-9360-z
TCMC2108
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 1 (ug/ml), Ref: 10.1007/s00044-011-9755-5
TCMC2108
TCMT1243 Aspergillus flavus Aspergillus flavus MIC: 0.7 (ug/ml), Ref: 10.1007/s00044-011-9755-5
TCMC2108
TCMT1329 Bacillus fortis Bacillus fortis MIC: 0.9 (ug/ml), Ref: 10.1007/s00044-011-9755-5
TCMC2108
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 12 (ug/ml), Ref: 10.1007/s00044-006-0015-z
TCMC2108
TCMT1275 Erwinia chrysanthemi Erwinia chrysanthemi MIC: 4.6 (ug/ml), Ref: 23229055
TCMC2108
TCMT1179 Escherichia coli ATCC 8739 Escherichia coli ATCC 8739 MIC: 5 (ug/ml), Ref: 10.1007/s00044-013-0728-8
TCMC2108
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 1.25 (ug/ml), Ref: 10.1007/s00044-013-0737-7
TCMC2108
TCMT1280 Salmonella sp. Salmonella sp. MIC: 15.63 (ug/ml), Ref: 24144849
TCMC2108
TCMT1185 Mycobacterium phlei Mycobacterium phlei MIC: 6.25 (ug/ml), Ref: 24463645
MIC: 0.5 (ug/ml), Ref: 24835198
TCMC2108
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 7.81 (ug/ml), Ref: 24480358
TCMC2108
TCMT1330 Salmonella enterica subsp. enterica serovar Paratyphi B Salmonella enterica subsp. enterica serovar Paratyphi B MIC: 62.5 (ug/ml), Ref: 24894558
MIC: 30 (ug/ml), Ref: 26296475
TCMC2108
TCMT1279 Staphylococcus aureus subsp. aureus Staphylococcus aureus subsp. aureus MIC: 5 (ug/ml), Ref: 25356913
TCMC2108
TCMT1331 Acinetobacter sp. Acinetobacter sp. MIC: 10 (ug/ml), Ref: 25356913
TCMC1803
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 23369537
TCMC884
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC795
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.6 (ug/ml), Ref: 15844943
TCMC2382
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 20022753
TCMC2382
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 12.5 (ug/ml), Ref: 20022753
TCMC2383
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 37.96 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2385
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 12502328
MIC: 50 (ug/ml), Ref: 12502328
TCMC2385
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 50 (ug/ml), Ref: 12502328
TCMC2385
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 12502328
TCMC2388
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 3.13 (ug/ml), Ref: 12502328
TCMC2388
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 3.13 (ug/ml), Ref: 12502328
TCMC2388
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1.56 (ug/ml), Ref: 12502328
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC2398
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.557 (ug/ml), Ref: 3286870
IC50: 2.008 (ug/ml), Ref: 3286870
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2402
TCMT1251 Candida albicans Candida albicans MIC: 31.25 (ug/ml), Ref: 8254344
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC895
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.2 (ug/ml), Ref: 6492075
TCMC895
TCMT1246 Escherichia coli Escherichia coli MIC: 0.5 (ug/ml), Ref: 6492075
MIC: 1 (ug/ml), Ref: 6492075
MIC: 2 (ug/ml), Ref: 19770280
MIC: 4 (ug/ml), Ref: 19770280
TCMC895
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 3.9 (ug/ml), Ref: 6492075
TCMC895
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 15.6 (ug/ml), Ref: 6492075
TCMC895
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 15.6 (ug/ml), Ref: 6492075
MIC: 10 (ug/ml), Ref: 18838593
MIC: 2.5 (ug/ml), Ref: 18838593
MIC: 1.25 (ug/ml), Ref: 18838593
MIC: 0.625 (ug/ml), Ref: 18838593
MIC: 5 (ug/ml), Ref: 18838593
MIC: 20 (ug/ml), Ref: 18838593
TCMC895
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 2 (ug/ml), Ref: 17220400
MIC: 0.312 (ug/ml), Ref: 10543897
TCMC895
TCMT1251 Candida albicans Candida albicans MIC: 1.5 (ug/ml), Ref: 19841146
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1424
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 27.95 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC1210
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC2434
TCMT1251 Candida albicans Candida albicans MIC: 31.25 (ug/ml), Ref: 17007965
MIC: 62.5 (ug/ml), Ref: 17007965
TCMC2434
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 18584918
MIC: 32 (ug/ml), Ref: 22727643
MIC: 64 (ug/ml), Ref: 22727643
TCMC2177
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 1.56 (ug/ml), Ref: 1453180
MIC: 0.6 (ug/ml), Ref: 25791674
TCMC2177
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1.56 (ug/ml), Ref: 1453180
MIC: 0.78 (ug/ml), Ref: 1453180
MIC: 2.5 (ug/ml), Ref: 17664318
MIC: 1.25 (ug/ml), Ref: 17664318
MIC: 16 (ug/ml), Ref: 17664318
MIC: 2 (ug/ml), Ref: 17664318
MIC: 1.5 (ug/ml), Ref: 25791674
TCMC2177
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 0.78 (ug/ml), Ref: 1453180
TCMC2177
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 16 (ug/ml), Ref: 25791674
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC2439
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 2 (ug/ml), Ref: 9784148
TCMC845
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 1522419
MIC: 6.25 (ug/ml), Ref: 1522419
TCMC845
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 1522419
MIC: 1.57 (ug/ml), Ref: 1522419
TCMC2442
TCMT1251 Candida albicans Candida albicans MIC: 50 (ug/ml), Ref: 10924184
TCMC2442
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 50 (ug/ml), Ref: 10924184
TCMC2442
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10924184
TCMC2442
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10924184
TCMC2444
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 5.8 (ug/ml), Ref: 8786363
IC50: 3.65 (ug/ml), Ref: 8786363
TCMC2444
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.8 (ug/ml), Ref: 8786363
IC50: 3.65 (ug/ml), Ref: 8786363
TCMC2444
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 25372601
TCMC2447
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 18 (ug/ml), Ref: 19904996
TCMC2454
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 19.6 (ug/ml), Ref: 10425115
TCMC2459
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 37.5 (ug/ml), Ref: 9748372
TCMC1113
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 15863332
TCMC1163
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 93.8 (ug/ml), Ref: 6512542
TCMC2003
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1251 Candida albicans Candida albicans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1246 Escherichia coli Escherichia coli MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12036362
TCMC2003
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
TCMC2003
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 25 (ug/ml), Ref: 20022753
TCMC2468
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 5 (ug/ml), Ref: 10654410
TCMC2468
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 2.5 (ug/ml), Ref: 10654410
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2477
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 72.5 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1986
TCMT1442 Leishmania donovani Leishmania donovani IC50: 17.7 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2479
TCMT1251 Candida albicans Candida albicans MIC: 6.25 (ug/ml), Ref: 11170676
TCMC2479
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 11170676
TCMC2481
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 12.5 (ug/ml), Ref: 17027268
TCMC2482
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1251 Candida albicans Candida albicans MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1102
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.103 (ug/ml), Ref: 11374952
IC50: 0.145 (ug/ml), Ref: 11374952
TCMC1102
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 5.5 (ug/ml), Ref: 12502337
TCMC1248
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 6.25 (ug/ml), Ref: 17959274
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC887
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 10395496
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC2506
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 1.99 (ug/ml), Ref: 8786363
IC50: 1.9 (ug/ml), Ref: 8786363
TCMC2506
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 1.99 (ug/ml), Ref: 8786363
IC50: 1.9 (ug/ml), Ref: 8786363
TCMC1515
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1767
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 60 (ug/ml), Ref: 20384293
TCMC1767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0419-x
TCMC1425
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.422 (ug/ml), Ref: 3286870
IC50: 1.607 (ug/ml), Ref: 3286870
TCMC614
TCMT1454 Bacillus subtilis Bacillus subtilis IC50: 98.5 (ug/ml), Ref: 25981688
TCMC934
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.73 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2045
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC2045
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 59 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 51 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC1186
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 3430167
TCMC1186
TCMT1284 Penicillium expansum Penicillium expansum MIC: 50 (ug/ml), Ref: 3430167
TCMC2532
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 20 (ug/ml), Ref: 19904996
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1768
TCMT1286 Bacillus cereus Bacillus cereus MIC: 4 (ug/ml), Ref: 18293924
TCMC1768
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 4 (ug/ml), Ref: 18293924
TCMC1768
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 4 (ug/ml), Ref: 18293924
TCMC1768
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 4 (ug/ml), Ref: 18293924
TCMC1768
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 4 (ug/ml), Ref: 18293924
TCMC1768
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 4 (ug/ml), Ref: 18293924
TCMC2546
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 10 (ug/ml), Ref: 10654410
TCMC2546
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 10 (ug/ml), Ref: 10654410
TCMC2547
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 6.25 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
TCMC2547
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 6.25 (ug/ml), Ref: 12502328
TCMC2547
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1.56 (ug/ml), Ref: 12502328
TCMC858
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.555 (ug/ml), Ref: 3286870
IC50: 1.739 (ug/ml), Ref: 3286870
TCMC858
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 42.71 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC1117
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 100 (ug/ml), Ref: 10425115
TCMC1117
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.89 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2556
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 10 (ug/ml), Ref: 10654410
TCMC2556
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 10 (ug/ml), Ref: 10654410
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC1936
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 14 (ug/ml), Ref: 10425115
TCMC1572
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC2565
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7 (ug/ml), Ref: 17845001
TCMC2566
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2571
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 13.4 (ug/ml), Ref: 15104489
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC2578
TCMT1251 Candida albicans Candida albicans IC50: 82.98 (ug/ml), Ref: 25686593
TCMC915
TCMT1246 Escherichia coli Escherichia coli MIC: 1 (ug/ml), Ref: 25791674
TCMC915
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 0.5 (ug/ml), Ref: 25791674
TCMC915
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.25 (ug/ml), Ref: 25791674
TCMC2580
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 12398535
TCMC2580
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 17.2 (ug/ml), Ref: 10425115
TCMC2581
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC755
TCMT1251 Candida albicans Candida albicans IC50: 6 (ug/ml), Ref: 12502337
TCMC755
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC755
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 6.46 (ug/ml), Ref: 25564380
TCMC1329
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2591
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 6.25 (ug/ml), Ref: 8864235
TCMC2591
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 0.78 (ug/ml), Ref: 8864235
TCMC2591
TCMT1210 Streptococcus sobrinus Streptococcus sobrinus MIC: 1.56 (ug/ml), Ref: 8864235
TCMC2591
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 0.39 (ug/ml), Ref: 8864235
TCMC2591
TCMT1370 Prevotella melaninogenica Prevotella melaninogenica MIC: 0.78 (ug/ml), Ref: 8864235
TCMC2596
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 17845001
TCMC2069
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 12502328
MIC: 50 (ug/ml), Ref: 12502328
TCMC2069
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 50 (ug/ml), Ref: 12502328
TCMC2069
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 12502328
TCMC1168
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 9392889
MIC: 2.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 9392889
TCMC1168
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
MIC: 25 (ug/ml), Ref: 10217726
TCMC1168
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1251 Candida albicans Candida albicans MIC: 25 (ug/ml), Ref: 9392889
TCMC1168
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.2 (ug/ml), Ref: 20218656
TCMC969
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 3.125 (ug/ml), Ref: 20605657
MIC: 3.125 (ug/ml), Ref: 21489661
MIC: 3.125 (ug/ml), Ref: 10.1007/s00044-012-9978-0
MIC: 3.125 (ug/ml), Ref: 23318903
TCMC1105
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 51.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 50.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1105
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 23534483
TCMC1105
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 1 (ug/ml), Ref: 23534483
TCMC1105
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 23534483
MIC: 4 (ug/ml), Ref: 23534483
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2040
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.03 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2612
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 4 (ug/ml), Ref: 12932139
TCMC2612
TCMT1251 Candida albicans Candida albicans MIC: 16 (ug/ml), Ref: 12932139
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2613
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 15 (ug/ml), Ref: 9748372
TCMC348
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 62 (ug/ml), Ref: 25813159
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC732
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 9 (ug/ml), Ref: 9748372
TCMC2617
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 29.9 (ug/ml), Ref: 10425115
TCMC1203
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 22.6 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC804
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC946
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 14510592
TCMC2628
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 19.45 (ug/ml), Ref: 24549242
IC50: 30.05 (ug/ml), Ref: 24549242
IC50: 57.67 (ug/ml), Ref: 24549242
TCMC1033
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC2633
TCMT1286 Bacillus cereus Bacillus cereus MIC: 100 (ug/ml), Ref: 10425115
TCMC2633
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 5.8 (ug/ml), Ref: 10425115
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC2640
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2.5 (ug/ml), Ref: 10654410
TCMC2640
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 2.5 (ug/ml), Ref: 10654410
TCMC2640
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 10 (ug/ml), Ref: 10654410
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1939
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 4.3 (ug/ml), Ref: 10425115
TCMC1977
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 19232493
TCMC1977
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 19232493
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2228
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 18 (ug/ml), Ref: 18597896
TCMC2228
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 9 (ug/ml), Ref: 18597896
TCMC2228
TCMT1246 Escherichia coli Escherichia coli MIC: 16 (ug/ml), Ref: 18597896
TCMC2228
TCMT1251 Candida albicans Candida albicans MIC: 11 (ug/ml), Ref: 18597896
TCMC2660
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2660
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 6.25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2661
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 11 (ug/ml), Ref: 19904996
TCMC2014
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 10 (ug/ml), Ref: 17220400
TCMC1523
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 18611050
MIC: 25 (ug/ml), Ref: 21131198
MIC: 25 (ug/ml), Ref: 21401117
MIC: 16 (ug/ml), Ref: 22424614
MIC: 32 (ug/ml), Ref: 22424614
MBC: 32 (ug/ml), Ref: 22424614
TCMC1523
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 6.25 (ug/ml), Ref: 18611050
MIC: 12.5 (ug/ml), Ref: 21131198
TCMC1523
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 12.5 (ug/ml), Ref: 18611050
MIC: 12.5 (ug/ml), Ref: 21131198
MIC: 12.5 (ug/ml), Ref: 21401117
TCMC1523
TCMT1201 Staphylococcus epidermidis ATCC 12228 Staphylococcus epidermidis ATCC 12228 MIC: 12.5 (ug/ml), Ref: 21401117
TCMC1523
TCMT1286 Bacillus cereus Bacillus cereus MIC: 12.5 (ug/ml), Ref: 21401117
TCMC1523
TCMT1219 Enterococcus Enterococcus MIC: 32 (ug/ml), Ref: 22424614
MBC: 32 (ug/ml), Ref: 22424614
TCMC2667
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 15104489
MIC: 100 (ug/ml), Ref: 20542692
TCMC1551
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 20832915
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC865
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.238 (ug/ml), Ref: 14575431
TCMC865
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 23 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC865
TCMT1286 Bacillus cereus Bacillus cereus MIC: 7.81 (ug/ml), Ref: 26681509
TCMC865
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 31.25 (ug/ml), Ref: 26681509
TCMC2675
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 8.3 (ug/ml), Ref: 10425115
TCMC1733
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.2 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1123
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1123
TCMT1442 Leishmania donovani Leishmania donovani IC50: 25 (ug/ml), Ref: 15679330
TCMC2086
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC2086
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC785
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.36 (ug/ml), Ref: 10.1016/S0960-894X(00)80357-1
IC50: 0.141 (ug/ml), Ref: 3286870
IC50: 0.148 (ug/ml), Ref: 3286870
TCMC785
TCMT1246 Escherichia coli Escherichia coli MIC: 5 (ug/ml), Ref: 16359864
MIC: 31.25 (ug/ml), Ref: 18591276
TCMC785
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 64 (ug/ml), Ref: 16730982
MIC: 31.3 (ug/ml), Ref: 16872133
TCMC785
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 17716892
MIC: 50 (ug/ml), Ref: 9784149
MIC: 60 (ug/ml), Ref: 15568768
MBC: 64 (ug/ml), Ref: 10.1007/s00044-013-0844-5
MIC: 32 (ug/ml), Ref: 10.1007/s00044-013-0844-5
TCMC785
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 100 (ug/ml), Ref: 9784149
TCMC785
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 25 (ug/ml), Ref: 9784149
TCMC785
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 9784149
MIC: 31.3 (ug/ml), Ref: 16872133
MIC: 15.6 (ug/ml), Ref: 16872133
TCMC785
TCMT1385 Candida shehatae Candida shehatae MIC: 7.8 (ug/ml), Ref: 16872133
TCMC1892
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC1892
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC624
TCMT1229 Enterococcus faecalis Enterococcus faecalis MBC: 6.25 (ug/ml), Ref: 12502328
MIC: 6.25 (ug/ml), Ref: 12502328
MBC: 3.13 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
TCMC624
TCMT1214 Enterococcus faecium Enterococcus faecium MBC: 6.25 (ug/ml), Ref: 12502328
MIC: 6.25 (ug/ml), Ref: 12502328
TCMC624
TCMT1218 Staphylococcus aureus Staphylococcus aureus MBC: 1.56 (ug/ml), Ref: 12502328
MIC: 1.56 (ug/ml), Ref: 12502328
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2681
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 16 (ug/ml), Ref: 19904996
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC2688
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 14969530
TCMC2688
TCMT1282 Colletotrichum orbiculare Colletotrichum orbiculare MIC: 30 (ug/ml), Ref: 14969530
TCMC1491
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 0.92 (ug/ml), Ref: 21334901
TCMC1491
TCMT1318 Human T-lymphotropic virus 1 Human T-lymphotropic virus 1 IC50: 1.07 (ug/ml), Ref: 21334901
TCMC1828
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.281 (ug/ml), Ref: 3286870
IC50: 0.163 (ug/ml), Ref: 3286870
TCMC2693
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 5 (ug/ml), Ref: 10654410
TCMC2693
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 5 (ug/ml), Ref: 10654410
TCMC2696
TCMT1354 Streptococcus mutans UA159 Streptococcus mutans UA159 MIC: 80 (ug/ml), Ref: 10.1007/s00044-011-9658-5
TCMC2699
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 6.3 (ug/ml), Ref: 14995101
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC1889
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2706
TCMT1229 Enterococcus faecalis Enterococcus faecalis MBC: 6.25 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
MBC: 3.13 (ug/ml), Ref: 12502328
TCMC2706
TCMT1214 Enterococcus faecium Enterococcus faecium MBC: 3.13 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
TCMC2706
TCMT1218 Staphylococcus aureus Staphylococcus aureus MBC: 3.13 (ug/ml), Ref: 12502328
MIC: 1.56 (ug/ml), Ref: 12502328
MBC: 1.56 (ug/ml), Ref: 12502328
TCMC2709
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 59.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1236
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (ug/ml), Ref: 19299148
TCMC2714
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 1.4 (ug/ml), Ref: 22280816
TCMC2714
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25.3 (ug/ml), Ref: 22280816
TCMC2718
TCMT1229 Enterococcus faecalis Enterococcus faecalis MBC: 3.13 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
TCMC2718
TCMT1214 Enterococcus faecium Enterococcus faecium MBC: 3.13 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
TCMC2718
TCMT1218 Staphylococcus aureus Staphylococcus aureus MBC: 3.13 (ug/ml), Ref: 12502328
MIC: 3.13 (ug/ml), Ref: 12502328
MBC: 1.56 (ug/ml), Ref: 12502328
MIC: 1.56 (ug/ml), Ref: 12502328
TCMC1519
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 22280816
TCMC2044
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 15 (ug/ml), Ref: 9644074
MIC: 15 (ug/ml), Ref: 8904847
TCMC2044
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 15 (ug/ml), Ref: 8904847
TCMC2044
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC90: 16 (ug/ml), Ref: 23127490
MIC90: 8 (ug/ml), Ref: 23127490
MIC: 16 (ug/ml), Ref: 23314053
MIC: 8 (ug/ml), Ref: 23314053
TCMC2044
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC90: 2 (ug/ml), Ref: 23127490
MIC: 2 (ug/ml), Ref: 23314053
MBC: 0.034 (nM), Ref: 22182580
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1961
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 6.25 (ug/ml), Ref: 20832915
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1064
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 15 (ug/ml), Ref: 11170636
TCMC784
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2806
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.5 (ug/ml), Ref: 18524594
TCMC2808
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 27 (ug/ml), Ref: 10425115
TCMC2811
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 37.35 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1113
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 16 (nM), Ref: 17263522
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC1117
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 17.56 (nM), Ref: 17263522
TCMC1118
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 79 (nM), Ref: 17263522
Ki: 8 (nM), Ref: 17263522
TCMC4
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 40 (nM), Ref: 16722653
TCMC2338
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 8.8 (nM), Ref: 17503850
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850
TCMC1047
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 50 (nM), Ref: 24549242
TCMC2514
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 8.9 (nM), Ref: 17503850
TCMC2542
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 8.8 (nM), Ref: 17503850
TCMC1118
TCMT1222 Plasmodium falciparum D6 Plasmodium falciparum D6 IC50: 73 (nM), Ref: 25488841
TCMC969
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 100 (nM), Ref: 17060533
TCMC969
TCMT1353 Plasmodium yoelii Plasmodium yoelii IC50: 78.1 (nM), Ref: 22096101
TCMC2044
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MBC: 0.034 (nM), Ref: 22182580
TCMC2771
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 8.9 (nM), Ref: 17503850