TCM Putative Target References: TCMF6446


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC61
TCMT193 Nuclear factor NF-kappa-B p65 subunit Homo sapiens IC50: 250 (nM), Ref: 21513293
TCMC61
TCMT194 Mitogen-activated protein kinase kinase kinase 7 Homo sapiens IC50: 80 (nM), Ref: 25529738
IC50: 11 (nM), Ref: 26481152
IC50: 8.1 (nM), Ref: 26481152
IC50: 9 (nM), Ref: 27448772
TCMC61
TCMT80 MAP kinase ERK2 Homo sapiens IC50: 6800 (nM), Ref: 25529738
TCMC61
TCMT195 Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens IC50: 80 (nM), Ref: 25529738
TCMC61
TCMT196 Dual specificity mitogen-activated protein kinase kinase 7 Homo sapiens IC50: 1300 (nM), Ref: 25529738
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC1851
TCMT560 Coagulation factor X Homo sapiens IC50: 170 (nM), Ref: 9834152
Ki: 570 (nM), Ref: 9834152
TCMC1851
TCMT207 Beta-secretase 1 Homo sapiens IC50: 3760 (nM), Ref: 24835197
Ki: 5130 (nM), Ref: 24835197
TCMC1851
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 2350 (nM), Ref: 26395057
Ki: 2600 (nM), Ref: 26395057
TCMC962
TCMT45 Beta amyloid A4 protein Homo sapiens Ki: 0.208 (nM), Ref: 17004725
IC50: 800 (nM), Ref: 17270435
IC50: 3900 (nM), Ref: 26099993
TCMC962
TCMT566 Nitric oxide synthase, inducible Homo sapiens IC50: 6000 (nM), Ref: 18077363
TCMC962
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 4300 (nM), Ref: 18249473
TCMC962
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 8500 (nM), Ref: 19128977
TCMC962
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2410 (nM), Ref: 20674354
TCMC962
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 380 (nM), Ref: 20674354
TCMC962
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4970 (nM), Ref: 20674354
TCMC962
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9460 (nM), Ref: 20674354
TCMC962
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 9940 (nM), Ref: 20674354
TCMC962
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9300 (nM), Ref: 20674354
TCMC962
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4050 (nM), Ref: 20674354
TCMC962
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3480 (nM), Ref: 20674354
TCMC962
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 6850 (nM), Ref: 20674354
TCMC962
TCMT44 Glyoxalase I Homo sapiens Ki: 10000 (nM), Ref: 21237663
TCMC962
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 7410 (nM), Ref:
TCMC962
TCMT46 Coagulation factor III Homo sapiens IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5
IC50: 199.63 (nM), Ref: 23199480
TCMC962
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 8600 (nM), Ref: 23245570
TCMC962
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 4501 (nM), Ref: 23800686
TCMC962
TCMT570 Aminopeptidase N Homo sapiens IC50: 10000 (nM), Ref: 23860593
TCMC962
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 3900 (nM), Ref: 24920381
IC50: 500 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
TCMC962
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 8100 (nM), Ref: 24920381
TCMC962
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 600 (nM), Ref: 24920381
IC50: 1200 (nM), Ref: 24920381
TCMC962
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 1200 (nM), Ref: 24920381
TCMC962
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5300 (nM), Ref: 25088549
TCMC962
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 25730130
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC1285
TCMT33 Cytochrome P450 3A4 Homo sapiens Ki: 399 (nM), Ref: 16248836
TCMC891
TCMT598 DNA topoisomerase I Homo sapiens IC50: 50 (nM), Ref: 1324981
IC50: 100 (nM), Ref: 1324981
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC42
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 8390 (nM), Ref: 26696252
TCMC42
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2540 (nM), Ref: 26696252
TCMC694
TCMT230 Estradiol 17-beta-dehydrogenase 3 Homo sapiens IC50: 758 (nM), Ref: 11086723
IC50: 758 (nM), Ref: 16078844
TCMC694
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 20 (nM), Ref: 8035427
Ki: 35 (nM), Ref: 26469743
TCMC1376
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 40 (nM), Ref: 11678654
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC43
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 220 (nM), Ref: 26588603
IC50: 200 (nM), Ref: 10.1039/C5MD00278H
TCMC43
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 26701186
TCMC43
TCMT208 Monoamine oxidase A Homo sapiens Ki: 710 (nM), Ref: 26819666
TCMC43
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3100 (nM), Ref: 27190601
IC50: 1500 (nM), Ref: 27190601
TCMC2142
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 600 (nM), Ref: 6827528
TCMC2142
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 10000 (nM), Ref: 14552748
TCMC2142
TCMT187 Androgen Receptor Homo sapiens IC50: 3.9 (nM), Ref: 15456242
IC50: 2.7 (nM), Ref: 16309907
IC50: 4.571 (nM), Ref: 22746350
IC50: 4.17 (nM), Ref: 25646649
IC50: 4.27 (nM), Ref: 25646649
TCMC2142
TCMT99 Testis-specific androgen-binding protein Homo sapiens IC50: 14 (nM), Ref: 17149875
TCMC2142
TCMT725 Voltage-gated L-type calcium channel alpha-1C subunit Homo sapiens IC50: 34 (nM), Ref: 22761000
IC50: 38.4 (nM), Ref: 22761000
TCMC156
TCMT327 Vanilloid receptor Homo sapiens IC50: 35 (nM), Ref: 16000002
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC2048
TCMT771 Serine-protein kinase ATR Homo sapiens IC50: 7300 (nM), Ref: 22835870
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC2189
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 400 (nM), Ref: 19097799
Ki: 60 (nM), Ref: 19097799
TCMC1015
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 4320 (nM), Ref:
TCMC2196
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 64 (nM), Ref: 22819942
IC50: 64 (nM), Ref: 23146282
TCMC2196
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 150 (nM), Ref: 22819942
TCMC2196
TCMT336 Indoleamine 2,3-dioxygenase Homo sapiens IC50: 53.7 (nM), Ref: 24099220
IC50: 7150 (nM), Ref: 24099220
Ki: 4810 (nM), Ref: 24099220
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC124
TCMT194 Mitogen-activated protein kinase kinase kinase 7 Homo sapiens IC50: 1300 (nM), Ref: 26481152
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1757
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 130 (nM), Ref: 17378609
IC50: 110 (nM), Ref: 19848434
IC50: 25 (nM), Ref: 21958737
IC50: 120 (nM), Ref: 21958738
TCMC1757
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 110 (nM), Ref: 12608855
IC50: 1100 (nM), Ref: 19848434
IC50: 5100 (nM), Ref: 21739938
IC50: 110 (nM), Ref: 24684213
TCMC1757
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens IC50: 180 (nM), Ref: 12608855
IC50: 5900 (nM), Ref: 19848434
IC50: 110 (nM), Ref: 21739938
TCMC1757
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 11 (nM), Ref: 20413308
TCMC183
TCMT188 Dihydrofolate reductase Homo sapiens IC50: 500 (nM), Ref: 26979156
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC1919
TCMT613 Glucocorticoid receptor Homo sapiens IC50: 14 (nM), Ref: 19364854
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1377
TCMT186 Monoamine oxidase B Homo sapiens Ki: 3000 (nM), Ref: 16137882
Ki: 3000 (nM), Ref: 19342233
IC50: 7943.28 (nM), Ref: 20934874
Ki: 5340 (nM), Ref: 21134756
Ki: 3000 (nM), Ref: 21778064
Ki: 2000 (nM), Ref: 24140951
TCMC1377
TCMT208 Monoamine oxidase A Homo sapiens Ki: 8380 (nM), Ref: 21134756
TCMC1400
TCMT223 Aldose reductase Homo sapiens IC50: 720 (nM), Ref: 22261024
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC804
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 2000 (nM), Ref: 21561086
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC1371
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 4 (nM), Ref: 26562543
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1365
TCMT307 HERG Homo sapiens IC50: 100 (nM), Ref: 21185626
TCMC1365
TCMT903 Glutamate [NMDA] receptor subunit epsilon 2 Homo sapiens IC50: 20 (nM), Ref: 24411196
Ki: 10 (nM), Ref: 25458498
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1851
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28 (ug/ml), Ref: 9461665
TCMC962
TCMT1104 Sortase Staphylococcus aureus IC50: 13.8 (ug/ml), Ref: 19269184
TCMC962
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 51.3 (ug/ml), Ref: 16643034
TCMC962
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 1 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC2189
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum IC50: 0.014 (ug/ml), Ref: 17765547
IC50: 73 (nM), Ref: 16198563
IC50: 73 (nM), Ref: 16466916
Ki: 7.29 (nM), Ref: 17263522
Ki: 28.31 (nM), Ref: 17263522
Ki: 52.71 (nM), Ref: 17263522
Ki: 30.54 (nM), Ref: 17263522
Ki: 71.02 (nM), Ref: 17263522
Ki: 0.0019 (nM), Ref: 17263522
Ki: 0.109 (nM), Ref: 17263522
Ki: 0.05206 (nM), Ref: 17263522
Ki: 0.2806 (nM), Ref: 17263522
Ki: 0.7983 (nM), Ref: 17263522
Ki: 1 (nM), Ref: 17263522
Ki: 8.25 (nM), Ref: 17263522
Ki: 8 (nM), Ref: 17263522
Ki: 10 (nM), Ref: 17263522
Ki: 13.72 (nM), Ref: 17263522
IC50: 66 (nM), Ref: 17477517
IC50: 73 (nM), Ref: 17567585
IC50: 70 (nM), Ref: 17485508
IC50: 73 (nM), Ref: 19217192
Ki: 50 (nM), Ref: 19217192
IC50: 70 (nM), Ref: 22082562
TCMC2189
TCMT1105 Enoyl-ACP reductase Plasmodium falciparum IC50: 0.014 (ug/ml), Ref: 20855214
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC1801
TCMT1136 Neuraminidase Influenza A virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2329
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 25.3 (ug/ml), Ref: 8946749
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC962
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
IC50: 3.5 (ug/ml), Ref: 19299148
TCMC962
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 4.2 (ug/ml), Ref: 19299148
IC50: 3.5 (ug/ml), Ref: 19299148
TCMC962
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC962
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 5 (ug/ml), Ref: 19204190
MIC: 15 (ug/ml), Ref: 19204190
MIC: 50 (ug/ml), Ref: 19204190
MIC: 30 (ug/ml), Ref: 19204190
TCMC962
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 30 (ug/ml), Ref: 18284200
TCMC962
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 25938986
MIC: 32 (ug/ml), Ref: 25938986
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC1322
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2189
TCMT1246 Escherichia coli Escherichia coli MIC: 0.3 (ug/ml), Ref: 14736233
MIC: 0.2 (ug/ml), Ref: 19933806
MIC: 3 (ug/ml), Ref: 19933806
MIC: 4 (ug/ml), Ref: 19933806
MIC: 0.2 (ug/ml), Ref: 18180352
MIC: 0.125 (ug/ml), Ref: 23092194
MIC: 2 (ug/ml), Ref: 23466234
TCMC2189
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.06 (ug/ml), Ref: 12109908
MIC: 0.03 (ug/ml), Ref: 11514139
MIC: 0.125 (ug/ml), Ref: 17095231
MIC: 0.063 (ug/ml), Ref: 17713898
MIC: 20 (ug/ml), Ref: 21821415
MIC: 0.031 (ug/ml), Ref: 23092194
MIC: 4 (ug/ml), Ref: 23466234
MIC: 0.01 (ug/ml), Ref: 24332629
MIC: 0.391 (ug/ml), Ref: 26343826
TCMC2189
TCMT1177 Haemophilus influenzae Haemophilus influenzae MIC: 0.06 (ug/ml), Ref: 12109908
TCMC2189
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 16 (ug/ml), Ref: 17220400
MIC: 4 (ug/ml), Ref: 20427099
TCMC2189
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 3.1 (ug/ml), Ref: 18499454
TCMC2189
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 5 (ug/ml), Ref: 18538450
MIC: 5 (ug/ml), Ref: 22079026
TCMC2189
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 4 (ug/ml), Ref: 20427099
TCMC2189
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 4 (ug/ml), Ref: 20427099
TCMC2189
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 2 (ug/ml), Ref: 20427099
TCMC2189
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 1 (ug/ml), Ref: 19933806
TCMC2189
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 0.2 (ug/ml), Ref: 18180352
MIC: 40 (ug/ml), Ref: 18180352
MIC: 2 (ug/ml), Ref: 18180352
MIC: 5 (ug/ml), Ref: 18180352
MIC: 0.1 (ug/ml), Ref: 18180352
MIC: 20 (ug/ml), Ref: 18180352
MIC: 10 (ug/ml), Ref: 18180352
MIC: 0.8 (ug/ml), Ref: 18180352
TCMC2189
TCMT1174 Mycobacterium bovis BCG Mycobacterium bovis BCG MIC: 8 (ug/ml), Ref: 19564371
TCMC2189
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 5 (ug/ml), Ref: 18538450
MIC: 5 (ug/ml), Ref: 22079026
TCMC2189
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 2 (ug/ml), Ref: 23092194
TCMC2189
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 10 (ug/ml), Ref: 24292339
MIC: 10 (ug/ml), Ref: 25771110
TCMC2189
TCMT1286 Bacillus cereus Bacillus cereus MIC: 0.01 (ug/ml), Ref: 24332629
TCMC2189
TCMT1172 Staphylococcus aureus subsp. aureus RN4220 Staphylococcus aureus subsp. aureus RN4220 MIC: 0.01 (ug/ml), Ref: 24332629
TCMC2196
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 10 (ug/ml), Ref: 22819942
MIC: 0.5 (ug/ml), Ref: 26253635
TCMC2196
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 1 (ug/ml), Ref: 23360475
MIC: 1 (ug/ml), Ref: 26253635
TCMC2196
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 6 (ug/ml), Ref: 26253635
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2040
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.03 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC804
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 0.087 (ug/ml), Ref: 9249972
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1915
TCMT1347 Human rhinovirus 16 Human rhinovirus 16 IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1333 Human rhinovirus 1A Human rhinovirus 1A IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1241 Human rhinovirus 14 Human rhinovirus 14 IC50: 0.02 (ug/ml), Ref: 17116681
IC50: 100 (nM), Ref: 23977995
TCMC1801
TCMT1449 Influenza A virus Influenza A virus IC50: 1 (ug/ml), Ref: 14987066
IC50: 2.4 (nM), Ref: 19919060
IC50: 3.41 (nM), Ref: 15974612
IC50: 3.79 (nM), Ref: 16532013
IC50: 7.03 (nM), Ref: 19101157
IC50: 30 (nM), Ref: 25305333
IC50: 1.08 (nM), Ref: 9784165
IC50: 0.85 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 2.27 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 93.92 (nM), Ref: 20430633
IC50: 99.57 (nM), Ref: 20430633
IC50: 0.54 (nM), Ref: 20430633
IC50: 94.4 (nM), Ref: 20430633
IC50: 0.49 (nM), Ref: 20411974
IC50: 0.25 (nM), Ref: 20384296
IC50: 1 (nM), Ref: IC50: 95.43 (nM), Ref: 9461668
IC50: 78.12 (nM), Ref: 9461668
IC50: 75.29 (nM), Ref: 9461668
IC50: 1.84 (nM), Ref: 20166736
IC50: 1.59 (nM), Ref: 24673739
IC50: 0.34 (nM), Ref: 23675610
IC50: 0.25 (nM), Ref: 1431945
IC50: 3.64 (nM), Ref: 11170656
TCMC1915
TCMT1348 Human rhinovirus 2 Human rhinovirus 2 IC50: 0.01 (ug/ml), Ref: 23920485
IC50: 100 (nM), Ref: 23977995
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC2189
TCMT1140 Enoyl-[acyl-carrier-protein] reductase Staphylococcus aureus IC50: 70 (nM), Ref: 12699381
TCMC2189
TCMT1142 Enoyl-[acyl-carrier-protein] reductase [NADPH] Staphylococcus aureus IC50: 59 (nM), Ref: 23092194
TCMC1801
TCMT1162 Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1)) Ki: 1.1 (nM), Ref: IC50: 0.1 (nM), Ref: 23398362
IC50: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1164 Neuraminidase Influenza A virus (A/chicken/Yogjakarta/BBVet-IX/2004(H5N1)) Ki: 4.9 (nM), Ref: 20579892
IC50: 4.9 (nM), Ref: 19708637
IC50: 3.7 (nM), Ref:
TCMC1801
TCMT1161 Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1)) Ki: 7.9 (nM), Ref: 20579892
IC50: 10.8 (nM), Ref: 10.6019/CHEMBL1201861
TCMC1801
TCMT1163 Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1)) IC50: 0.3 (nM), Ref: 9322359
IC50: 0.2 (nM), Ref: Ki: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/swine/Belzig/2/2001(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/New Caledonia/20/1999(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Yamagata/32/1989(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC1801
TCMT1151 Neuraminidase Influenza B virus IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Hong Kong/1/1968(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1160 Neuraminidase Influenza A virus (A/Aichi/2/1968(H3N2)) IC50: 1.55 (nM), Ref: 20185316
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/whooper swan/Mongolia/1/2009(H5N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Wisconsin/67/2005(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Shandong/LY/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/Perth/16/2009(H3N2)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1151 Neuraminidase Influenza B virus (B/Memphis/3/89) IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Sandong/Li/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC2333
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 11 (nM), Ref: 9834179
TCMC962
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 10.2 (nM), Ref: 17503850
TCMC962
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 37 (nM), Ref: 20034711
TCMC962
TCMT1313 Human immunodeficiency virus 2 Human immunodeficiency virus type 2 (ISOLATE ROD) IC50: 37 (nM), Ref: 20034711
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850
TCMC1919
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 MIC: 10 (nM), Ref: 11311065
IC50: 50 (nM), Ref: 9834179
TCMC1919
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 MIC: 10 (nM), Ref: 11311065
TCMC1919
TCMT1250 Vesicular stomatitis virus Vesicular stomatitis virus IC50: 100 (nM), Ref: 9834179
TCMC1801
TCMT1296 Influenza A virus H3N2 Influenza A virus H3N2 IC50: 18.5 (nM), Ref: 12542349
TCMC1915
TCMT1285 Human coxsackievirus B3 Human coxsackievirus B3 IC50: 2.5 (nM), Ref: 13678412