TCM Putative Target References: TCMFx911


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC957
TCMT191 Signal transducer and activator of transcription 3 Homo sapiens IC50: 4600 (nM), Ref: 22650325
TCMC957
TCMT131 Acetylcholinesterase Homo sapiens Ki: 6410 (nM), Ref: 23286284
TCMC957
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 290 (nM), Ref: 23286284
Ki: 141 (nM), Ref: 23286284
TCMC957
TCMT211 Acyl coenzyme A:cholesterol acyltransferase Homo sapiens Ki: 544 (nM), Ref: 23286284
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1372
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2330 (nM), Ref: 22245047
TCMC1372
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 3630 (nM), Ref: 22245047
TCMC1107
TCMT290 Muscarinic acetylcholine receptor M5 Homo sapiens Ki: 0.14 (nM), Ref: 23707254
Ki: 0.3388 (nM), Ref: 24365159
Ki: 0.34 (nM), Ref: 24365159
Ki: 3.02 (nM), Ref: 25051097
TCMC1107
TCMT291 Muscarinic acetylcholine receptor M3 Homo sapiens Ki: 0.2692 (nM), Ref: 24365159
Ki: 0.27 (nM), Ref: 24365159
TCMC1107
TCMT292 Muscarinic acetylcholine receptor M1 Homo sapiens Ki: 0.2692 (nM), Ref: 24365159
Ki: 0.27 (nM), Ref: 24365159
TCMC1107
TCMT293 Muscarinic acetylcholine receptor M2 Homo sapiens Ki: 5.012 (nM), Ref: 25051097
Ki: 12.88 (nM), Ref: 25051097
Ki: 3.631 (nM), Ref: 25051097
Ki: 2.818 (nM), Ref: 25051097
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1957
TCMT34 Cytochrome P450 2D6 Homo sapiens Ki: 78 (nM), Ref: 26125082
TCMC602
TCMT302 HMG-CoA reductase Homo sapiens IC50: 5000 (nM), Ref: 10.1021/np50061a020
TCMC244
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 7900 (nM), Ref: 15916432
TCMC244
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 8300 (nM), Ref: 15658857
IC50: 8298.51 (nM), Ref: 19110342
TCMC820
TCMT187 Androgen Receptor Homo sapiens IC50: 5900 (nM), Ref: 23768907
TCMC2126
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 1410 (nM), Ref: 23286284
TCMC2126
TCMT171 Protein-tyrosine phosphatase 1C Homo sapiens IC50: 1970 (nM), Ref: 23957426
TCMC2126
TCMT233 Protein-tyrosine phosphatase 2C Homo sapiens IC50: 2570 (nM), Ref: 23957426
TCMC1180
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5210 (nM), Ref: 22487176
Ki: 5100 (nM), Ref: 22487176
TCMC1180
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9300 (nM), Ref: 22487176
Ki: 9200 (nM), Ref: 22487176
TCMC1180
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5540 (nM), Ref: 22487176
Ki: 5630 (nM), Ref: 22487176
TCMC1180
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 6590 (nM), Ref: 22487176
Ki: 6650 (nM), Ref: 22487176
TCMC2052
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9110 (nM), Ref: 22892213
TCMC2052
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8720 (nM), Ref: 22892213
TCMC2052
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 8430 (nM), Ref: 22892213
TCMC2052
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5930 (nM), Ref: 22892213
TCMC2052
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 780 (nM), Ref: 22892213
TCMC1806
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9600 (nM), Ref: 22137345
TCMC1806
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3660 (nM), Ref: 22137345
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC1364
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 4000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1364
TCMT308 Oxoeicosanoid receptor 1 Homo sapiens IC50: 2000 (nM), Ref: 24351031
TCMC1285
TCMT33 Cytochrome P450 3A4 Homo sapiens Ki: 399 (nM), Ref: 16248836
TCMC2188
TCMT223 Aldose reductase Homo sapiens IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC2079
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1490 (nM), Ref: 20674354
TCMC2079
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2510 (nM), Ref: 20674354
TCMC2079
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6430 (nM), Ref: 20674354
TCMC2079
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 8960 (nM), Ref: 20674354
TCMC2079
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20674354
TCMC2079
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4560 (nM), Ref: 20674354
TCMC2079
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 9700 (nM), Ref: 20674354
TCMC2079
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4710 (nM), Ref: 20674354
TCMC2079
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9050 (nM), Ref: 20674354
TCMC2079
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4820 (nM), Ref: 20674354
TCMC2079
TCMT87 Cytochrome P450 2C9 Homo sapiens Ki: 5000 (nM), Ref: 16248836
TCMC2079
TCMT278 Solute carrier organic anion transporter family member 1B1 Homo sapiens IC50: 9700 (nM), Ref: 23401473
TCMC2079
TCMT277 Solute carrier organic anion transporter family member 1B3 Homo sapiens IC50: 2700 (nM), Ref: 23401473
TCMC2079
TCMT276 Solute carrier organic anion transporter family member 2B1 Homo sapiens IC50: 4500 (nM), Ref: 23401473
TCMC1620
TCMT223 Aldose reductase Homo sapiens IC50: 88 (nM), Ref: 22236472
TCMC1620
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 130 (nM), Ref: 22236472
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC2025
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2025.72 (nM), Ref:
TCMC680
TCMT666 Transitional endoplasmic reticulum ATPase Homo sapiens IC50: 8984 (nM), Ref:
TCMC680
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 1634.07 (nM), Ref:
TCMC680
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7400 (nM), Ref: 25907369
Ki: 7800 (nM), Ref: 25907369
TCMC1413
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7370 (nM), Ref: 22892213
TCMC1413
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 5270 (nM), Ref: 22892213
TCMC1413
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4140 (nM), Ref: 22892213
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1506
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 101.2 (nM), Ref: 26498393
TCMC1506
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 268.3 (nM), Ref: 26498393
TCMC1506
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.8 (nM), Ref: 26498393
TCMC845
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 630 (nM), Ref: 19231207
TCMC1189
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9890 (nM), Ref: 22892213
TCMC1189
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7840 (nM), Ref: 22892213
TCMC1189
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5560 (nM), Ref: 22892213
TCMC1189
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 850 (nM), Ref: 22892213
TCMC837
TCMT690 Histone deacetylase 3 Homo sapiens IC50: 9000 (nM), Ref: 21874153
TCMC1594
TCMT197 Phosphodiesterase 4D Homo sapiens IC50: 2900 (nM), Ref: 22483586
IC50: 2910 (nM), Ref: 26473791
TCMC1594
TCMT698 Phosphodiesterase 4B Homo sapiens IC50: 4500 (nM), Ref: 22483586
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1567
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 890 (nM), Ref: 22668600
TCMC1567
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 960 (nM), Ref: 22668600
TCMC1567
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 790 (nM), Ref: 22668600
TCMC1567
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 810 (nM), Ref: 22668600
TCMC1567
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 580 (nM), Ref: 22668600
TCMC1567
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 710 (nM), Ref: 22668600
TCMC2025
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 5600 (nM), Ref: 23353736
TCMC2003
TCMT82 Estrogen receptor alpha Homo sapiens Ki: 785 (nM), Ref: 15634023
TCMC2003
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 2840 (nM), Ref: 16814546
IC50: 4120 (nM), Ref: 18063374
IC50: 625 (nM), Ref:
TCMC2003
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 996 (nM), Ref: 17604631
IC50: 750 (nM), Ref: 20527891
IC50: 996 (nM), Ref: 26850006
TCMC2003
TCMT329 Quinone reductase 2 Homo sapiens IC50: 960 (nM), Ref: 19265439
IC50: 450 (nM), Ref: 20036559
IC50: 450 (nM), Ref: 20356739
IC50: 960 (nM), Ref: 21261296
IC50: 6900 (nM), Ref: 23953689
Ki: 88 (nM), Ref: 23953689
IC50: 1400 (nM), Ref: 26854376
IC50: 913 (nM), Ref: 26854376
TCMC2003
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2210 (nM), Ref: 20674354
TCMC2003
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2770 (nM), Ref: 20674354
TCMC2003
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 9090 (nM), Ref: 20674354
TCMC2003
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4470 (nM), Ref: 20674354
TCMC2003
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4750 (nM), Ref: 20674354
TCMC2003
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4640 (nM), Ref: 20674354
TCMC2003
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8070 (nM), Ref: 20674354
TCMC2003
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4350 (nM), Ref: 20674354
TCMC2003
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 20674354
TCMC2003
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 950 (nM), Ref: 20674354
TCMC2003
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 4090 (nM), Ref: 20674354
TCMC2003
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 830 (nM), Ref: 20674354
TCMC2003
TCMT729 PI3-kinase p110-alpha subunit Homo sapiens IC50: 250 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT730 PI3-kinase p110-beta subunit Homo sapiens IC50: 500 (nM), Ref: 10.1039/C2MD20044A
TCMC2003
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4100 (nM), Ref: 27190601
IC50: 2600 (nM), Ref: 27190601
TCMC156
TCMT327 Vanilloid receptor Homo sapiens IC50: 35 (nM), Ref: 16000002
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC1568
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3580 (nM), Ref: 22658537
TCMC1568
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 610 (nM), Ref: 22658537
TCMC1568
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 2750 (nM), Ref: 22658537
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC2025
TCMT359 Tyrosine-protein kinase FYN Homo sapiens IC50: 1300 (nM), Ref: 17315853
IC50: 3600 (nM), Ref: 17315853
Ki: 7500 (nM), Ref: 17315853
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC910
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1118 (nM), Ref: 20696580
TCMC910
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 95 (nM), Ref: 20696580
TCMC910
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 20 (nM), Ref: 20696580
TCMC2048
TCMT771 Serine-protein kinase ATR Homo sapiens IC50: 7300 (nM), Ref: 22835870
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1201
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 3150 (nM), Ref: 8576921
TCMC1201
TCMT132 Butyrylcholinesterase Homo sapiens Ki: 6900 (nM), Ref: 19879672
TCMC1201
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1201
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 40 (nM), Ref: 20696580
TCMC1201
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1201
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1201
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 568.3 (nM), Ref: 26498393
TCMC1201
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 24.5 (nM), Ref: 26498393
TCMC1201
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 41.8 (nM), Ref: 26498393
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC2098
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1400 (nM), Ref: 20590092
TCMC2098
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1110 (nM), Ref: 20590092
TCMC2098
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 112 (nM), Ref: 20590092
TCMC2098
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 1220 (nM), Ref: 20590092
TCMC2098
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 1440 (nM), Ref: 20590092
TCMC2098
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 1410 (nM), Ref: 20590092
TCMC2098
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 1230 (nM), Ref: 20590092
TCMC2098
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 1370 (nM), Ref: 20590092
TCMC2098
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 1000 (nM), Ref: 20590092
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC614
TCMT151 Protein kinase C alpha Homo sapiens IC50: 9300 (nM), Ref: 9834166
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1886
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 670 (nM), Ref: 26498394
TCMC1886
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 770 (nM), Ref: 26498394
TCMC1886
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 620 (nM), Ref: 26498394
TCMC1886
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 810 (nM), Ref: 26498394
TCMC1886
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8470 (nM), Ref: 26498394
TCMC1886
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 720 (nM), Ref: 26498394
TCMC1597
TCMT807 Solute carrier family 22 member 12 Homo sapiens IC50: 2000 (nM), Ref: 17325024
Ki: 5740 (nM), Ref: 17325024
TCMC1597
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2927.18 (nM), Ref:
TCMC1597
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2988.26 (nM), Ref:
TCMC1597
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 1600 (nM), Ref: 24900447
TCMC1597
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 1600 (nM), Ref: 26322379
TCMC1597
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 4300 (nM), Ref: 26602279
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2128
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 3900 (nM), Ref: 23286284
TCMC1757
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 130 (nM), Ref: 17378609
IC50: 110 (nM), Ref: 19848434
IC50: 25 (nM), Ref: 21958737
IC50: 120 (nM), Ref: 21958738
TCMC1757
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 110 (nM), Ref: 12608855
IC50: 1100 (nM), Ref: 19848434
IC50: 5100 (nM), Ref: 21739938
IC50: 110 (nM), Ref: 24684213
TCMC1757
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens IC50: 180 (nM), Ref: 12608855
IC50: 5900 (nM), Ref: 19848434
IC50: 110 (nM), Ref: 21739938
TCMC1757
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 11 (nM), Ref: 20413308
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC1919
TCMT613 Glucocorticoid receptor Homo sapiens IC50: 14 (nM), Ref: 19364854
TCMC1153
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7700 (nM), Ref: 22668600
TCMC1153
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8600 (nM), Ref: 22668600
TCMC1153
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 22668600
TCMC1153
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8700 (nM), Ref: 22668600
TCMC1153
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4800 (nM), Ref: 22668600
TCMC1153
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 7900 (nM), Ref: 22668600
TCMC1587
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 83.7 (nM), Ref: 23286284
Ki: 40 (nM), Ref: 23286284
TCMC1587
TCMT211 Acyl coenzyme A:cholesterol acyltransferase Homo sapiens Ki: 2530 (nM), Ref: 23286284
TCMC1428
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 509 (nM), Ref: 20696580
TCMC1428
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 88 (nM), Ref: 20696580
TCMC1428
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1898
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 7906 (nM), Ref: 20696580
TCMC1898
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1679 (nM), Ref: 20696580
TCMC1898
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1491 (nM), Ref: 20696580
TCMC1898
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 900 (nM), Ref: 10.1039/C3MD00166K
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC1168
TCMT117 Kappa opioid receptor Homo sapiens Ki: 2515 (nM), Ref: 18166466
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC378
TCMT848 Serine/threonine-protein kinase/endoribonuclease IRE1 Homo sapiens IC50: 2370 (nM), Ref: IC50: 5750 (nM), Ref:
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC804
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 2000 (nM), Ref: 21561086
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC392
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 2400 (nM), Ref: 15658857
IC50: 2398.83 (nM), Ref: 19110342
TCMC1179
TCMT187 Androgen Receptor Homo sapiens IC50: 5900 (nM), Ref: 19592245
IC50: 5900 (nM), Ref: 19592245
TCMC1179
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8 (nM), Ref: 20413308
IC50: 10000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1179
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1890 (nM), Ref: 22487176
Ki: 1880 (nM), Ref: 22487176
TCMC1179
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8710 (nM), Ref: 22487176
Ki: 8800 (nM), Ref: 22487176
TCMC1179
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4130 (nM), Ref: 22487176
Ki: 4220 (nM), Ref: 22487176
TCMC1179
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7220 (nM), Ref: 22487176
Ki: 7330 (nM), Ref: 22487176
TCMC2127
TCMT223 Aldose reductase Homo sapiens IC50: 8690 (nM), Ref: 22261024
TCMC2127
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 5000 (nM), Ref: 22044621
IC50: 500 (nM), Ref: 22044621
TCMC1179
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 1380.38 (nM), Ref: 23574272
IC50: 1400 (nM), Ref: 23574272
TCMC2127
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 69.4 (nM), Ref: 23286284
Ki: 2450 (nM), Ref: 23286284
TCMC2127
TCMT211 Acyl coenzyme A:cholesterol acyltransferase Homo sapiens Ki: 6890 (nM), Ref: 23286284
TCMC2127
TCMT171 Protein-tyrosine phosphatase 1C Homo sapiens IC50: 2140 (nM), Ref: 23957426
TCMC2127
TCMT233 Protein-tyrosine phosphatase 2C Homo sapiens IC50: 2590 (nM), Ref: 23957426
TCMC1179
TCMT128 Tankyrase-2 Homo sapiens IC50: 147.91 (nM), Ref: 23574272
IC50: 140 (nM), Ref: 23574272
TCMC1179
TCMT129 Tankyrase-1 Homo sapiens IC50: 323.59 (nM), Ref: 23574272
IC50: 320 (nM), Ref: 23574272
IC50: 323.59 (nM), Ref: 24116873
IC50: 330 (nM), Ref: 24116873
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC1551
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 1900 (nM), Ref: 16248836
Ki: 1900 (nM), Ref: 16248836
Ki: 800 (nM), Ref: 16248836
Ki: 250 (nM), Ref: 22696418
TCMC1551
TCMT131 Acetylcholinesterase Homo sapiens IC50: 760 (nM), Ref: 23746477
TCMC1551
TCMT268 Cytochrome P450 2A13 Homo sapiens Ki: 40 (nM), Ref: 22696418
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC1892
TCMT508 Tyrosine-protein kinase SYK Homo sapiens IC50: 10000 (nM), Ref: 23917087
TCMC2201
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8700 (nM), Ref: 21332115
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1742
TCMT637 NAD-dependent deacetylase sirtuin 3 Homo sapiens IC50: 6200 (nM), Ref: 25275824
TCMC1742
TCMT638 NAD-dependent deacetylase sirtuin 2 Homo sapiens IC50: 6300 (nM), Ref: 25549554
IC50: 1200 (nM), Ref: 26696402
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC1175
TCMT186 Monoamine oxidase B Homo sapiens IC50: 2870 (nM), Ref: 20045650
TCMC1175
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 8000 (nM), Ref: 24345481
IC50: 8000 (nM), Ref: 26301554
TCMC2041
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9594.4 (nM), Ref: 26498393
TCMC2041
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 66.6 (nM), Ref: 26498393
TCMC2041
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 71.4 (nM), Ref: 26498393
TCMC2041
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 39.8 (nM), Ref: 26498393
TCMC1236
TCMT236 Estrogen receptor beta Homo sapiens IC50: 10 (nM), Ref: 15341953
IC50: 10 (nM), Ref: 15456246
IC50: 98.7 (nM), Ref: 15887952
IC50: 98.7 (nM), Ref: 15887952
IC50: 9.7 (nM), Ref: 15943471
IC50: 10 (nM), Ref: 16098741
IC50: 1.3 (nM), Ref: 16219463
IC50: 61 (nM), Ref: 16610787
IC50: 25 (nM), Ref: 17149865
IC50: 395 (nM), Ref: 17049855
IC50: 9.7 (nM), Ref: 17188490
IC50: 6.8 (nM), Ref: 17574424
IC50: 18 (nM), Ref: 12502307
IC50: 98.7 (nM), Ref:
TCMC1236
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 395 (nM), Ref: 15341953
IC50: 395 (nM), Ref: 15456246
IC50: 4660 (nM), Ref: 15887952
IC50: 4660 (nM), Ref: 15887952
IC50: 395 (nM), Ref: 15943471
IC50: 395 (nM), Ref: 16098741
IC50: 29.4 (nM), Ref: 16219463
IC50: 1973 (nM), Ref: 16610787
IC50: 1145 (nM), Ref: 17149865
IC50: 2150 (nM), Ref: 17696335
IC50: 9.7 (nM), Ref: 17049855
IC50: 395 (nM), Ref: 17188490
IC50: 580 (nM), Ref: 17574424
IC50: 300 (nM), Ref: 12502307
IC50: 4680 (nM), Ref:
TCMC1236
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 10 (nM), Ref: 17482813
TCMC1236
TCMT910 Estrogen-related receptor beta Homo sapiens IC50: 395 (nM), Ref: 17482813
TCMC1236
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 2210 (nM), Ref: 18533708
TCMC1236
TCMT344 Aldehyde oxidase Homo sapiens IC50: 340 (nM), Ref: 20853847
TCMC1236
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 7720 (nM), Ref:
TCMC950
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 75.7 (nM), Ref: 15887952
IC50: 75.7 (nM), Ref: 15887952
IC50: 75.7 (nM), Ref:
TCMC950
TCMT236 Estrogen receptor beta Homo sapiens IC50: 18.6 (nM), Ref: 15887952
IC50: 18.6 (nM), Ref: 15887952
IC50: 18.6 (nM), Ref:
TCMC1183
TCMT247 Alpha-2a adrenergic receptor Homo sapiens Ki: 6.31 (nM), Ref: 11262089
TCMC1183
TCMT307 HERG Homo sapiens IC50: 1513.56 (nM), Ref: 12873512
IC50: 1513.56 (nM), Ref: 18448342
IC50: 3100 (nM), Ref: 20637635
IC50: 457.09 (nM), Ref: 21185626
IC50: 10 (nM), Ref: 23919353
TCMC1183
TCMT633 Serotonin transporter Homo sapiens Ki: 48 (nM), Ref: 16220969
Ki: 0.72 (nM), Ref: 16162005
IC50: 39.4 (nM), Ref: 16854086
IC50: 16 (nM), Ref: 16750363
IC50: 16 (nM), Ref: 16750359
Ki: 2 (nM), Ref: 17107798
Ki: 2.2 (nM), Ref: 17616397
Ki: 2.2 (nM), Ref: 17127059
Ki: 2.2 (nM), Ref: 17307358
IC50: 47 (nM), Ref: 18667309
Ki: 1.1 (nM), Ref: 19014888
IC50: 7 (nM), Ref: 19014888
IC50: 47 (nM), Ref: 18550369
IC50: 9.4 (nM), Ref: 18557608
IC50: 39.4 (nM), Ref: 18834188
IC50: 10 (nM), Ref: 18771916
IC50: 10 (nM), Ref: 19329313
IC50: 9.4 (nM), Ref: 18951020
Ki: 1.1 (nM), Ref: 19256502
IC50: 7.3 (nM), Ref: 19256502
IC50: 9.4 (nM), Ref: 19722525
IC50: 9.4 (nM), Ref: 19713106
IC50: 9.4 (nM), Ref: 19632110
IC50: 2.5 (nM), Ref: 20034793
IC50: 9.4 (nM), Ref: 20131864
IC50: 9.4 (nM), Ref: 20378347
IC50: 9.4 (nM), Ref: 20462211
IC50: 3.1 (nM), Ref: 20724153
IC50: 5.2 (nM), Ref: 21093273
IC50: 5.012 (nM), Ref: 21310612
IC50: 9.4 (nM), Ref: 21916421
Ki: 98 (nM), Ref: 23602445
IC50: 281.84 (nM), Ref: 23602445
Ki: 1.4 (nM), Ref: 23403082
IC50: 8.6 (nM), Ref: 23403082
IC50: 7.2 (nM), Ref: 24012181
IC50: 150 (nM), Ref: 24974340
IC50: 150 (nM), Ref: 25221656
IC50: 4410 (nM), Ref: 25221656
TCMC1183
TCMT634 Norepinephrine transporter Homo sapiens Ki: 2000 (nM), Ref: 16220969
Ki: 440 (nM), Ref: 16162005
IC50: 5200 (nM), Ref: 16750363
IC50: 5200 (nM), Ref: 16750359
IC50: 2000 (nM), Ref: 18667309
Ki: 1560 (nM), Ref: 19014888
IC50: 1020 (nM), Ref: 19014888
IC50: 2000 (nM), Ref: 18550369
IC50: 563 (nM), Ref: 18771916
IC50: 563 (nM), Ref: 19329313
Ki: 1560 (nM), Ref: 19256502
IC50: 1020 (nM), Ref: 19256502
Ki: 1394 (nM), Ref: 23602445
IC50: 6309.57 (nM), Ref: 23602445
IC50: 4410 (nM), Ref: 24974340
TCMC1183
TCMT635 Dopamine transporter Homo sapiens Ki: 6000 (nM), Ref: 16220969
Ki: 1900 (nM), Ref: 16162005
IC50: 4400 (nM), Ref: 16750363
IC50: 4400 (nM), Ref: 16750359
IC50: 6000 (nM), Ref: 18667309
Ki: 6670 (nM), Ref: 19014888
IC50: 6000 (nM), Ref: 18550369
Ki: 6670 (nM), Ref: 19256502
Ki: 3764 (nM), Ref: 23602445
IC50: 9120.11 (nM), Ref: 23602445
TCMC1183
TCMT242 Histamine H3 receptor Homo sapiens Ki: 7300 (nM), Ref: 17107798
Ki: 7300 (nM), Ref: 17616397
Ki: 7300 (nM), Ref: 17127059
Ki: 7300 (nM), Ref: 17307358
TCMC1183
TCMT31 Cytochrome P450 2C19 Homo sapiens IC50: 40 (nM), Ref: 26355532
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC987
TCMT885 Lysine-specific demethylase 2A Homo sapiens Ki: 1970 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 22724510
IC50: 1500 (nM), Ref: 23964788
TCMC987
TCMT965 Lysine-specific demethylase 7 Homo sapiens IC50: 2100 (nM), Ref: 22724510
TCMC987
TCMT884 Histone lysine demethylase PHF8 Homo sapiens IC50: 550 (nM), Ref: 22724510
IC50: 550 (nM), Ref: 23964788
TCMC1922
TCMT634 Norepinephrine transporter Homo sapiens IC50: 6040 (nM), Ref: 17573162
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC1053
TCMT131 Acetylcholinesterase Homo sapiens Ki: 1950 (nM), Ref: 23286284
IC50: 1000 (nM), Ref: 24900610
Ki: 600 (nM), Ref: 24900610
TCMC1053
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 1830 (nM), Ref: 23286284
Ki: 118 (nM), Ref: 23286284
TCMC1053
TCMT211 Acyl coenzyme A:cholesterol acyltransferase Homo sapiens Ki: 398 (nM), Ref: 23286284
TCMC1053
TCMT171 Protein-tyrosine phosphatase 1C Homo sapiens IC50: 3670 (nM), Ref: 23957426
TCMC1053
TCMT233 Protein-tyrosine phosphatase 2C Homo sapiens IC50: 3940 (nM), Ref: 23957426
TCMC1961
TCMT206 Cytochrome P450 2A6 Homo sapiens Ki: 600 (nM), Ref: 16248836
TCMC1961
TCMT131 Acetylcholinesterase Homo sapiens IC50: 6480 (nM), Ref: 23746477
TCMC1174
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 850 (nM), Ref: 15689157
IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1174
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC2216
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3600 (nM), Ref: 17489632
IC50: 3100 (nM), Ref: 18798681
IC50: 3600 (nM), Ref: 19008110
IC50: 3600 (nM), Ref: 17125223
IC50: 3800 (nM), Ref: 19846295
IC50: 3900 (nM), Ref: 19632832
IC50: 3600 (nM), Ref: 19836230
IC50: 3100 (nM), Ref: 21555221
IC50: 3600 (nM), Ref: 21571537
IC50: 3100 (nM), Ref: 22940448
IC50: 2300 (nM), Ref: 21453996
Ki: 3400 (nM), Ref: 21453996
IC50: 3600 (nM), Ref: 23022281
IC50: 3080 (nM), Ref: 23141910
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3080 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2750 (nM), Ref: 23387824
IC50: 4120 (nM), Ref: 24224843
IC50: 4000 (nM), Ref: 24953600
IC50: 3500 (nM), Ref: 25559759
IC50: 3400 (nM), Ref: 25907369
Ki: 6400 (nM), Ref: 25907369
IC50: 5200 (nM), Ref: 26841168
TCMC2216
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 1900 (nM), Ref: 20100662
TCMC2216
TCMT102 Low molecular weight phosphotyrosine protein phosphatase Homo sapiens IC50: 7200 (nM), Ref: 21453996
TCMC2216
TCMT103 Receptor-type tyrosine-protein phosphatase F (LAR) Homo sapiens IC50: 3800 (nM), Ref: 21453996
TCMC2216
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 21561086
Ki: 3700 (nM), Ref: 21561086
Ki: 2100 (nM), Ref: 21561086
Ki: 2800 (nM), Ref: 21561086
Ki: 2000 (nM), Ref: 21561086
IC50: 4000 (nM), Ref: 21561086
TCMC2216
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 2400 (nM), Ref: 23387824
TCMC2216
TCMT150 Nuclear receptor ROR-gamma Homo sapiens IC50: 680 (nM), Ref: 10.1039/C3MD00005B
IC50: 130 (nM), Ref: 24704616
IC50: 1060 (nM), Ref: 24704616
IC50: 9410 (nM), Ref: 24704616
TCMC2180
TCMT302 HMG-CoA reductase Homo sapiens IC50: 5860 (nM), Ref: 25311563
IC50: 36.31 (nM), Ref: 25311563
TCMC1403
TCMT223 Aldose reductase Homo sapiens IC50: 1910 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC1834
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9060 (nM), Ref: 21402476
TCMC1834
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8030 (nM), Ref: 21402476
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755
TCMC1378
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 8960 (nM), Ref: 22658537
TCMC1378
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 8220 (nM), Ref: 22658537

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1620
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 0.66 (ug/ml), Ref: 11430019
IC50: 5.9 (ug/ml), Ref: 16643034
TCMC2177
TCMT1120 Cell division protein ftsZ Staphylococcus aureus MIC: 4 (ug/ml), Ref: 25791674
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2257
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 15.46 (ug/ml), Ref: 20116898
TCMC2264
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 13.01 (ug/ml), Ref: 22552195
IC50: 11.54 (ug/ml), Ref: 22552195
IC50: 22.45 (ug/ml), Ref: 22552195
IC50: 23.54 (ug/ml), Ref: 22552195
TCMC2264
TCMT1136 Neuraminidase Influenza A virus IC50: 13.01 (ug/ml), Ref: 22552195
IC50: 11.54 (ug/ml), Ref: 22552195
IC50: 22.45 (ug/ml), Ref: 22552195
IC50: 23.54 (ug/ml), Ref: 22552195
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC2233
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.85 (ug/ml), Ref: 20116898
TCMC2277
TCMT1136 Neuraminidase influenza A virus IC50: 89.81 (ug/ml), Ref: 26774928
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC1236
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.84 (ug/ml), Ref: 20116898
TCMC2305
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 12.8 (ug/ml), Ref: 22552195
IC50: 9.33 (ug/ml), Ref: 22552195
IC50: 25.59 (ug/ml), Ref: 22552195
IC50: 28.42 (ug/ml), Ref: 22552195
TCMC2305
TCMT1136 Neuraminidase Influenza A virus IC50: 12.8 (ug/ml), Ref: 22552195
IC50: 9.33 (ug/ml), Ref: 22552195
IC50: 25.59 (ug/ml), Ref: 22552195
IC50: 28.42 (ug/ml), Ref: 22552195
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2313
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2313
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC1793
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
TCMC1793
TCMT1251 Candida albicans Candida albicans MIC: 12.5 (ug/ml), Ref: 9392889
TCMC1793
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 61.5 (ug/ml), Ref: 20218656
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC2325
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 71.7 (ug/ml), Ref: 15104496
TCMC2325
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 53.8 (ug/ml), Ref: 15104496
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2329
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 25.3 (ug/ml), Ref: 8946749
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC1957
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.13 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1395
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 23369537
TCMC2351
TCMT1190 Plasmodium falciparum (isolate FcB1 / Columbia) Plasmodium falciparum FcB1/Columbia IC50: 16.7 (ug/ml), Ref: 21985060
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC2363
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 22537683
TCMC2366
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.8 (ug/ml), Ref: 17845001
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC2395
TCMT1292 Japanese encephalitis virus Japanese encephalitis virus IC50: 0.022 (ug/ml), Ref: 1336040
TCMC2395
TCMT1336 Yellow fever virus Yellow fever virus IC50: 0.016 (ug/ml), Ref: 1336040
TCMC2395
TCMT1337 Dengue virus type 4 Dengue virus 4 IC50: 0.063 (ug/ml), Ref: 1336040
TCMC2395
TCMT1338 Rift Valley fever virus Rift Valley fever virus IC50: 0.16 (ug/ml), Ref: 1336040
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC2404
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 100 (ug/ml), Ref: 18710283
MIC: 28 (ug/ml), Ref: 22280816
TCMC2079
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 11170636
TCMC2411
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 16 (ug/ml), Ref: 11141098
TCMC2411
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 64 (ug/ml), Ref: 12608857
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC1322
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC2177
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 1.56 (ug/ml), Ref: 1453180
MIC: 0.6 (ug/ml), Ref: 25791674
TCMC2177
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1.56 (ug/ml), Ref: 1453180
MIC: 0.78 (ug/ml), Ref: 1453180
MIC: 2.5 (ug/ml), Ref: 17664318
MIC: 1.25 (ug/ml), Ref: 17664318
MIC: 16 (ug/ml), Ref: 17664318
MIC: 2 (ug/ml), Ref: 17664318
MIC: 1.5 (ug/ml), Ref: 25791674
TCMC2177
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 0.78 (ug/ml), Ref: 1453180
TCMC2177
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 16 (ug/ml), Ref: 25791674
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC2257
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 15.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 37.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 59.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC845
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 1522419
MIC: 6.25 (ug/ml), Ref: 1522419
TCMC845
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 25 (ug/ml), Ref: 1522419
MIC: 1.57 (ug/ml), Ref: 1522419
TCMC1594
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 25461329
TCMC1594
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 25461329
MIC: 12.5 (ug/ml), Ref: 25461329
TCMC1594
TCMT1246 Escherichia coli Escherichia coli MIC: 78 (ug/ml), Ref: 25461329
TCMC1594
TCMT1289 Shigella dysenteriae Shigella dysenteriae MIC: 78 (ug/ml), Ref: 25461329
TCMC1594
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 78 (ug/ml), Ref: 25461329
TCMC2003
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1251 Candida albicans Candida albicans MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1246 Escherichia coli Escherichia coli MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 0 (ug/ml), Ref: 12036362
TCMC2003
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12036362
TCMC2003
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
TCMC2003
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 25 (ug/ml), Ref: 20022753
TCMC2472
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 23792320
TCMC2472
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 25 (ug/ml), Ref: 23792320
TCMC2472
TCMT1286 Bacillus cereus Bacillus cereus MIC: 12.5 (ug/ml), Ref: 23792320
TCMC2472
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 12.5 (ug/ml), Ref: 23792320
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2477
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 72.5 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2481
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 12.5 (ug/ml), Ref: 17027268
TCMC2482
TCMT1246 Escherichia coli Escherichia coli MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2482
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 3.1 (ug/ml), Ref: 9392889
TCMC2482
TCMT1251 Candida albicans Candida albicans MIC: 6.25 (ug/ml), Ref: 9392889
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC2487
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 11.4 (ug/ml), Ref: 23294378
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC887
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 62.5 (ug/ml), Ref: 10395496
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1515
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1767
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 60 (ug/ml), Ref: 20384293
TCMC1767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0419-x
TCMC614
TCMT1454 Bacillus subtilis Bacillus subtilis IC50: 98.5 (ug/ml), Ref: 25981688
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC1186
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 3430167
TCMC1186
TCMT1284 Penicillium expansum Penicillium expansum MIC: 50 (ug/ml), Ref: 3430167
TCMC2528
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 50 (ug/ml), Ref: 20476748
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC1572
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC319
TCMT1286 Bacillus cereus Bacillus cereus MIC: 46.9 (ug/ml), Ref: 22014830
TCMC319
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 22014830
TCMC319
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 31.3 (ug/ml), Ref: 22014830
TCMC319
TCMT1251 Candida albicans Candida albicans MIC: 31.3 (ug/ml), Ref: 22014830
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC2578
TCMT1251 Candida albicans Candida albicans IC50: 82.98 (ug/ml), Ref: 25686593
TCMC2182
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 12.5 (ug/ml), Ref: 22280816
TCMC2581
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1428
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1428
TCMT1286 Bacillus cereus Bacillus cereus MIC: 25 (ug/ml), Ref: 12762812
TCMC1428
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 32.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 26 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1898
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 12.5 (ug/ml), Ref: 22280816
TCMC1898
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 80.76 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1898
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 73 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 63.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1168
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 9392889
MIC: 2.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 9392889
TCMC1168
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
MIC: 25 (ug/ml), Ref: 10217726
TCMC1168
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 6.25 (ug/ml), Ref: 9392889
MIC: 12.5 (ug/ml), Ref: 10217726
TCMC1168
TCMT1251 Candida albicans Candida albicans MIC: 25 (ug/ml), Ref: 9392889
TCMC1168
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.2 (ug/ml), Ref: 20218656
TCMC2603
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 7714539
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC804
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 25 (ug/ml), Ref: 22280816
TCMC804
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 32 (ug/ml), Ref: 15387646
MIC: 62 (ug/ml), Ref: 23356207
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1033
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10924184
TCMC1033
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 30 (ug/ml), Ref: 18564877
TCMC54
TCMT1246 Escherichia coli Escherichia coli MIC: 64 (ug/ml), Ref: 23994872
TCMC54
TCMT1172 Staphylococcus aureus subsp. aureus RN4220 Staphylococcus aureus subsp. aureus RN4220 MIC: 16 (ug/ml), Ref: 23994872
TCMC54
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 23994872
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2655
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 IC50: 7 (ug/ml), Ref: 2828553
TCMC2655
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 IC50: 7 (ug/ml), Ref: 2828553
TCMC2025
TCMT1218 Staphylococcus aureus Staphylococcus aureus MBC: 0.12 (ug/ml), Ref: 18004816
TCMC2667
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 15104489
MIC: 100 (ug/ml), Ref: 20542692
TCMC1551
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 20832915
TCMC2025
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MBC: 0.12 (ug/ml), Ref: 18004816
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC2025
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MBC: 0.12 (ug/ml), Ref: 18004816
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1733
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.2 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1892
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC1892
TCMT1182 Streptococcus sanguinis Streptococcus sanguinis MIC: 50 (ug/ml), Ref: 20022753
MBC: 100 (ug/ml), Ref: 20022753
TCMC2025
TCMT1246 Escherichia coli Escherichia coli MBC: 0.12 (ug/ml), Ref: 18004816
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC2688
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 14969530
TCMC2688
TCMT1282 Colletotrichum orbiculare Colletotrichum orbiculare MIC: 30 (ug/ml), Ref: 14969530
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC1236
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (ug/ml), Ref: 19299148
TCMC2714
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 1.4 (ug/ml), Ref: 22280816
TCMC2714
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25.3 (ug/ml), Ref: 22280816
TCMC1183
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 18061311
TCMC1183
TCMT1168 Trichomonas vaginalis Trichomonas vaginalis MIC: 28 (ug/ml), Ref: 18061311
TCMC1183
TCMT1251 Candida albicans Candida albicans MIC: 50 (ug/ml), Ref: 18061311
TCMC1183
TCMT1243 Aspergillus flavus Aspergillus flavus MIC: 6.25 (ug/ml), Ref: 21194811
TCMC1183
TCMT1405 Penicillium citrinum Penicillium citrinum MIC: 6.25 (ug/ml), Ref: 21194811
TCMC582
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 16680159
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC582
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 1602301
TCMC582
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 24927000
MIC: 62.5 (ug/ml), Ref: 24927000
TCMC582
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 24927000
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1961
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 6.25 (ug/ml), Ref: 20832915
TCMC1174
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 55 (ug/ml), Ref: 25564380
TCMC1174
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.6 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2216
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 6.5 (ug/ml), Ref: 9748372
TCMC2216
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 32 (ug/ml), Ref: 15387646
MIC: 100 (ug/ml), Ref: 20542692
TCMC2216
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1403
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1246 Escherichia coli Escherichia coli MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC1403
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC2821
TCMT1251 Candida albicans Candida albicans MIC: 1.56 (ug/ml), Ref: 7760078
MFC: 3.12 (ug/ml), Ref: 7760078
MFC: 6.25 (ug/ml), Ref: 7760078
MIC: 3.125 (ug/ml), Ref: 10346966
MFC: 6.25 (ug/ml), Ref: 10346966
MIC: 6.25 (ug/ml), Ref: 18611050
MIC: 6.25 (ug/ml), Ref: 21131198
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC2333
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 11 (nM), Ref: 9834179
TCMC791
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 12.7 (nM), Ref: 17503850
TCMC1919
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 MIC: 10 (nM), Ref: 11311065
IC50: 50 (nM), Ref: 9834179
TCMC1919
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 MIC: 10 (nM), Ref: 11311065
TCMC1919
TCMT1250 Vesicular stomatitis virus Vesicular stomatitis virus IC50: 100 (nM), Ref: 9834179
TCMC2605
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 8.8 (nM), Ref: 17503850
TCMC1179
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (nM), Ref: 19097788