Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 6000 (nM), Ref: 15689157 IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 2600 (nM), Ref: 15267241 IC50: 1 (nM), Ref: 20413308 IC50: 800 (nM), Ref: 10.1039/C3MD00166K IC50: 500 (nM), Ref: 26301554 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8500 (nM), Ref: 18165015 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
IC50: 670 (nM), Ref: 19097799 Ki: 110 (nM), Ref: 19097799 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 153 (nM), Ref: 20696580 IC50: 1290 (nM), Ref: 23600958 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 84 (nM), Ref: 20696580 IC50: 54 (nM), Ref: 20832301 IC50: 570 (nM), Ref: 23600958 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 24 (nM), Ref: 20696580 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 5225 (nM), Ref: 20832301 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 5490 (nM), Ref: 22487176 Ki: 5420 (nM), Ref: 22487176 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 4380 (nM), Ref: 22487176 Ki: 4310 (nM), Ref: 22487176 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 2650 (nM), Ref: 22487176 Ki: 2710 (nM), Ref: 22487176 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8960 (nM), Ref: 22487176 Ki: 9070 (nM), Ref: 22487176 Ki: 34.7 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 537.75 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 171.41 (nM), Ref: 26498393 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 4630 (nM), Ref: 15270556 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 5405 (nM), Ref: |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2940 (nM), Ref: 19231207 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 4000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT308 | Oxoeicosanoid receptor 1 | Homo sapiens |
IC50: 2000 (nM), Ref: 24351031 |
|
TCMT107 | Glutamate receptor ionotropic kainate 2 | Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
|
TCMT108 | Glutamate receptor ionotropic, AMPA 1 | Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
|
TCMT109 | Glutamate receptor ionotropic, AMPA 2 | Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
|
TCMT110 | Glutamate receptor ionotropic, AMPA 4 | Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
|
TCMT111 | Glutamate receptor ionotropic kainate 5 | Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
|
TCMT660 | Metabotropic glutamate receptor 8 | Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
|
TCMT653 | Metabotropic glutamate receptor 1 | Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT654 | Metabotropic glutamate receptor 5 | Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT657 | Metabotropic glutamate receptor 4 | Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT655 | Metabotropic glutamate receptor 2 | Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT664 | Excitatory amino acid transporter 3 | Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
|
TCMT656 | Metabotropic glutamate receptor 3 | Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
IC50: 140 (nM), Ref: 17994679 IC50: 140 (nM), Ref: 18029181 Ki: 50 (nM), Ref: 18665582 IC50: 150 (nM), Ref: 18752940 IC50: 140 (nM), Ref: 19307116 IC50: 130 (nM), Ref: 18760600 IC50: 140 (nM), Ref: 19309152 IC50: 140 (nM), Ref: 19592242 IC50: 140 (nM), Ref: 19592242 Ki: 82 (nM), Ref: 20184326 Ki: 104 (nM), Ref: 20184326 IC50: 140 (nM), Ref: 20444602 IC50: 140 (nM), Ref: 20615702 IC50: 249 (nM), Ref: 25737085 |
|
TCMT594 | Platelet activating factor receptor | Homo sapiens |
Ki: 1000 (nM), Ref: 1404229 |
|
TCMT318 | Putative hexokinase HKDC1 | Homo sapiens | IC50: 4320 (nM), Ref: |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT174 | 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens |
IC50: 11.78 (nM), Ref: 18242087 IC50: 13 (nM), Ref: 18653260 IC50: 778 (nM), Ref: 20851614 IC50: 778 (nM), Ref: 21376605 IC50: 8.6 (nM), Ref: 21873057 IC50: 29.1 (nM), Ref: 23747808 IC50: 29.1 (nM), Ref: 25590374 |
|
TCMT209 | 11-beta-hydroxysteroid dehydrogenase 2 | Homo sapiens |
IC50: 257 (nM), Ref: 20851614 IC50: 257 (nM), Ref: 21376605 IC50: 1.22 (nM), Ref: 23747808 IC50: 1.2 (nM), Ref: 25590374 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4900 (nM), Ref: 21561086 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 509 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 88 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8700 (nM), Ref: 21332115 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT302 | HMG-CoA reductase | Homo sapiens |
IC50: 5860 (nM), Ref: 25311563 IC50: 36.31 (nM), Ref: 25311563 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |