Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 8710 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4050 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
Ki: 3000 (nM), Ref: 18565755 IC50: 2600 (nM), Ref: 18565755 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
Ki: 78 (nM), Ref: 26125082 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 6.9 (nM), Ref: 19027293 Ki: 3.9 (nM), Ref: 20055417 |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 180 (nM), Ref: 19027293 Ki: 49 (nM), Ref: 20055417 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 3 (nM), Ref: 19027293 Ki: 2.2 (nM), Ref: 20055417 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 3400 (nM), Ref: 11678652 |
|
TCMT37 | Serotonin 2a (5-HT2a) receptor | Homo sapiens |
Ki: 966 (nM), Ref: 25695425 |
|
TCMT160 | Serotonin 7 (5-HT7) receptor | Homo sapiens |
Ki: 43 (nM), Ref: 25695425 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 171 (nM), Ref: 25695425 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
Ki: 3900 (nM), Ref: 18565755 IC50: 8400 (nM), Ref: 18565755 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 260 (nM), Ref: 22439881 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 9.5 (nM), Ref: 22439881 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2700 (nM), Ref: 17378609 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 1050 (nM), Ref: 18533708 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 360 (nM), Ref: 18533708 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 9700 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 716 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 632 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 47 (nM), Ref: 20696580 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 10000 (nM), Ref: 22261024 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 2320 (nM), Ref: 23411073 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 9640 (nM), Ref: 23656512 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 10000 (nM), Ref: 26322379 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9525.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 25 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 145.9 (nM), Ref: 26498393 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 1000 (nM), Ref: 26841168 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 286 (nM), Ref: 17616524 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8900 (nM), Ref: 19911821 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 48 (nM), Ref: 19911821 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9100 (nM), Ref: 19911821 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3300 (nM), Ref: 19911821 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 2000 (nM), Ref: 19911821 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 5200 (nM), Ref: 19911821 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9400 (nM), Ref: 19911821 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 6800 (nM), Ref: 19911821 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 5600 (nM), Ref: 19911821 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3100 (nM), Ref: 19911821 Ki: 3100 (nM), Ref: 21067924 Ki: 3100 (nM), Ref: 22137345 Ki: 3100 (nM), Ref: 22077347 Ki: 3100 (nM), Ref: 22365761 Ki: 3100 (nM), Ref: 22377674 Ki: 3100 (nM), Ref: 23241068 Ki: 3100 (nM), Ref: 22892213 Ki: 3100 (nM), Ref: 26688270 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 9200 (nM), Ref: 21067924 Ki: 9200 (nM), Ref: 22137345 Ki: 9200 (nM), Ref: 22077347 Ki: 9200 (nM), Ref: 22365761 Ki: 9200 (nM), Ref: 22377674 Ki: 9200 (nM), Ref: 23241068 Ki: 9200 (nM), Ref: 22892213 Ki: 9200 (nM), Ref: 26688270 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3900 (nM), Ref: 16580200 IC50: 7600 (nM), Ref: 18798681 IC50: 4200 (nM), Ref: 19702283 IC50: 3840 (nM), Ref: 22044245 IC50: 5600 (nM), Ref: 22690646 IC50: 9500 (nM), Ref: 21453996 Ki: 6000 (nM), Ref: 21453996 IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5 IC50: 2600 (nM), Ref: 23357636 IC50: 1100 (nM), Ref: 23434422 IC50: 3020 (nM), Ref: 23942421 IC50: 2010 (nM), Ref: 24090912 IC50: 1900 (nM), Ref: 24684845 IC50: 3020 (nM), Ref: 25497963 IC50: 9500 (nM), Ref: 25264584 Ki: 6000 (nM), Ref: 25264584 IC50: 1030 (nM), Ref: 25595683 IC50: 1170 (nM), Ref: 25600405 IC50: 3020 (nM), Ref: 25872983 IC50: 1000 (nM), Ref: 26083682 IC50: 1536 (nM), Ref: 26100442 IC50: 700 (nM), Ref: 26115570 IC50: 700 (nM), Ref: 26253631 IC50: 1536 (nM), Ref: 26481657 IC50: 730 (nM), Ref: 26711144 IC50: 3020 (nM), Ref: 26774579 IC50: 1536 (nM), Ref: 27123900 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 4000 (nM), Ref: 21561086 Ki: 3560 (nM), Ref: 21561086 Ki: 660 (nM), Ref: 21561086 Ki: 940 (nM), Ref: 21561086 Ki: 160 (nM), Ref: 21561086 Ki: 72 (nM), Ref: 21561086 IC50: 90 (nM), Ref: 21561086 |
|
TCMT190 | T-cell protein-tyrosine phosphatase | Homo sapiens |
IC50: 4230 (nM), Ref: 24684845 IC50: 4440 (nM), Ref: 25497963 IC50: 5460 (nM), Ref: 26100442 IC50: 5460 (nM), Ref: 26481657 IC50: 5460 (nM), Ref: 27123900 |
|
TCMT563 | Dual specificity phosphatase Cdc25B | Homo sapiens |
IC50: 980 (nM), Ref: 25497963 |
|
TCMT615 | Sentrin-specific protease 8 | Homo sapiens | IC50: 2470 (nM), Ref: |
|
TCMT616 | Sentrin-specific protease 7 | Homo sapiens | IC50: 1670 (nM), Ref: |
|
TCMT617 | Sentrin-specific protease 6 | Homo sapiens | IC50: 805 (nM), Ref: |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2100 (nM), Ref: 18042388 IC50: 340 (nM), Ref: 18778944 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 320 (nM), Ref: 22261024 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 150 (nM), Ref: 18165015 IC50: 2000 (nM), Ref: 22261024 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 4500 (nM), Ref: 22261024 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 75.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3.8 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 7400 (nM), Ref: 17616524 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 43 (nM), Ref: 16302800 IC50: 500 (nM), Ref: 24328302 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 790 (nM), Ref: 17378609 IC50: 4000 (nM), Ref: 24368208 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2200 (nM), Ref: 18165015 IC50: 14.8 (nM), Ref: 18976928 IC50: 2200 (nM), Ref: 22261024 IC50: 2900 (nM), Ref: 25152999 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 3200 (nM), Ref: 18258440 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 1540 (nM), Ref: 18533708 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7890 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8100 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2540 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2680 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6170 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4840 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7000 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9390 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 5410 (nM), Ref: 20185318 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 12 (nM), Ref: 20413308 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 4097 (nM), Ref: 20696580 IC50: 1550 (nM), Ref: 22328583 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1191 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 6680 (nM), Ref: 22658537 |
|
TCMT320 | Matrix metalloproteinase 3 | Homo sapiens |
IC50: 5570 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 1610 (nM), Ref: 22658537 |
|
TCMT322 | Matrix metalloproteinase 13 | Homo sapiens |
IC50: 8460 (nM), Ref: 22658537 |
|
TCMT422 | CaM kinase II beta | Homo sapiens |
IC50: 3000 (nM), Ref: 21798748 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y IC50: 6500 (nM), Ref: 26003344 |
|
TCMT784 | Vasopressin V2 receptor | Homo sapiens |
IC50: 7000 (nM), Ref: 23437772 IC50: 6309.57 (nM), Ref: 23437772 |
|
TCMT785 | Interleukin-8 receptor A | Homo sapiens |
IC50: 4500 (nM), Ref: 23437772 IC50: 5011.87 (nM), Ref: 23437772 |
|
TCMT786 | C-C chemokine receptor type 4 | Homo sapiens |
IC50: 10000 (nM), Ref: 23437772 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 590 (nM), Ref: 23411073 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 22 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 214 (nM), Ref: 23332346 |
|
TCMT601 | Thrombin | Homo sapiens |
IC50: 1500 (nM), Ref: 24610996 |
|
TCMT789 | Phosphodiesterase 3A | Homo sapiens |
Ki: 279 (nM), Ref: 17228859 |
|
TCMT790 | Phosphodiesterase 3B | Homo sapiens |
Ki: 417 (nM), Ref: 17228859 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 280 (nM), Ref: 24328302 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 120 (nM), Ref: 24328302 |
|
TCMT791 | Protein kinase N1 | Homo sapiens |
IC50: 5800 (nM), Ref: 24328302 |
|
TCMT792 | Phosphodiesterase 10A | Homo sapiens |
IC50: 56.9 (nM), Ref: 20450197 IC50: 76 (nM), Ref: 20450197 IC50: 17 (nM), Ref: 21087867 IC50: 21 (nM), Ref: 21705115 IC50: 36 (nM), Ref: 22321214 IC50: 210 (nM), Ref: 23978358 IC50: 36 (nM), Ref: 24721831 IC50: 36 (nM), Ref: 25592707 IC50: 92.3 (nM), Ref: 10.1039/C5MD00419E |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 5750 (nM), Ref: 24328302 |
|
TCMT462 | Serine/threonine-protein kinase NEK6 | Homo sapiens |
IC50: 4230 (nM), Ref: 24328302 |
|
TCMT445 | Serine/threonine-protein kinase NEK2 | Homo sapiens |
IC50: 5730 (nM), Ref: 24328302 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 24328302 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 300 (nM), Ref: 24328302 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 1200 (nM), Ref: 24328302 |
|
TCMT307 | HERG | Homo sapiens |
IC50: 7244.36 (nM), Ref: 21185626 |
|
TCMT388 | Tyrosine-protein kinase receptor UFO | Homo sapiens |
IC50: 960 (nM), Ref: 24328302 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 910 (nM), Ref: 24328302 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 5090 (nM), Ref: 24328302 |
|
TCMT402 | ALK tyrosine kinase receptor | Homo sapiens |
IC50: 3320 (nM), Ref: 24328302 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 5390 (nM), Ref: 24328302 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 280 (nM), Ref: 25060641 IC50: 3500 (nM), Ref: 27162124 |
|
TCMT793 | Liver glycogen phosphorylase | Homo sapiens |
IC50: 4800 (nM), Ref: 25092521 |
|
TCMT33 | Cytochrome P450 3A4 | Homo sapiens |
IC50: 2110 (nM), Ref: 22328583 |
|
TCMT217 | Cytochrome P450 2C8 | Homo sapiens |
IC50: 1390 (nM), Ref: 22328583 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 8900 (nM), Ref: 26322379 |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 41 (nM), Ref: 10741545 Ki: 33 (nM), Ref: 14643346 Ki: 33 (nM), Ref: 17149859 Ki: 33 (nM), Ref: 17149858 Ki: 76 (nM), Ref: 17407276 IC50: 138 (nM), Ref: 17388627 IC50: 138 (nM), Ref: 17451272 IC50: 138 (nM), Ref: 18039010 Ki: 33 (nM), Ref: 18313920 Ki: 120 (nM), Ref: 19027293 IC50: 138 (nM), Ref: 16989522 Ki: 51 (nM), Ref: 20055417 Ki: 38 (nM), Ref: 21482470 Ki: 21.38 (nM), Ref: 19527931 Ki: 103 (nM), Ref: 25062506 Ki: 1516 (nM), Ref: 25268943 Ki: 30 (nM), Ref: 26035635 Ki: 103 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 1.2 (nM), Ref: 10741545 Ki: 9.2 (nM), Ref: 17149859 Ki: 9.2 (nM), Ref: 17149858 Ki: 1.1 (nM), Ref: 17407276 IC50: 320 (nM), Ref: 17407276 Ki: 9.2 (nM), Ref: 18313920 Ki: 1.2 (nM), Ref: 19027293 Ki: 3 (nM), Ref: 20055417 Ki: 14.7 (nM), Ref: 20441176 Ki: 0.25 (nM), Ref: 21482470 Ki: 4.467 (nM), Ref: 19527931 Ki: 362 (nM), Ref: 25268943 Ki: 15 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
IC50: 7.3 (nM), Ref: 14643346 Ki: 3.7 (nM), Ref: 17149859 IC50: 7.3 (nM), Ref: 17149859 Ki: 3.7 (nM), Ref: 17149858 IC50: 7.3 (nM), Ref: 17149858 Ki: 0.79 (nM), Ref: 17407276 IC50: 23 (nM), Ref: 17407276 Ki: 3.7 (nM), Ref: 18313920 IC50: 7.3 (nM), Ref: 18313920 Ki: 0.66 (nM), Ref: 19027293 Ki: 0.98 (nM), Ref: 20055417 Ki: 0.23 (nM), Ref: 21482470 Ki: 0.5623 (nM), Ref: 19527931 IC50: 1.87 (nM), Ref: 24171469 Ki: 2.3 (nM), Ref: 25062506 Ki: 354 (nM), Ref: 25268943 Ki: 1.148 (nM), Ref: 26632862 Ki: 1.259 (nM), Ref: 26632862 Ki: 2.3 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.6 (nM), Ref: 16250647 |
|
TCMT309 | Solute carrier family 22 member 2 | Homo sapiens |
IC50: 2600 (nM), Ref: 23241029 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 105 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 6.6 (nM), Ref: 23332346 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 459 (nM), Ref: 17616524 |
|
TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT238 | Sodium/glucose cotransporter 2 | Homo sapiens |
IC50: 4100 (nM), Ref: 17374486 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
Ki: 1100 (nM), Ref: 18565755 IC50: 5200 (nM), Ref: 18565755 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 4410 (nM), Ref: 15658857 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 3.96 (nM), Ref: 12372519 Ki: 0.88 (nM), Ref: 16392810 Ki: 1.1 (nM), Ref: 16913723 Ki: 1.1 (nM), Ref: 17887741 Ki: 4 (nM), Ref: 17616524 Ki: 2.55 (nM), Ref: 19627147 Ki: 2.55 (nM), Ref: 21684752 Ki: 2.6 (nM), Ref: 21570305 Ki: 2.6 (nM), Ref: 22341895 Ki: 2.2 (nM), Ref: 24900459 Ki: 0.88 (nM), Ref: 22439881 IC50: 4.3 (nM), Ref: 22995061 Ki: 2.6 (nM), Ref: 23618710 Ki: 2.6 (nM), Ref: 23880358 IC50: 2.5 (nM), Ref: 24171469 Ki: 5.2 (nM), Ref: 25062506 Ki: 2.6 (nM), Ref: 25599950 Ki: 22 (nM), Ref: 25494650 IC50: 6.3 (nM), Ref: 26789491 Ki: 0.53 (nM), Ref: 26390077 Ki: 5.2 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 140 (nM), Ref: 16392810 Ki: 140 (nM), Ref: 16913723 Ki: 140 (nM), Ref: 17887741 Ki: 605 (nM), Ref: 22341895 Ki: 140 (nM), Ref: 22439881 Ki: 605 (nM), Ref: 23618710 Ki: 605 (nM), Ref: 23880358 Ki: 605 (nM), Ref: 25599950 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 24 (nM), Ref: 16392810 Ki: 46.9 (nM), Ref: 16913723 Ki: 46.9 (nM), Ref: 17887741 Ki: 6.9 (nM), Ref: 19932964 Ki: 299 (nM), Ref: 22341895 Ki: 24 (nM), Ref: 22439881 Ki: 60.9 (nM), Ref: 23419026 Ki: 299 (nM), Ref: 23618710 Ki: 299 (nM), Ref: 23880358 Ki: 299 (nM), Ref: 25599950 Ki: 120 (nM), Ref: 26390077 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 6700 (nM), Ref: 18565755 |
|
TCMT614 | Egl nine homolog 1 | Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2710 (nM), Ref: 26275107 |
|
TCMT683 | Macrophage migration inhibitory factor | Homo sapiens |
Ki: 38 (nM), Ref: 19090668 IC50: 38 (nM), Ref: 27156768 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 0.38 (nM), Ref: 19027293 Ki: 2 (nM), Ref: 26390077 |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 120 (nM), Ref: 19027293 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 0.19 (nM), Ref: 19027293 Ki: 0.36 (nM), Ref: 26390077 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270 |
|
TCMT226 | 3-phosphoinositide dependent protein kinase-1 | Homo sapiens |
IC50: 6600 (nM), Ref: 22537682 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2100 (nM), Ref: 26918635 IC50: 2900 (nM), Ref: 26918635 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 529 (nM), Ref: 23332346 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT853 | Sigma opioid receptor | Homo sapiens |
Ki: 36 (nM), Ref: 24617836 IC50: 8.24 (nM), Ref: 26717207 IC50: 7.59 (nM), Ref: 26717207 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 7700 (nM), Ref: 18258440 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 3370 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1249 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 79 (nM), Ref: 20696580 |
|
TCMT83 | Lymphocyte differentiation antigen CD38 | Homo sapiens |
IC50: 8200 (nM), Ref: 21641214 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 3610 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 5620 (nM), Ref: 22658537 |
|
TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 980 (nM), Ref: 22658537 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 830 (nM), Ref: 23411073 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 1600 (nM), Ref: 24368208 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 6400 (nM), Ref: 24878198 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677 |
|
TCMT100 | Transthyretin | Homo sapiens |
IC50: 7000 (nM), Ref: 26214366 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3691.6 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 60.3 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 293 (nM), Ref: 26498393 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 9200 (nM), Ref: 26529431 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 7410 (nM), Ref: 21669522 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 540 (nM), Ref: 21669522 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 520 (nM), Ref: 21669522 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 2030 (nM), Ref: 19097799 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 9900 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10.2 (nM), Ref: 20413308 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7078.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 371.5 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 52.5 (nM), Ref: 26498393 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT210 | Carboxylesterase 2 | Homo sapiens |
Ki: 1840 (nM), Ref: 15828829 Ki: 1840 (nM), Ref: 21733699 |
|
TCMT211 | Acyl coenzyme A:cholesterol acyltransferase | Homo sapiens |
Ki: 5270 (nM), Ref: 15828829 Ki: 5270 (nM), Ref: 21733699 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 1.585 (nM), Ref: 26632862 |
|
TCMT615 | Sentrin-specific protease 8 | Homo sapiens | IC50: 5470 (nM), Ref: |
|
TCMT616 | Sentrin-specific protease 7 | Homo sapiens | IC50: 4630 (nM), Ref: |
|
TCMT617 | Sentrin-specific protease 6 | Homo sapiens | IC50: 1860 (nM), Ref: |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 6300 (nM), Ref: 17616524 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 91 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 4.5 (nM), Ref: 23332346 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 90 (nM), Ref: 18501600 Ki: 90 (nM), Ref: 18579385 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7800 (nM), Ref: 18579385 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8200 (nM), Ref: 18579385 |
|
TCMT853 | Sigma opioid receptor | Homo sapiens |
Ki: 36 (nM), Ref: 27156565 |