Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 7585.78 (nM), Ref: 23574272 IC50: 7500 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 870.96 (nM), Ref: 23574272 IC50: 870 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 645.65 (nM), Ref: 23574272 IC50: 630 (nM), Ref: 23574272 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 2000 (nM), Ref: 24368208 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 6000 (nM), Ref: 15689157 IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 2600 (nM), Ref: 15267241 IC50: 1 (nM), Ref: 20413308 IC50: 800 (nM), Ref: 10.1039/C3MD00166K IC50: 500 (nM), Ref: 26301554 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8500 (nM), Ref: 18165015 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
IC50: 670 (nM), Ref: 19097799 Ki: 110 (nM), Ref: 19097799 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 153 (nM), Ref: 20696580 IC50: 1290 (nM), Ref: 23600958 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 84 (nM), Ref: 20696580 IC50: 54 (nM), Ref: 20832301 IC50: 570 (nM), Ref: 23600958 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 24 (nM), Ref: 20696580 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 5225 (nM), Ref: 20832301 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 5490 (nM), Ref: 22487176 Ki: 5420 (nM), Ref: 22487176 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 4380 (nM), Ref: 22487176 Ki: 4310 (nM), Ref: 22487176 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 2650 (nM), Ref: 22487176 Ki: 2710 (nM), Ref: 22487176 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8960 (nM), Ref: 22487176 Ki: 9070 (nM), Ref: 22487176 Ki: 34.7 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 537.75 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 171.41 (nM), Ref: 26498393 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
Ki: 78 (nM), Ref: 26125082 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 6.9 (nM), Ref: 19027293 Ki: 3.9 (nM), Ref: 20055417 |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 180 (nM), Ref: 19027293 Ki: 49 (nM), Ref: 20055417 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 3 (nM), Ref: 19027293 Ki: 2.2 (nM), Ref: 20055417 |
|
TCMT37 | Serotonin 2a (5-HT2a) receptor | Homo sapiens |
Ki: 966 (nM), Ref: 25695425 |
|
TCMT160 | Serotonin 7 (5-HT7) receptor | Homo sapiens |
Ki: 43 (nM), Ref: 25695425 |
|
TCMT36 | Serotonin 1a (5-HT1a) receptor | Homo sapiens |
Ki: 171 (nM), Ref: 25695425 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 260 (nM), Ref: 22439881 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 9.5 (nM), Ref: 22439881 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 452.6 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 515 (nM), Ref: 26498393 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 286 (nM), Ref: 17616524 |
|
TCMT240 | Salivary alpha-amylase | Homo sapiens |
IC50: 9640 (nM), Ref: 18507367 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 6610 (nM), Ref: |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 600 (nM), Ref: 26602279 |
|
TCMT615 | Sentrin-specific protease 8 | Homo sapiens | IC50: 2470 (nM), Ref: |
|
TCMT616 | Sentrin-specific protease 7 | Homo sapiens | IC50: 1670 (nM), Ref: |
|
TCMT617 | Sentrin-specific protease 6 | Homo sapiens | IC50: 805 (nM), Ref: |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 7400 (nM), Ref: 17616524 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 22 (nM), Ref: 23332346 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 214 (nM), Ref: 23332346 |
|
TCMT789 | Phosphodiesterase 3A | Homo sapiens |
Ki: 279 (nM), Ref: 17228859 |
|
TCMT790 | Phosphodiesterase 3B | Homo sapiens |
Ki: 417 (nM), Ref: 17228859 |
|
TCMT792 | Phosphodiesterase 10A | Homo sapiens |
IC50: 56.9 (nM), Ref: 20450197 IC50: 76 (nM), Ref: 20450197 IC50: 17 (nM), Ref: 21087867 IC50: 21 (nM), Ref: 21705115 IC50: 36 (nM), Ref: 22321214 IC50: 210 (nM), Ref: 23978358 IC50: 36 (nM), Ref: 24721831 IC50: 36 (nM), Ref: 25592707 IC50: 92.3 (nM), Ref: 10.1039/C5MD00419E |
|
TCMT307 | HERG | Homo sapiens |
IC50: 7244.36 (nM), Ref: 21185626 |
|
TCMT151 | Protein kinase C alpha | Homo sapiens |
IC50: 9300 (nM), Ref: 9834166 |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 41 (nM), Ref: 10741545 Ki: 33 (nM), Ref: 14643346 Ki: 33 (nM), Ref: 17149859 Ki: 33 (nM), Ref: 17149858 Ki: 76 (nM), Ref: 17407276 IC50: 138 (nM), Ref: 17388627 IC50: 138 (nM), Ref: 17451272 IC50: 138 (nM), Ref: 18039010 Ki: 33 (nM), Ref: 18313920 Ki: 120 (nM), Ref: 19027293 IC50: 138 (nM), Ref: 16989522 Ki: 51 (nM), Ref: 20055417 Ki: 38 (nM), Ref: 21482470 Ki: 21.38 (nM), Ref: 19527931 Ki: 103 (nM), Ref: 25062506 Ki: 1516 (nM), Ref: 25268943 Ki: 30 (nM), Ref: 26035635 Ki: 103 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 1.2 (nM), Ref: 10741545 Ki: 9.2 (nM), Ref: 17149859 Ki: 9.2 (nM), Ref: 17149858 Ki: 1.1 (nM), Ref: 17407276 IC50: 320 (nM), Ref: 17407276 Ki: 9.2 (nM), Ref: 18313920 Ki: 1.2 (nM), Ref: 19027293 Ki: 3 (nM), Ref: 20055417 Ki: 14.7 (nM), Ref: 20441176 Ki: 0.25 (nM), Ref: 21482470 Ki: 4.467 (nM), Ref: 19527931 Ki: 362 (nM), Ref: 25268943 Ki: 15 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
IC50: 7.3 (nM), Ref: 14643346 Ki: 3.7 (nM), Ref: 17149859 IC50: 7.3 (nM), Ref: 17149859 Ki: 3.7 (nM), Ref: 17149858 IC50: 7.3 (nM), Ref: 17149858 Ki: 0.79 (nM), Ref: 17407276 IC50: 23 (nM), Ref: 17407276 Ki: 3.7 (nM), Ref: 18313920 IC50: 7.3 (nM), Ref: 18313920 Ki: 0.66 (nM), Ref: 19027293 Ki: 0.98 (nM), Ref: 20055417 Ki: 0.23 (nM), Ref: 21482470 Ki: 0.5623 (nM), Ref: 19527931 IC50: 1.87 (nM), Ref: 24171469 Ki: 2.3 (nM), Ref: 25062506 Ki: 354 (nM), Ref: 25268943 Ki: 1.148 (nM), Ref: 26632862 Ki: 1.259 (nM), Ref: 26632862 Ki: 2.3 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.6 (nM), Ref: 16250647 |
|
TCMT309 | Solute carrier family 22 member 2 | Homo sapiens |
IC50: 2600 (nM), Ref: 23241029 |
|
TCMT318 | Putative hexokinase HKDC1 | Homo sapiens | IC50: 4320 (nM), Ref: |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 105 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 6.6 (nM), Ref: 23332346 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 459 (nM), Ref: 17616524 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 251 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 86 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 12 (nM), Ref: 20696580 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 3.96 (nM), Ref: 12372519 Ki: 0.88 (nM), Ref: 16392810 Ki: 1.1 (nM), Ref: 16913723 Ki: 1.1 (nM), Ref: 17887741 Ki: 4 (nM), Ref: 17616524 Ki: 2.55 (nM), Ref: 19627147 Ki: 2.55 (nM), Ref: 21684752 Ki: 2.6 (nM), Ref: 21570305 Ki: 2.6 (nM), Ref: 22341895 Ki: 2.2 (nM), Ref: 24900459 Ki: 0.88 (nM), Ref: 22439881 IC50: 4.3 (nM), Ref: 22995061 Ki: 2.6 (nM), Ref: 23618710 Ki: 2.6 (nM), Ref: 23880358 IC50: 2.5 (nM), Ref: 24171469 Ki: 5.2 (nM), Ref: 25062506 Ki: 2.6 (nM), Ref: 25599950 Ki: 22 (nM), Ref: 25494650 IC50: 6.3 (nM), Ref: 26789491 Ki: 0.53 (nM), Ref: 26390077 Ki: 5.2 (nM), Ref: 10.1039/C5MD00414D |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 140 (nM), Ref: 16392810 Ki: 140 (nM), Ref: 16913723 Ki: 140 (nM), Ref: 17887741 Ki: 605 (nM), Ref: 22341895 Ki: 140 (nM), Ref: 22439881 Ki: 605 (nM), Ref: 23618710 Ki: 605 (nM), Ref: 23880358 Ki: 605 (nM), Ref: 25599950 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 24 (nM), Ref: 16392810 Ki: 46.9 (nM), Ref: 16913723 Ki: 46.9 (nM), Ref: 17887741 Ki: 6.9 (nM), Ref: 19932964 Ki: 299 (nM), Ref: 22341895 Ki: 24 (nM), Ref: 22439881 Ki: 60.9 (nM), Ref: 23419026 Ki: 299 (nM), Ref: 23618710 Ki: 299 (nM), Ref: 23880358 Ki: 299 (nM), Ref: 25599950 Ki: 120 (nM), Ref: 26390077 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
Ki: 600 (nM), Ref: 21739938 |
|
TCMT81 | Arachidonate 12-lipoxygenase | Homo sapiens |
Ki: 1600 (nM), Ref: 21739938 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 8700 (nM), Ref: |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2710 (nM), Ref: 26275107 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 0.38 (nM), Ref: 19027293 Ki: 2 (nM), Ref: 26390077 |
|
TCMT113 | Delta opioid receptor | Homo sapiens |
Ki: 120 (nM), Ref: 19027293 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 0.19 (nM), Ref: 19027293 Ki: 0.36 (nM), Ref: 26390077 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 529 (nM), Ref: 23332346 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT232 | P-glycoprotein 1 | Homo sapiens |
IC50: 11.5 (nM), Ref: 23332369 IC50: 6.6 (nM), Ref: 23895532 |
|
TCMT801 | Tubulin beta-3 chain | Homo sapiens |
IC50: 5.2 (nM), Ref: 23332369 IC50: 5.7 (nM), Ref: 23895532 |
|
TCMT853 | Sigma opioid receptor | Homo sapiens |
Ki: 36 (nM), Ref: 24617836 IC50: 8.24 (nM), Ref: 26717207 IC50: 7.59 (nM), Ref: 26717207 |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1480 (nM), Ref: 23411073 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1284 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 72.8 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 31.1 (nM), Ref: 26498393 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 1.585 (nM), Ref: 26632862 |
|
TCMT615 | Sentrin-specific protease 8 | Homo sapiens | IC50: 5470 (nM), Ref: |
|
TCMT616 | Sentrin-specific protease 7 | Homo sapiens | IC50: 4630 (nM), Ref: |
|
TCMT617 | Sentrin-specific protease 6 | Homo sapiens | IC50: 1860 (nM), Ref: |
|
TCMT116 | Mu opioid receptor | Homo sapiens |
Ki: 6300 (nM), Ref: 17616524 |
|
TCMT747 | ATP-binding cassette sub-family G member 2 | Homo sapiens |
IC50: 10000 (nM), Ref: 22822035 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 91 (nM), Ref: 23332346 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 4.5 (nM), Ref: 23332346 |
|
TCMT853 | Sigma opioid receptor | Homo sapiens |
Ki: 36 (nM), Ref: 27156565 |