Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT151 | Protein kinase C alpha | Homo sapiens |
Ki: 2.5 (nM), Ref: 11327599 Ki: 6.4 (nM), Ref: 21596562 |
|
TCMT152 | Protein kinase C beta | Homo sapiens |
Ki: 1.8 (nM), Ref: 11327599 |
|
TCMT153 | Protein kinase C gamma | Homo sapiens |
Ki: 4.9 (nM), Ref: 11327599 |
|
TCMT154 | Protein kinase C delta | Homo sapiens |
Ki: 0.8 (nM), Ref: 11327599 |
|
TCMT155 | Protein kinase C epsilon | Homo sapiens |
Ki: 0.45 (nM), Ref: 11327599 |
|
TCMT186 | Monoamine oxidase B | Homo sapiens |
IC50: 1410 (nM), Ref: 19378991 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 8710 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4050 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 6000 (nM), Ref: 15689157 IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
Ki: 2600 (nM), Ref: 15267241 IC50: 1 (nM), Ref: 20413308 IC50: 800 (nM), Ref: 10.1039/C3MD00166K IC50: 500 (nM), Ref: 26301554 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 8500 (nM), Ref: 18165015 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
IC50: 670 (nM), Ref: 19097799 Ki: 110 (nM), Ref: 19097799 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 153 (nM), Ref: 20696580 IC50: 1290 (nM), Ref: 23600958 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 84 (nM), Ref: 20696580 IC50: 54 (nM), Ref: 20832301 IC50: 570 (nM), Ref: 23600958 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 24 (nM), Ref: 20696580 |
|
TCMT87 | Cytochrome P450 2C9 | Homo sapiens |
IC50: 5225 (nM), Ref: 20832301 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 5490 (nM), Ref: 22487176 Ki: 5420 (nM), Ref: 22487176 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 4380 (nM), Ref: 22487176 Ki: 4310 (nM), Ref: 22487176 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 2650 (nM), Ref: 22487176 Ki: 2710 (nM), Ref: 22487176 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8960 (nM), Ref: 22487176 Ki: 9070 (nM), Ref: 22487176 Ki: 34.7 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 537.75 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 171.41 (nM), Ref: 26498393 |
|
TCMT290 | Muscarinic acetylcholine receptor M5 | Homo sapiens |
Ki: 0.14 (nM), Ref: 23707254 Ki: 0.3388 (nM), Ref: 24365159 Ki: 0.34 (nM), Ref: 24365159 Ki: 3.02 (nM), Ref: 25051097 |
|
TCMT291 | Muscarinic acetylcholine receptor M3 | Homo sapiens |
Ki: 0.2692 (nM), Ref: 24365159 Ki: 0.27 (nM), Ref: 24365159 |
|
TCMT292 | Muscarinic acetylcholine receptor M1 | Homo sapiens |
Ki: 0.2692 (nM), Ref: 24365159 Ki: 0.27 (nM), Ref: 24365159 |
|
TCMT293 | Muscarinic acetylcholine receptor M2 | Homo sapiens |
Ki: 5.012 (nM), Ref: 25051097 Ki: 12.88 (nM), Ref: 25051097 Ki: 3.631 (nM), Ref: 25051097 Ki: 2.818 (nM), Ref: 25051097 |
|
TCMT303 | Voltage-gated potassium channel subunit Kv1.3 | Homo sapiens |
IC50: 740 (nM), Ref: 20971642 IC50: 2 (nM), Ref: 20971642 |
|
TCMT34 | Cytochrome P450 2D6 | Homo sapiens |
IC50: 4630 (nM), Ref: 15270556 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 5405 (nM), Ref: |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9140 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9010 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8200 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7810 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7550 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6340 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8580 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3190 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 4150 (nM), Ref: 20185318 |
|
TCMT588 | D-amino-acid oxidase | Homo sapiens |
IC50: 2000 (nM), Ref: 23683589 |
|
TCMT159 | Tyrosinase | Homo sapiens |
IC50: 9150 (nM), Ref: 26386819 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 1720 (nM), Ref: 8576921 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 320 (nM), Ref: 22261024 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 3150 (nM), Ref: 8576921 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
Ki: 6900 (nM), Ref: 19879672 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 77 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 40 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 568.3 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 24.5 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 41.8 (nM), Ref: 26498393 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1400 (nM), Ref: 20590092 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1110 (nM), Ref: 20590092 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 112 (nM), Ref: 20590092 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 1220 (nM), Ref: 20590092 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 1440 (nM), Ref: 20590092 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 1410 (nM), Ref: 20590092 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 1230 (nM), Ref: 20590092 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 1370 (nM), Ref: 20590092 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 1000 (nM), Ref: 20590092 |
|
TCMT287 | Taste receptor type 2 member 31 | Homo sapiens |
IC50: 3600 (nM), Ref: 21650152 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref: |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 7300 (nM), Ref: 21030469 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 718.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.2 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 56.4 (nM), Ref: 26498393 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2710 (nM), Ref: 26275107 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 7906 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 1679 (nM), Ref: 20696580 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1491 (nM), Ref: 20696580 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 900 (nM), Ref: 10.1039/C3MD00166K |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 3430 (nM), Ref: 19097799 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 4960 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 2.9 (nM), Ref: 20413308 IC50: 230 (nM), Ref: 22115839 IC50: 230 (nM), Ref: 23142320 IC50: 1200 (nM), Ref: 23994869 IC50: 3300 (nM), Ref: 24074257 IC50: 1200 (nM), Ref: 24992702 IC50: 5100 (nM), Ref: 27155469 IC50: 1000 (nM), Ref: 27155469 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 3656 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 79.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.3 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 44.3 (nM), Ref: 26498393 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8700 (nM), Ref: 21332115 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 500 (nM), Ref: 20590092 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 52 (nM), Ref: 20590092 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 44 (nM), Ref: 20590092 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 540 (nM), Ref: 20590092 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 740 (nM), Ref: 20590092 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 420 (nM), Ref: 20590092 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 380 (nM), Ref: 20590092 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 450 (nM), Ref: 20590092 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 500 (nM), Ref: 20590092 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 10 (nM), Ref: 15341953 IC50: 10 (nM), Ref: 15456246 IC50: 98.7 (nM), Ref: 15887952 IC50: 98.7 (nM), Ref: 15887952 IC50: 9.7 (nM), Ref: 15943471 IC50: 10 (nM), Ref: 16098741 IC50: 1.3 (nM), Ref: 16219463 IC50: 61 (nM), Ref: 16610787 IC50: 25 (nM), Ref: 17149865 IC50: 395 (nM), Ref: 17049855 IC50: 9.7 (nM), Ref: 17188490 IC50: 6.8 (nM), Ref: 17574424 IC50: 18 (nM), Ref: 12502307 IC50: 98.7 (nM), Ref: |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 395 (nM), Ref: 15341953 IC50: 395 (nM), Ref: 15456246 IC50: 4660 (nM), Ref: 15887952 IC50: 4660 (nM), Ref: 15887952 IC50: 395 (nM), Ref: 15943471 IC50: 395 (nM), Ref: 16098741 IC50: 29.4 (nM), Ref: 16219463 IC50: 1973 (nM), Ref: 16610787 IC50: 1145 (nM), Ref: 17149865 IC50: 2150 (nM), Ref: 17696335 IC50: 9.7 (nM), Ref: 17049855 IC50: 395 (nM), Ref: 17188490 IC50: 580 (nM), Ref: 17574424 IC50: 300 (nM), Ref: 12502307 IC50: 4680 (nM), Ref: |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 10 (nM), Ref: 17482813 |
|
TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 395 (nM), Ref: 17482813 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 2210 (nM), Ref: 18533708 |
|
TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 340 (nM), Ref: 20853847 |
|
TCMT291 | Muscarinic acetylcholine receptor M3 | Homo sapiens |
Ki: 0.5 (nM), Ref: 11831911 Ki: 0.9 (nM), Ref: 20684563 Ki: 2.18 (nM), Ref: 23523385 |
|
TCMT292 | Muscarinic acetylcholine receptor M1 | Homo sapiens |
Ki: 0.25 (nM), Ref: 11831911 Ki: 1.202 (nM), Ref: 22329602 Ki: 0.5754 (nM), Ref: 22329602 Ki: 0.922 (nM), Ref: 23523385 |
|
TCMT293 | Muscarinic acetylcholine receptor M2 | Homo sapiens |
Ki: 1.5 (nM), Ref: 11831911 Ki: 1.9 (nM), Ref: 20684563 Ki: 1.44 (nM), Ref: 23523385 |
|
TCMT551 | Muscarinic acetylcholine receptor M4 | Homo sapiens |
Ki: 0.34 (nM), Ref: 11831911 Ki: 3 (nM), Ref: 20684563 Ki: 1.39 (nM), Ref: 23523385 |
|
TCMT290 | Muscarinic acetylcholine receptor M5 | Homo sapiens |
Ki: 0.54 (nM), Ref: 11831911 Ki: 0.21 (nM), Ref: 19438238 Ki: 1 (nM), Ref: 20684563 Ki: 1.47 (nM), Ref: 25147929 |
|
TCMT289 | Thromboxane-A synthase | Homo sapiens | IC50: 7720 (nM), Ref: |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 7500 (nM), Ref: 15916432 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: 15887952 IC50: 75.7 (nM), Ref: |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: 15887952 IC50: 18.6 (nM), Ref: |
|
TCMT601 | Thrombin | Homo sapiens |
IC50: 250 (nM), Ref: 24610996 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2420 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1840 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 3580 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4900 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4210 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4020 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4910 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 450 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5030 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4720 (nM), Ref: 20674354 |