Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2940 (nM), Ref: 19231207 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 500 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT571 | Adenosine A2b receptor | Homo sapiens |
Ki: 8200 (nM), Ref: 15084123 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
Ki: 680 (nM), Ref: 15084123 |
|
TCMT683 | Macrophage migration inhibitory factor | Homo sapiens |
IC50: 250 (nM), Ref: 25743213 IC50: 1100 (nM), Ref: 25743213 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1118 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 95 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 20 (nM), Ref: 20696580 |
|
TCMT151 | Protein kinase C alpha | Homo sapiens |
IC50: 9300 (nM), Ref: 9834166 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 7700 (nM), Ref: 18258440 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 3370 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1249 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 79 (nM), Ref: 20696580 |
|
TCMT83 | Lymphocyte differentiation antigen CD38 | Homo sapiens |
IC50: 8200 (nM), Ref: 21641214 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 3610 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 5620 (nM), Ref: 22658537 |
|
TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 980 (nM), Ref: 22658537 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 830 (nM), Ref: 23411073 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 1600 (nM), Ref: 24368208 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 6400 (nM), Ref: 24878198 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677 |
|
TCMT100 | Transthyretin | Homo sapiens |
IC50: 7000 (nM), Ref: 26214366 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3691.6 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 60.3 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 293 (nM), Ref: 26498393 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 9200 (nM), Ref: 26529431 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 4 (nM), Ref: 26562543 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT637 | NAD-dependent deacetylase sirtuin 3 | Homo sapiens |
IC50: 6200 (nM), Ref: 25275824 |
|
TCMT638 | NAD-dependent deacetylase sirtuin 2 | Homo sapiens |
IC50: 6300 (nM), Ref: 25549554 IC50: 1200 (nM), Ref: 26696402 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 3400 (nM), Ref: 23388705 IC50: 5400 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 5200 (nM), Ref: 23388705 IC50: 5800 (nM), Ref: 23388705 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
IC50: 1.3 (nM), Ref: 15203155 IC50: 3 (nM), Ref: 10673099 IC50: 1.3 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 5.9 (nM), Ref: 10447957 IC50: 1.3 (nM), Ref: 15745820 IC50: 1.3 (nM), Ref: 15664843 IC50: 1.3 (nM), Ref: 15582421 IC50: 1.3 (nM), Ref: 15225685 IC50: 1.3 (nM), Ref: 15225686 IC50: 3.2 (nM), Ref: 15341953 IC50: 3.2 (nM), Ref: 15456246 IC50: 3.2 (nM), Ref: 15876535 IC50: 3.2 (nM), Ref: 15943471 IC50: 28 (nM), Ref: 15658851 Ki: 1.995 (nM), Ref: 15771467 IC50: 3.2 (nM), Ref: 16098741 IC50: 0.75 (nM), Ref: 16219463 IC50: 1.4 (nM), Ref: 16309907 IC50: 1.35 (nM), Ref: 16412638 IC50: 10 (nM), Ref: 16610787 IC50: 1.3 (nM), Ref: 16632357 IC50: 1.3 (nM), Ref: 16730987 IC50: 46 (nM), Ref: 16942012 IC50: 1.6 (nM), Ref: 16942012 IC50: 1.3 (nM), Ref: 16777408 IC50: 1.2 (nM), Ref: 17149865 IC50: 4.7 (nM), Ref: 17696335 IC50: 3.6 (nM), Ref: 17049855 IC50: 3.2 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.4 (nM), Ref: 17448656 IC50: 1.4 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 12.5 (nM), Ref: 19836949 IC50: 3.2 (nM), Ref: 19705860 Ki: 0.16 (nM), Ref: 20621492 IC50: 21.04 (nM), Ref: 20812681 IC50: 46 (nM), Ref: 20875743 IC50: 1.3 (nM), Ref: 24315190 IC50: 5.7 (nM), Ref: 25369367 IC50: 0.9 (nM), Ref: 26183544 Ki: 0.21 (nM), Ref: Ki: 0.21 (nM), Ref: IC50: 1.7 (nM), Ref: 27407030 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 1.1 (nM), Ref: 15203155 IC50: 4 (nM), Ref: 10673099 IC50: 1.1 (nM), Ref: 15203156 Ki: 100 (nM), Ref: 12954056 IC50: 2 (nM), Ref: 12749898 IC50: 1.1 (nM), Ref: 15745820 IC50: 1.1 (nM), Ref: 15664843 IC50: 1.1 (nM), Ref: 15993065 IC50: 1.1 (nM), Ref: 15582421 IC50: 1.1 (nM), Ref: 15225685 IC50: 1.1 (nM), Ref: 15225686 IC50: 3.6 (nM), Ref: 15341953 IC50: 3.6 (nM), Ref: 15456246 IC50: 3.6 (nM), Ref: 15876535 IC50: 3.6 (nM), Ref: 15943471 IC50: 24 (nM), Ref: 15658851 Ki: 3.162 (nM), Ref: 15771467 IC50: 3.6 (nM), Ref: 16098741 IC50: 1.18 (nM), Ref: 16219463 IC50: 1.2 (nM), Ref: 16309907 IC50: 1.2 (nM), Ref: 16412638 IC50: 11 (nM), Ref: 16610787 IC50: 1.2 (nM), Ref: 16632357 IC50: 1.2 (nM), Ref: 16730987 IC50: 1.4 (nM), Ref: 16942012 IC50: 1.1 (nM), Ref: 16777408 IC50: 1.4 (nM), Ref: 17149865 IC50: 16.7 (nM), Ref: 17696335 IC50: 3.2 (nM), Ref: 17049855 IC50: 3.6 (nM), Ref: 17188490 IC50: 1 (nM), Ref: 17289385 IC50: 1.2 (nM), Ref: 17448656 IC50: 1.2 (nM), Ref: 17890084 IC50: 4 (nM), Ref: 18760603 Ki: 2 (nM), Ref: 18722117 IC50: 2.9 (nM), Ref: 19705860 IC50: 10.74 (nM), Ref: 20812681 IC50: 0.046 (nM), Ref: 24315190 IC50: 5.6 (nM), Ref: 25369367 Ki: 0.015 (nM), Ref: Ki: 0.015 (nM), Ref: IC50: 3 (nM), Ref: 27407030 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 19.1 (nM), Ref: 16309907 |
|
TCMT99 | Testis-specific androgen-binding protein | Homo sapiens |
IC50: 50 (nM), Ref: 17149875 |
|
TCMT591 | Estrogen-related receptor alpha | Homo sapiens |
IC50: 3.6 (nM), Ref: 17482813 IC50: 6 (nM), Ref: 23448346 |
|
TCMT910 | Estrogen-related receptor beta | Homo sapiens |
IC50: 3.2 (nM), Ref: 17482813 IC50: 8.7 (nM), Ref: 23448346 |
|
TCMT344 | Aldehyde oxidase | Homo sapiens |
IC50: 80 (nM), Ref: 20853847 Ki: 4400 (nM), Ref: 22996261 Ki: 870 (nM), Ref: 22996261 |
|
TCMT974 | G-protein coupled estrogen receptor 1 | Homo sapiens |
Ki: 5.7 (nM), Ref: 23672690 Ki: 2.7 (nM), Ref: 10.1039/C5MD00455A |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 2437 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 140 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 29 (nM), Ref: 20696580 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 8960 (nM), Ref: 22658537 |
|
TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 8220 (nM), Ref: 22658537 |