TCM Putative Target References: TCMFx2615


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC417
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 7585.78 (nM), Ref: 23574272
IC50: 7500 (nM), Ref: 23574272
TCMC417
TCMT128 Tankyrase-2 Homo sapiens IC50: 870.96 (nM), Ref: 23574272
IC50: 870 (nM), Ref: 23574272
TCMC417
TCMT129 Tankyrase-1 Homo sapiens IC50: 645.65 (nM), Ref: 23574272
IC50: 630 (nM), Ref: 23574272
TCMC417
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2000 (nM), Ref: 24368208
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC616
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 800 (nM), Ref: 16759088
IC50: 3450 (nM), Ref: 16759088
IC50: 7138 (nM), Ref: 20851614
IC50: 7100 (nM), Ref: 21376605
TCMC616
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 201 (nM), Ref: 16759088
IC50: 6430 (nM), Ref: 16759088
IC50: 750 (nM), Ref: 20851614
IC50: 750 (nM), Ref: 21376605
TCMC616
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 3780 (nM), Ref: 16759088
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC761
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 3920 (nM), Ref: 15658857
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC1447
TCMT207 Beta-secretase 1 Homo sapiens Ki: 3000 (nM), Ref: 18565755
IC50: 2600 (nM), Ref: 18565755
TCMC332
TCMT231 Beta-glucosidase Homo sapiens Ki: 200 (nM), Ref: 10.1039/C3MD00033H
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1366
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 8800 (nM), Ref: 26965864
TCMC88
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 3400 (nM), Ref: 11678652
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC87
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 400 (nM), Ref: 11678652
TCMC1397
TCMT34 Cytochrome P450 2D6 Homo sapiens IC50: 4630 (nM), Ref: 15270556
TCMC1397
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 5405 (nM), Ref:
TCMC1464
TCMT207 Beta-secretase 1 Homo sapiens Ki: 3900 (nM), Ref: 18565755
IC50: 8400 (nM), Ref: 18565755
TCMC2093
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 57 (nM), Ref: 17149865
TCMC2093
TCMT236 Estrogen receptor beta Homo sapiens IC50: 68 (nM), Ref: 17149865
TCMC795
TCMT223 Aldose reductase Homo sapiens IC50: 8000 (nM), Ref: 24341381
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1293
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2940 (nM), Ref: 19231207
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC1255
TCMT33 Cytochrome P450 3A4 Homo sapiens Ki: 7000 (nM), Ref: 16248836
TCMC2188
TCMT223 Aldose reductase Homo sapiens IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC1411
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1261 (nM), Ref: 20696580
TCMC1411
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 56 (nM), Ref: 20696580
TCMC1411
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 17 (nM), Ref: 20696580
TCMC1411
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 212.9 (nM), Ref: 26498393
TCMC1411
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.4 (nM), Ref: 26498393
TCMC1411
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 54.9 (nM), Ref: 26498393
Ki: 220 (nM), Ref: 26498393
TCMC1411
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 440 (nM), Ref: 26498393
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC2054
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 9640 (nM), Ref: 18507367
TCMC2054
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 6610 (nM), Ref:
TCMC2054
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 600 (nM), Ref: 26602279
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC1584
TCMT571 Adenosine A2b receptor Homo sapiens Ki: 8200 (nM), Ref: 15084123
TCMC1584
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 680 (nM), Ref: 15084123
TCMC949
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8900 (nM), Ref: 19911821
TCMC949
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 48 (nM), Ref: 19911821
TCMC949
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9100 (nM), Ref: 19911821
TCMC949
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3300 (nM), Ref: 19911821
TCMC949
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 2000 (nM), Ref: 19911821
TCMC949
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 5200 (nM), Ref: 19911821
TCMC949
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9400 (nM), Ref: 19911821
TCMC949
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 6800 (nM), Ref: 19911821
TCMC949
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 5600 (nM), Ref: 19911821
TCMC949
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3100 (nM), Ref: 19911821
Ki: 3100 (nM), Ref: 21067924
Ki: 3100 (nM), Ref: 22137345
Ki: 3100 (nM), Ref: 22077347
Ki: 3100 (nM), Ref: 22365761
Ki: 3100 (nM), Ref: 22377674
Ki: 3100 (nM), Ref: 23241068
Ki: 3100 (nM), Ref: 22892213
Ki: 3100 (nM), Ref: 26688270
TCMC949
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9200 (nM), Ref: 21067924
Ki: 9200 (nM), Ref: 22137345
Ki: 9200 (nM), Ref: 22077347
Ki: 9200 (nM), Ref: 22365761
Ki: 9200 (nM), Ref: 22377674
Ki: 9200 (nM), Ref: 23241068
Ki: 9200 (nM), Ref: 22892213
Ki: 9200 (nM), Ref: 26688270
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC315
TCMT46 Coagulation factor III Homo sapiens IC50: 14.98 (nM), Ref: 23199480
TCMC1376
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 40 (nM), Ref: 11678654
TCMC1501
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2100 (nM), Ref: 18042388
IC50: 340 (nM), Ref: 18778944
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1113
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1399
TCMT223 Aldose reductase Homo sapiens IC50: 320 (nM), Ref: 22261024
TCMC575
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 2400 (nM), Ref: 26704263
Ki: 2500 (nM), Ref: 26704263
TCMC584
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2 (nM), Ref: 20413308
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC910
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1118 (nM), Ref: 20696580
TCMC910
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 95 (nM), Ref: 20696580
TCMC910
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 20 (nM), Ref: 20696580
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC405
TCMT506 Protein tyrosine kinase 2 beta Homo sapiens IC50: 2324 (nM), Ref:
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1201
TCMT112 Adenosine A3 receptor Homo sapiens Ki: 3150 (nM), Ref: 8576921
TCMC1201
TCMT132 Butyrylcholinesterase Homo sapiens Ki: 6900 (nM), Ref: 19879672
TCMC1201
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1201
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 40 (nM), Ref: 20696580
TCMC1201
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC1201
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1201
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 568.3 (nM), Ref: 26498393
TCMC1201
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 24.5 (nM), Ref: 26498393
TCMC1201
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 41.8 (nM), Ref: 26498393
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC614
TCMT151 Protein kinase C alpha Homo sapiens IC50: 9300 (nM), Ref: 9834166
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC1398
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 100 (nM), Ref: 11678652
TCMC1281
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 10 (nM), Ref: 19564108
IC50: 18.6 (nM), Ref: 22148241
IC50: 6 (nM), Ref: 22360639
TCMC1281
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 1 (nM), Ref: 19564108
IC50: 0.7 (nM), Ref: 22148241
IC50: 0.4 (nM), Ref: 22360639
TCMC1380
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3000 (nM), Ref: 26841168
TCMC533
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 9300 (nM), Ref: 26704263
Ki: 9600 (nM), Ref: 26704263
TCMC916
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens Ki: 4900 (nM), Ref: 21167710
TCMC1015
TCMT318 Putative hexokinase HKDC1 Homo sapiens IC50: 4320 (nM), Ref:
TCMC2196
TCMT30 Cyclooxygenase-2 Homo sapiens IC50: 64 (nM), Ref: 22819942
IC50: 64 (nM), Ref: 23146282
TCMC2196
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 150 (nM), Ref: 22819942
TCMC2196
TCMT336 Indoleamine 2,3-dioxygenase Homo sapiens IC50: 53.7 (nM), Ref: 24099220
IC50: 7150 (nM), Ref: 24099220
Ki: 4810 (nM), Ref: 24099220
TCMC2105
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2105
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1597
TCMT807 Solute carrier family 22 member 12 Homo sapiens IC50: 2000 (nM), Ref: 17325024
Ki: 5740 (nM), Ref: 17325024
TCMC1597
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2927.18 (nM), Ref:
TCMC1597
TCMT61 Induced myeloid leukemia cell differentiation protein Mcl-1 Homo sapiens IC50: 2988.26 (nM), Ref:
TCMC1597
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 1600 (nM), Ref: 24900447
TCMC1597
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 1600 (nM), Ref: 26322379
TCMC1597
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 4300 (nM), Ref: 26602279
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC596
TCMT39 Phosphodiesterase 5A Homo sapiens IC50: 1290 (nM), Ref: 18778098
TCMC2094
TCMT238 Sodium/glucose cotransporter 2 Homo sapiens IC50: 4100 (nM), Ref: 17374486
TCMC2094
TCMT207 Beta-secretase 1 Homo sapiens Ki: 1100 (nM), Ref: 18565755
IC50: 5200 (nM), Ref: 18565755
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1869
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 4410 (nM), Ref: 15658857
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC587
TCMT131 Acetylcholinesterase Homo sapiens IC50: 9900 (nM), Ref: 26841168
TCMC1111
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 11.78 (nM), Ref: 18242087
IC50: 13 (nM), Ref: 18653260
IC50: 778 (nM), Ref: 20851614
IC50: 778 (nM), Ref: 21376605
IC50: 8.6 (nM), Ref: 21873057
IC50: 29.1 (nM), Ref: 23747808
IC50: 29.1 (nM), Ref: 25590374
TCMC1111
TCMT209 11-beta-hydroxysteroid dehydrogenase 2 Homo sapiens IC50: 257 (nM), Ref: 20851614
IC50: 257 (nM), Ref: 21376605
IC50: 1.22 (nM), Ref: 23747808
IC50: 1.2 (nM), Ref: 25590374
TCMC1111
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4900 (nM), Ref: 21561086
TCMC983
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2800 (nM), Ref: 15887952
IC50: 2800 (nM), Ref: 15887952
IC50: 1200 (nM), Ref: 12502307
IC50: 2800 (nM), Ref:
TCMC983
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 7300 (nM), Ref: 21030469
TCMC983
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 718.7 (nM), Ref: 26498393
TCMC983
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.2 (nM), Ref: 26498393
TCMC983
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 56.4 (nM), Ref: 26498393
TCMC84
TCMT207 Beta-secretase 1 Homo sapiens IC50: 6700 (nM), Ref: 18565755
TCMC183
TCMT188 Dihydrofolate reductase Homo sapiens IC50: 500 (nM), Ref: 26979156
TCMC755
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens Ki: 600 (nM), Ref: 21739938
TCMC755
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens Ki: 1600 (nM), Ref: 21739938
TCMC755
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4400 (nM), Ref: 21030469
IC50: 7000 (nM), Ref: 21030469
TCMC755
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 8700 (nM), Ref:
TCMC1329
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2710 (nM), Ref: 26275107
TCMC412
TCMT683 Macrophage migration inhibitory factor Homo sapiens Ki: 38 (nM), Ref: 19090668
IC50: 38 (nM), Ref: 27156768
TCMC1898
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 7906 (nM), Ref: 20696580
TCMC1898
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1679 (nM), Ref: 20696580
TCMC1898
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1491 (nM), Ref: 20696580
TCMC1898
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 900 (nM), Ref: 10.1039/C3MD00166K
TCMC2204
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 482 (nM), Ref: 21067924
Ki: 478 (nM), Ref: 22077347
Ki: 480 (nM), Ref: 26688270
TCMC2204
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 754 (nM), Ref: 22077347
Ki: 750 (nM), Ref: 26688270
TCMC2239
TCMT226 3-phosphoinositide dependent protein kinase-1 Homo sapiens IC50: 6600 (nM), Ref: 22537682
TCMC2239
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2100 (nM), Ref: 26918635
IC50: 2900 (nM), Ref: 26918635
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1377
TCMT186 Monoamine oxidase B Homo sapiens Ki: 3000 (nM), Ref: 16137882
Ki: 3000 (nM), Ref: 19342233
IC50: 7943.28 (nM), Ref: 20934874
Ki: 5340 (nM), Ref: 21134756
Ki: 3000 (nM), Ref: 21778064
Ki: 2000 (nM), Ref: 24140951
TCMC1377
TCMT208 Monoamine oxidase A Homo sapiens Ki: 8380 (nM), Ref: 21134756
TCMC1105
TCMT752 Casein kinase II alpha Homo sapiens IC50: 2000 (nM), Ref: 19414254
TCMC1105
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 2500 (nM), Ref: 27173800
TCMC1400
TCMT223 Aldose reductase Homo sapiens IC50: 720 (nM), Ref: 22261024
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC937
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 11.5 (nM), Ref: 23332369
IC50: 6.6 (nM), Ref: 23895532
TCMC937
TCMT801 Tubulin beta-3 chain Homo sapiens IC50: 5.2 (nM), Ref: 23332369
IC50: 5.7 (nM), Ref: 23895532
TCMC1489
TCMT223 Aldose reductase Homo sapiens IC50: 560 (nM), Ref: 22261024
TCMC1516
TCMT44 Glyoxalase I Homo sapiens IC50: 7700 (nM), Ref: 18258440
TCMC1516
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 3370 (nM), Ref: 20696580
TCMC1516
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1249 (nM), Ref: 20696580
TCMC1516
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 79 (nM), Ref: 20696580
TCMC1516
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 8200 (nM), Ref: 21641214
TCMC1516
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 3610 (nM), Ref: 22658537
TCMC1516
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 5620 (nM), Ref: 22658537
TCMC1516
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 980 (nM), Ref: 22658537
TCMC1516
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1516
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 830 (nM), Ref: 23411073
TCMC1516
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 4265.8 (nM), Ref: 23574272
IC50: 4200 (nM), Ref: 23574272
TCMC1516
TCMT128 Tankyrase-2 Homo sapiens IC50: 1071.52 (nM), Ref: 23574272
IC50: 1100 (nM), Ref: 23574272
TCMC1516
TCMT129 Tankyrase-1 Homo sapiens IC50: 2398.83 (nM), Ref: 23574272
IC50: 2400 (nM), Ref: 23574272
TCMC1516
TCMT223 Aldose reductase Homo sapiens IC50: 600 (nM), Ref: 23683835
IC50: 3200 (nM), Ref: 26529431
TCMC1516
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 1600 (nM), Ref: 24368208
TCMC1516
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 6400 (nM), Ref: 24878198
TCMC1516
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 2900 (nM), Ref: 25019478
IC50: 7800 (nM), Ref: 26096677
TCMC1516
TCMT100 Transthyretin Homo sapiens IC50: 7000 (nM), Ref: 26214366
TCMC1516
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3691.6 (nM), Ref: 26498393
TCMC1516
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1516
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 60.3 (nM), Ref: 26498393
TCMC1516
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 293 (nM), Ref: 26498393
TCMC1516
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 9200 (nM), Ref: 26529431
TCMC1734
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 3430 (nM), Ref: 19097799
TCMC1734
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 4960 (nM), Ref: 18533708
TCMC1734
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 2.9 (nM), Ref: 20413308
IC50: 230 (nM), Ref: 22115839
IC50: 230 (nM), Ref: 23142320
IC50: 1200 (nM), Ref: 23994869
IC50: 3300 (nM), Ref: 24074257
IC50: 1200 (nM), Ref: 24992702
IC50: 5100 (nM), Ref: 27155469
IC50: 1000 (nM), Ref: 27155469
TCMC1734
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 3656 (nM), Ref: 20696580
TCMC1734
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 79.5 (nM), Ref: 26498393
TCMC1734
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1734
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 44.3 (nM), Ref: 26498393
TCMC1798
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1480 (nM), Ref: 23411073
TCMC811
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 2030 (nM), Ref: 19097799
TCMC811
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 9900 (nM), Ref: 18533708
TCMC811
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10.2 (nM), Ref: 20413308
TCMC811
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7078.5 (nM), Ref: 26498393
TCMC811
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 371.5 (nM), Ref: 26498393
TCMC811
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.5 (nM), Ref: 26498393
TCMC1496
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1496
TCMT164 Cyclooxygenase-1 Homo sapiens Ki: 4000 (nM), Ref: 24088053
TCMC1123
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1284 (nM), Ref: 20696580
TCMC1123
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 72.8 (nM), Ref: 26498393
TCMC1123
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1123
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 31.1 (nM), Ref: 26498393
TCMC1562
TCMT210 Carboxylesterase 2 Homo sapiens IC50: 5610 (nM), Ref: 26900660
TCMC778
TCMT683 Macrophage migration inhibitory factor Homo sapiens IC50: 540 (nM), Ref: 25743213
IC50: 530 (nM), Ref: 25743213
TCMC1873
TCMT210 Carboxylesterase 2 Homo sapiens Ki: 1840 (nM), Ref: 15828829
Ki: 1840 (nM), Ref: 21733699
TCMC1873
TCMT211 Acyl coenzyme A:cholesterol acyltransferase Homo sapiens Ki: 5270 (nM), Ref: 15828829
Ki: 5270 (nM), Ref: 21733699
TCMC1371
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 4 (nM), Ref: 26562543
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1320
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 2786 (nM), Ref: 20696580
TCMC1320
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 511 (nM), Ref: 20696580
TCMC1320
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 102.1 (nM), Ref: 26498393
TCMC1320
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.3 (nM), Ref: 26498393
TCMC1320
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 454.1 (nM), Ref: 26498393
TCMC1832
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1832
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1742
TCMT637 NAD-dependent deacetylase sirtuin 3 Homo sapiens IC50: 6200 (nM), Ref: 25275824
TCMC1742
TCMT638 NAD-dependent deacetylase sirtuin 2 Homo sapiens IC50: 6300 (nM), Ref: 25549554
IC50: 1200 (nM), Ref: 26696402
TCMC1267
TCMT159 Tyrosinase Homo sapiens IC50: 154 (nM), Ref: 26841168
TCMC1236
TCMT236 Estrogen receptor beta Homo sapiens IC50: 10 (nM), Ref: 15341953
IC50: 10 (nM), Ref: 15456246
IC50: 98.7 (nM), Ref: 15887952
IC50: 98.7 (nM), Ref: 15887952
IC50: 9.7 (nM), Ref: 15943471
IC50: 10 (nM), Ref: 16098741
IC50: 1.3 (nM), Ref: 16219463
IC50: 61 (nM), Ref: 16610787
IC50: 25 (nM), Ref: 17149865
IC50: 395 (nM), Ref: 17049855
IC50: 9.7 (nM), Ref: 17188490
IC50: 6.8 (nM), Ref: 17574424
IC50: 18 (nM), Ref: 12502307
IC50: 98.7 (nM), Ref:
TCMC1236
TCMT82 Estrogen receptor alpha Homo sapiens IC50: 395 (nM), Ref: 15341953
IC50: 395 (nM), Ref: 15456246
IC50: 4660 (nM), Ref: 15887952
IC50: 4660 (nM), Ref: 15887952
IC50: 395 (nM), Ref: 15943471
IC50: 395 (nM), Ref: 16098741
IC50: 29.4 (nM), Ref: 16219463
IC50: 1973 (nM), Ref: 16610787
IC50: 1145 (nM), Ref: 17149865
IC50: 2150 (nM), Ref: 17696335
IC50: 9.7 (nM), Ref: 17049855
IC50: 395 (nM), Ref: 17188490
IC50: 580 (nM), Ref: 17574424
IC50: 300 (nM), Ref: 12502307
IC50: 4680 (nM), Ref:
TCMC1236
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 10 (nM), Ref: 17482813
TCMC1236
TCMT910 Estrogen-related receptor beta Homo sapiens IC50: 395 (nM), Ref: 17482813
TCMC1236
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 2210 (nM), Ref: 18533708
TCMC1236
TCMT344 Aldehyde oxidase Homo sapiens IC50: 340 (nM), Ref: 20853847
TCMC1236
TCMT289 Thromboxane-A synthase Homo sapiens IC50: 7720 (nM), Ref:
TCMC2055
TCMT747 ATP-binding cassette sub-family G member 2 Homo sapiens IC50: 10000 (nM), Ref: 22822035
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC1174
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 850 (nM), Ref: 15689157
IC50: 850 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1174
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1064
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 2437 (nM), Ref: 20696580
TCMC1064
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 140 (nM), Ref: 20696580
TCMC1064
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 29 (nM), Ref: 20696580
TCMC1266
TCMT159 Tyrosinase Homo sapiens IC50: 177 (nM), Ref: 26841168
TCMC700
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 400 (nM), Ref: 26841168
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755
TCMC1378
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 8960 (nM), Ref: 22658537
TCMC1378
TCMT734 Matrix metalloproteinase 12 Homo sapiens IC50: 8220 (nM), Ref: 22658537

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC2254
TCMT1121 Sialidase Clostridium perfringens IC50: 0.44 (ug/ml), Ref: 21123068
TCMC2254
TCMT1136 Neuraminidase Influenza A virus IC50: 52.96 (ug/ml), Ref: 21123068
IC50: 75.38 (ug/ml), Ref: 21123068
IC50: 83.14 (ug/ml), Ref: 21123068
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC2054
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 14.48 (ug/ml), Ref: 20116898
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2263
TCMT1121 Sialidase Clostridium perfringens IC50: 1.18 (ug/ml), Ref: 21123068
TCMC2263
TCMT1136 Neuraminidase Influenza A virus IC50: 28.62 (ug/ml), Ref: 21123068
IC50: 35.21 (ug/ml), Ref: 21123068
IC50: 36.52 (ug/ml), Ref: 21123068
TCMC1399
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 3.42 (ug/ml), Ref: 21123068
IC50: 3.48 (ug/ml), Ref: 21123068
IC50: 8.41 (ug/ml), Ref: 21123068
IC50: 9.69 (ug/ml), Ref: 21123068
IC50: 10.56 (ug/ml), Ref: 21123068
TCMC1399
TCMT1136 Neuraminidase Influenza A virus IC50: 3.42 (ug/ml), Ref: 21123068
IC50: 3.48 (ug/ml), Ref: 21123068
IC50: 8.41 (ug/ml), Ref: 21123068
IC50: 9.69 (ug/ml), Ref: 21123068
IC50: 10.56 (ug/ml), Ref: 21123068
TCMC1399
TCMT1121 Sialidase Clostridium perfringens IC50: 11.28 (ug/ml), Ref: 21123068
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC1482
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 4.2 (ug/ml), Ref: 21123068
IC50: 5.42 (ug/ml), Ref: 21123068
IC50: 17.98 (ug/ml), Ref: 21123068
IC50: 18.23 (ug/ml), Ref: 21123068
IC50: 19.09 (ug/ml), Ref: 21123068
TCMC1482
TCMT1121 Sialidase Clostridium perfringens IC50: 6.9 (ug/ml), Ref: 21123068
TCMC1482
TCMT1136 Neuraminidase Influenza A virus IC50: 4.2 (ug/ml), Ref: 21123068
IC50: 5.42 (ug/ml), Ref: 21123068
IC50: 17.98 (ug/ml), Ref: 21123068
IC50: 18.23 (ug/ml), Ref: 21123068
IC50: 19.09 (ug/ml), Ref: 21123068
TCMC983
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.43 (ug/ml), Ref: 20116898
TCMC1329
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.9 (ug/ml), Ref: 20116898
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1095
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 2.19 (ug/ml), Ref: 21123068
IC50: 2.49 (ug/ml), Ref: 21123068
IC50: 5.7 (ug/ml), Ref: 21123068
IC50: 5.8 (ug/ml), Ref: 21123068
IC50: 8.23 (ug/ml), Ref: 21123068
TCMC1095
TCMT1136 Neuraminidase Influenza A virus IC50: 2.19 (ug/ml), Ref: 21123068
IC50: 2.49 (ug/ml), Ref: 21123068
IC50: 5.7 (ug/ml), Ref: 21123068
IC50: 5.8 (ug/ml), Ref: 21123068
IC50: 8.23 (ug/ml), Ref: 21123068
TCMC1095
TCMT1121 Sialidase Clostridium perfringens IC50: 8.13 (ug/ml), Ref: 21123068
TCMC1516
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.65 (ug/ml), Ref: 20116898
TCMC2292
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.15 (ug/ml), Ref: 20116898
TCMC1236
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 20.84 (ug/ml), Ref: 20116898
TCMC2304
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.3 (ug/ml), Ref: 9461665
TCMC1801
TCMT1136 Neuraminidase Influenza A virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC2316
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 7381508
TCMC2316
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 3.12 (ug/ml), Ref: 7381508
TCMC1381
TCMT1251 Candida albicans Candida albicans IC50: 3 (ug/ml), Ref: 17112640
IC50: 2 (ug/ml), Ref: 12502337
TCMC1381
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 7 (ug/ml), Ref: 17112640
IC50: 45 (ug/ml), Ref: 12502337
TCMC1381
TCMT1286 Bacillus cereus Bacillus cereus MIC: 31.2 (ug/ml), Ref: 18951808
TCMC1381
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 31.2 (ug/ml), Ref: 18951808
MIC: 31.25 (ug/ml), Ref: 22169259
MIC: 62.5 (ug/ml), Ref: 22169259
MIC: 15.62 (ug/ml), Ref: 22169259
TCMC1381
TCMT1246 Escherichia coli Escherichia coli MIC: 2 (ug/ml), Ref: 20160051
MIC: 64 (ug/ml), Ref: 20160051
MIC: 0.5 (ug/ml), Ref: 20160051
MIC: 16 (ug/ml), Ref: 20160051
MIC: 0.25 (ug/ml), Ref: 20160051
MIC: 8 (ug/ml), Ref: 20160051
TCMC1381
TCMT1179 Escherichia coli ATCC 8739 Escherichia coli ATCC 8739 MIC: 8 (ug/ml), Ref: 20160051
TCMC1381
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 16 (ug/ml), Ref: 20160051
MIC: 32 (ug/ml), Ref: 20160051
MIC: 0.5 (ug/ml), Ref: 20160051
MIC: 8 (ug/ml), Ref: 20160051
MIC: 64 (ug/ml), Ref: 20160051
TCMC1381
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 32 (ug/ml), Ref: 20160051
MIC: 4 (ug/ml), Ref: 20160051
MIC: 16 (ug/ml), Ref: 20160051
MIC: 0.5 (ug/ml), Ref: 20160051
TCMC1381
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 64 (ug/ml), Ref: 20160051
MIC: 16 (ug/ml), Ref: 20160051
TCMC1381
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 64 (ug/ml), Ref: 20160051
MIC: 4 (ug/ml), Ref: 20160051
TCMC1381
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 8 (ug/ml), Ref: 20160051
MIC: 64 (ug/ml), Ref: 20160051
MIC: 1 (ug/ml), Ref: 20160051
TCMC1381
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 18 (ug/ml), Ref: 22280816
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC2251
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 7381508
TCMC2251
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 3.12 (ug/ml), Ref: 7381508
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC2351
TCMT1190 Plasmodium falciparum (isolate FcB1 / Columbia) Plasmodium falciparum FcB1/Columbia IC50: 16.7 (ug/ml), Ref: 21985060
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC1488
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 12.5 (ug/ml), Ref: 24479468
TCMC1901
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1236 Mycobacterium bovis Mycobacterium bovis BCG MIC: 26 (ug/ml), Ref: 18849164
TCMC1901
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1191 Bacillus megaterium Bacillus megaterium MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1286 Bacillus cereus Bacillus cereus MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1260 Streptococcus agalactiae Streptococcus agalactiae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1322 Streptococcus mitis Streptococcus mitis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1323 Corynebacterium pseudodiphtheriticum Corynebacterium pseudodiphtheriticum MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1324 Corynebacterium diphtheriae Corynebacterium diphtheriae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1319 Corynebacterium xerosis Corynebacterium xerosis MIC: 16 (ug/ml), Ref: 18849164
TCMC2365
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 34 (ug/ml), Ref: 18068371
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC2093
TCMT1251 Candida albicans Candida albicans MIC: 64 (ug/ml), Ref: 12932139
TCMC2093
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 64 (ug/ml), Ref: 12932139
TCMC795
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.6 (ug/ml), Ref: 15844943
TCMC2107
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 37.5 (ug/ml), Ref: 11678648
TCMC2107
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 20542692
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1255
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 7381508
MIC: 3.125 (ug/ml), Ref: 10.1039/C5MD00527B
MIC: 12.5 (ug/ml), Ref: 10.1039/C5MD00527B
MIC: 62.5 (ug/ml), Ref: 10.1039/C5MD00527B
TCMC1255
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 6.25 (ug/ml), Ref: 7381508
TCMC1255
TCMT1251 Candida albicans Candida albicans MIC: 25 (ug/ml), Ref: 7381508
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC2420
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 7381508
TCMC2420
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 25 (ug/ml), Ref: 7381508
TCMC2432
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 12.5 (ug/ml), Ref: 10360733
MIC: 6.25 (ug/ml), Ref: 10360733
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC2441
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 50 (ug/ml), Ref: 24479468
TCMC1256
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 1.56 (ug/ml), Ref: 7381508
TCMC1256
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 1.56 (ug/ml), Ref: 7381508
TCMC1113
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 15863332
TCMC2468
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 5 (ug/ml), Ref: 10654410
TCMC2468
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 2.5 (ug/ml), Ref: 10654410
TCMC1399
TCMT1286 Bacillus cereus Bacillus cereus MIC: 62.5 (ug/ml), Ref: 18951808
TCMC1399
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 18951808
MIC: 31.25 (ug/ml), Ref: 22169259
MIC: 62.5 (ug/ml), Ref: 22169259
MIC: 15.6 (ug/ml), Ref: 25137491
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2274
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 18171023
TCMC614
TCMT1454 Bacillus subtilis Bacillus subtilis IC50: 98.5 (ug/ml), Ref: 25981688
TCMC2196
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 10 (ug/ml), Ref: 22819942
MIC: 0.5 (ug/ml), Ref: 26253635
TCMC2196
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 1 (ug/ml), Ref: 23360475
MIC: 1 (ug/ml), Ref: 26253635
TCMC2196
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 6 (ug/ml), Ref: 26253635
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC1186
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 3430167
TCMC1186
TCMT1284 Penicillium expansum Penicillium expansum MIC: 50 (ug/ml), Ref: 3430167
TCMC2530
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 6.25 (ug/ml), Ref: 24479468
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2556
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 10 (ug/ml), Ref: 10654410
TCMC2556
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 10 (ug/ml), Ref: 10654410
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC1482
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.2 (ug/ml), Ref: 16153842
IC50: 1.43 (ug/ml), Ref: 25137491
IC50: 1.4 (ug/ml), Ref: 10.1039/C5MD00481K
IC50: 4.2 (nM), Ref: 19269069
TCMC1482
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 2 (ug/ml), Ref: 17112640
TCMC1482
TCMT1234 Bacillus coagulans Bacillus coagulans MIC: 2 (ug/ml), Ref: 17112640
TCMC1482
TCMT1235 Clostridium sporogenes Clostridium sporogenes MIC: 8 (ug/ml), Ref: 17112640
TCMC1482
TCMT1286 Bacillus cereus Bacillus cereus MIC: 3 (ug/ml), Ref: 17112640
TCMC1482
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3 (ug/ml), Ref: 17112640
MIC: 16 (ug/ml), Ref: 17112640
MIC: 6.25 (ug/ml), Ref: 17112640
MIC: 3.13 (ug/ml), Ref: 17112640
TCMC1482
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 6 (ug/ml), Ref: 17112640
TCMC1482
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 6 (ug/ml), Ref: 17112640
TCMC1482
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 5 (ug/ml), Ref: 17112640
TCMC1482
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 17112640
TCMC1482
TCMT1236 Mycobacterium bovis Mycobacterium bovis MIC: 20 (ug/ml), Ref: 17112640
TCMC1482
TCMT1237 Mycobacterium kansasii Mycobacterium kansasii MIC: 20 (ug/ml), Ref: 17112640
TCMC1482
TCMT1238 Mycobacterium xenopi Mycobacterium xenopi MIC: 20 (ug/ml), Ref: 17112640
TCMC1482
TCMT1239 Mycobacterium marinum Mycobacterium marinum MIC: 20 (ug/ml), Ref: 17112640
TCMC1482
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 20 (ug/ml), Ref: 17112640
MIC: 7.1 (ug/ml), Ref: 23369537
TCMC1482
TCMT1457 Leishmania major Leishmania major IC50: 2.5 (ug/ml), Ref: 26778149
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC915
TCMT1246 Escherichia coli Escherichia coli MIC: 1 (ug/ml), Ref: 25791674
TCMC915
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 0.5 (ug/ml), Ref: 25791674
TCMC915
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.25 (ug/ml), Ref: 25791674
TCMC2283
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 30 (ug/ml), Ref: 22280816
TCMC755
TCMT1251 Candida albicans Candida albicans IC50: 6 (ug/ml), Ref: 12502337
TCMC755
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC755
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 6.46 (ug/ml), Ref: 25564380
TCMC1329
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1898
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 12.5 (ug/ml), Ref: 22280816
TCMC1898
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 80.76 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1898
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 73 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 63.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2589
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 7381508
TCMC2589
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 6.25 (ug/ml), Ref: 7381508
TCMC2592
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3.12 (ug/ml), Ref: 7381508
TCMC2592
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 3.12 (ug/ml), Ref: 7381508
TCMC1105
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 51.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 50.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC1105
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 23534483
TCMC1105
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 1 (ug/ml), Ref: 23534483
TCMC1105
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 2 (ug/ml), Ref: 23534483
MIC: 4 (ug/ml), Ref: 23534483
TCMC2040
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 50.03 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2612
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 4 (ug/ml), Ref: 12932139
TCMC2612
TCMT1251 Candida albicans Candida albicans MIC: 16 (ug/ml), Ref: 12932139
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC2035
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2089
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 17210767
MIC: 50 (ug/ml), Ref: 19770280
MIC: 5 (ug/ml), Ref: 19770280
MIC: 31.25 (ug/ml), Ref: 20855745
MIC: 8 (ug/ml), Ref: 20855745
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC1516
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 64 (ug/ml), Ref: 12608861
MIC: 4 (ug/ml), Ref: 22677320
TCMC1516
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
MIC: 50 (ug/ml), Ref: 18313801
MIC: 18 (ug/ml), Ref: 22677320
MIC: 9 (ug/ml), Ref: 22677320
TCMC1516
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 25 (ug/ml), Ref: 17027268
TCMC1516
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 25 (ug/ml), Ref: 18313801
TCMC1516
TCMT1213 Neisseria gonorrhoeae Neisseria gonorrhoeae MIC: 16 (ug/ml), Ref: 12608861
TCMC1516
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 7 (ug/ml), Ref: 17394331
TCMC1516
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.8 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1516
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1516
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.8 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.063 (ug/ml), Ref: 9249972
IC50: 0.108 (ug/ml), Ref: 9249972
TCMC2654
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 0.087 (ug/ml), Ref: 9249972
TCMC1734
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 92.24 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC395
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC395
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC2673
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 7381508
TCMC2673
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 12.5 (ug/ml), Ref: 7381508
TCMC1733
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 17.2 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1123
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1123
TCMT1442 Leishmania donovani Leishmania donovani IC50: 25 (ug/ml), Ref: 15679330
TCMC2678
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 5 (ug/ml), Ref: 12444686
TCMC2680
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 16 (ug/ml), Ref: 19566082
TCMC2680
TCMT1251 Candida albicans Candida albicans MIC: 8 (ug/ml), Ref: 19566082
MIC: 64 (ug/ml), Ref: 19566082
TCMC2680
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 16 (ug/ml), Ref: 19566082
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC2693
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 5 (ug/ml), Ref: 10654410
TCMC2693
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 5 (ug/ml), Ref: 10654410
TCMC872
TCMT1444 Fusarium oxysporum Fusarium oxysporum MIC: 64 (ug/ml), Ref: 22850211
TCMC2703
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 25462220
TCMC1236
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2 (ug/ml), Ref: 19299148
TCMC1519
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 50 (ug/ml), Ref: 22280816
TCMC1792
TCMT1227 Streptococcus Streptococcus MIC: 25 (ug/ml), Ref: 9182126
TCMC2777
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 3430167
TCMC2777
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 3430167
TCMC1915
TCMT1347 Human rhinovirus 16 Human rhinovirus 16 IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1333 Human rhinovirus 1A Human rhinovirus 1A IC50: 0.02 (ug/ml), Ref: 17116681
TCMC1915
TCMT1241 Human rhinovirus 14 Human rhinovirus 14 IC50: 0.02 (ug/ml), Ref: 17116681
IC50: 100 (nM), Ref: 23977995
TCMC1801
TCMT1449 Influenza A virus Influenza A virus IC50: 1 (ug/ml), Ref: 14987066
IC50: 2.4 (nM), Ref: 19919060
IC50: 3.41 (nM), Ref: 15974612
IC50: 3.79 (nM), Ref: 16532013
IC50: 7.03 (nM), Ref: 19101157
IC50: 30 (nM), Ref: 25305333
IC50: 1.08 (nM), Ref: 9784165
IC50: 0.85 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 2.27 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 93.92 (nM), Ref: 20430633
IC50: 99.57 (nM), Ref: 20430633
IC50: 0.54 (nM), Ref: 20430633
IC50: 94.4 (nM), Ref: 20430633
IC50: 0.49 (nM), Ref: 20411974
IC50: 0.25 (nM), Ref: 20384296
IC50: 1 (nM), Ref: IC50: 95.43 (nM), Ref: 9461668
IC50: 78.12 (nM), Ref: 9461668
IC50: 75.29 (nM), Ref: 9461668
IC50: 1.84 (nM), Ref: 20166736
IC50: 1.59 (nM), Ref: 24673739
IC50: 0.34 (nM), Ref: 23675610
IC50: 0.25 (nM), Ref: 1431945
IC50: 3.64 (nM), Ref: 11170656
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC1915
TCMT1348 Human rhinovirus 2 Human rhinovirus 2 IC50: 0.01 (ug/ml), Ref: 23920485
IC50: 100 (nM), Ref: 23977995
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1174
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1174
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 55 (ug/ml), Ref: 25564380
TCMC1174
TCMT1442 Leishmania donovani Leishmania donovani IC50: 0.6 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1064
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 15 (ug/ml), Ref: 11170636
TCMC2812
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 7381508
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1113
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 16 (nM), Ref: 17263522
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC2274
TCMT1121 Sialidase Clostridium perfringens IC50: 90 (nM), Ref: 21911291
TCMC1801
TCMT1162 Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1)) Ki: 1.1 (nM), Ref: IC50: 0.1 (nM), Ref: 23398362
IC50: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1164 Neuraminidase Influenza A virus (A/chicken/Yogjakarta/BBVet-IX/2004(H5N1)) Ki: 4.9 (nM), Ref: 20579892
IC50: 4.9 (nM), Ref: 19708637
IC50: 3.7 (nM), Ref:
TCMC1801
TCMT1161 Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1)) Ki: 7.9 (nM), Ref: 20579892
IC50: 10.8 (nM), Ref: 10.6019/CHEMBL1201861
TCMC1801
TCMT1163 Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1)) IC50: 0.3 (nM), Ref: 9322359
IC50: 0.2 (nM), Ref: Ki: 0.1 (nM), Ref: 17067157
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/swine/Belzig/2/2001(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/New Caledonia/20/1999(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Yamagata/32/1989(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1099 Neuraminidase Influenza A virus IC50: 0.000681 (ug/ml), Ref: PubChem BioAssay data set
IC50: 1 (nM), Ref: 23993676
IC50: 7.09 (nM), Ref: 16936720
TCMC1801
TCMT1151 Neuraminidase Influenza B virus IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Hong Kong/1/1968(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1160 Neuraminidase Influenza A virus (A/Aichi/2/1968(H3N2)) IC50: 1.55 (nM), Ref: 20185316
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/whooper swan/Mongolia/1/2009(H5N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/Wisconsin/67/2005(H3N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Shandong/LY/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1085 Neuraminidase Influenza A virus (A/Perth/16/2009(H3N2)) IC50: 2.57 (nM), Ref: IC50: 1.39 (nM), Ref:
TCMC1801
TCMT1151 Neuraminidase Influenza B virus (B/Memphis/3/89) IC50: 5 (nM), Ref: 23993676
Ki: 1.1 (nM), Ref: 22705001
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/California/07/2009(H1N1)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC1801
TCMT1136 Neuraminidase Influenza A virus (A/chicken/Sandong/Li/2008(H9N2)) IC50: 0.03974 (ug/ml), Ref: 17958396
IC50: 0.00494 (ug/ml), Ref: 20359898
IC50: 0.00494 (ug/ml), Ref: 17536859
IC50: 0.03974 (ug/ml), Ref: 19115838
IC50: 0.02109 (ug/ml), Ref: 18212108
IC50: 5.13 (ug/ml), Ref: 18077363
IC50: 0.02109 (ug/ml), Ref: 21741130
IC50: 5.13 (ug/ml), Ref: 19159272
IC50: 0.03974 (ug/ml), Ref: 20308368
IC50: 0.00494 (ug/ml), Ref: 24900628
IC50: 10 (nM), Ref: 2746258
IC50: 20 (nM), Ref: 17536859
IC50: 2.81 (nM), Ref: 25530833
IC50: 1.43 (nM), Ref: 12729671
IC50: 2.17 (nM), Ref: 11454459
IC50: 2.12 (nM), Ref: 11000047
IC50: 2.56 (nM), Ref: 11000047
IC50: 1.78 (nM), Ref: 18163588
IC50: 1.25 (nM), Ref: 8289060
IC50: 3.65 (nM), Ref: 24195447
IC50: 0.3 (nM), Ref: 7964782
IC50: 0.2 (nM), Ref: IC50: 1.12 (nM), Ref: 23270663
IC50: 0.925 (nM), Ref: 23270663
IC50: 2.39 (nM), Ref: 23270663
IC50: 0.658 (nM), Ref: 23270663
IC50: 1.26 (nM), Ref: 23270663
IC50: 1.6 (nM), Ref: 23270663
IC50: 1.71 (nM), Ref: 23270663
IC50: 0.2 (nM), Ref: 10.6019/CHEMBL1201861
IC50: 0.925 (nM), Ref: 21924611
IC50: 0.885 (nM), Ref: 15043409
IC50: 50 (nM), Ref: 7528786
Ki: 0.1 (nM), Ref: 19651906
IC50: 1.9 (nM), Ref: 23189988
IC50: 1.99 (nM), Ref: 20553004
IC50: 1.56 (nM), Ref: 24582402
IC50: 16 (nM), Ref: 19734910
IC50: 1.58 (nM), Ref: 20945914
IC50: 1.54 (nM), Ref: IC50: 2.39 (nM), Ref: IC50: 1.08 (nM), Ref: IC50: 1.34 (nM), Ref: IC50: 0.2 (nM), Ref: 26034885
IC50: 50 (nM), Ref: 12088425
IC50: 0.06 (nM), Ref: IC50: 4.95 (nM), Ref: 19734910
IC50: 0.87 (nM), Ref: IC50: 1.2 (nM), Ref: IC50: 80 (nM), Ref: 22276679
Ki: 0.9 (nM), Ref: 17844994
IC50: 1.08 (nM), Ref: 11975486
IC50: 0.711 (nM), Ref: 11575942
IC50: 3.44 (nM), Ref: 15730251
IC50: 0.981 (nM), Ref: 16248836
IC50: 1.09 (nM), Ref: 12828461
IC50: 1.59 (nM), Ref: 16933872
IC50: 1 (nM), Ref: 17724156
IC50: 8 (nM), Ref: 19349512
IC50: 1.5 (nM), Ref: IC50: 0.5 (nM), Ref: IC50: 0.16 (nM), Ref: IC50: 0.19 (nM), Ref: IC50: 1.7 (nM), Ref: IC50: 2.28 (nM), Ref: IC50: 2.8 (nM), Ref: 18077425
IC50: 0.706 (nM), Ref: 24582402
IC50: 1.33 (nM), Ref: 24582402
IC50: 0.785 (nM), Ref: 19700225
IC50: 1.86 (nM), Ref: 19856923
IC50: 10 (nM), Ref: 14510595
IC50: 1.7 (nM), Ref: 15043424
IC50: 37.2 (nM), Ref: 17296744
IC50: 24.9 (nM), Ref: 18955520
IC50: 2.94 (nM), Ref: 18955520
IC50: 1.18 (nM), Ref:
TCMC2338
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 8.8 (nM), Ref: 17503850
TCMC1482
TCMT1186 Plasmodium yoelii yoelii Plasmodium yoelii yoelii IC50: 0.927 (nM), Ref: 18212104
IC50: 0.927 (nM), Ref: 22122518
TCMC2089
TCMT1229 Enterococcus faecalis Enterococcus faecalis MBC: 0.5 (nM), Ref: 21794958
TCMC1801
TCMT1296 Influenza A virus H3N2 Influenza A virus H3N2 IC50: 18.5 (nM), Ref: 12542349
TCMC1915
TCMT1285 Human coxsackievirus B3 Human coxsackievirus B3 IC50: 2.5 (nM), Ref: 13678412