Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 8710 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4050 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6680 (nM), Ref: 20185318 Ki: 6680 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8010 (nM), Ref: 20185318 Ki: 8010 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 5330 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 5230 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6720 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7760 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 5960 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9600 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7570 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 980 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1070 (nM), Ref: 20185318 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 5157.65 (nM), Ref: |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 1261 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 56 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 17 (nM), Ref: 20696580 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 212.9 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.4 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 54.9 (nM), Ref: 26498393 Ki: 220 (nM), Ref: 26498393 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 440 (nM), Ref: 26498393 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 168 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 5591.2 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 423.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4.9 (nM), Ref: 26498393 |
|
TCMT107 | Glutamate receptor ionotropic kainate 2 | Homo sapiens |
Ki: 1106 (nM), Ref: 10821708 |
|
TCMT108 | Glutamate receptor ionotropic, AMPA 1 | Homo sapiens |
Ki: 1360 (nM), Ref: 9357531 |
|
TCMT109 | Glutamate receptor ionotropic, AMPA 2 | Homo sapiens |
Ki: 940 (nM), Ref: 9357531 |
|
TCMT110 | Glutamate receptor ionotropic, AMPA 4 | Homo sapiens |
Ki: 868 (nM), Ref: 9357531 |
|
TCMT111 | Glutamate receptor ionotropic kainate 5 | Homo sapiens |
Ki: 701 (nM), Ref: 9357531 |
|
TCMT660 | Metabotropic glutamate receptor 8 | Homo sapiens |
IC50: 5.7 (nM), Ref: 15603952 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 613 (nM), Ref: 16250647 |
|
TCMT653 | Metabotropic glutamate receptor 1 | Homo sapiens |
Ki: 250 (nM), Ref: 17725337 Ki: 570 (nM), Ref: 19042134 Ki: 1584.89 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT654 | Metabotropic glutamate receptor 5 | Homo sapiens |
Ki: 390 (nM), Ref: 17725337 Ki: 1160 (nM), Ref: 19042134 Ki: 4677.35 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT657 | Metabotropic glutamate receptor 4 | Homo sapiens |
Ki: 2400 (nM), Ref: 17725337 Ki: 1400 (nM), Ref: 19042134 Ki: 3235.94 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT655 | Metabotropic glutamate receptor 2 | Homo sapiens |
Ki: 6400 (nM), Ref: 19042134 Ki: 1819.7 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT664 | Excitatory amino acid transporter 3 | Homo sapiens |
Ki: 51 (nM), Ref: 18578477 |
|
TCMT656 | Metabotropic glutamate receptor 3 | Homo sapiens |
Ki: 57.54 (nM), Ref: 10.1039/C1MD00186H |
|
TCMT599 | Ubiquitin-conjugating enzyme E2 N | Homo sapiens | IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref: |
|
TCMT38 | Dopamine D2 receptor | Homo sapiens |
Ki: 1.89 (nM), Ref: 10465538 Ki: 759 (nM), Ref: 10465538 Ki: 572 (nM), Ref: 8893836 Ki: 20 (nM), Ref: 10691700 Ki: 17 (nM), Ref: 10691700 Ki: 450 (nM), Ref: 18834111 Ki: 360 (nM), Ref: 18834111 Ki: 2100 (nM), Ref: 20155917 Ki: 2.9 (nM), Ref: 20155917 Ki: 2100 (nM), Ref: 22846798 Ki: 422 (nM), Ref: 23134120 Ki: 110 (nM), Ref: 23428965 Ki: 190 (nM), Ref: 23428965 Ki: 2100 (nM), Ref: 23727194 Ki: 8 (nM), Ref: 24138311 Ki: 8.73 (nM), Ref: 27035329 Ki: 3690 (nM), Ref: 27035329 Ki: 48 (nM), Ref: 27132867 |
|
TCMT651 | Dopamine D3 receptor | Homo sapiens |
Ki: 13.2 (nM), Ref: 8893836 Ki: 50 (nM), Ref: 10691700 Ki: 240 (nM), Ref: 18834111 Ki: 72 (nM), Ref: 18834111 Ki: 15 (nM), Ref: 22846798 Ki: 20 (nM), Ref: 23134120 Ki: 21 (nM), Ref: 23428965 Ki: 15 (nM), Ref: 23727194 Ki: 7.58 (nM), Ref: 27035329 Ki: 293 (nM), Ref: 27035329 |
|
TCMT635 | Dopamine transporter | Homo sapiens |
Ki: 6400 (nM), Ref: 14592523 IC50: 460 (nM), Ref: 14592523 |
|
TCMT634 | Norepinephrine transporter | Homo sapiens |
IC50: 6.63 (nM), Ref: 14592523 |
|
TCMT648 | Dopamine D4 receptor | Homo sapiens |
Ki: 1.2 (nM), Ref: 10691700 Ki: 6.2 (nM), Ref: 18834111 Ki: 8.9 (nM), Ref: 23428965 |
|
TCMT316 | Melatonin receptor 1A | Homo sapiens |
Ki: 7100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
|
TCMT317 | Melatonin receptor 1B | Homo sapiens |
Ki: 9100 (nM), Ref: 10.1016/S0960-894X(97)00444-7 |
|
TCMT27 | Dopamine D1 receptor | Homo sapiens |
Ki: 4470 (nM), Ref: 23134120 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 320 (nM), Ref: 22261024 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT22 | Intestinal alkaline phosphatase | Homo sapiens | IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 4500 (nM), Ref: 22261024 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 6211.2 (nM), Ref: 26498393 Ki: 410 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 75.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 3.8 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 52.1 (nM), Ref: 26498393 Ki: 170 (nM), Ref: 26498393 |
|
TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens |
IC50: 2800 (nM), Ref: 15887952 IC50: 2800 (nM), Ref: 15887952 IC50: 1200 (nM), Ref: 12502307 IC50: 2800 (nM), Ref: |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 7300 (nM), Ref: 21030469 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 718.7 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.2 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 56.4 (nM), Ref: 26498393 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT254 | Carbonyl reductase [NADPH] 1 | Homo sapiens |
Ki: 2030 (nM), Ref: 19097799 |
|
TCMT66 | Estradiol 17-beta-dehydrogenase 2 | Homo sapiens |
IC50: 9900 (nM), Ref: 18533708 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10.2 (nM), Ref: 20413308 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7078.5 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 371.5 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 52.5 (nM), Ref: 26498393 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 5200 (nM), Ref: 18558747 |