TCM Putative Target References: TCMF525


Targeted Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.
.
Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC879
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 230 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC417
TCMT127 Poly [ADP-ribose] polymerase-1 Homo sapiens IC50: 7585.78 (nM), Ref: 23574272
IC50: 7500 (nM), Ref: 23574272
TCMC417
TCMT128 Tankyrase-2 Homo sapiens IC50: 870.96 (nM), Ref: 23574272
IC50: 870 (nM), Ref: 23574272
TCMC417
TCMT129 Tankyrase-1 Homo sapiens IC50: 645.65 (nM), Ref: 23574272
IC50: 630 (nM), Ref: 23574272
TCMC417
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2000 (nM), Ref: 24368208
TCMC1173
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9430 (nM), Ref: 20185318
Ki: 9430 (nM), Ref: 26498394
TCMC1173
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9780 (nM), Ref: 20185318
Ki: 9780 (nM), Ref: 26498394
TCMC1173
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 9870 (nM), Ref: 20185318
TCMC1173
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7410 (nM), Ref: 20185318
TCMC1173
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 8450 (nM), Ref: 20185318
TCMC1173
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 7040 (nM), Ref: 20185318
TCMC1173
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2400 (nM), Ref: 20185318
TCMC1173
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2890 (nM), Ref: 20185318
TCMC943
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 810 (nM), Ref: 20100662
TCMC943
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 7000 (nM), Ref: 22940448
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 5490 (nM), Ref: 10.1007/s00044-010-9529-5
TCMC61
TCMT193 Nuclear factor NF-kappa-B p65 subunit Homo sapiens IC50: 250 (nM), Ref: 21513293
TCMC61
TCMT194 Mitogen-activated protein kinase kinase kinase 7 Homo sapiens IC50: 80 (nM), Ref: 25529738
IC50: 11 (nM), Ref: 26481152
IC50: 8.1 (nM), Ref: 26481152
IC50: 9 (nM), Ref: 27448772
TCMC61
TCMT80 MAP kinase ERK2 Homo sapiens IC50: 6800 (nM), Ref: 25529738
TCMC61
TCMT195 Dual specificity mitogen-activated protein kinase kinase 1 Homo sapiens IC50: 80 (nM), Ref: 25529738
TCMC61
TCMT196 Dual specificity mitogen-activated protein kinase kinase 7 Homo sapiens IC50: 1300 (nM), Ref: 25529738
TCMC2051
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 8710 (nM), Ref: 22892213
TCMC2051
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4050 (nM), Ref: 22892213
TCMC2051
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 960 (nM), Ref: 22892213
TCMC908
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 6000 (nM), Ref: 15689157
IC50: 6000 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC908
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 2600 (nM), Ref: 15267241
IC50: 1 (nM), Ref: 20413308
IC50: 800 (nM), Ref: 10.1039/C3MD00166K
IC50: 500 (nM), Ref: 26301554
TCMC908
TCMT223 Aldose reductase Homo sapiens IC50: 8500 (nM), Ref: 18165015
TCMC908
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens IC50: 670 (nM), Ref: 19097799
Ki: 110 (nM), Ref: 19097799
TCMC908
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 153 (nM), Ref: 20696580
IC50: 1290 (nM), Ref: 23600958
TCMC908
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 84 (nM), Ref: 20696580
IC50: 54 (nM), Ref: 20832301
IC50: 570 (nM), Ref: 23600958
TCMC908
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 24 (nM), Ref: 20696580
TCMC908
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 5225 (nM), Ref: 20832301
TCMC908
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 5490 (nM), Ref: 22487176
Ki: 5420 (nM), Ref: 22487176
TCMC908
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4380 (nM), Ref: 22487176
Ki: 4310 (nM), Ref: 22487176
TCMC908
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 2650 (nM), Ref: 22487176
Ki: 2710 (nM), Ref: 22487176
TCMC908
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8960 (nM), Ref: 22487176
Ki: 9070 (nM), Ref: 22487176
Ki: 34.7 (nM), Ref: 26498393
TCMC908
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 537.75 (nM), Ref: 26498393
TCMC908
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 171.41 (nM), Ref: 26498393
TCMC903
TCMT175 G-protein coupled bile acid receptor 1 Homo sapiens IC50: 6000 (nM), Ref: 20801037
TCMC948
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6680 (nM), Ref: 20185318
Ki: 6680 (nM), Ref: 26498394
TCMC948
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8010 (nM), Ref: 20185318
Ki: 8010 (nM), Ref: 26498394
TCMC948
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5330 (nM), Ref: 20185318
TCMC948
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 5230 (nM), Ref: 20185318
TCMC948
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6720 (nM), Ref: 20185318
TCMC948
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7760 (nM), Ref: 20185318
TCMC948
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 5960 (nM), Ref: 20185318
TCMC948
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9600 (nM), Ref: 20185318
TCMC948
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7570 (nM), Ref: 20185318
TCMC948
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 980 (nM), Ref: 20185318
TCMC948
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1070 (nM), Ref: 20185318
TCMC948
TCMT223 Aldose reductase Homo sapiens IC50: 140 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1495
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 1000 (nM), Ref: 20471252
IC50: 1000 (nM), Ref: 25461324
IC50: 1000 (nM), Ref: 25461324
Ki: 9300 (nM), Ref: 27460668
TCMC1495
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 1000 (nM), Ref: 20471252
Ki: 6800 (nM), Ref: 27460668
TCMC1495
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1495
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC2013
TCMT223 Aldose reductase Homo sapiens IC50: 2700 (nM), Ref: 22261024
TCMC1433
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6863.3 (nM), Ref: 26498393
TCMC1433
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 62.2 (nM), Ref: 26498393
TCMC1433
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 26.6 (nM), Ref: 26498393
TCMC1433
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 399.7 (nM), Ref: 26498393
TCMC2037
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9920 (nM), Ref: 18501600
Ki: 9900 (nM), Ref: 18579385
Ki: 9900 (nM), Ref: 26520662
TCMC2037
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 7120 (nM), Ref: 18501600
Ki: 7100 (nM), Ref: 18579385
Ki: 7100 (nM), Ref: 26520662
TCMC2037
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 8800 (nM), Ref: 18579385
TCMC1871
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9200 (nM), Ref: 20185318
Ki: 9200 (nM), Ref: 20590092
Ki: 9200 (nM), Ref: 20674354
Ki: 9200 (nM), Ref: 21282059
Ki: 9200 (nM), Ref: 23265898
Ki: 9200 (nM), Ref: 23010455
Ki: 9200 (nM), Ref: 24189056
TCMC1871
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8800 (nM), Ref: 20185318
Ki: 8800 (nM), Ref: 20590092
Ki: 8800 (nM), Ref: 20674354
Ki: 8800 (nM), Ref: 21282059
Ki: 8800 (nM), Ref: 23265898
Ki: 8800 (nM), Ref: 23010455
Ki: 8800 (nM), Ref: 24189056
Ki: 8800 (nM), Ref: 26520662
TCMC1871
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9500 (nM), Ref: 20185318
Ki: 9500 (nM), Ref: 20590092
Ki: 9500 (nM), Ref: 20674354
Ki: 9500 (nM), Ref: 23010455
TCMC1871
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 2700 (nM), Ref: 20185318
Ki: 2700 (nM), Ref: 20590092
Ki: 2700 (nM), Ref: 20674354
Ki: 2700 (nM), Ref: 23010455
TCMC1871
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 5500 (nM), Ref: 20185318
Ki: 5500 (nM), Ref: 20590092
Ki: 5500 (nM), Ref: 20674354
Ki: 5500 (nM), Ref: 21282059
Ki: 5500 (nM), Ref: 21332115
Ki: 5500 (nM), Ref: 23265898
Ki: 5500 (nM), Ref: 23265903
Ki: 5500 (nM), Ref: 23010455
Ki: 5500 (nM), Ref: 24189056
Ki: 5500 (nM), Ref: 26073005
Ki: 5500 (nM), Ref: 26520662
TCMC962
TCMT45 Beta amyloid A4 protein Homo sapiens Ki: 0.208 (nM), Ref: 17004725
IC50: 800 (nM), Ref: 17270435
IC50: 3900 (nM), Ref: 26099993
TCMC962
TCMT566 Nitric oxide synthase, inducible Homo sapiens IC50: 6000 (nM), Ref: 18077363
TCMC962
TCMT87 Cytochrome P450 2C9 Homo sapiens IC50: 4300 (nM), Ref: 18249473
TCMC962
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 8500 (nM), Ref: 19128977
TCMC962
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2410 (nM), Ref: 20674354
TCMC962
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 380 (nM), Ref: 20674354
TCMC962
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4970 (nM), Ref: 20674354
TCMC962
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9460 (nM), Ref: 20674354
TCMC962
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 9940 (nM), Ref: 20674354
TCMC962
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 9300 (nM), Ref: 20674354
TCMC962
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4050 (nM), Ref: 20674354
TCMC962
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 3480 (nM), Ref: 20674354
TCMC962
TCMT225 Carbonic anhydrase XIII Homo sapiens Ki: 6850 (nM), Ref: 20674354
TCMC962
TCMT44 Glyoxalase I Homo sapiens Ki: 10000 (nM), Ref: 21237663
TCMC962
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 7410 (nM), Ref:
TCMC962
TCMT46 Coagulation factor III Homo sapiens IC50: 199.63 (nM), Ref: 10.1007/s00044-012-0330-5
IC50: 199.63 (nM), Ref: 23199480
TCMC962
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 8600 (nM), Ref: 23245570
TCMC962
TCMT174 11-beta-hydroxysteroid dehydrogenase 1 Homo sapiens IC50: 4501 (nM), Ref: 23800686
TCMC962
TCMT570 Aminopeptidase N Homo sapiens IC50: 10000 (nM), Ref: 23860593
TCMC962
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 3900 (nM), Ref: 24920381
IC50: 500 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
IC50: 600 (nM), Ref: 24920381
TCMC962
TCMT164 Cyclooxygenase-1 Homo sapiens IC50: 8100 (nM), Ref: 24920381
TCMC962
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 600 (nM), Ref: 24920381
IC50: 1200 (nM), Ref: 24920381
TCMC962
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 1200 (nM), Ref: 24920381
TCMC962
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5300 (nM), Ref: 25088549
TCMC962
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 25730130
TCMC2119
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 9140 (nM), Ref: 20185318
TCMC2119
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9010 (nM), Ref: 20185318
TCMC2119
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8200 (nM), Ref: 20185318
TCMC2119
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7810 (nM), Ref: 20185318
TCMC2119
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7550 (nM), Ref: 20185318
TCMC2119
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6340 (nM), Ref: 20185318
TCMC2119
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8580 (nM), Ref: 20185318
TCMC2119
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 3190 (nM), Ref: 20185318
TCMC2119
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4150 (nM), Ref: 20185318
TCMC1429
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 2700 (nM), Ref: 17378609
TCMC1429
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 1050 (nM), Ref: 18533708
TCMC1429
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 360 (nM), Ref: 18533708
TCMC1429
TCMT187 Androgen Receptor Homo sapiens IC50: 9700 (nM), Ref: 19592245
TCMC1429
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 716 (nM), Ref: 20696580
TCMC1429
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 632 (nM), Ref: 20696580
TCMC1429
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 47 (nM), Ref: 20696580
TCMC1429
TCMT223 Aldose reductase Homo sapiens IC50: 10000 (nM), Ref: 22261024
TCMC1429
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 2320 (nM), Ref: 23411073
TCMC1429
TCMT591 Estrogen-related receptor alpha Homo sapiens IC50: 9640 (nM), Ref: 23656512
TCMC1429
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 10000 (nM), Ref: 26322379
TCMC1429
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 9525.7 (nM), Ref: 26498393
TCMC1429
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 25 (nM), Ref: 26498393
TCMC1429
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 145.9 (nM), Ref: 26498393
TCMC1429
TCMT159 Tyrosinase Homo sapiens IC50: 1000 (nM), Ref: 26841168
TCMC1285
TCMT33 Cytochrome P450 3A4 Homo sapiens Ki: 399 (nM), Ref: 16248836
TCMC2188
TCMT223 Aldose reductase Homo sapiens IC50: 2030 (nM), Ref: 10.1007/s00044-010-9412-4
TCMC1965
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 452.6 (nM), Ref: 26498393
TCMC1965
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 515 (nM), Ref: 26498393
TCMC1411
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 1261 (nM), Ref: 20696580
TCMC1411
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 56 (nM), Ref: 20696580
TCMC1411
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 17 (nM), Ref: 20696580
TCMC1411
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 212.9 (nM), Ref: 26498393
TCMC1411
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.4 (nM), Ref: 26498393
TCMC1411
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 54.9 (nM), Ref: 26498393
Ki: 220 (nM), Ref: 26498393
TCMC1411
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 440 (nM), Ref: 26498393
TCMC13
TCMT23 Alkaline phosphatase, tissue-nonspecific isozyme Homo sapiens IC50: 407 (nM), Ref:
TCMC1620
TCMT223 Aldose reductase Homo sapiens IC50: 88 (nM), Ref: 22236472
TCMC1620
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 130 (nM), Ref: 22236472
TCMC1424
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2100 (nM), Ref: 17994701
TCMC42
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 8390 (nM), Ref: 26696252
TCMC42
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2540 (nM), Ref: 26696252
TCMC2054
TCMT240 Salivary alpha-amylase Homo sapiens IC50: 9640 (nM), Ref: 18507367
TCMC2054
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 6610 (nM), Ref:
TCMC2054
TCMT283 Receptor-type tyrosine-protein phosphatase S Homo sapiens IC50: 600 (nM), Ref: 26602279
TCMC737
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 168 (nM), Ref: 26498393
TCMC737
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 5591.2 (nM), Ref: 26498393
TCMC737
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 423.7 (nM), Ref: 26498393
TCMC737
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4.9 (nM), Ref: 26498393
TCMC694
TCMT230 Estradiol 17-beta-dehydrogenase 3 Homo sapiens IC50: 758 (nM), Ref: 11086723
IC50: 758 (nM), Ref: 16078844
TCMC694
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 20 (nM), Ref: 8035427
Ki: 35 (nM), Ref: 26469743
TCMC1786
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3900 (nM), Ref: 16580200
IC50: 7600 (nM), Ref: 18798681
IC50: 4200 (nM), Ref: 19702283
IC50: 3840 (nM), Ref: 22044245
IC50: 5600 (nM), Ref: 22690646
IC50: 9500 (nM), Ref: 21453996
Ki: 6000 (nM), Ref: 21453996
IC50: 5050.1 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 3370 (nM), Ref: 10.1007/s00044-010-9529-5
IC50: 2600 (nM), Ref: 23357636
IC50: 1100 (nM), Ref: 23434422
IC50: 3020 (nM), Ref: 23942421
IC50: 2010 (nM), Ref: 24090912
IC50: 1900 (nM), Ref: 24684845
IC50: 3020 (nM), Ref: 25497963
IC50: 9500 (nM), Ref: 25264584
Ki: 6000 (nM), Ref: 25264584
IC50: 1030 (nM), Ref: 25595683
IC50: 1170 (nM), Ref: 25600405
IC50: 3020 (nM), Ref: 25872983
IC50: 1000 (nM), Ref: 26083682
IC50: 1536 (nM), Ref: 26100442
IC50: 700 (nM), Ref: 26115570
IC50: 700 (nM), Ref: 26253631
IC50: 1536 (nM), Ref: 26481657
IC50: 730 (nM), Ref: 26711144
IC50: 3020 (nM), Ref: 26774579
IC50: 1536 (nM), Ref: 27123900
TCMC1786
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 4000 (nM), Ref: 21561086
Ki: 3560 (nM), Ref: 21561086
Ki: 660 (nM), Ref: 21561086
Ki: 940 (nM), Ref: 21561086
Ki: 160 (nM), Ref: 21561086
Ki: 72 (nM), Ref: 21561086
IC50: 90 (nM), Ref: 21561086
TCMC1786
TCMT190 T-cell protein-tyrosine phosphatase Homo sapiens IC50: 4230 (nM), Ref: 24684845
IC50: 4440 (nM), Ref: 25497963
IC50: 5460 (nM), Ref: 26100442
IC50: 5460 (nM), Ref: 26481657
IC50: 5460 (nM), Ref: 27123900
TCMC1786
TCMT563 Dual specificity phosphatase Cdc25B Homo sapiens IC50: 980 (nM), Ref: 25497963
TCMC1735
TCMT599 Ubiquitin-conjugating enzyme E2 N Homo sapiens IC50: 8695 (nM), Ref: IC50: 5771 (nM), Ref: IC50: 6662 (nM), Ref:
TCMC315
TCMT46 Coagulation factor III Homo sapiens IC50: 14.98 (nM), Ref: 23199480
TCMC1844
TCMT113 Delta opioid receptor Homo sapiens Ki: 8400 (nM), Ref: 26035635
TCMC1844
TCMT510 Stem cell growth factor receptor Homo sapiens IC50: 600 (nM), Ref: 26807861
IC50: 1500 (nM), Ref: 26807861
TCMC632
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 2100 (nM), Ref: 23388705
IC50: 3300 (nM), Ref: 23388705
TCMC632
TCMT709 Sodium/nucleoside cotransporter 2 Homo sapiens Ki: 5300 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 1800 (nM), Ref: 23388705
IC50: 5500 (nM), Ref: 23388705
TCMC632
TCMT296 Adenosine A1 receptor Homo sapiens IC50: 2.344 (nM), Ref: 26756468
TCMC632
TCMT112 Adenosine A3 receptor Homo sapiens IC50: 1.148 (nM), Ref: 26756468
TCMC1956
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 1080 (nM), Ref: 21282059
TCMC1956
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 470 (nM), Ref: 21282059
TCMC1956
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 4450 (nM), Ref: 21282059
TCMC1956
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4090 (nM), Ref: 21282059
TCMC1956
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4720 (nM), Ref: 21669522
Ki: 4720 (nM), Ref: 22687439
TCMC1956
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 2450 (nM), Ref: 22687439
TCMC1956
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 690 (nM), Ref: 22668600
TCMC1956
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7870 (nM), Ref: 22668600
TCMC1113
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 400 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC43
TCMT301 Prostaglandin E synthase Homo sapiens IC50: 220 (nM), Ref: 26588603
IC50: 200 (nM), Ref: 10.1039/C5MD00278H
TCMC43
TCMT565 Histone acetyltransferase p300 Homo sapiens IC50: 6500 (nM), Ref: 26701186
TCMC43
TCMT208 Monoamine oxidase A Homo sapiens Ki: 710 (nM), Ref: 26819666
TCMC43
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3100 (nM), Ref: 27190601
IC50: 1500 (nM), Ref: 27190601
TCMC2142
TCMT156 Cytochrome P450 19A1 Homo sapiens Ki: 600 (nM), Ref: 6827528
TCMC2142
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 10000 (nM), Ref: 14552748
TCMC2142
TCMT187 Androgen Receptor Homo sapiens IC50: 3.9 (nM), Ref: 15456242
IC50: 2.7 (nM), Ref: 16309907
IC50: 4.571 (nM), Ref: 22746350
IC50: 4.17 (nM), Ref: 25646649
IC50: 4.27 (nM), Ref: 25646649
TCMC2142
TCMT99 Testis-specific androgen-binding protein Homo sapiens IC50: 14 (nM), Ref: 17149875
TCMC2142
TCMT725 Voltage-gated L-type calcium channel alpha-1C subunit Homo sapiens IC50: 34 (nM), Ref: 22761000
IC50: 38.4 (nM), Ref: 22761000
TCMC876
TCMT560 Coagulation factor X Homo sapiens IC50: 720 (nM), Ref: 9834152
Ki: 450 (nM), Ref: 9834152
TCMC156
TCMT327 Vanilloid receptor Homo sapiens IC50: 35 (nM), Ref: 16000002
TCMC1624
TCMT560 Coagulation factor X Homo sapiens IC50: 280 (nM), Ref: 9834152
Ki: 690 (nM), Ref: 9834152
TCMC1741
TCMT161 Hydroxycarboxylic acid receptor 2 Homo sapiens IC50: 140 (nM), Ref: 17994679
IC50: 140 (nM), Ref: 18029181
Ki: 50 (nM), Ref: 18665582
IC50: 150 (nM), Ref: 18752940
IC50: 140 (nM), Ref: 19307116
IC50: 130 (nM), Ref: 18760600
IC50: 140 (nM), Ref: 19309152
IC50: 140 (nM), Ref: 19592242
IC50: 140 (nM), Ref: 19592242
Ki: 82 (nM), Ref: 20184326
Ki: 104 (nM), Ref: 20184326
IC50: 140 (nM), Ref: 20444602
IC50: 140 (nM), Ref: 20615702
IC50: 249 (nM), Ref: 25737085
TCMC1446
TCMT83 Lymphocyte differentiation antigen CD38 Homo sapiens IC50: 6300 (nM), Ref: 21641214
TCMC1758
TCMT247 Alpha-2a adrenergic receptor Homo sapiens Ki: 66 (nM), Ref: 8632424
TCMC1758
TCMT243 Alpha-2c adrenergic receptor Homo sapiens Ki: 63 (nM), Ref: 8632424
TCMC1758
TCMT559 Beta-2 adrenergic receptor Homo sapiens Ki: 3300 (nM), Ref: 27132867
TCMC1758
TCMT38 Dopamine D2 receptor Homo sapiens Ki: 1300 (nM), Ref: 27132867
TCMC1609
TCMT44 Glyoxalase I Homo sapiens IC50: 560 (nM), Ref: 18258440
IC50: 560 (nM), Ref: 21669529
TCMC1609
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18778944
TCMC1609
TCMT737 DNA dC->dU-editing enzyme APOBEC-3G Homo sapiens IC50: 2390 (nM), Ref:
TCMC1609
TCMT739 G-protein coupled receptor 35 Homo sapiens IC50: 2120 (nM), Ref: 24900447
TCMC1609
TCMT558 DNA topoisomerase II alpha Homo sapiens IC50: 390 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1609
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2800 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1609
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1690 (nM), Ref: 23411073
TCMC1609
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1200 (nM), Ref: 23484434
IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC1609
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 3000 (nM), Ref: 25086914
TCMC1609
TCMT740 PI3-kinase p110-gamma subunit Homo sapiens IC50: 4720 (nM), Ref: 25050878
TCMC1609
TCMT13 DNA-(apurinic or apyrimidinic site) lyase Homo sapiens IC50: 320 (nM), Ref: 25280182
TCMC1399
TCMT223 Aldose reductase Homo sapiens IC50: 320 (nM), Ref: 22261024
TCMC2031
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1409
TCMT22 Intestinal alkaline phosphatase Homo sapiens IC50: 5250 (nM), Ref: IC50: 8960 (nM), Ref:
TCMC1409
TCMT223 Aldose reductase Homo sapiens IC50: 4500 (nM), Ref: 22261024
TCMC1409
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6211.2 (nM), Ref: 26498393
Ki: 410 (nM), Ref: 26498393
TCMC1409
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 75.7 (nM), Ref: 26498393
TCMC1409
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 3.8 (nM), Ref: 26498393
TCMC1409
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.1 (nM), Ref: 26498393
Ki: 170 (nM), Ref: 26498393
TCMC2048
TCMT771 Serine-protein kinase ATR Homo sapiens IC50: 7300 (nM), Ref: 22835870
TCMC1982
TCMT239 Serine/threonine-protein kinase PIM1 Homo sapiens IC50: 43 (nM), Ref: 16302800
IC50: 500 (nM), Ref: 24328302
TCMC1982
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 790 (nM), Ref: 17378609
IC50: 4000 (nM), Ref: 24368208
TCMC1982
TCMT223 Aldose reductase Homo sapiens IC50: 2200 (nM), Ref: 18165015
IC50: 14.8 (nM), Ref: 18976928
IC50: 2200 (nM), Ref: 22261024
IC50: 2900 (nM), Ref: 25152999
TCMC1982
TCMT44 Glyoxalase I Homo sapiens IC50: 3200 (nM), Ref: 18258440
TCMC1982
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 1540 (nM), Ref: 18533708
TCMC1982
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7890 (nM), Ref: 20185318
TCMC1982
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 8100 (nM), Ref: 20185318
TCMC1982
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2540 (nM), Ref: 20185318
TCMC1982
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2680 (nM), Ref: 20185318
TCMC1982
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6810 (nM), Ref: 20185318
TCMC1982
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6170 (nM), Ref: 20185318
TCMC1982
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4840 (nM), Ref: 20185318
TCMC1982
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7000 (nM), Ref: 20185318
TCMC1982
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9390 (nM), Ref: 20185318
TCMC1982
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 5410 (nM), Ref: 20185318
TCMC1982
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 12 (nM), Ref: 20413308
TCMC1982
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 4097 (nM), Ref: 20696580
IC50: 1550 (nM), Ref: 22328583
TCMC1982
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 1191 (nM), Ref: 20696580
TCMC1982
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 77 (nM), Ref: 20696580
TCMC1982
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 6680 (nM), Ref: 22658537
TCMC1982
TCMT320 Matrix metalloproteinase 3 Homo sapiens IC50: 5570 (nM), Ref: 22658537
TCMC1982
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 1610 (nM), Ref: 22658537
TCMC1982
TCMT322 Matrix metalloproteinase 13 Homo sapiens IC50: 8460 (nM), Ref: 22658537
TCMC1982
TCMT422 CaM kinase II beta Homo sapiens IC50: 3000 (nM), Ref: 21798748
TCMC1982
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 2000 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC1982
TCMT207 Beta-secretase 1 Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0353-y
IC50: 6500 (nM), Ref: 26003344
TCMC1982
TCMT784 Vasopressin V2 receptor Homo sapiens IC50: 7000 (nM), Ref: 23437772
IC50: 6309.57 (nM), Ref: 23437772
TCMC1982
TCMT785 Interleukin-8 receptor A Homo sapiens IC50: 4500 (nM), Ref: 23437772
IC50: 5011.87 (nM), Ref: 23437772
TCMC1982
TCMT786 C-C chemokine receptor type 4 Homo sapiens IC50: 10000 (nM), Ref: 23437772
TCMC1982
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 590 (nM), Ref: 23411073
TCMC1982
TCMT601 Thrombin Homo sapiens IC50: 1500 (nM), Ref: 24610996
TCMC1982
TCMT370 Vascular endothelial growth factor receptor 2 Homo sapiens IC50: 280 (nM), Ref: 24328302
TCMC1982
TCMT212 Tyrosine-protein kinase SRC Homo sapiens IC50: 120 (nM), Ref: 24328302
TCMC1982
TCMT791 Protein kinase N1 Homo sapiens IC50: 5800 (nM), Ref: 24328302
TCMC1982
TCMT484 Serine/threonine-protein kinase PLK1 Homo sapiens IC50: 5750 (nM), Ref: 24328302
TCMC1982
TCMT462 Serine/threonine-protein kinase NEK6 Homo sapiens IC50: 4230 (nM), Ref: 24328302
TCMC1982
TCMT445 Serine/threonine-protein kinase NEK2 Homo sapiens IC50: 5730 (nM), Ref: 24328302
TCMC1982
TCMT401 Hepatocyte growth factor receptor Homo sapiens IC50: 580 (nM), Ref: 24328302
TCMC1982
TCMT369 Insulin-like growth factor I receptor Homo sapiens IC50: 300 (nM), Ref: 24328302
TCMC1982
TCMT441 Focal adhesion kinase 1 Homo sapiens IC50: 1200 (nM), Ref: 24328302
TCMC1982
TCMT388 Tyrosine-protein kinase receptor UFO Homo sapiens IC50: 960 (nM), Ref: 24328302
TCMC1982
TCMT374 Serine/threonine-protein kinase Aurora-B Homo sapiens IC50: 910 (nM), Ref: 24328302
TCMC1982
TCMT436 NUAK family SNF1-like kinase 1 Homo sapiens IC50: 5090 (nM), Ref: 24328302
TCMC1982
TCMT402 ALK tyrosine kinase receptor Homo sapiens IC50: 3320 (nM), Ref: 24328302
TCMC1982
TCMT479 Serine/threonine-protein kinase AKT Homo sapiens IC50: 5390 (nM), Ref: 24328302
TCMC1982
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 280 (nM), Ref: 25060641
IC50: 3500 (nM), Ref: 27162124
TCMC1982
TCMT793 Liver glycogen phosphorylase Homo sapiens IC50: 4800 (nM), Ref: 25092521
TCMC1982
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 2110 (nM), Ref: 22328583
TCMC1982
TCMT217 Cytochrome P450 2C8 Homo sapiens IC50: 1390 (nM), Ref: 22328583
TCMC1477
TCMT273 Bile acid receptor FXR Homo sapiens IC50: 7860 (nM), Ref: 23688559
TCMC1477
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 5600 (nM), Ref: 21030469
IC50: 4900 (nM), Ref: 21030469
TCMC614
TCMT151 Protein kinase C alpha Homo sapiens IC50: 9300 (nM), Ref: 9834166
TCMC1982
TCMT261 Death-associated protein kinase 1 Homo sapiens IC50: 8900 (nM), Ref: 26322379
TCMC469
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 100 (nM), Ref: 22921742
TCMC2150
TCMT46 Coagulation factor III Homo sapiens IC50: 22.78 (nM), Ref: 23199480
TCMC2150
TCMT27 Dopamine D1 receptor Homo sapiens Ki: 231 (nM), Ref: 23332346
TCMC124
TCMT194 Mitogen-activated protein kinase kinase kinase 7 Homo sapiens IC50: 1300 (nM), Ref: 26481152
TCMC1830
TCMT297 Fatty acid binding protein adipocyte Homo sapiens IC50: 930 (nM), Ref: 15357969
TCMC1830
TCMT298 Fatty acid binding protein muscle Homo sapiens IC50: 2600 (nM), Ref: 15357969
TCMC1830
TCMT808 Fatty acid binding protein epidermal Homo sapiens IC50: 1200 (nM), Ref: 15357969
TCMC1830
TCMT809 Fatty acid binding protein intestinal Homo sapiens IC50: 1700 (nM), Ref: 15357969
TCMC1830
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1830
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1830
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1432
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8790.2 (nM), Ref: 26498393
TCMC1432
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 344.2 (nM), Ref: 26498393
TCMC1432
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.7 (nM), Ref: 26498393
TCMC1432
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 408.9 (nM), Ref: 26498393
TCMC418
TCMT223 Aldose reductase Homo sapiens IC50: 78 (nM), Ref: 22236472
TCMC418
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 240 (nM), Ref: 22236472
TCMC418
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4700 (nM), Ref: 22921742
TCMC1202
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 7030 (nM), Ref: 20185318
TCMC1202
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1202
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6990 (nM), Ref: 20185318
TCMC1202
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6070 (nM), Ref: 20185318
TCMC1202
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 6130 (nM), Ref: 20185318
TCMC1202
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9970 (nM), Ref: 20185318
TCMC1202
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1202
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 9800 (nM), Ref: 20185318
TCMC1202
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 7490 (nM), Ref: 20185318
TCMC1202
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 2250 (nM), Ref: 20185318
TCMC1202
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 3200 (nM), Ref: 20185318
TCMC1202
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 60 (nM), Ref: 10.1039/C4MD00086B
TCMC1757
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 130 (nM), Ref: 17378609
IC50: 110 (nM), Ref: 19848434
IC50: 25 (nM), Ref: 21958737
IC50: 120 (nM), Ref: 21958738
TCMC1757
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens IC50: 110 (nM), Ref: 12608855
IC50: 1100 (nM), Ref: 19848434
IC50: 5100 (nM), Ref: 21739938
IC50: 110 (nM), Ref: 24684213
TCMC1757
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens IC50: 180 (nM), Ref: 12608855
IC50: 5900 (nM), Ref: 19848434
IC50: 110 (nM), Ref: 21739938
TCMC1757
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 11 (nM), Ref: 20413308
TCMC606
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 251 (nM), Ref: 20696580
TCMC606
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 86 (nM), Ref: 20696580
TCMC606
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 12 (nM), Ref: 20696580
TCMC983
TCMT236 Estrogen receptor beta Homo sapiens IC50: 2800 (nM), Ref: 15887952
IC50: 2800 (nM), Ref: 15887952
IC50: 1200 (nM), Ref: 12502307
IC50: 2800 (nM), Ref:
TCMC983
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 7300 (nM), Ref: 21030469
TCMC983
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 718.7 (nM), Ref: 26498393
TCMC983
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.2 (nM), Ref: 26498393
TCMC983
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 56.4 (nM), Ref: 26498393
TCMC2111
TCMT614 Egl nine homolog 1 Homo sapiens IC50: 3000 (nM), Ref: 18942826
TCMC1919
TCMT613 Glucocorticoid receptor Homo sapiens IC50: 14 (nM), Ref: 19364854
TCMC755
TCMT3 Arachidonate 15-lipoxygenase Homo sapiens Ki: 600 (nM), Ref: 21739938
TCMC755
TCMT81 Arachidonate 12-lipoxygenase Homo sapiens Ki: 1600 (nM), Ref: 21739938
TCMC755
TCMT8 Lysine-specific demethylase 4D-like Homo sapiens IC50: 3000 (nM), Ref: 10.1039/C1MD00199J
TCMC755
TCMT162 UDP-glucuronosyltransferase 1-1 Homo sapiens IC50: 4400 (nM), Ref: 21030469
IC50: 7000 (nM), Ref: 21030469
TCMC755
TCMT384 G protein-coupled receptor kinase 6 Homo sapiens IC50: 8700 (nM), Ref:
TCMC1118
TCMT304 Matrix metalloproteinase 14 Homo sapiens IC50: 6800 (nM), Ref: 19524436
TCMC1118
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 9600 (nM), Ref: 19524436
TCMC1118
TCMT207 Beta-secretase 1 Homo sapiens IC50: 757 (nM), Ref: 22225636
TCMC1118
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 1000 (nM), Ref: 22413845
IC50: 1080 (nM), Ref: 22413845
IC50: 1180 (nM), Ref: 22413845
IC50: 1000 (nM), Ref: 10.1039/C0MD00241K
TCMC1118
TCMT47 Apoptosis regulator Bcl-2 Homo sapiens Ki: 335 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC1118
TCMT2 Microtubule-associated protein tau Homo sapiens IC50: 1800 (nM), Ref: 23484434
TCMC1118
TCMT751 Dual-specificity tyrosine-phosphorylation regulated kinase 1A Homo sapiens IC50: 330 (nM), Ref: 24188002
TCMC1118
TCMT45 Beta amyloid A4 protein Homo sapiens IC50: 4600 (nM), Ref: 24878198
IC50: 3000 (nM), Ref: 24878198
IC50: 500 (nM), Ref: 25978520
TCMC1118
TCMT567 DNA (cytosine-5)-methyltransferase 1 Homo sapiens IC50: 500 (nM), Ref: 25406944
TCMC1118
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 124.1 (nM), Ref: 25985195
IC50: 122.6 (nM), Ref: 25985195
TCMC1839
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 9800 (nM), Ref: 18501600
Ki: 9800 (nM), Ref: 18579385
Ki: 920 (nM), Ref: 20185318
TCMC1839
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4800 (nM), Ref: 18579385
Ki: 6270 (nM), Ref: 20185318
TCMC1839
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 9200 (nM), Ref: 18579385
Ki: 3670 (nM), Ref: 20185318
TCMC1839
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 6160 (nM), Ref: 20185318
TCMC1839
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 3730 (nM), Ref: 20185318
TCMC1839
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4080 (nM), Ref: 20185318
TCMC1839
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 5700 (nM), Ref: 20185318
TCMC1839
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 7130 (nM), Ref: 20185318
TCMC1839
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7780 (nM), Ref: 20185318
TCMC1839
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 6610 (nM), Ref: 20185318
TCMC1839
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 870 (nM), Ref: 20185318
TCMC1788
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7
IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT64 Peroxisome proliferator-activated receptor delta Homo sapiens IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT67 Peroxisome proliferator-activated receptor gamma Homo sapiens IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1788
TCMT126 Telomerase reverse transcriptase Homo sapiens IC50: 8600 (nM), Ref: 10.1039/C0MD00241K
TCMC1788
TCMT297 Fatty acid binding protein adipocyte Homo sapiens Ki: 1500 (nM), Ref: 27460668
TCMC937
TCMT232 P-glycoprotein 1 Homo sapiens IC50: 11.5 (nM), Ref: 23332369
IC50: 6.6 (nM), Ref: 23895532
TCMC937
TCMT801 Tubulin beta-3 chain Homo sapiens IC50: 5.2 (nM), Ref: 23332369
IC50: 5.7 (nM), Ref: 23895532
TCMC732
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 5900 (nM), Ref: 21561086
TCMC1203
TCMT822 Alpha-(1,3)-fucosyltransferase 7 Homo sapiens IC50: 8000 (nM), Ref: 10.1039/C4MD00086B
TCMC453
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 156 (nM), Ref: 23391306
IC50: 943 (nM), Ref: 23391306
IC50: 440 (nM), Ref: 23391306
IC50: 34.67 (nM), Ref: 23631755
Ki: 13 (nM), Ref: 23631755
TCMC1204
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2500 (nM), Ref: 14592472
TCMC1504
TCMT273 Bile acid receptor FXR Homo sapiens IC50: 18.3 (nM), Ref: 24775917
TCMC1356
TCMT223 Aldose reductase Homo sapiens IC50: 3000 (nM), Ref: 22261024
TCMC1498
TCMT864 Thyroid hormone receptor alpha Homo sapiens IC50: 0.24 (nM), Ref: 16099653
IC50: 0.24 (nM), Ref: 17543524
Ki: 0.33 (nM), Ref: 18975928
Ki: 2.33 (nM), Ref: 22542282
Ki: 2.33 (nM), Ref: 23276448
IC50: 3.2 (nM), Ref: 24290064
TCMC1498
TCMT69 Thyroid hormone receptor beta-1 Homo sapiens IC50: 0.26 (nM), Ref: 16099653
IC50: 0.26 (nM), Ref: 17543524
IC50: 0.257 (nM), Ref: 17524652
Ki: 0.68 (nM), Ref: 18975928
Ki: 2.29 (nM), Ref: 22542282
Ki: 2.29 (nM), Ref: 23276448
IC50: 2.9 (nM), Ref: 24290064
TCMC1498
TCMT796 Proliferating cell nuclear antigen Homo sapiens IC50: 3600 (nM), Ref: 23395113
TCMC2228
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 6830 (nM), Ref: 21282059
TCMC2228
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 6180 (nM), Ref: 21282059
TCMC2228
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 8250 (nM), Ref: 21282059
TCMC2228
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 6700 (nM), Ref: 21282059
TCMC2228
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 6480 (nM), Ref: 22687439
TCMC2228
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 740 (nM), Ref: 22668600
TCMC2228
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 7150 (nM), Ref: 22668600
TCMC341
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 510 (nM), Ref: 19231207
TCMC2114
TCMT683 Macrophage migration inhibitory factor Homo sapiens IC50: 2200 (nM), Ref: 25743213
TCMC2114
TCMT423 Epidermal growth factor receptor erbB1 Homo sapiens IC50: 9000 (nM), Ref: 27135370
TCMC1798
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1480 (nM), Ref: 23411073
TCMC811
TCMT254 Carbonyl reductase [NADPH] 1 Homo sapiens Ki: 2030 (nM), Ref: 19097799
TCMC811
TCMT66 Estradiol 17-beta-dehydrogenase 2 Homo sapiens IC50: 9900 (nM), Ref: 18533708
TCMC811
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10.2 (nM), Ref: 20413308
TCMC811
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 7078.5 (nM), Ref: 26498393
TCMC811
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 371.5 (nM), Ref: 26498393
TCMC811
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 52.5 (nM), Ref: 26498393
TCMC1123
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 1284 (nM), Ref: 20696580
TCMC1123
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 72.8 (nM), Ref: 26498393
TCMC1123
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 4.3 (nM), Ref: 26498393
TCMC1123
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 31.1 (nM), Ref: 26498393
TCMC847
TCMT135 Carbonic anhydrase XIV Homo sapiens Ki: 8710 (nM), Ref: 20185318
Ki: 8710 (nM), Ref: 26498394
TCMC847
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 9060 (nM), Ref: 20185318
Ki: 9060 (nM), Ref: 26498394
TCMC847
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 7870 (nM), Ref: 20185318
TCMC847
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 6420 (nM), Ref: 20185318
TCMC847
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 7330 (nM), Ref: 20185318
TCMC847
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 9080 (nM), Ref: 20185318
TCMC847
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 6490 (nM), Ref: 20185318
TCMC847
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 10000 (nM), Ref: 20185318
TCMC847
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1610 (nM), Ref: 20185318
TCMC847
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2380 (nM), Ref: 20185318
TCMC847
TCMT101 Protein-tyrosine phosphatase 1B Homo sapiens IC50: 3060 (nM), Ref: 19476336
TCMC847
TCMT321 Matrix metalloproteinase 9 Homo sapiens IC50: 21.22 (nM), Ref: 23375794
IC50: 10 (nM), Ref: 23375794
TCMC847
TCMT306 Matrix metalloproteinase-2 Homo sapiens IC50: 24.26 (nM), Ref: 23375794
TCMC847
TCMT295 Matrix metalloproteinase-1 Homo sapiens IC50: 238.91 (nM), Ref: 23375794
TCMC847
TCMT130 Arachidonate 5-lipoxygenase Homo sapiens IC50: 8500 (nM), Ref: 26197161
TCMC785
TCMT131 Acetylcholinesterase Homo sapiens IC50: 610 (nM), Ref: 23062825
TCMC2201
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 8700 (nM), Ref: 21332115
TCMC1611
TCMT810 Toll-like receptor 2 Homo sapiens IC50: 5000 (nM), Ref: 16509590
TCMC1611
TCMT63 Peroxisome proliferator-activated receptor alpha Homo sapiens IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6
TCMC1003
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 15 (nM), Ref: 20413308
TCMC897
TCMT223 Aldose reductase Homo sapiens IC50: 300 (nM), Ref: 22236472
IC50: 1800 (nM), Ref: 22261024
TCMC897
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens IC50: 7900 (nM), Ref: 22236472
TCMC1828
TCMT33 Cytochrome P450 3A4 Homo sapiens IC50: 900 (nM), Ref: 17994701
TCMC1237
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 7300 (nM), Ref: 22668600
TCMC1237
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 6600 (nM), Ref: 22668600
TCMC1237
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 4100 (nM), Ref: 22668600
TCMC1237
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 4200 (nM), Ref: 22668600
TCMC273
TCMT332 Amine oxidase, copper containing Homo sapiens IC50: 4100 (nM), Ref: 23664164
TCMC90
TCMT207 Beta-secretase 1 Homo sapiens IC50: 2400 (nM), Ref: 14592472
TCMC2055
TCMT747 ATP-binding cassette sub-family G member 2 Homo sapiens IC50: 10000 (nM), Ref: 22822035
TCMC2209
TCMT597 Solute carrier family 28 member 3 Homo sapiens Ki: 3400 (nM), Ref: 23388705
IC50: 5400 (nM), Ref: 23388705
TCMC2209
TCMT710 Sodium/nucleoside cotransporter 1 Homo sapiens Ki: 5200 (nM), Ref: 23388705
IC50: 5800 (nM), Ref: 23388705
TCMC710
TCMT249 Cyclin-dependent kinase 6 Homo sapiens IC50: 1700 (nM), Ref: 15689157
IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5
TCMC710
TCMT156 Cytochrome P450 19A1 Homo sapiens IC50: 10000 (nM), Ref: 18192087
IC50: 900 (nM), Ref: 20413308
IC50: 1200 (nM), Ref: 26301554
TCMC710
TCMT65 Estradiol 17-beta-dehydrogenase 1 Homo sapiens IC50: 710 (nM), Ref: 18533708
TCMC710
TCMT752 Casein kinase II alpha Homo sapiens IC50: 800 (nM), Ref: 19414254
TCMC710
TCMT187 Androgen Receptor Homo sapiens IC50: 5200 (nM), Ref: 19592245
TCMC710
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 795 (nM), Ref: 20696580
TCMC710
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 427 (nM), Ref: 20696580
TCMC710
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 25 (nM), Ref: 20696580
TCMC710
TCMT265 Glycogen synthase kinase-3 beta Homo sapiens IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT131 Acetylcholinesterase Homo sapiens IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y
TCMC710
TCMT260 Tyrosine-protein kinase receptor FLT3 Homo sapiens IC50: 1450 (nM), Ref: 23411073
TCMC710
TCMT128 Tankyrase-2 Homo sapiens IC50: 2951.21 (nM), Ref: 23574272
IC50: 2900 (nM), Ref: 23574272
TCMC710
TCMT129 Tankyrase-1 Homo sapiens IC50: 3162.28 (nM), Ref: 23574272
IC50: 3100 (nM), Ref: 23574272
TCMC710
TCMT592 Xanthine dehydrogenase Homo sapiens Ki: 520 (nM), Ref: 25019478
IC50: 3200 (nM), Ref: 26022844
TCMC710
TCMT280 Aldo-keto reductase family 1 member B10 Homo sapiens Ki: 6000 (nM), Ref: 26529431
IC50: 6600 (nM), Ref: 26529431
TCMC1064
TCMT219 Cytochrome P450 1A2 Homo sapiens IC50: 2437 (nM), Ref: 20696580
TCMC1064
TCMT215 Cytochrome P450 1A1 Homo sapiens IC50: 140 (nM), Ref: 20696580
TCMC1064
TCMT257 Cytochrome P450 1B1 Homo sapiens IC50: 29 (nM), Ref: 20696580
TCMC784
TCMT131 Acetylcholinesterase Homo sapiens IC50: 100 (nM), Ref: 26003344
TCMC784
TCMT132 Butyrylcholinesterase Homo sapiens IC50: 1090 (nM), Ref: 26003344
TCMC702
TCMT206 Cytochrome P450 2A6 Homo sapiens IC50: 5150 (nM), Ref: 15658857
TCMC878
TCMT133 Carbonic anhydrase I Homo sapiens Ki: 2420 (nM), Ref: 20674354
TCMC878
TCMT134 Carbonic anhydrase II Homo sapiens Ki: 1840 (nM), Ref: 20674354
TCMC878
TCMT143 Carbonic anhydrase III Homo sapiens Ki: 3580 (nM), Ref: 20674354
TCMC878
TCMT142 Carbonic anhydrase IV Homo sapiens Ki: 4900 (nM), Ref: 20674354
TCMC878
TCMT141 Carbonic anhydrase VA Homo sapiens Ki: 4210 (nM), Ref: 20674354
TCMC878
TCMT140 Carbonic anhydrase VB Homo sapiens Ki: 4020 (nM), Ref: 20674354
TCMC878
TCMT139 Carbonic anhydrase VI Homo sapiens Ki: 4910 (nM), Ref: 20674354
TCMC878
TCMT138 Carbonic anhydrase VII Homo sapiens Ki: 450 (nM), Ref: 20674354
TCMC878
TCMT137 Carbonic anhydrase IX Homo sapiens Ki: 5030 (nM), Ref: 20674354
TCMC878
TCMT136 Carbonic anhydrase XII Homo sapiens Ki: 4720 (nM), Ref: 20674354
TCMC770
TCMT588 D-amino-acid oxidase Homo sapiens Ki: 7000 (nM), Ref: 23391306
IC50: 2089.3 (nM), Ref: 23631755
Ki: 2000 (nM), Ref: 23631755

Targeted Pathogenic Microbes or non-Human Proteins by the Ingredients of Prescription

References are linked to referred publications via PubMed ID or DOI.
There may be multiple activity records for a specific ingredient-target pair.

Ingredient ID & Structure Target ID Target Name Target Organism Activity Records & Reference
TCMC908
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 11.62 (ug/ml), Ref: 20116898
TCMC2252
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 19.4 (ug/ml), Ref: 16643034
TCMC962
TCMT1104 Sortase Staphylococcus aureus IC50: 13.8 (ug/ml), Ref: 19269184
TCMC962
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 51.3 (ug/ml), Ref: 16643034
TCMC962
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 1 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC1429
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 16.77 (ug/ml), Ref: 20116898
TCMC1620
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 0.66 (ug/ml), Ref: 11430019
IC50: 5.9 (ug/ml), Ref: 16643034
TCMC2054
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 14.48 (ug/ml), Ref: 20116898
TCMC1786
TCMT1107 Protease Human immunodeficiency virus 1 IC50: 10 (ug/ml), Ref: 10691716
TCMC2257
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 15.46 (ug/ml), Ref: 20116898
TCMC2259
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 47.4 (ug/ml), Ref: 16643034
TCMC2265
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 23.6 (ug/ml), Ref: 16643034
TCMC1399
TCMT1136 Neuraminidase H1N1 swine influenza virus IC50: 3.42 (ug/ml), Ref: 21123068
IC50: 3.48 (ug/ml), Ref: 21123068
IC50: 8.41 (ug/ml), Ref: 21123068
IC50: 9.69 (ug/ml), Ref: 21123068
IC50: 10.56 (ug/ml), Ref: 21123068
TCMC1399
TCMT1136 Neuraminidase Influenza A virus IC50: 3.42 (ug/ml), Ref: 21123068
IC50: 3.48 (ug/ml), Ref: 21123068
IC50: 8.41 (ug/ml), Ref: 21123068
IC50: 9.69 (ug/ml), Ref: 21123068
IC50: 10.56 (ug/ml), Ref: 21123068
TCMC1399
TCMT1121 Sialidase Clostridium perfringens IC50: 11.28 (ug/ml), Ref: 21123068
TCMC1609
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 26.29 (ug/ml), Ref: 20116898
TCMC2271
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 43.5 (ug/ml), Ref: 16643034
TCMC2031
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 31.14 (ug/ml), Ref: 20116898
TCMC1206
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 21.25 (ug/ml), Ref: 20116898
TCMC1982
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 17.65 (ug/ml), Ref: 20116898
TCMC1425
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 71 (ug/ml), Ref: 1710653
IC50: 71 (ug/ml), Ref: 21295891
TCMC2275
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 44.5 (ug/ml), Ref: 16643034
TCMC469
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 5.4 (ug/ml), Ref: 16643034
TCMC983
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 9.43 (ug/ml), Ref: 20116898
TCMC1858
TCMT1112 Quinolone resistance protein norA Staphylococcus aureus MIC: 4 (ug/ml), Ref: 10.1039/C4MD00196F
TCMC995
TCMT1104 Sortase Staphylococcus aureus IC50: 18.3 (ug/ml), Ref: 16154746
TCMC1118
TCMT1092 Fatty acid synthase Plasmodium falciparum IC50: 0.03 (ug/ml), Ref: 20855214
IC50: 30 (nM), Ref: 24063369
TCMC1118
TCMT1094 3-oxoacyl-acyl-carrier protein reductase Plasmodium falciparum IC50: 0.32 (ug/ml), Ref: 20855214
TCMC1203
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 28.5 (ug/ml), Ref: 9461665
TCMC1356
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 64.6 (ug/ml), Ref: 9461665
TCMC785
TCMT1104 Sortase Staphylococcus aureus IC50: 8.7 (ug/ml), Ref: 17716892
IC50: 8.7 (ug/ml), Ref: 19269184
TCMC785
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 100 (ug/ml), Ref: 1710653
IC50: 100 (ug/ml), Ref: 21295891
TCMC785
TCMT1154 Sortase Staphylococcus aureus IC50: 40.6 (ug/ml), Ref: 26551342
TCMC2292
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 13.15 (ug/ml), Ref: 20116898
TCMC1491
TCMT1109 Reverse transcriptase Human immunodeficiency virus 1 IC50: 0.00423 (ug/ml), Ref: 21334901
IC50: 0.00211 (ug/ml), Ref: 21334901
TCMC2299
TCMT1108 Integrase Human immunodeficiency virus 1 IC50: 20.1 (ug/ml), Ref: 16643034
TCMC710
TCMT1099 Neuraminidase Influenza A virus (A/Puerto Rico/8/1934(H1N1)) IC50: 8.54 (ug/ml), Ref: 20116898
TCMC943
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 8 (ug/ml), Ref: 9748372
TCMC943
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 21288041
MIC: 7 (ug/ml), Ref: 25794790
TCMC943
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 21288041
TCMC2322
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 20 (ug/ml), Ref: 3204384
TCMC2322
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 5 (ug/ml), Ref: 3204384
TCMC2324
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC2051
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 42 (ug/ml), Ref: 22280816
MIC: 42.1 (ug/ml), Ref: 26112067
TCMC908
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 11170636
MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 50 (ug/ml), Ref: 16213726
TCMC908
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 81 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2329
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 25.3 (ug/ml), Ref: 8946749
TCMC903
TCMT1251 Candida albicans Candida albicans MIC: 64 (ug/ml), Ref: 18805690
TCMC903
TCMT1246 Escherichia coli Escherichia coli MIC: 64 (ug/ml), Ref: 18805690
MIC: 7.81 (ug/ml), Ref: 20181416
MIC: 4 (ug/ml), Ref: 20038628
MIC: 8 (ug/ml), Ref: 20038628
MIC: 16 (ug/ml), Ref: 20038628
TCMC903
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 15.63 (ug/ml), Ref: 20181416
TCMC903
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 31.25 (ug/ml), Ref: 20181416
TCMC855
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
TCMC2013
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1395
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 64 (ug/ml), Ref: 23369537
TCMC2354
TCMT1251 Candida albicans Candida albicans IC50: 81.47 (ug/ml), Ref: 25686593
TCMC1901
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1214 Enterococcus faecium Enterococcus faecium MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1236 Mycobacterium bovis Mycobacterium bovis BCG MIC: 26 (ug/ml), Ref: 18849164
TCMC1901
TCMT1217 Bacillus anthracis Bacillus anthracis MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1191 Bacillus megaterium Bacillus megaterium MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1286 Bacillus cereus Bacillus cereus MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 8 (ug/ml), Ref: 18849164
TCMC1901
TCMT1260 Streptococcus agalactiae Streptococcus agalactiae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1322 Streptococcus mitis Streptococcus mitis MIC: 64 (ug/ml), Ref: 18849164
TCMC1901
TCMT1410 Listeria monocytogenes Listeria monocytogenes MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1323 Corynebacterium pseudodiphtheriticum Corynebacterium pseudodiphtheriticum MIC: 16 (ug/ml), Ref: 18849164
TCMC1901
TCMT1324 Corynebacterium diphtheriae Corynebacterium diphtheriae MIC: 32 (ug/ml), Ref: 18849164
TCMC1901
TCMT1319 Corynebacterium xerosis Corynebacterium xerosis MIC: 16 (ug/ml), Ref: 18849164
TCMC884
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC1172
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 6.25 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1172
TCMT1251 Candida albicans Candida albicans IC50: 2.82 (ug/ml), Ref: 11958988
TCMC1172
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 8 (ug/ml), Ref: 24641242
TCMC553
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0032-z
TCMC962
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 4.2 (ug/ml), Ref: 19299148
IC50: 3.5 (ug/ml), Ref: 19299148
TCMC962
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 4.2 (ug/ml), Ref: 19299148
IC50: 3.5 (ug/ml), Ref: 19299148
TCMC962
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC962
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 5 (ug/ml), Ref: 19204190
MIC: 15 (ug/ml), Ref: 19204190
MIC: 50 (ug/ml), Ref: 19204190
MIC: 30 (ug/ml), Ref: 19204190
TCMC962
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 30 (ug/ml), Ref: 18284200
TCMC962
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 16 (ug/ml), Ref: 25938986
MIC: 32 (ug/ml), Ref: 25938986
TCMC2383
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 37.96 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2398
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.557 (ug/ml), Ref: 3286870
IC50: 2.008 (ug/ml), Ref: 3286870
TCMC1429
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 7.93 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC885
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 3.1 (ug/ml), Ref: 7381838
MIC: 0.8 (ug/ml), Ref: 7381838
MIC: 4 (ug/ml), Ref: 2933519
MIC: 1 (ug/ml), Ref: 2933519
MIC: 0.5 (ug/ml), Ref: 3373488
MIC: 0.5 (ug/ml), Ref: 2502627
MIC: 4 (ug/ml), Ref: 3877809
MIC: 4 (ug/ml), Ref: 2933520
MIC: 0.3 (ug/ml), Ref: 3701783
MIC: 20 (ug/ml), Ref: 2724308
MIC: 10 (ug/ml), Ref: 17825955
MIC: 8 (ug/ml), Ref: 19027993
MIC: 2 (ug/ml), Ref: 19027993
MIC: 4 (ug/ml), Ref: 19027993
MIC: 1 (ug/ml), Ref: 19027993
MIC: 4.6 (ug/ml), Ref: 20211890
MIC: 3.9 (ug/ml), Ref: 20211890
MIC: 2.5 (ug/ml), Ref: 20211890
MIC: 10.7 (ug/ml), Ref: 20211890
MIC: 3.1 (ug/ml), Ref: 20211890
MIC: 3.3 (ug/ml), Ref: 20211890
MIC: 3.8 (ug/ml), Ref: 20211890
MIC: 14.7 (ug/ml), Ref: 20211890
MIC: 6.6 (ug/ml), Ref: 20211890
MIC: 10.6 (ug/ml), Ref: 20211890
MIC: 1.25 (ug/ml), Ref: 894680
MIC: 5 (ug/ml), Ref: 894680
MIC: 1.25 (ug/ml), Ref: 894679
MIC: 5 (ug/ml), Ref: 894679
MIC: 1.6 (ug/ml), Ref: 392100
MIC: 6.2 (ug/ml), Ref: 392100
MIC: 4.5 (ug/ml), Ref: 21963
TCMC885
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 1.6 (ug/ml), Ref: 7381838
MIC: 4 (ug/ml), Ref: 2933519
MIC: 0.5 (ug/ml), Ref: 3373488
MIC: 2 (ug/ml), Ref: 3877809
MIC: 2 (ug/ml), Ref: 2933520
TCMC885
TCMT1448 Enterobacter aerogenes Enterobacter aerogenes MIC: 25 (ug/ml), Ref: 7381838
MIC: 5 (ug/ml), Ref: 894680
MIC: 5 (ug/ml), Ref: 894679
MIC: 6.8 (ug/ml), Ref: 21963
TCMC885
TCMT1170 Enterobacter cloacae Enterobacter cloacae MIC: 25 (ug/ml), Ref: 7381838
TCMC885
TCMT1246 Escherichia coli Escherichia coli MIC: 6.2 (ug/ml), Ref: 7381838
MIC: 8 (ug/ml), Ref: 3373488
MIC: 1 (ug/ml), Ref: 3701783
MIC: 2 (ug/ml), Ref: 18180352
MIC: 12.5 (ug/ml), Ref: 894680
MIC: 12.5 (ug/ml), Ref: 894679
MIC: 6.2 (ug/ml), Ref: 392100
MIC: 8.5 (ug/ml), Ref: 21963
TCMC885
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 3.1 (ug/ml), Ref: 7381838
MIC: 16 (ug/ml), Ref: 3373488
MIC: 3.1 (ug/ml), Ref: 392100
MIC: 7 (ug/ml), Ref: 21963
TCMC885
TCMT1224 Proteus mirabilis Proteus mirabilis MIC: 12.5 (ug/ml), Ref: 7381838
MIC: 4 (ug/ml), Ref: 3373488
MIC: 6 (ug/ml), Ref: 18180352
MIC: 4 (ug/ml), Ref: 18180352
MIC: 3 (ug/ml), Ref: 18180352
MIC: 2 (ug/ml), Ref: 18180352
MIC: 1.5 (ug/ml), Ref: 18180352
MIC: 1 (ug/ml), Ref: 18180352
MIC: 12.5 (ug/ml), Ref: 894680
MIC: 12.5 (ug/ml), Ref: 894679
MIC: 25 (ug/ml), Ref: 392100
TCMC885
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 2933519
MIC: 32 (ug/ml), Ref: 3877809
MIC: 32 (ug/ml), Ref: 2933520
MIC: 12.5 (ug/ml), Ref: 392100
TCMC885
TCMT1177 Haemophilus influenzae Haemophilus influenzae MIC: 8 (ug/ml), Ref: 2933519
MIC: 4 (ug/ml), Ref: 3373488
MIC: 8 (ug/ml), Ref: 3877809
MIC: 8 (ug/ml), Ref: 2933520
TCMC885
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 32 (ug/ml), Ref: 3373488
MIC: 64 (ug/ml), Ref: 2502627
MIC: 64 (ug/ml), Ref: 19027993
TCMC885
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 1 (ug/ml), Ref: 3701783
MIC: 1 (ug/ml), Ref: 19027993
TCMC13
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 34.1 (ug/ml), Ref: 10425115
TCMC13
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1.92 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC885
TCMT1194 Shigella sonnei Shigella sonnei MIC: 5 (ug/ml), Ref: 894680
MIC: 5 (ug/ml), Ref: 894679
TCMC885
TCMT1195 Streptococcus pasteurianus Streptococcus pasteurianus MIC: 1.6 (ug/ml), Ref: 392100
TCMC885
TCMT1196 Salmonella Salmonella MIC: 6.2 (ug/ml), Ref: 392100
TCMC885
TCMT1197 Shigella sp. Shigella sp. MIC: 9 (ug/ml), Ref: 21963
TCMC1424
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 27.95 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2237
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4 (ug/ml), Ref: 24549242
TCMC737
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 26.9 (ug/ml), Ref: 15104496
TCMC737
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 35.8 (ug/ml), Ref: 15104496
TCMC737
TCMT1449 Influenza A virus Influenza A virus IC50: 24.5 (ug/ml), Ref: 15104496
TCMC1322
TCMT1181 Mycobacterium tuberculosis H37Ra Mycobacterium tuberculosis H37Ra MIC: 100 (ug/ml), Ref: 20691508
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC1786
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 21.8 (ug/ml), Ref: 9748372
TCMC1786
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 16 (ug/ml), Ref: 21288041
TCMC1786
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 50 (ug/ml), Ref: 11141098
MIC: 100 (ug/ml), Ref: 18798682
MIC: 64 (ug/ml), Ref: 15387646
MIC: 29 (ug/ml), Ref: 23356207
TCMC2257
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 15.3 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 37.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 59.7 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC2447
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 18 (ug/ml), Ref: 19904996
TCMC1113
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 0.5 (ug/ml), Ref: 15863332
TCMC1163
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 93.8 (ug/ml), Ref: 6512542
TCMC2463
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 1 (ug/ml), Ref: 15921418
TCMC2463
TCMT1251 Candida albicans Candida albicans MIC: 2 (ug/ml), Ref: 15921418
TCMC2463
TCMT1176 Streptococcus pneumoniae Streptococcus pneumoniae MIC: 16 (ug/ml), Ref: 15921418
TCMC1399
TCMT1286 Bacillus cereus Bacillus cereus MIC: 62.5 (ug/ml), Ref: 18951808
TCMC1399
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 18951808
MIC: 31.25 (ug/ml), Ref: 22169259
MIC: 62.5 (ug/ml), Ref: 22169259
MIC: 15.6 (ug/ml), Ref: 25137491
TCMC1609
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 0.88 (ug/ml), Ref: 24749980
TCMC1609
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1609
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC2481
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1246 Escherichia coli Escherichia coli MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1232 Pseudomonas aeruginosa Pseudomonas aeruginosa MIC: 50 (ug/ml), Ref: 17027268
TCMC2481
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 25 (ug/ml), Ref: 17027268
TCMC2481
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 12.5 (ug/ml), Ref: 17027268
TCMC2031
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 30 (ug/ml), Ref: 12502337
TCMC2031
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 80 (ug/ml), Ref: 17394331
TCMC1409
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 94 (ug/ml), Ref: 15104489
TCMC1409
TCMT1447 Respiratory syncytial virus Respiratory syncytial virus IC50: 5.9 (ug/ml), Ref: 15104496
TCMC1409
TCMT1294 Human parainfluenza virus 3 Human parainfluenza virus 3 IC50: 23.4 (ug/ml), Ref: 15104496
TCMC1409
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 12762812
TCMC1409
TCMT1443 Leishmania amazonensis Leishmania amazonensis IC50: 0.78 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC2491
TCMT1251 Candida albicans Candida albicans MIC: 3.2 (ug/ml), Ref: 9873584
TCMC1982
TCMT1246 Escherichia coli Escherichia coli MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 2 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 1 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 3.9 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
IC50: 3.8 (ug/ml), Ref: 24749980
TCMC1982
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 31.25 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC1982
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
MIC: 100 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC1982
TCMT1286 Bacillus cereus Bacillus cereus MIC: 50 (ug/ml), Ref: 12762812
TCMC1982
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 6.5 (ug/ml), Ref: 12398543
TCMC1982
TCMT1442 Leishmania donovani Leishmania donovani IC50: 29.5 (ug/ml), Ref: 12398543
IC50: 1 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1982
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 2.4 (ug/ml), Ref: 18855442
TCMC1206
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 44.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1982
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 64 (ug/ml), Ref: 20655215
MIC: 64 (ug/ml), Ref: 21534606
TCMC2506
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 1.99 (ug/ml), Ref: 8786363
IC50: 1.9 (ug/ml), Ref: 8786363
TCMC2506
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 1.99 (ug/ml), Ref: 8786363
IC50: 1.9 (ug/ml), Ref: 8786363
TCMC1982
TCMT1212 Verticillium dahliae Verticillium dahliae IC50: 6 (ug/ml), Ref: 17394331
TCMC1982
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC1767
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis H37Rv MIC: 60 (ug/ml), Ref: 20384293
TCMC1767
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-012-0419-x
TCMC1425
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.422 (ug/ml), Ref: 3286870
IC50: 1.607 (ug/ml), Ref: 3286870
TCMC614
TCMT1454 Bacillus subtilis Bacillus subtilis IC50: 98.5 (ug/ml), Ref: 25981688
TCMC934
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.73 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2045
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC2045
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 59 (ug/ml), Ref: 10.1007/s00044-013-0485-8
MIC: 51 (ug/ml), Ref: 10.1007/s00044-013-0485-8
TCMC60
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC60
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 12.5 (ug/ml), Ref: 10.1021/np50124a013
TCMC1186
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 3430167
TCMC1186
TCMT1284 Penicillium expansum Penicillium expansum MIC: 50 (ug/ml), Ref: 3430167
TCMC2532
TCMT1248 Hepatitis C virus Hepatitis C virus IC50: 20 (ug/ml), Ref: 19904996
TCMC2539
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 100 (ug/ml), Ref: 1517735
TCMC1830
TCMT1361 Neisseria meningitidis Neisseria meningitidis MIC: 50 (ug/ml), Ref: 19884363
TCMC1830
TCMT1382 Plasmodium falciparum (isolate K1 / Thailand) Plasmodium falciparum K1 IC50: 3.8 (ug/ml), Ref: 20855214
IC50: 3.8 (ug/ml), Ref: 25103602
TCMC1830
TCMT1442 Leishmania donovani Leishmania donovani IC50: 14.5 (ug/ml), Ref: 20855214
TCMC2550
TCMT1393 Vibrio sp. Vibrio sp. MIC: 15 (ug/ml), Ref: 21865038
TCMC913
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 65.55 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC913
TCMT1189 Pseudomonas fluorescens Pseudomonas fluorescens MIC: 1.6 (ug/ml), Ref: 14995101
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum D6 IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC495
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 7.33 (ug/ml), Ref: 8759172
IC50: 5.56 (ug/ml), Ref: 8759172
TCMC1117
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 100 (ug/ml), Ref: 10425115
TCMC1117
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.89 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1202
TCMT1178 Actinomyces viscosus Actinomyces viscosus MIC: 78 (ug/ml), Ref: 8904847
TCMC1202
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 14.8 (ug/ml), Ref: 15844943
TCMC801
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 32 (ug/ml), Ref: 15844943
TCMC801
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 52.3 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC924
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC606
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 5.5 (ug/ml), Ref: 19299148
TCMC755
TCMT1251 Candida albicans Candida albicans IC50: 6 (ug/ml), Ref: 12502337
TCMC755
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 50 (ug/ml), Ref: 10.1007/s00044-012-0268-7
TCMC755
TCMT1249 Dengue virus 2 Dengue virus 2 IC50: 6.46 (ug/ml), Ref: 25564380
TCMC1238
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 64 (ug/ml), Ref: 24641242
TCMC2166
TCMT1211 Fusobacterium nucleatum Fusobacterium nucleatum MIC: 50 (ug/ml), Ref: 8864235
TCMC2166
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1321 Staphylococcus hominis Staphylococcus hominis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1223 Staphylococcus epidermidis Staphylococcus epidermidis MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
MIC: 32.25 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1209 Staphylococcus haemolyticus Staphylococcus haemolyticus MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1343 Staphylococcus simulans Staphylococcus simulans MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1344 Staphylococcus sciuri Staphylococcus sciuri MIC: 32 (ug/ml), Ref: 19651906
MIC50: 64 (ug/ml), Ref: 19651906
MBC: 64 (ug/ml), Ref: 19651906
MIC: 4 (ug/ml), Ref: 19651906
MIC90: 64 (ug/ml), Ref: 19651906
TCMC2166
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1229 Enterococcus faecalis Enterococcus faecalis MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1246 Escherichia coli Escherichia coli MIC: 100 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC2166
TCMT1462 Streptococcus mutans Streptococcus mutans MIC: 62.5 (ug/ml), Ref: 10.1007/s00044-013-0809-8
TCMC1788
TCMT1455 Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC: 100 (ug/ml), Ref: 24103427
TCMC732
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 9 (ug/ml), Ref: 9748372
TCMC1203
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 22.6 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC1955
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 4.17 (ug/ml), Ref: 24549242
TCMC2644
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1356
TCMT1215 Pseudomonas aeruginosa PAO1 Pseudomonas aeruginosa PAO1 MIC: 32 (ug/ml), Ref: 21534606
TCMC1356
TCMT1208 Escherichia coli K12 Escherichia coli K-12 MIC: 16 (ug/ml), Ref: 21534606
TCMC912
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 6.21 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2228
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 18 (ug/ml), Ref: 18597896
TCMC2228
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 9 (ug/ml), Ref: 18597896
TCMC2228
TCMT1246 Escherichia coli Escherichia coli MIC: 16 (ug/ml), Ref: 18597896
TCMC2228
TCMT1251 Candida albicans Candida albicans MIC: 11 (ug/ml), Ref: 18597896
TCMC2671
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC2671
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 50 (ug/ml), Ref: 10.1021/np50124a013
TCMC1578
TCMT1408 Colletotrichum gloeosporioides Colletotrichum gloeosporioides IC50: 0.09 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1578
TCMT1245 Phytophthora cactorum Phytophthora cactorum IC50: 0.052 (ug/ml), Ref: 10.1016/j.cropro.2009.12.007
TCMC1123
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 50 (ug/ml), Ref: 12762812
TCMC1123
TCMT1442 Leishmania donovani Leishmania donovani IC50: 25 (ug/ml), Ref: 15679330
TCMC785
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.36 (ug/ml), Ref: 10.1016/S0960-894X(00)80357-1
IC50: 0.141 (ug/ml), Ref: 3286870
IC50: 0.148 (ug/ml), Ref: 3286870
TCMC785
TCMT1246 Escherichia coli Escherichia coli MIC: 5 (ug/ml), Ref: 16359864
MIC: 31.25 (ug/ml), Ref: 18591276
TCMC785
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans MIC: 64 (ug/ml), Ref: 16730982
MIC: 31.3 (ug/ml), Ref: 16872133
TCMC785
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 100 (ug/ml), Ref: 17716892
MIC: 50 (ug/ml), Ref: 9784149
MIC: 60 (ug/ml), Ref: 15568768
MBC: 64 (ug/ml), Ref: 10.1007/s00044-013-0844-5
MIC: 32 (ug/ml), Ref: 10.1007/s00044-013-0844-5
TCMC785
TCMT1226 Klebsiella pneumoniae Klebsiella pneumoniae MIC: 100 (ug/ml), Ref: 9784149
TCMC785
TCMT1439 Mycobacterium smegmatis Mycobacterium smegmatis MIC: 25 (ug/ml), Ref: 9784149
TCMC785
TCMT1251 Candida albicans Candida albicans MIC: 100 (ug/ml), Ref: 9784149
MIC: 31.3 (ug/ml), Ref: 16872133
MIC: 15.6 (ug/ml), Ref: 16872133
TCMC785
TCMT1385 Candida shehatae Candida shehatae MIC: 7.8 (ug/ml), Ref: 16872133
TCMC1776
TCMT1253 Penicillium chrysogenum Penicillium chrysogenum MIC: 100 (ug/ml), Ref: 10.1021/np50124a013
TCMC897
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 6.25 (ug/ml), Ref: 12762812
TCMC1491
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 0.92 (ug/ml), Ref: 21334901
TCMC1491
TCMT1318 Human T-lymphotropic virus 1 Human T-lymphotropic virus 1 IC50: 1.07 (ug/ml), Ref: 21334901
TCMC1828
TCMT1438 Plasmodium falciparum Plasmodium falciparum IC50: 0.281 (ug/ml), Ref: 3286870
IC50: 0.163 (ug/ml), Ref: 3286870
TCMC1792
TCMT1227 Streptococcus Streptococcus MIC: 25 (ug/ml), Ref: 9182126
TCMC710
TCMT1246 Escherichia coli Escherichia coli MIC: 7.8 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1412 Salmonella typhimurium Salmonella enterica subsp. enterica serovar Typhimurium MIC: 15.6 (ug/ml), Ref: 10.1016/S0960-894X(01)80881-7
TCMC710
TCMT1458 Filobasidiella neoformans Cryptococcus neoformans IC50: 20 (ug/ml), Ref: 12502337
TCMC710
TCMT1251 Candida albicans Candida albicans MIC: 3 (ug/ml), Ref: 10395518
TCMC710
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 12.7 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC710
TCMT1346 Helicobacter pylori Helicobacter pylori MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1349 Helicobacter pylori SS1 Helicobacter pylori SS1 MIC: 25 (ug/ml), Ref: 10.1007/s00044-012-0207-7
TCMC710
TCMT1442 Leishmania donovani Leishmania donovani IC50: 1.9 (ug/ml), Ref: 10.1039/C5MD00481K
TCMC1738
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 50 (ug/ml), Ref: 10.1016/S0960-894X(00)80336-4
TCMC1064
TCMT1218 Staphylococcus aureus Staphylococcus aureus MIC: 15 (ug/ml), Ref: 11170636
TCMC784
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 1 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2808
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 27 (ug/ml), Ref: 10425115
TCMC2811
TCMT1465 Entamoeba histolytica Entamoeba histolytica IC50: 37.35 (ug/ml), Ref: 10.1007/s00044-011-9767-1
TCMC2815
TCMT1454 Bacillus subtilis Bacillus subtilis MIC: 50 (ug/ml), Ref: 1517735
TCMC2821
TCMT1251 Candida albicans Candida albicans MIC: 1.56 (ug/ml), Ref: 7760078
MFC: 3.12 (ug/ml), Ref: 7760078
MFC: 6.25 (ug/ml), Ref: 7760078
MIC: 3.125 (ug/ml), Ref: 10346966
MFC: 6.25 (ug/ml), Ref: 10346966
MIC: 6.25 (ug/ml), Ref: 18611050
MIC: 6.25 (ug/ml), Ref: 21131198
TCMC2822
TCMT1463 Mycobacterium tuberculosis Mycobacterium tuberculosis MIC: 6.25 (ug/ml), Ref: 17845001
TCMC1113
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 16 (nM), Ref: 17263522
TCMC1982
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 22 (nM), Ref: 17263522
TCMC1117
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 17.56 (nM), Ref: 17263522
TCMC1118
TCMT1093 Enoyl-acyl-carrier protein reductase Plasmodium falciparum Ki: 79 (nM), Ref: 17263522
Ki: 8 (nM), Ref: 17263522
TCMC2333
TCMT1175 Human immunodeficiency virus Human immunodeficiency virus IC50: 11 (nM), Ref: 9834179
TCMC962
TCMT1221 Human herpesvirus 4 Human herpesvirus 4 IC50: 10.2 (nM), Ref: 17503850
TCMC962
TCMT1255 Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50: 37 (nM), Ref: 20034711
TCMC962
TCMT1313 Human immunodeficiency virus 2 Human immunodeficiency virus type 2 (ISOLATE ROD) IC50: 37 (nM), Ref: 20034711
TCMC1047
TCMT1464 Hepatitis B virus Hepatitis B virus IC50: 50 (nM), Ref: 24549242
TCMC1919
TCMT1247 Human herpesvirus 1 Human herpesvirus 1 MIC: 10 (nM), Ref: 11311065
IC50: 50 (nM), Ref: 9834179
TCMC1919
TCMT1180 Human herpesvirus 2 Human herpesvirus 2 MIC: 10 (nM), Ref: 11311065
TCMC1919
TCMT1250 Vesicular stomatitis virus Vesicular stomatitis virus IC50: 100 (nM), Ref: 9834179
TCMC1118
TCMT1222 Plasmodium falciparum D6 Plasmodium falciparum D6 IC50: 73 (nM), Ref: 25488841