Ingredient ID & Structure | Target ID | Target Name | Target Organism | Activity Records & Reference |
---|---|---|---|---|
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 270 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 270 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 750 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 2200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 9430 (nM), Ref: 20185318 Ki: 9430 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9780 (nM), Ref: 20185318 Ki: 9780 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7410 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8450 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7040 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2400 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2890 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 8710 (nM), Ref: 22892213 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4050 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 960 (nM), Ref: 22892213 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 3920 (nM), Ref: 15658857 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2330 (nM), Ref: 22245047 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 3630 (nM), Ref: 22245047 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 IC50: 1000 (nM), Ref: 25461324 IC50: 1000 (nM), Ref: 25461324 Ki: 9300 (nM), Ref: 27460668 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 1000 (nM), Ref: 20471252 Ki: 6800 (nM), Ref: 27460668 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 10000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 7900 (nM), Ref: 15916432 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 8300 (nM), Ref: 15658857 IC50: 8298.51 (nM), Ref: 19110342 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 3100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 1600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
Ki: 2200 (nM), Ref: 21511472 IC50: 3400 (nM), Ref: 21511472 |
|
TCMT132 | Butyrylcholinesterase | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
Ki: 3100 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 36 (nM), Ref: 16005223 Ki: 3.3 (nM), Ref: 17531479 Ki: 36 (nM), Ref: 17919913 Ki: 41 (nM), Ref: 18522867 Ki: 36 (nM), Ref: 20621488 Ki: 36 (nM), Ref: 20943404 IC50: 9.5 (nM), Ref: 21999614 Ki: 24 (nM), Ref: 22284817 Ki: 36 (nM), Ref: 22341572 Ki: 71.6 (nM), Ref: 23679955 Ki: 71.6 (nM), Ref: 10.1039/C3MD00394A Ki: 36.4 (nM), Ref: 23865723 Ki: 46 (nM), Ref: 25072877 Ki: 42 (nM), Ref: 26000707 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 17 (nM), Ref: 17531479 Ki: 2.9 (nM), Ref: 18522867 IC50: 2.8 (nM), Ref: 21999614 Ki: 10 (nM), Ref: 22284817 Ki: 3.88 (nM), Ref: 23679955 Ki: 3.88 (nM), Ref: 10.1039/C3MD00394A Ki: 40.7 (nM), Ref: 23865723 Ki: 22 (nM), Ref: 25072877 Ki: 18 (nM), Ref: 26000707 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
IC50: 3270 (nM), Ref: 21902175 Ki: 750 (nM), Ref: 21902175 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
IC50: 710 (nM), Ref: 21902175 Ki: 180 (nM), Ref: 21902175 |
|
TCMT327 | Vanilloid receptor | Homo sapiens |
IC50: 5700 (nM), Ref: 21902175 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9920 (nM), Ref: 18501600 Ki: 9900 (nM), Ref: 18579385 Ki: 9900 (nM), Ref: 26520662 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 7120 (nM), Ref: 18501600 Ki: 7100 (nM), Ref: 18579385 Ki: 7100 (nM), Ref: 26520662 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8800 (nM), Ref: 18579385 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9200 (nM), Ref: 20185318 Ki: 9200 (nM), Ref: 20590092 Ki: 9200 (nM), Ref: 20674354 Ki: 9200 (nM), Ref: 21282059 Ki: 9200 (nM), Ref: 23265898 Ki: 9200 (nM), Ref: 23010455 Ki: 9200 (nM), Ref: 24189056 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 8800 (nM), Ref: 20185318 Ki: 8800 (nM), Ref: 20590092 Ki: 8800 (nM), Ref: 20674354 Ki: 8800 (nM), Ref: 21282059 Ki: 8800 (nM), Ref: 23265898 Ki: 8800 (nM), Ref: 23010455 Ki: 8800 (nM), Ref: 24189056 Ki: 8800 (nM), Ref: 26520662 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9500 (nM), Ref: 20185318 Ki: 9500 (nM), Ref: 20590092 Ki: 9500 (nM), Ref: 20674354 Ki: 9500 (nM), Ref: 23010455 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 2700 (nM), Ref: 20185318 Ki: 2700 (nM), Ref: 20590092 Ki: 2700 (nM), Ref: 20674354 Ki: 2700 (nM), Ref: 23010455 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 5500 (nM), Ref: 20185318 Ki: 5500 (nM), Ref: 20590092 Ki: 5500 (nM), Ref: 20674354 Ki: 5500 (nM), Ref: 21282059 Ki: 5500 (nM), Ref: 21332115 Ki: 5500 (nM), Ref: 23265898 Ki: 5500 (nM), Ref: 23265903 Ki: 5500 (nM), Ref: 23010455 Ki: 5500 (nM), Ref: 24189056 Ki: 5500 (nM), Ref: 26073005 Ki: 5500 (nM), Ref: 26520662 |
|
TCMT560 | Coagulation factor X | Homo sapiens |
IC50: 170 (nM), Ref: 9834152 Ki: 570 (nM), Ref: 9834152 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3760 (nM), Ref: 24835197 Ki: 5130 (nM), Ref: 24835197 |
|
TCMT240 | Salivary alpha-amylase | Homo sapiens |
IC50: 2350 (nM), Ref: 26395057 Ki: 2600 (nM), Ref: 26395057 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2940 (nM), Ref: 19231207 |
|
TCMT690 | Histone deacetylase 3 | Homo sapiens |
IC50: 9000 (nM), Ref: 21874153 |
|
TCMT597 | Solute carrier family 28 member 3 | Homo sapiens |
Ki: 2100 (nM), Ref: 23388705 IC50: 3300 (nM), Ref: 23388705 |
|
TCMT709 | Sodium/nucleoside cotransporter 2 | Homo sapiens |
Ki: 5300 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT710 | Sodium/nucleoside cotransporter 1 | Homo sapiens |
Ki: 1800 (nM), Ref: 23388705 IC50: 5500 (nM), Ref: 23388705 |
|
TCMT296 | Adenosine A1 receptor | Homo sapiens |
IC50: 2.344 (nM), Ref: 26756468 |
|
TCMT112 | Adenosine A3 receptor | Homo sapiens |
IC50: 1.148 (nM), Ref: 26756468 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 1080 (nM), Ref: 21282059 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 470 (nM), Ref: 21282059 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 4450 (nM), Ref: 21282059 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4090 (nM), Ref: 21282059 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 4720 (nM), Ref: 21669522 Ki: 4720 (nM), Ref: 22687439 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 2450 (nM), Ref: 22687439 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 690 (nM), Ref: 22668600 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 7870 (nM), Ref: 22668600 |
|
TCMT82 | Estrogen receptor alpha | Homo sapiens |
Ki: 785 (nM), Ref: 15634023 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
IC50: 2840 (nM), Ref: 16814546 IC50: 4120 (nM), Ref: 18063374 IC50: 625 (nM), Ref: |
|
TCMT30 | Cyclooxygenase-2 | Homo sapiens |
IC50: 996 (nM), Ref: 17604631 IC50: 750 (nM), Ref: 20527891 IC50: 996 (nM), Ref: 26850006 |
|
TCMT329 | Quinone reductase 2 | Homo sapiens |
IC50: 960 (nM), Ref: 19265439 IC50: 450 (nM), Ref: 20036559 IC50: 450 (nM), Ref: 20356739 IC50: 960 (nM), Ref: 21261296 IC50: 6900 (nM), Ref: 23953689 Ki: 88 (nM), Ref: 23953689 IC50: 1400 (nM), Ref: 26854376 IC50: 913 (nM), Ref: 26854376 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2210 (nM), Ref: 20674354 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2770 (nM), Ref: 20674354 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 9090 (nM), Ref: 20674354 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 4470 (nM), Ref: 20674354 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4750 (nM), Ref: 20674354 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 4640 (nM), Ref: 20674354 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 8070 (nM), Ref: 20674354 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4350 (nM), Ref: 20674354 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 810 (nM), Ref: 20674354 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 950 (nM), Ref: 20674354 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4090 (nM), Ref: 20674354 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 830 (nM), Ref: 20674354 |
|
TCMT729 | PI3-kinase p110-alpha subunit | Homo sapiens |
IC50: 250 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT730 | PI3-kinase p110-beta subunit | Homo sapiens |
IC50: 500 (nM), Ref: 10.1039/C2MD20044A |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 4100 (nM), Ref: 27190601 IC50: 2600 (nM), Ref: 27190601 |
|
TCMT161 | Hydroxycarboxylic acid receptor 2 | Homo sapiens |
IC50: 140 (nM), Ref: 17994679 IC50: 140 (nM), Ref: 18029181 Ki: 50 (nM), Ref: 18665582 IC50: 150 (nM), Ref: 18752940 IC50: 140 (nM), Ref: 19307116 IC50: 130 (nM), Ref: 18760600 IC50: 140 (nM), Ref: 19309152 IC50: 140 (nM), Ref: 19592242 IC50: 140 (nM), Ref: 19592242 Ki: 82 (nM), Ref: 20184326 Ki: 104 (nM), Ref: 20184326 IC50: 140 (nM), Ref: 20444602 IC50: 140 (nM), Ref: 20615702 IC50: 249 (nM), Ref: 25737085 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 7500 (nM), Ref: 16610779 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 40 (nM), Ref: 19414254 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2320 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2180 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 7590 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7060 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6320 (nM), Ref: 20185318 Ki: 8790 (nM), Ref: 22892213 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 9370 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8910 (nM), Ref: 20185318 |
|
TCMT753 | Mothers against decapentaplegic homolog 3 | Homo sapiens | IC50: 142 (nM), Ref: |
|
TCMT721 | Heat shock 70 kDa protein 1 | Homo sapiens | IC50: 760 (nM), Ref: |
|
TCMT189 | Dual specificity protein phosphatase 3 | Homo sapiens | IC50: 1230 (nM), Ref: IC50: 980 (nM), Ref: |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 200 (nM), Ref: 22261024 |
|
TCMT479 | Serine/threonine-protein kinase AKT | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT436 | NUAK family SNF1-like kinase 1 | Homo sapiens |
IC50: 510 (nM), Ref: 22377675 |
|
TCMT354 | Serine/threonine-protein kinase Aurora-A | Homo sapiens |
IC50: 2480 (nM), Ref: 22377675 |
|
TCMT374 | Serine/threonine-protein kinase Aurora-B | Homo sapiens |
IC50: 2500 (nM), Ref: 22377675 |
|
TCMT626 | Serine/threonine-protein kinase B-raf | Homo sapiens |
IC50: 1760 (nM), Ref: 22377675 |
|
TCMT423 | Epidermal growth factor receptor erbB1 | Homo sapiens |
IC50: 690 (nM), Ref: 22377675 |
|
TCMT418 | Ephrin type-B receptor 4 | Homo sapiens |
IC50: 1830 (nM), Ref: 22377675 |
|
TCMT704 | Receptor protein-tyrosine kinase erbB-2 | Homo sapiens |
IC50: 3540 (nM), Ref: 22377675 |
|
TCMT441 | Focal adhesion kinase 1 | Homo sapiens |
IC50: 3110 (nM), Ref: 22377675 |
|
TCMT369 | Insulin-like growth factor I receptor | Homo sapiens |
IC50: 250 (nM), Ref: 22377675 |
|
TCMT212 | Tyrosine-protein kinase SRC | Homo sapiens |
IC50: 800 (nM), Ref: 22377675 |
|
TCMT370 | Vascular endothelial growth factor receptor 2 | Homo sapiens |
IC50: 790 (nM), Ref: 22377675 |
|
TCMT457 | Vascular endothelial growth factor receptor 3 | Homo sapiens |
IC50: 1540 (nM), Ref: 22377675 |
|
TCMT377 | Insulin receptor | Homo sapiens |
IC50: 340 (nM), Ref: 22377675 |
|
TCMT401 | Hepatocyte growth factor receptor | Homo sapiens |
IC50: 580 (nM), Ref: 22377675 |
|
TCMT536 | Platelet-derived growth factor receptor beta | Homo sapiens |
IC50: 1300 (nM), Ref: 22377675 |
|
TCMT484 | Serine/threonine-protein kinase PLK1 | Homo sapiens |
IC50: 3340 (nM), Ref: 22377675 |
|
TCMT755 | Serine/threonine-protein kinase PLK4 | Homo sapiens |
IC50: 2970 (nM), Ref: 22377675 |
|
TCMT502 | Tyrosine-protein kinase TIE-2 | Homo sapiens |
IC50: 260 (nM), Ref: 22377675 |
|
TCMT756 | Mitogen-activated protein kinase kinase kinase 8 | Homo sapiens |
IC50: 2370 (nM), Ref: 22377675 |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 100 (nM), Ref: 24900447 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8150 (nM), Ref: 22892213 |
|
TCMT225 | Carbonic anhydrase XIII | Homo sapiens |
Ki: 4240 (nM), Ref: 22892213 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3900 (nM), Ref: 24835197 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 3100 (nM), Ref: 24835197 Ki: 6840 (nM), Ref: 24835197 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
IC50: 3310 (nM), Ref: 21902175 Ki: 760 (nM), Ref: 21902175 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
IC50: 3460 (nM), Ref: 21902175 Ki: 880 (nM), Ref: 21902175 |
|
TCMT327 | Vanilloid receptor | Homo sapiens |
IC50: 2600 (nM), Ref: 21902175 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 810 (nM), Ref: 26498394 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 670 (nM), Ref: 26498394 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 770 (nM), Ref: 26498394 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 620 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 810 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 8470 (nM), Ref: 26498394 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 720 (nM), Ref: 26498394 |
|
TCMT807 | Solute carrier family 22 member 12 | Homo sapiens |
IC50: 2000 (nM), Ref: 17325024 Ki: 5740 (nM), Ref: 17325024 |
|
TCMT236 | Estrogen receptor beta | Homo sapiens | IC50: 2927.18 (nM), Ref: |
|
TCMT61 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | IC50: 2988.26 (nM), Ref: |
|
TCMT739 | G-protein coupled receptor 35 | Homo sapiens |
IC50: 1600 (nM), Ref: 24900447 |
|
TCMT261 | Death-associated protein kinase 1 | Homo sapiens |
IC50: 1600 (nM), Ref: 26322379 |
|
TCMT283 | Receptor-type tyrosine-protein phosphatase S | Homo sapiens |
IC50: 4300 (nM), Ref: 26602279 |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
IC50: 930 (nM), Ref: 15357969 |
|
TCMT298 | Fatty acid binding protein muscle | Homo sapiens |
IC50: 2600 (nM), Ref: 15357969 |
|
TCMT808 | Fatty acid binding protein epidermal | Homo sapiens |
IC50: 1200 (nM), Ref: 15357969 |
|
TCMT809 | Fatty acid binding protein intestinal | Homo sapiens |
IC50: 1700 (nM), Ref: 15357969 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 7400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 7030 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 6990 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6070 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 6130 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9970 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 9800 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 7490 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 2250 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 3200 (nM), Ref: 20185318 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 60 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT614 | Egl nine homolog 1 | Homo sapiens |
IC50: 3000 (nM), Ref: 18942826 |
|
TCMT3 | Arachidonate 15-lipoxygenase | Homo sapiens |
Ki: 600 (nM), Ref: 21739938 |
|
TCMT81 | Arachidonate 12-lipoxygenase | Homo sapiens |
Ki: 1600 (nM), Ref: 21739938 |
|
TCMT8 | Lysine-specific demethylase 4D-like | Homo sapiens |
IC50: 3000 (nM), Ref: 10.1039/C1MD00199J |
|
TCMT162 | UDP-glucuronosyltransferase 1-1 | Homo sapiens |
IC50: 4400 (nM), Ref: 21030469 IC50: 7000 (nM), Ref: 21030469 |
|
TCMT384 | G protein-coupled receptor kinase 6 | Homo sapiens | IC50: 8700 (nM), Ref: |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 482 (nM), Ref: 21067924 Ki: 478 (nM), Ref: 22077347 Ki: 480 (nM), Ref: 26688270 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 754 (nM), Ref: 22077347 Ki: 750 (nM), Ref: 26688270 |
|
TCMT117 | Kappa opioid receptor | Homo sapiens |
Ki: 2515 (nM), Ref: 18166466 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9800 (nM), Ref: 18501600 Ki: 9800 (nM), Ref: 18579385 Ki: 920 (nM), Ref: 20185318 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 4800 (nM), Ref: 18579385 Ki: 6270 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 9200 (nM), Ref: 18579385 Ki: 3670 (nM), Ref: 20185318 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 6160 (nM), Ref: 20185318 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 3730 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4080 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 5700 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 7130 (nM), Ref: 20185318 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 7780 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 6610 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 870 (nM), Ref: 20185318 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 2000 (nM), Ref: 19414254 |
|
TCMT239 | Serine/threonine-protein kinase PIM1 | Homo sapiens |
IC50: 2500 (nM), Ref: 27173800 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 600 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 5300 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 4100 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT126 | Telomerase reverse transcriptase | Homo sapiens |
IC50: 8600 (nM), Ref: 10.1039/C0MD00241K |
|
TCMT297 | Fatty acid binding protein adipocyte | Homo sapiens |
Ki: 1500 (nM), Ref: 27460668 |
|
TCMT822 | Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens |
IC50: 8000 (nM), Ref: 10.1039/C4MD00086B |
|
TCMT44 | Glyoxalase I | Homo sapiens |
IC50: 7700 (nM), Ref: 18258440 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 3370 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 1249 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 79 (nM), Ref: 20696580 |
|
TCMT83 | Lymphocyte differentiation antigen CD38 | Homo sapiens |
IC50: 8200 (nM), Ref: 21641214 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 3610 (nM), Ref: 22658537 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 5620 (nM), Ref: 22658537 |
|
TCMT734 | Matrix metalloproteinase 12 | Homo sapiens |
IC50: 980 (nM), Ref: 22658537 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1500 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 830 (nM), Ref: 23411073 |
|
TCMT127 | Poly [ADP-ribose] polymerase-1 | Homo sapiens |
IC50: 4265.8 (nM), Ref: 23574272 IC50: 4200 (nM), Ref: 23574272 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 1071.52 (nM), Ref: 23574272 IC50: 1100 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 2398.83 (nM), Ref: 23574272 IC50: 2400 (nM), Ref: 23574272 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 600 (nM), Ref: 23683835 IC50: 3200 (nM), Ref: 26529431 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 1600 (nM), Ref: 24368208 |
|
TCMT45 | Beta amyloid A4 protein | Homo sapiens |
IC50: 6400 (nM), Ref: 24878198 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 2900 (nM), Ref: 25019478 IC50: 7800 (nM), Ref: 26096677 |
|
TCMT100 | Transthyretin | Homo sapiens |
IC50: 7000 (nM), Ref: 26214366 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 3691.6 (nM), Ref: 26498393 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 4.7 (nM), Ref: 26498393 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 60.3 (nM), Ref: 26498393 |
|
TCMT142 | Carbonic anhydrase IV | Homo sapiens |
Ki: 293 (nM), Ref: 26498393 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 9200 (nM), Ref: 26529431 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
IC50: 2400 (nM), Ref: 15658857 IC50: 2398.83 (nM), Ref: 19110342 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 7410 (nM), Ref: 21669522 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 540 (nM), Ref: 21669522 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 520 (nM), Ref: 21669522 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 1900 (nM), Ref: 16248836 Ki: 1900 (nM), Ref: 16248836 Ki: 800 (nM), Ref: 16248836 Ki: 250 (nM), Ref: 22696418 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 760 (nM), Ref: 23746477 |
|
TCMT268 | Cytochrome P450 2A13 | Homo sapiens |
Ki: 40 (nM), Ref: 22696418 |
|
TCMT292 | Muscarinic acetylcholine receptor M1 | Homo sapiens |
Ki: 56 (nM), Ref: 10891110 |
|
TCMT293 | Muscarinic acetylcholine receptor M2 | Homo sapiens |
Ki: 25 (nM), Ref: 10891110 Ki: 72 (nM), Ref: 10891110 Ki: 75 (nM), Ref: 9622546 IC50: 449 (nM), Ref: 9622546 IC50: 3900 (nM), Ref: 9622546 Ki: 489.78 (nM), Ref: 18182302 |
|
TCMT551 | Muscarinic acetylcholine receptor M4 | Homo sapiens |
Ki: 1400 (nM), Ref: 10891110 Ki: 23 (nM), Ref: 10891110 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1200 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1200 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6000 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT164 | Cyclooxygenase-1 | Homo sapiens |
Ki: 4000 (nM), Ref: 24088053 |
|
TCMT135 | Carbonic anhydrase XIV | Homo sapiens |
Ki: 8710 (nM), Ref: 20185318 Ki: 8710 (nM), Ref: 26498394 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 9060 (nM), Ref: 20185318 Ki: 9060 (nM), Ref: 26498394 |
|
TCMT137 | Carbonic anhydrase IX | Homo sapiens |
Ki: 7870 (nM), Ref: 20185318 |
|
TCMT138 | Carbonic anhydrase VII | Homo sapiens |
Ki: 6420 (nM), Ref: 20185318 |
|
TCMT139 | Carbonic anhydrase VI | Homo sapiens |
Ki: 7330 (nM), Ref: 20185318 |
|
TCMT140 | Carbonic anhydrase VB | Homo sapiens |
Ki: 9080 (nM), Ref: 20185318 |
|
TCMT141 | Carbonic anhydrase VA | Homo sapiens |
Ki: 6490 (nM), Ref: 20185318 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 10000 (nM), Ref: 20185318 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 1610 (nM), Ref: 20185318 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 2380 (nM), Ref: 20185318 |
|
TCMT101 | Protein-tyrosine phosphatase 1B | Homo sapiens |
IC50: 3060 (nM), Ref: 19476336 |
|
TCMT321 | Matrix metalloproteinase 9 | Homo sapiens |
IC50: 21.22 (nM), Ref: 23375794 IC50: 10 (nM), Ref: 23375794 |
|
TCMT306 | Matrix metalloproteinase-2 | Homo sapiens |
IC50: 24.26 (nM), Ref: 23375794 |
|
TCMT295 | Matrix metalloproteinase-1 | Homo sapiens |
IC50: 238.91 (nM), Ref: 23375794 |
|
TCMT130 | Arachidonate 5-lipoxygenase | Homo sapiens |
IC50: 8500 (nM), Ref: 26197161 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 10000 (nM), Ref: 20218623 Ki: 2860 (nM), Ref: 23865723 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 2400 (nM), Ref: 20218623 Ki: 4350 (nM), Ref: 23865723 |
|
TCMT810 | Toll-like receptor 2 | Homo sapiens |
IC50: 5000 (nM), Ref: 16509590 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 5400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT223 | Aldose reductase | Homo sapiens |
IC50: 300 (nM), Ref: 22236472 IC50: 1800 (nM), Ref: 22261024 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
IC50: 7900 (nM), Ref: 22236472 |
|
TCMT63 | Peroxisome proliferator-activated receptor alpha | Homo sapiens |
IC50: 1700 (nM), Ref: 10.1007/s00044-008-9102-7 IC50: 1700 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT64 | Peroxisome proliferator-activated receptor delta | Homo sapiens |
IC50: 9600 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT67 | Peroxisome proliferator-activated receptor gamma | Homo sapiens |
IC50: 6400 (nM), Ref: 10.1007/s00044-012-0285-6 |
|
TCMT314 | Serotonin 2c (5-HT2c) receptor | Homo sapiens |
Ki: 10 (nM), Ref: 24491146 |
|
TCMT207 | Beta-secretase 1 | Homo sapiens |
IC50: 2400 (nM), Ref: 14592472 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 30 (nM), Ref: 25282650 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 3274 (nM), Ref: 25282650 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 3219 (nM), Ref: 25218910 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 88 (nM), Ref: 25218910 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 912 (nM), Ref: 25173852 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 2143 (nM), Ref: 25218910 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 129 (nM), Ref: 25218910 |
|
TCMT114 | Cannabinoid CB2 receptor | Homo sapiens |
Ki: 335 (nM), Ref: 25218910 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 224 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 117 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 5668 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 47 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 65 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 1906 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 830 (nM), Ref: 19969457 |
|
TCMT115 | Cannabinoid CB1 receptor | Homo sapiens |
Ki: 31 (nM), Ref: 19969457 |
|
TCMT249 | Cyclin-dependent kinase 6 | Homo sapiens |
IC50: 1700 (nM), Ref: 15689157 IC50: 1700 (nM), Ref: 10.1007/s00044-009-9233-5 |
|
TCMT156 | Cytochrome P450 19A1 | Homo sapiens |
IC50: 10000 (nM), Ref: 18192087 IC50: 900 (nM), Ref: 20413308 IC50: 1200 (nM), Ref: 26301554 |
|
TCMT65 | Estradiol 17-beta-dehydrogenase 1 | Homo sapiens |
IC50: 710 (nM), Ref: 18533708 |
|
TCMT752 | Casein kinase II alpha | Homo sapiens |
IC50: 800 (nM), Ref: 19414254 |
|
TCMT187 | Androgen Receptor | Homo sapiens |
IC50: 5200 (nM), Ref: 19592245 |
|
TCMT219 | Cytochrome P450 1A2 | Homo sapiens |
IC50: 795 (nM), Ref: 20696580 |
|
TCMT215 | Cytochrome P450 1A1 | Homo sapiens |
IC50: 427 (nM), Ref: 20696580 |
|
TCMT257 | Cytochrome P450 1B1 | Homo sapiens |
IC50: 25 (nM), Ref: 20696580 |
|
TCMT265 | Glycogen synthase kinase-3 beta | Homo sapiens |
IC50: 1900 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 12 (nM), Ref: 10.1007/s00044-012-0353-y |
|
TCMT260 | Tyrosine-protein kinase receptor FLT3 | Homo sapiens |
IC50: 1450 (nM), Ref: 23411073 |
|
TCMT128 | Tankyrase-2 | Homo sapiens |
IC50: 2951.21 (nM), Ref: 23574272 IC50: 2900 (nM), Ref: 23574272 |
|
TCMT129 | Tankyrase-1 | Homo sapiens |
IC50: 3162.28 (nM), Ref: 23574272 IC50: 3100 (nM), Ref: 23574272 |
|
TCMT592 | Xanthine dehydrogenase | Homo sapiens |
Ki: 520 (nM), Ref: 25019478 IC50: 3200 (nM), Ref: 26022844 |
|
TCMT280 | Aldo-keto reductase family 1 member B10 | Homo sapiens |
Ki: 6000 (nM), Ref: 26529431 IC50: 6600 (nM), Ref: 26529431 |
|
TCMT206 | Cytochrome P450 2A6 | Homo sapiens |
Ki: 600 (nM), Ref: 16248836 |
|
TCMT131 | Acetylcholinesterase | Homo sapiens |
IC50: 6480 (nM), Ref: 23746477 |
|
TCMT133 | Carbonic anhydrase I | Homo sapiens |
Ki: 9060 (nM), Ref: 21402476 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 8030 (nM), Ref: 21402476 |
|
TCMT588 | D-amino-acid oxidase | Homo sapiens |
Ki: 7000 (nM), Ref: 23391306 IC50: 2089.3 (nM), Ref: 23631755 Ki: 2000 (nM), Ref: 23631755 |
|
TCMT134 | Carbonic anhydrase II | Homo sapiens |
Ki: 90 (nM), Ref: 18501600 Ki: 90 (nM), Ref: 18579385 |
|
TCMT136 | Carbonic anhydrase XII | Homo sapiens |
Ki: 7800 (nM), Ref: 18579385 |
|
TCMT143 | Carbonic anhydrase III | Homo sapiens |
Ki: 8200 (nM), Ref: 18579385 |