Plant ingredients against the target with activities between 10uM and 50uM
Ingredient ID | Target (Gene Symbol) | No. of Activity Values | Activity Value (nM) | Activity Type | Activity Reference |
---|---|---|---|---|---|
NPC100551 | CA14 | 1 | 49800 | Ki |
PMID: 18579385 |
NPC100551 | ALDH1A1 | 2 |
Median: 39810.7 Range: 39810.7 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC100551 | SMN1;SMN2 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC100551 | KDM4E | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC100551 | HPGD | 2 |
Median: 29903.3 Range: 28183.8 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC1075 | CYP2C9 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC110899 | CA5B | 1 | 35400 | Ki |
PMID: 20185318 |
NPC116775 | BCHE | 1 | 43100 | Ki |
PMID: 19879672 |
NPC116775 | ALDH1A1 | 2 |
Median: 35716.75 Range: 31622.8 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | HPGD | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | CDK6 | 2 |
Median: 22000 Range: 22000 to 22000 |
IC50 |
PMID: 15689157 DOI: 10.1007/s00044-009-9233-5 |
NPC116775 | GLO1 | 1 | 20600 | IC50 |
PMID: 18258440 |
NPC116775 | KDM4E | 2 |
Median: 27829.8 Range: 15848.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | HSD17B10 | 2 |
Median: 15848.9 Range: 15848.9 to 15848.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC116775 | BACE1 | 1 | 14700 | IC50 |
DOI: 10.1007/s00044-012-0353-y |
NPC142415 | ACP1 | 4 |
Median: 22050 Range: 21200 to 22900 |
IC50 |
PMID: 21453996 PMID: 21453996 PMID: 25264584 PMID: 25264584 |
NPC142415 | PTPN6 | 2 |
Median: 22760 Range: 14190 to 31330 |
IC50 |
PMID: 18707891 PMID: 27123900 |
NPC156654 | L3MBTL1 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC156654 | KDM4E | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC156654 | POLB | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC173555 | GLA | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC176740 | MAPT | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC176740 | EPHX2 | 1 | 24300 | IC50 |
PMID: 24679441 |
NPC176740 | KDM4E | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CYP2C9 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CYP2C19 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | THRB | 2 |
Median: 32464.8 Range: 25118.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CARM1 | 1 | 25000 | IC50 |
DOI: 10.1039/C1MD00199J |
NPC178134 | GSR | 1 | 22800 | IC50 |
PMID: 19015351 |
NPC178134 | EPHX2 | 1 | 20700 | IC50 |
PMID: 24679441 |
NPC178134 | ATM | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | MAPK1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC181465 | XDH | 1 | 14800 | IC50 |
PMID: 9461655 |
NPC20791 | PMP22 | 1 | 47754.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | THRB | 1 | 44668.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | GALK1 | 1 | 42128.5 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CDK2 | 1 | 40000 | IC50 |
PMID: 17178224 |
NPC20791 | CD38 | 1 | 37900 | IC50 |
PMID: 21641214 |
NPC20791 | SORD | 2 |
Median: 106300 Range: 35600 to 177000 |
IC50 |
PMID: 8893834 PMID: 12672241 |
NPC20791 | SMN1;SMN2 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | EPHX2 | 1 | 33540 | IC50 |
PMID: 24679441 |
NPC20791 | DPP4 | 2 |
Median: 81365 Range: 32730 to 130000 |
IC50 |
PMID: 18650094 DOI: 10.1039/C0MD00245C |
NPC20791 | MAPK1 | 2 |
Median: 35716.75 Range: 31622.8 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | ADORA3 | 1 | 30000 | Ki |
PMID: 8576921 |
NPC20791 | PTGS2 | 1 | 28600 | IC50 |
PMID: 17378609 |
NPC20791 | BLM | 3 |
Median: 28183.8 Range: 28183.8 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | TDP1 | 2 |
Median: 26651.35 Range: 25118.9 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | ALDH1A1 | 6 |
Median: 37646 Range: 25118.9 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CDK6 | 2 |
Median: 25000 Range: 25000 to 25000 |
IC50 |
PMID: 15689157 DOI: 10.1007/s00044-009-9233-5 |
NPC20791 | PTPN1 | 2 |
Median: 23300 Range: 23300 to 23300 |
IC50 |
PMID: 12419367 PMID: 19297174 |
NPC20791 | KMT2A | 1 | 22387.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | AMY1A;AMY1B;AMY1C | 1 | 21400 | IC50 |
PMID: 18507367 |
NPC20791 | SYK | 1 | 20000 | IC50 |
PMID: 22257213 |
NPC20791 | HPGD | 2 |
Median: 21169.9 Range: 19952.6 to 22387.2 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | APEX1 | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | CYP2D6 | 1 | 18800 | IC50 |
PMID: 22328583 |
NPC20791 | USP2 | 2 |
Median: 25057.75 Range: 18492.7 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | GPR35 | 1 | 15400 | IC50 |
PMID: 24900447 |
NPC20791 | APP | 1 | 15300 | IC50 |
PMID: 26719209 |
NPC209970 | ALOX15 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC209970 | PPARG | 1 | 30000 | IC50 |
DOI: 10.1007/s00044-012-0285-6 |
NPC209970 | TDP1 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC209970 | HSD17B10 | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | HSD17B10 | 1 | 39810.7 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | PTGS1 | 2 |
Median: 58350 Range: 36700 to 80000 |
IC50 |
PMID: 11858749 PMID: 16038536 |
NPC219876 | SMN1;SMN2 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | NPSR1 | 1 | 31622.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | BLM | 2 |
Median: 28183.8 Range: 28183.8 to 28183.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | ALDH1A1 | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | RECQL | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | MAPT | 2 |
Median: 19952.6 Range: 19952.6 to 19952.6 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | APEX1 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | SELL | 1 | 27600 | IC50 |
PMID: 17302397 |
NPC225710 | GAPDH | 1 | 25118.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | MAPK1 | 2 |
Median: 23753.05 Range: 22387.2 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | SELP | 1 | 19100 | IC50 |
PMID: 17302397 |
NPC225710 | SMN1;SMN2 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC230301 | DPP4 | 1 | 28840 | IC50 |
DOI: 10.1039/C0MD00245C |
NPC230301 | POLB | 1 | 26300 | IC50 |
PMID: 14640519 |
NPC243728 | POLB | 1 | 26500 | IC50 |
PMID: 15165161 |
NPC294902 | HPGD | 3 |
Median: 39810.7 Range: 39810.7 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | ALDH1A1 | 2 |
Median: 39810.7 Range: 39810.7 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | APEX1 | 1 | 35481.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | APP | 1 | 32800 | IC50 |
PMID: 22921742 |
NPC294902 | AKR1B1 | 1 | 32000 | IC50 |
PMID: 22236472 |
NPC294902 | CYP3A4 | 2 |
Median: 25118.9 Range: 25118.9 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | POLB | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC51700 | PPARA | 1 | 41310 | EC50 |
PMID: 21855333 |
NPC51700 | AKR1B1 | 1 | 41000 | IC50 |
PMID: 21561086 |
NPC51700 | CYP19A1 | 1 | 32000 | IC50 |
PMID: 18192087 |
NPC51700 | PTPN6 | 1 | 25780 | IC50 |
PMID: 18707891 |
NPC51700 | POLB | 1 | 18600 | IC50 |
PMID: 15165161 |
NPC51700 | CTSD | 1 | 18200 | IC50 |
DOI: 10.1007/s00044-012-0397-z |
NPC51700 | SLCO1B1 | 1 | 15848.93 | IC50 |
PMID: 23571415 |
NPC61477 | HPGD | 1 | 19952.6 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | MAPK1 | 1 | 15848.9 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | RECQL | 2 |
Median: 77689.6 Range: 14125.4 to 141253.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC70744 | KDM4E | 1 | 28183.8 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC81010 | ESR1 | 1 | 16120 | EC50 |
PMID: 23608764 |
NPC84319 | PYGM | 1 | 28000 | IC50 |
PMID: 16169219 |
NPC84319 | PTPN2 | 1 | 19470 | IC50 |
PMID: 19846303 |
NPC100551 | CA6 | 2 |
Median: 1165950 Range: 11900 to 2320000 |
Ki |
PMID: 18579385 PMID: 21669522 |
NPC100551 | CA4 | 1 | 11100 | Ki |
PMID: 18579385 |
NPC1075 | KDM4E | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC110899 | CA4 | 1 | 10600 | Ki |
PMID: 20185318 |
NPC116775 | MAPT | 2 |
Median: 14219.1 Range: 12589.3 to 15848.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC142415 | PTPRF | 2 |
Median: 17055 Range: 11800 to 22310 |
IC50 |
PMID: 21453996 PMID: 27123900 |
NPC142415 | PTPN11 | 1 | 11620 | IC50 |
PMID: 27123900 |
NPC173555 | SLCO1B3 | 1 | 13182.57 | IC50 |
PMID: 23571415 |
NPC178134 | CA5B | 1 | 12700 | Ki |
PMID: 20185318 |
NPC178134 | MAPT | 8 |
Median: 21169.9 Range: 12589.3 to 39810.7 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | TP53 | 2 |
Median: 22106.05 Range: 12589.3 to 31622.8 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | KMT2A | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC178134 | CA3 | 1 | 10500 | Ki |
PMID: 20185318 |
NPC20791 | LMNA | 1 | 14125.4 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC20791 | PIK3CG | 1 | 13790 | IC50 |
PMID: 25050878 |
NPC20791 | PREP | 1 | 13000 | IC50 |
PMID: 18650094 |
NPC20791 | LCK | 2 |
Median: 13000 Range: 13000 to 13000 |
IC50 |
PMID: 1995903 PMID: 16441060 |
NPC20791 | CALM1;CALM2;CALM3 | 1 | 12970 | IC50 |
PMID: 21129983 |
NPC20791 | PLAU | 1 | 12100 | IC50 |
PMID: 24610996 |
NPC20791 | CA5B | 1 | 11900 | Ki |
PMID: 20185318 |
NPC20791 | CYP2C19 | 1 | 10500 | IC50 |
PMID: 22328583 |
NPC20791 | MMP12 | 1 | 10230 | IC50 |
PMID: 22658537 |
NPC20791 | HIF1AN | 1 | 10200 | IC50 |
PMID: 19822432 |
NPC20791 | CYP2C9 | 1 | 10200 | IC50 |
PMID: 22328583 |
NPC219876 | KDM4E | 2 |
Median: 19622.15 Range: 14125.4 to 25118.9 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC219876 | POLB | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC225710 | FUT4 | 1 | 14000 | IC50 |
DOI: 10.1039/C4MD00086B |
NPC294902 | THRB | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC294902 | CA4 | 1 | 10100 | Ki |
PMID: 20185318 |
NPC29883 | CA2 | 2 |
Median: 10600 Range: 10600 to 10600 |
Ki |
PMID: 18501600 PMID: 18579385 |
NPC51700 | SLCO1B3 | 1 | 11481.54 | IC50 |
PMID: 23571415 |
NPC61477 | MAPT | 2 |
Median: 14125.4 Range: 14125.4 to 14125.4 |
Potency |
PubChem BioAssay data set CHEMBL1201862 PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | ALOX15 | 1 | 12589.3 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | CA14 | 1 | 11550 | Ki |
PMID: 20674354 |
NPC61477 | KDM4E | 1 | 11220.2 | Potency |
PubChem BioAssay data set CHEMBL1201862 |
NPC61477 | CA13 | 1 | 10510 | Ki |
PMID: 20674354 |
NPC70744 | CA3 | 1 | 11100 | Ki |
PMID: 20185318 |
NPC70744 | CA4 | 1 | 10800 | Ki |
PMID: 20185318 |
NPC70744 | CA5B | 1 | 10500 | Ki |
PMID: 20185318 |
NPC81010 | HCAR2 | 1 | 14000 | Ki |
PMID: 21167710 |